Works matching AU Venugopala, Katharigatta N.


Results: 97
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    Anti-tubercular Potency and Computationally-assessed Drug-likeness and Toxicology of Diversely Substituted Indolizines.

    Published in:
    Indian Journal of Pharmaceutical Education & Research, 2019, v. 53, n. 3, p. 545, doi. 10.5530/ijper.53.3.87
    By:
    • Venugopala, Katharigatta N.;
    • Tratrat, Christophe;
    • Chandrashekharappa, Sandeep;
    • Attimarad, Mahesh;
    • Sreeharsha, Nagaraja;
    • Nair, Anroop B.;
    • Pottathil, Shinu;
    • Venugopala, Rashmi;
    • Al-Attraqchi, Omar Husham Ahmed;
    • Morsy, Mohamed A.;
    • Haroun, Michelyne;
    • Odhav, Bharti
    Publication type:
    Article
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    An Approach to Enhance Dissolution Rate of Tamoxifen Citrate.

    Published in:
    BioMed Research International, 2019, p. 1, doi. 10.1155/2019/2161348
    By:
    • SreeHarsha, Nagaraja;
    • Hiremath, Jagadeesh G.;
    • Chilukuri, Swathi;
    • Aitha, Rajesh Kumar;
    • Al-Dhubiab, Bandar E.;
    • Venugopala, Katharigatta N.;
    • Alzahrani, Abdullah Mossa;
    • Meravanige, Girish
    Publication type:
    Article
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    Identification of Novel Cyclooxygenase-1 Selective Inhibitors of Thiadiazole-Based Scaffold as Potent Anti-Inflammatory Agents with Safety Gastric and Cytotoxic Profile.

    Published in:
    Molecules, 2023, v. 28, n. 8, p. 3416, doi. 10.3390/molecules28083416
    By:
    • Haroun, Michelyne;
    • Fesatidou, Maria;
    • Petrou, Anthi;
    • Tratrat, Christophe;
    • Zagaliotis, Panagiotis;
    • Gavalas, Antonis;
    • Venugopala, Katharigatta N.;
    • Kochkar, Hafedh;
    • Emeka, Promise M.;
    • Younis, Nancy S.;
    • Elmaghraby, Dalia Ahmed;
    • Almostafa, Mervt M.;
    • Chohan, Muhammad Shahzad;
    • Vizirianakis, Ioannis S.;
    • Papadimitriou-Tsantarliotou, Aliki;
    • Geronikaki, Athina
    Publication type:
    Article
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    Computational Design, Synthesis, and Pharmacological Evaluation of Naproxen-Guaiacol Chimera for Gastro-Sparing Anti-Inflammatory Response by Selective COX2 Inhibition.

    Published in:
    Molecules, 2022, v. 27, n. 20, p. 6905, doi. 10.3390/molecules27206905
    By:
    • Shinu, Pottathil;
    • Sharma, Manu;
    • Gupta, Girdhari Lal;
    • Mujwar, Somdutt;
    • Kandeel, Mahmoud;
    • Kumar, Manish;
    • Nair, Anroop B.;
    • Goyal, Manoj;
    • Singh, Purna;
    • Attimarad, Mahesh;
    • Venugopala, Katharigatta N.;
    • Nagaraja, Sreeharsha;
    • Telsang, Mallikarjun;
    • Aldhubiab, Bandar E.;
    • Morsy, Mohamed A.
    Publication type:
    Article
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    Thiazole: A Versatile Standalone Moiety Contributing to the Development of Various Drugs and Biologically Active Agents.

    Published in:
    Molecules, 2022, v. 27, n. 13, p. 3994, doi. 10.3390/molecules27133994
    By:
    • Arshad, Mohammed F.;
    • Alam, Aftab;
    • Alshammari, Abdullah Ayed;
    • Alhazza, Mohammed Bader;
    • Alzimam, Ibrahim Mohammed;
    • Alam, Md Anish;
    • Mustafa, Gulam;
    • Ansari, Md Salahuddin;
    • Alotaibi, Abdulelah M.;
    • Alotaibi, Abdullah A.;
    • Kumar, Suresh;
    • Asdaq, Syed Mohammed Basheeruddin;
    • Imran, Mohd.;
    • Deb, Pran Kishore;
    • Venugopala, Katharigatta N.;
    • Jomah, Shahamah
    Publication type:
    Article
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    1,5-Benzothiazepine Derivatives: Green Synthesis, In Silico and In Vitro Evaluation as Anticancer Agents.

    Published in:
    Molecules, 2022, v. 27, n. 12, p. 3757, doi. 10.3390/molecules27123757
    By:
    • Haroun, Michelyne;
    • Chobe, Santosh S.;
    • Alavala, Rajasekhar Reddy;
    • Mathure, Savita M.;
    • Jamullamudi, Risy Namratha;
    • Nerkar, Charushila K.;
    • Gugulothu, Vijay Kumar;
    • Tratrat, Christophe;
    • Islam, Mohammed Monirul;
    • Venugopala, Katharigatta N.;
    • Habeebuddin, Mohammed;
    • Telsang, Mallikarjun;
    • Sreeharsha, Nagaraja;
    • Anwer, Md. Khalid
    Publication type:
    Article
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    1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector Anopheles arabiensis and In Silico Molecular Docking Study.

    Published in:
    Molecules, 2022, v. 27, n. 9, p. 2676, doi. 10.3390/molecules27092676
    By:
    • Venugopala, Katharigatta N.;
    • Shinu, Pottathil;
    • Tratrat, Christophe;
    • Deb, Pran Kishore;
    • Gleiser, Raquel M.;
    • Chandrashekharappa, Sandeep;
    • Chopra, Deepak;
    • Attimarad, Mahesh;
    • Nair, Anroop B.;
    • Sreeharsha, Nagaraja;
    • Mahomoodally, Fawzi M.;
    • Haroun, Michelyne;
    • Kandeel, Mahmoud;
    • Asdaq, Syed Mohammed Basheeruddin;
    • Mohanlall, Viresh;
    • Al-Shar'i, Nizar A.;
    • Morsy, Mohamed A.
    Publication type:
    Article
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    Crystallography, Molecular Modeling, and COX-2 Inhibition Studies on Indolizine Derivatives.

    Published in:
    Molecules, 2021, v. 26, n. 12, p. 3550, doi. 10.3390/molecules26123550
    By:
    • Venugopala, Katharigatta N.;
    • Chandrashekharappa, Sandeep;
    • Tratrat, Christophe;
    • Deb, Pran Kishore;
    • Nagdeve, Rahul D.;
    • Nayak, Susanta K.;
    • Morsy, Mohamed A.;
    • Borah, Pobitra;
    • Mahomoodally, Fawzi M.;
    • Mailavaram, Raghu Prasad;
    • Attimarad, Mahesh;
    • Aldhubiab, Bandar E.;
    • Sreeharsha, Nagaraja;
    • Nair, Anroop B.;
    • Alwassil, Osama I.;
    • Haroun, Michelyne;
    • Mohanlall, Viresh;
    • Shinu, Pottathil;
    • Venugopala, Rashmi;
    • Kandeel, Mahmoud
    Publication type:
    Article
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    Investigation of Antifungal Properties of Synthetic Dimethyl-4-Bromo-1-(Substituted Benzoyl) Pyrrolo[1,2-a] Quinoline-2,3-Dicarboxylates Analogues: Molecular Docking Studies and Conceptual DFT-Based Chemical Reactivity Descriptors and Pharmacokinetics Evaluation

    Published in:
    Molecules, 2021, v. 26, n. 9, p. 2722, doi. 10.3390/molecules26092722
    By:
    • Uppar, Vijayakumar;
    • Chandrashekharappa, Sandeep;
    • Shivamallu, Chandan;
    • P, Sushma;
    • Kollur, Shiva Prasad;
    • Ortega-Castro, Joaquín;
    • Frau, Juan;
    • Flores-Holguín, Norma;
    • Basarikatti, Atiyaparveen I.;
    • Chougala, Mallikarjun;
    • Mohan M, Mrudula;
    • Banuprakash, Govindappa;
    • Jayadev;
    • Venugopala, Katharigatta N.;
    • Nandeshwarappa, Belakatte P.;
    • Veerapur, Ravindra;
    • Al-Kheraif, Abdulaziz A.;
    • Elgorban, Abdallah M.;
    • Syed, Asad;
    • Mudnakudu-Nagaraju, Kiran K.
    Publication type:
    Article
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    Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target Investigation.

    Published in:
    Molecules, 2020, v. 25, n. 6, p. 1316, doi. 10.3390/molecules25061316
    By:
    • Venugopala, Katharigatta N.;
    • Ramachandra, Pushpalatha;
    • Tratrat, Christophe;
    • Gleiser, Raquel M.;
    • Bhandary, Subhrajyoti;
    • Chopra, Deepak;
    • Morsy, Mohamed A.;
    • Aldhubiab, Bandar E.;
    • Attimarad, Mahesh;
    • Nair, Anroop B.;
    • Sreeharsha, Nagaraja;
    • Venugopala, Rashmi;
    • Deb, Pran Kishore;
    • Chandrashekharappa, Sandeep;
    • Khalil, Hany Ezzat;
    • Alwassil, Osama I.;
    • Abed, Sara Nidal;
    • Bataineh, Yazan A.;
    • Palenge, Ramachandra;
    • Haroun, Michelyne
    Publication type:
    Article
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    In silico Design and Synthesis of Tetrahydropyrimidinones and Tetrahydropyrimidinethiones as Potential Thymidylate Kinase Inhibitors Exerting Anti-TB Activity Against Mycobacterium tuberculosis.

    Published in:
    Drug Design, Development & Therapy, 2020, v. 14, p. 1027, doi. 10.2147/DDDT.S228381
    By:
    • Venugopala, Katharigatta N;
    • Tratrat, Christophe;
    • Pillay, Melendhran;
    • Chandrashekharappa, Sandeep;
    • Al-Attraqchi, Omar Husham Ahmed;
    • Aldhubiab, Bandar E;
    • Attimarad, Mahesh;
    • Alwassil, Osama I;
    • Nair, Anroop B;
    • Sreeharsha, Nagaraja;
    • Venugopala, Rashmi;
    • Morsy, Mohamed A;
    • Haroun, Michelyne;
    • Kumalo, Hezekiel M;
    • Odhav, Bharti;
    • Mlisana, Koleka
    Publication type:
    Article
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    An Efficient, Lung-Targeted, Drug-Delivery System To Treat Asthma Via Microparticles.

    Published in:
    Drug Design, Development & Therapy, 2019, v. 13, p. 4389, doi. 10.2147/DDDT.S216660
    By:
    • SreeHarsha, Nagaraja;
    • Venugopala, Katharigatta N;
    • Nair, Anroop B;
    • Roopashree, Teeka S;
    • Attimarad, Mahesh;
    • Hiremath, Jagadeesh G;
    • Al-Dhubiab, Bandar E;
    • Ramnarayanan, Chandramouli;
    • Shinu, Pottathil;
    • Handral, Mukund;
    • Haroun, Micheline;
    • Tratrat, Christophe
    Publication type:
    Article
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    Synthesis, biological evaluation, and computational investigation of ethyl 2,4,6-trisubstituted-1,4-dihydropyrimidine-5-carboxylates as potential larvicidal agents against Anopheles arabiensis.

    Published in:
    Journal of Biomolecular Structure & Dynamics, 2024, v. 42, n. 8, p. 4016, doi. 10.1080/07391102.2023.2217929
    By:
    • Duraisamy, Ramasamy;
    • Al-Shar'i, Nizar A.;
    • Chandrashekharappa, Sandeep;
    • Deb, Pran Kishore;
    • Gleiser, Raquel M.;
    • Tratrat, Christophe;
    • Chopra, Deepak;
    • Muthukurpalya Bhojegowd, Madhusudana Reddy;
    • Thirumalai, Dhakshanamurthy;
    • Morsy, Mohamed A.;
    • Ibrahim, Yasmine F.;
    • Mohanlall, Viresh;
    • Venugopala, Katharigatta N.
    Publication type:
    Article
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    Nanotechnology Integration for SARS-CoV-2 Diagnosis and Treatment: An Approach to Preventing Pandemic.

    Published in:
    Nanomaterials (2079-4991), 2021, v. 11, n. 7, p. 1841, doi. 10.3390/nano11071841
    By:
    • Asdaq, Syed Mohammed Basheeruddin;
    • Ikbal, Abu Md Ashif;
    • Sahu, Ram Kumar;
    • Bhattacharjee, Bedanta;
    • Paul, Tirna;
    • Deka, Bhargab;
    • Fattepur, Santosh;
    • Widyowati, Retno;
    • Vijaya, Joshi;
    • Al mohaini, Mohammed;
    • Alsalman, Abdulkhaliq J.;
    • Imran, Mohd.;
    • Nagaraja, Sreeharsha;
    • Nair, Anroop B.;
    • Attimarad, Mahesh;
    • Venugopala, Katharigatta N.
    Publication type:
    Article
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    Reinforced electrospun nanofiber composites for drug delivery applications.

    Published in:
    Journal of Biomedical Materials Research, Part A, 2021, v. 109, n. 10, p. 2036, doi. 10.1002/jbm.a.37187
    By:
    • Anup, Neelima;
    • Chavan, Tejas;
    • Chavan, Shruti;
    • Polaka, Suryanarayana;
    • Kalyane, Dnyaneshwar;
    • Abed, Sara Nidal;
    • Venugopala, Katharigatta N.;
    • Kalia, Kiran;
    • Tekade, Rakesh K.
    Publication type:
    Article
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    Novel Series of Methyl 3-(Substituted Benzoyl)-7-Substituted-2-Phenylindolizine-1-Carboxylates as Promising Anti-Inflammatory Agents: Molecular Modeling Studies.

    Published in:
    Biomolecules (2218-273X), 2019, v. 9, n. 11, p. 661, doi. 10.3390/biom9110661
    By:
    • Venugopala, Katharigatta N.;
    • Al-Attraqchi, Omar H.A.;
    • Tratrat, Christophe;
    • Nayak, Susanta K.;
    • Morsy, Mohamed A.;
    • Aldhubiab, Bandar E.;
    • Attimarad, Mahesh;
    • Nair, Anroop B.;
    • Sreeharsha, Nagaraja;
    • Venugopala, Rashmi;
    • Haroun, Michelyne;
    • Girish, Meravanige B.;
    • Chandrashekharappa, Sandeep;
    • Alwassil, Osama I.;
    • Odhav, Bharti
    Publication type:
    Article
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    Multifunctional Mesoporous Silica Nanoparticles for Oral Drug Delivery.

    Published in:
    Coatings (2079-6412), 2022, v. 12, n. 3, p. 358, doi. 10.3390/coatings12030358
    By:
    • Sreeharsha, Nagaraja;
    • Philip, Manish;
    • Krishna, Sivadas Swathi;
    • Viswanad, Vidya;
    • Sahu, Ram Kumar;
    • Shiroorkar, Predeepkumar Narayanappa;
    • Aasif, Afzal Haq;
    • Fattepur, Santosh;
    • Asdaq, Syed Mohammed Basheeruddin;
    • Nair, Anroop B.;
    • Attimarad, Mahesh;
    • Venugopala, Katharigatta N.
    Publication type:
    Article
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    Paclitaxel loaded poly (DL lactic acid co castor oil) 60:40 with poloxamer‐F68 rod shape cylindrical nanoparticle preparation and in vitro cytotoxicity studies.

    Published in:
    Polymers for Advanced Technologies, 2019, v. 30, n. 10, p. 2613, doi. 10.1002/pat.4719
    By:
    • SreeHarsha, Nagaraja;
    • Hiremath, Jagadeesh G.;
    • Aitha, Rajesh Kumar;
    • Domb, Abraham J.;
    • Al‐Dhubiab, Bandar E.;
    • Ramnarayanan, Chandramouli;
    • Alzahrani, Abdullah Mossa;
    • Venugopala, Katharigatta N.;
    • Akrawi, Sabah H.;
    • Attimarad, Mahesh;
    • Nair, Anroop B.
    Publication type:
    Article
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