Works matching AU Volcho, Konstantin


Results: 68
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    Structure-Based Design, Synthesis, and Biological Evaluation of the Cage–Amide Derived Orthopox Virus Replication Inhibitors.

    Published in:
    Viruses (1999-4915), 2023, v. 15, n. 1, p. 29, doi. 10.3390/v15010029
    By:
    • Mozhaitsev, Evgenii S.;
    • Suslov, Evgeniy V.;
    • Rastrepaeva, Daria A.;
    • Yarovaya, Olga I.;
    • Borisevich, Sophia S.;
    • Khamitov, Edward M.;
    • Kolybalov, Dmitry S.;
    • Arkhipov, Sergey G.;
    • Bormotov, Nikolai I.;
    • Shishkina, Larisa N.;
    • Serova, Olga A.;
    • Brunilin, Roman V.;
    • Vernigora, Andrey A.;
    • Nawrozkij, Maxim B.;
    • Agafonov, Alexander P.;
    • Maksyutov, Rinat A.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.
    Publication type:
    Article
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    Key Enzymes of the Serotonergic System – Tryptophan Hydroxylase 2 and Monoamine Oxidase A – In the Brain of Rats Selectively Bred for a Reaction toward Humans: Effects of Benzopentathiepin TC-2153.

    Published in:
    Biochemistry (00062979), 2024, v. 89, n. 6, p. 1109, doi. 10.1134/S0006297924060105
    By:
    • Moskaliuk, Vitalii S.;
    • Kozhemyakina, Rimma V.;
    • Khomenko, Tatyana M.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Kulikov, Alexander V.;
    • Naumenko, Vladimir S.;
    • Kulikova, Elizabeth A.
    Publication type:
    Article
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    Diverse Biological Activity of Benzofuroxan/Sterically Hindered Phenols Hybrids.

    Published in:
    Pharmaceuticals (14248247), 2023, v. 16, n. 4, p. 499, doi. 10.3390/ph16040499
    By:
    • Chugunova, Elena;
    • Gibadullina, Elmira;
    • Matylitsky, Kirill;
    • Bazarbayev, Baurat;
    • Neganova, Margarita;
    • Volcho, Konstantin;
    • Rogachev, Artem;
    • Akylbekov, Nurgali;
    • Nguyen, Hoang Bao Tran;
    • Voloshina, Alexandra;
    • Lyubina, Anna;
    • Amerhanova, Syumbelya;
    • Syakaev, Victor;
    • Burilov, Alexander;
    • Appazov, Nurbol;
    • Zhanakov, Mukhtar;
    • Kuhn, Leah;
    • Sinyashin, Oleg;
    • Alabugin, Igor
    Publication type:
    Article
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    Biotransformation of (–)-Isopulegol by Rhodococcus rhodochrous.

    Published in:
    Pharmaceuticals (14248247), 2022, v. 15, n. 8, p. 964, doi. 10.3390/ph15080964
    By:
    • Ivshina, Irina B.;
    • Luchnikova, Natalia A.;
    • Maltseva, Polina Yu.;
    • Ilyina, Irina V.;
    • Volcho, Konstantin P.;
    • Gatilov, Yurii V.;
    • Korchagina, Dina V.;
    • Kostrikina, Nadezhda A.;
    • Sorokin, Vladimir V.;
    • Mulyukin, Andrey L.;
    • Salakhutdinov, Nariman F.
    Publication type:
    Article
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    Rational Design of New Monoterpene-Containing Azoles and Their Antifungal Activity.

    Published in:
    Antibiotics (2079-6382), 2023, v. 12, n. 5, p. 818, doi. 10.3390/antibiotics12050818
    By:
    • Li-Zhulanov, Nikolai S.;
    • Zaikova, Nadezhda P.;
    • Sari, Suat;
    • Gülmez, Dolunay;
    • Sabuncuoğlu, Suna;
    • Ozadali-Sari, Keriman;
    • Arikan-Akdagli, Sevtap;
    • Nefedov, Andrey A.;
    • Rybalova, Tatyana V.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.
    Publication type:
    Article
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    MPTP-Treated Zebrafish Recapitulate 'Late-Stage' Parkinson's-like Cognitive Decline.

    Published in:
    Toxics, 2022, v. 10, n. 2, p. N.PAG, doi. 10.3390/toxics10020069
    By:
    • Bashirzade, Alim A. O.;
    • Cheresiz, Sergey V.;
    • Belova, Alisa S.;
    • Drobkov, Alexey V.;
    • Korotaeva, Anastasiia D.;
    • Azizi-Arani, Soheil;
    • Azimirad, Amirhossein;
    • Odle, Eric;
    • Gild, Emma-Yanina V.;
    • Ardashov, Oleg V.;
    • Volcho, Konstantin P.;
    • Bozhko, Dmitrii V.;
    • Myrov, Vladislav O.;
    • Kolchanova, Sofia M.;
    • Polovian, Aleksander I.;
    • Galumov, Georgii K.;
    • Salakhutdinov, Nariman F.;
    • Amstislavskaya, Tamara G.;
    • Kalueff, Allan V.
    Publication type:
    Article
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    Identification and Study of the Action Mechanism of Small Compound That Inhibits Replication of Respiratory Syncytial Virus.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 16, p. 12933, doi. 10.3390/ijms241612933
    By:
    • Shtro, Anna A.;
    • Klabukov, Artem M.;
    • Garshinina, Anzhelika V.;
    • Galochkina, Anastasia V.;
    • Nikolaeva, Yulia V.;
    • Khomenko, Tatyana M.;
    • Bobkov, Danila E.;
    • Lozhkov, Aleksey A.;
    • Sivak, Konstantin V.;
    • Yakovlev, Kirill S.;
    • Komissarov, Andrey B.;
    • Borisevich, Sophia S.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.
    Publication type:
    Article
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    Hybrids of Sterically Hindered Phenols and Diaryl Ureas: Synthesis, Switch from Antioxidant Activity to ROS Generation and Induction of Apoptosis.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 16, p. 12637, doi. 10.3390/ijms241612637
    By:
    • Gibadullina, Elmira;
    • Neganova, Margarita;
    • Aleksandrova, Yulia;
    • Nguyen, Hoang Bao Tran;
    • Voloshina, Alexandra;
    • Khrizanforov, Mikhail;
    • Nguyen, Thi Thu;
    • Vinyukova, Ekaterina;
    • Volcho, Konstantin;
    • Tsypyshev, Dmitry;
    • Lyubina, Anna;
    • Amerhanova, Syumbelya;
    • Strelnik, Anna;
    • Voronina, Julia;
    • Islamov, Daut;
    • Zhapparbergenov, Rakhmetulla;
    • Appazov, Nurbol;
    • Chabuka, Beauty;
    • Christopher, Kimberley;
    • Burilov, Alexander
    Publication type:
    Article
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    New 5-Hydroxycoumarin-Based Tyrosyl-DNA Phosphodiesterase I Inhibitors Sensitize Tumor Cell Line to Topotecan.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 11, p. 9155, doi. 10.3390/ijms24119155
    By:
    • Khomenko, Tatyana M.;
    • Zakharenko, Alexandra L.;
    • Kornienko, Tatyana E.;
    • Chepanova, Arina A.;
    • Dyrkheeva, Nadezhda S.;
    • Artemova, Anastasia O.;
    • Korchagina, Dina V.;
    • Achara, Chigozie;
    • Curtis, Anthony;
    • Reynisson, Jóhannes;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    Novel TDP1 Inhibitors: Disubstituted Thiazolidine-2,4-Diones Containing Monoterpene Moieties.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 4, p. 3834, doi. 10.3390/ijms24043834
    By:
    • Ivankin, Dmitry I.;
    • Kornienko, Tatyana E.;
    • Mikhailova, Marina A.;
    • Dyrkheeva, Nadezhda S.;
    • Zakharenko, Alexandra L.;
    • Achara, Chigozie;
    • Reynisson, Jóhannes;
    • Golyshev, Victor M.;
    • Luzina, Olga A.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    The First Berberine-Based Inhibitors of Tyrosyl-DNA Phosphodiesterase 1 (Tdp1), an Important DNA Repair Enzyme.

    Published in:
    International Journal of Molecular Sciences, 2020, v. 21, n. 19, p. 7162, doi. 10.3390/ijms21197162
    By:
    • Gladkova, Elizaveta D.;
    • Nechepurenko, Ivan V.;
    • Bredikhin, Roman A.;
    • Chepanova, Arina A.;
    • Zakharenko, Alexandra L.;
    • Luzina, Olga A.;
    • Ilina, Ekaterina S.;
    • Dyrkheeva, Nadezhda S.;
    • Mamontova, Evgeniya M.;
    • Anarbaev, Rashid O.;
    • Reynisson, Jóhannes;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    Promising New Inhibitors of Tyrosyl-DNA Phosphodiesterase I (Tdp 1) Combining 4-Arylcoumarin and Monoterpenoid Moieties as Components of Complex Antitumor Therapy.

    Published in:
    International Journal of Molecular Sciences, 2020, v. 21, n. 1, p. 126, doi. 10.3390/ijms21010126
    By:
    • Khomenko, Tatyana M.;
    • Zakharenko, Alexandra L.;
    • Chepanova, Arina A.;
    • Ilina, Ekaterina S.;
    • Zakharova, Olga D.;
    • Kaledin, Vasily I.;
    • Nikolin, Valeriy P.;
    • Popova, Nelly A.;
    • Korchagina, Dina V.;
    • Reynisson, Jóhannes;
    • Chand, Raina;
    • Ayine-Tora, Daniel M.;
    • Patel, Jinal;
    • Leung, Ivanhoe K. H.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    The Development of Tyrosyl-DNA Phosphodiesterase 1 Inhibitors. Combination of Monoterpene and Adamantine Moieties via Amide or Thioamide Bridges.

    Published in:
    Applied Sciences (2076-3417), 2019, v. 9, n. 13, p. 2767, doi. 10.3390/app9132767
    By:
    • Chepanova, Arina A.;
    • Mozhaitsev, Evgenii S.;
    • Munkuev, Aldar A.;
    • Suslov, Evgeniy V.;
    • Korchagina, Dina V.;
    • Zakharova, Olga D.;
    • Zakharenko, Alexandra L.;
    • Patel, Jinal;
    • Ayine-Tora, Daniel M.;
    • Reynisson, Jóhannes;
    • Leung, Ivanhoe K. H.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    MEMORY-IMPROVING EFFECTS OF MYRTENAL-ADAMANTANE CONJUGATES.

    Published in:
    Journal of Chemical Technology & Metallurgy, 2023, v. 58, n. 3, p. 627, doi. 10.59957/jctm.v58i3.95
    By:
    • Dragomanova, Stela;
    • Andonova, Velichka;
    • Lazarova, Maria;
    • Munkuev, Aldar;
    • Suslov, Evgeny;
    • Volcho, Konstantin;
    • Salakhutdinov, Neriman;
    • Stefanova, Miroslava;
    • Gavrilova, Petya;
    • Uzunova, Diamara;
    • Kalfin, Reni;
    • Tancheva, Lyubka
    Publication type:
    Article
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    New Hybrid Compounds Combining Fragments of Usnic Acid and Monoterpenoids for Effective Tyrosyl-DNA Phosphodiesterase 1 Inhibition.

    Published in:
    Biomolecules (2218-273X), 2021, v. 11, n. 7, p. 973, doi. 10.3390/biom11070973
    By:
    • Dyrkheeva, Nadezhda S.;
    • Filimonov, Aleksandr S.;
    • Luzina, Olga A.;
    • Zakharenko, Alexandra L.;
    • Ilina, Ekaterina S.;
    • Malakhova, Anastasia A.;
    • Medvedev, Sergey P.;
    • Reynisson, Jóhannes;
    • Volcho, Konstantin P.;
    • Zakian, Suren M.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    Sulfide, Sulfoxide, and Sulfone Derivatives of Usnic Acid as Inhibitors of Human TDP1 and TDP2 Enzymes.

    Published in:
    Chemistry (2624-8549), 2024, v. 6, n. 6, p. 1658, doi. 10.3390/chemistry6060101
    By:
    • Filimonov, Aleksandr S.;
    • Mikhailova, Marina A.;
    • Dyrkheeva, Nadezhda S.;
    • Chernyshova, Irina A.;
    • Kornienko, Tatyana E.;
    • Naumenko, Konstantin A.;
    • Anarbaev, Rashid O.;
    • Nefedov, Andrey A.;
    • Achara, Chigozie;
    • Curtis, Anthony D. M.;
    • Luzina, Olga A.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.;
    • Reynisson, Jóhannes
    Publication type:
    Article
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    Novel Peptide–Drug Conjugates with Dual Anticancer Activity.

    Published in:
    International Journal of Molecular Sciences, 2024, v. 25, n. 22, p. 12411, doi. 10.3390/ijms252212411
    By:
    • O'Flaherty, Siobhán;
    • Luzina, Olga A.;
    • Dyrkheeva, Nadezhda S.;
    • Krier, Ysaline;
    • Leprince, Jérôme;
    • Zakharenko, Alexandra L.;
    • Pokrovsky, Mikhail A.;
    • Pokrovsky, Andrey G.;
    • Lavrik, Olga I.;
    • Salakhutdinov, Nariman F.;
    • Varbanov, Mihayl;
    • Devocelle, Marc;
    • Volcho, Konstantin P.
    Publication type:
    Article
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    Stereoselectivity Inversion by Water Addition in the −SO<sub>3</sub>H‐catalyzed Tandem Prins‐Ritter Reaction for Synthesis of 4‐amidotetrahydropyran Derivatives.

    Published in:
    ChemCatChem, 2020, v. 12, n. 9, p. 2605, doi. 10.1002/cctc.202000070
    By:
    • Sidorenko, Alexander Yu.;
    • Li‐Zhulanov, Nikolai S.;
    • Mäki‐Arvela, Päivi;
    • Sandberg, Thomas;
    • Kravtsova, Anna V.;
    • Peixoto, Andreia F.;
    • Freire, Cristina;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Agabekov, Vladimir E.;
    • Murzin, Dmitry Yu.
    Publication type:
    Article
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