Works by Van Der Veken, Pieter

Results: 39

Dipeptidyl Peptidase 9 in Human Leukocytes: Novel Inhibitors Induce Caspase‐1‐ and Gasdermin‐Dependent Cell Death.

Published in:

European Journal of Immunology, 2025, v. 55, n. 6, p. 1, doi. 10.1002/eji.202451526

By:

De Loose, Joni;
Mertens, Kathleen;
Filippi, Nicolò;
Corthaut, Sam;
Benramdane, Siham;
Sim, Yani;
Van Rymenant, Yentl;
Claesen, Karen;
Vliegen, Gwendolyn;
Berg, Maya;
Gomard, Tiphanie;
Caljon, Guy;
Pintelon, Isabel;
Van Der Veken, Pieter;
De Meester, Ingrid

Publication type:

Article

Repositioning the Substrate Activity Screening (SAS) Approach as a Fragment-Based Method for Identification of Weak Binders.

Published in:

ChemBioChem, 2014, v. 15, n. 15, p. 2238, doi. 10.1002/cbic.201402192

By:

Gladysz, Rafaela;
Cleenewerck, Matthias;
Joossens, Jurgen;
Lambeir, Anne‐Marie;
Augustyns, Koen;
Van der Veken, Pieter

Publication type:

Article

The Dipeptidyl Peptidases 4, 8, and 9 in Mouse Monocytes and Macrophages: DPP8/9 Inhibition Attenuates M1 Macrophage Activation in Mice.

Published in:

Inflammation, 2016, v. 39, n. 1, p. 413, doi. 10.1007/s10753-015-0263-5

By:

Waumans, Yannick;
Vliegen, Gwendolyn;
Maes, Lynn;
Rombouts, Miche;
Declerck, Ken;
Van Der Veken, Pieter;
Vanden Berghe, Wim;
De Meyer, Guido;
Schrijvers, Dorien;
De Meester, Ingrid

Publication type:

Article

Mass spectrometric characterization of organosulfates related to secondary organic aerosol from isoprene.

Published in:

Rapid Communications in Mass Spectrometry: RCM, 2013, v. 27, n. 7, p. 784, doi. 10.1002/rcm.6511

By:

Safi Shalamzari, Mohammad;
Ryabtsova, Oxana;
Kahnt, Ariane;
Vermeylen, Reinhilde;
Hérent, Marie‐France;
Quetin‐Leclercq, Joëlle;
Van der Veken, Pieter;
Maenhaut, Willy;
Claeys, Magda

Publication type:

Article

Targeting fibroblast activation protein (FAP): next generation PET radiotracers using squaramide coupled bifunctional DOTA and DATA5m chelators.

Published in:

EJNMMI Radiopharmacy & Chemistry, 2020, v. 5, n. 1, p. 1, doi. 10.1186/s41181-020-00102-z

By:

Moon, Euy Sung;
Elvas, Filipe;
Vliegen, Gwendolyn;
De Lombaerde, Stef;
Vangestel, Christel;
De Bruycker, Sven;
Bracke, An;
Eppard, Elisabeth;
Greifenstein, Lukas;
Klasen, Benedikt;
Kramer, Vasko;
Staelens, Steven;
De Meester, Ingrid;
Van der Veken, Pieter;
Rösch, Frank

Publication type:

Article

ATG4B Inhibitor UAMC-2526 Potentiates the Chemotherapeutic Effect of Gemcitabine in a Panc02 Mouse Model of Pancreatic Ductal Adenocarcinoma.

Published in:

Frontiers in Oncology, 2021, v. 11, p. 1, doi. 10.3389/fonc.2021.750259

By:

Takhsha, Farnaz Sedigheh;
Vangestel, Christel;
Tanc, Muhammet;
De Bruycker, Sven;
Berg, Maya;
Pintelon, Isabel;
Stroobants, Sigrid;
De Meyer, Guido R. Y.;
Van Der Veken, Pieter;
Martinet, Wim

Publication type:

Article

Expression and spatial heterogeneity of dipeptidyl peptidases in endothelial cells of conduct vessels and capillaries.

Published in:

Biological Chemistry, 2011, v. 392, n. 3, p. 189, doi. 10.1515/BC.2011.002

By:

Matheeussen, Veerle;
Baerts, Lesley;
De Meyer, Guido;
De Keulenaer, Gilles;
Van der Veken, Pieter;
Augustyns, Koen;
Dubois, Véronique;
Scharpé, Simon;
De Meester, Ingrid

Publication type:

Article

Evaluation of [18F]BR420 and [18F]BR351 as radiotracers for MMP-9 imaging in colorectal cancer.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2017, v. 60, n. 1, p. 69, doi. 10.1002/jlcr.3476

By:

Vazquez, Naiara;
Missault, Stephan;
Vangestel, Christel;
Deleye, Steven;
Thomae, David;
Van der Veken, Pieter;
Augustyns, Koen;
Staelens, Steven;
Dedeurwaerdere, Stefanie;
wyffels, Leonie

Publication type:

Article

Selective Glucocorticoid Receptor Properties of GSK866 Analogs with Cysteine Reactive Warheads.

Published in:

Frontiers in Immunology, 2017, p. 1, doi. 10.3389/fimmu.2017.01324

By:

Chirumamilla, Chandra S.;
Palagani, Ajay;
Kamaraj, Balu;
Declerck, Ken;
Verbeek, Marinus W. C.;
Oksana, Ryabtsova;
De Bosscher, Karolien;
Bougarne, Nadia;
Ruttens, Bart;
Gevaert, Kris;
Houtman, René;
De Vos, Winnok H.;
Joossens, Jurgen;
Van Der Veken, Pieter;
Augustyns, Koen;
Van Ostade, Xaveer;
Bogaerts, Annemie;
De Winter, Hans;
Berghe, Wim Vanden

Publication type:

Article

Design and Synthesis of 1,3-Diarylpyrazoles and Investigation of Their Cytotoxicity and Antiparasitic Profile.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 9, p. 4693, doi. 10.3390/ijms25094693

By:

Bozdag, Murat;
Mertens, Freke;
Matheeussen, An;
Van Pelt, Natascha;
Foubert, Kenn;
Hermans, Nina;
De Meyer, Guido R. Y.;
Augustyns, Koen;
Martinet, Wim;
Caljon, Guy;
Van der Veken, Pieter

Publication type:

Article

Prolyl Carboxypeptidase Mediates the C-Terminal Cleavage of (Pyr)-Apelin-13 in Human Umbilical Vein and Aortic Endothelial Cells.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 13, p. 6698, doi. 10.3390/ijms22136698

By:

De Hert, Emilie;
Bracke, An;
Pintelon, Isabel;
Janssens, Eline;
Lambeir, Anne-Marie;
Van Der Veken, Pieter;
De Meester, Ingrid

Publication type:

Article

Molecular Imaging of Apoptosis: The Case of Caspase-3 Radiotracers.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 8, p. 3948, doi. 10.3390/ijms22083948

By:

Beroske, Lucas;
Van den Wyngaert, Tim;
Stroobants, Sigrid;
Van der Veken, Pieter;
Elvas, Filipe

Publication type:

Article

ClpP Protease, a Promising Antimicrobial Target.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 9, p. 2232, doi. 10.3390/ijms20092232

By:

Moreno-Cinos, Carlos;
Goossens, Kenneth;
Salado, Irene G.;
Van Der Veken, Pieter;
De Winter, Hans;
Augustyns, Koen

Publication type:

Article

Synthesis and Evaluation of a Zr-89-Labeled Monoclonal Antibody for Immuno-PET Imaging of Amyloid-β Deposition in the Brain.

Published in:

2016

By:

Fissers, Jens;
Waldron, Ann-Marie;
De Vijlder, Thomas;
Van Broeck, Bianca;
Pemberton, Darrel;
Mercken, Marc;
Van Der Veken, Pieter;
Joossens, Jurgen;
Augustyns, Koen;
Dedeurwaerdere, Stefanie;
Stroobants, Sigrid;
Staelens, Steven;
wyffels, Leonie;
Pemberton, Darrel J

Publication type:

journal article

Development of caspase-3-selective activity-based probes for PET imaging of apoptosis.

Published in:

EJNMMI Radiopharmacy & Chemistry, 2024, v. 9, n. 1, p. 1, doi. 10.1186/s41181-024-00291-x

By:

Lauwerys, Louis;
Beroske, Lucas;
Solania, Angelo;
Vangestel, Christel;
Miranda, Alan;
Van Giel, Nele;
Adhikari, Karuna;
Lambeir, Anne-Marie;
wyffels, Leonie;
Wolan, Dennis;
Van der Veken, Pieter;
Elvas, Filipe

Publication type:

Article

Newly developed serine protease inhibitors decrease visceral hypersensitivity in a post-inflammatory rat model for irritable bowel syndrome.

Published in:

2018

By:

Ceuleers, Hannah;
Hanning, Nikita;
Heirbaut, Jelena;
Van Remoortel, Samuel;
Joossens, Jurgen;
Van Der Veken, Pieter;
Francque, Sven M.;
De bruyn, Michelle;
Lambeir, Anne‐Marie;
De Man, Joris G.;
Timmermans, Jean‐Pierre;
Augustyns, Koen;
De Meester, Ingrid;
De Winter, Benedicte Y.;
Lambeir, Anne-Marie;
Timmermans, Jean-Pierre

Publication type:

journal article

Synthesis of γ,δ-Aziridino α-Amino Acid Derivatives and their Stereoselective Ring Transformation to 2-(Aminomethyl)-1-aminocyclopropanecarboxylic Acid Derivatives.

Published in:

European Journal of Organic Chemistry, 2014, v. 2014, n. 6, p. 1220, doi. 10.1002/ejoc.201301030

By:

De Brabandere, Stijn;
Mangelinckx, Sven;
Kadam, Santosh T.;
Nural, Yahya;
Augustyns, Koen;
Van der Veken, Pieter;
Törnroos, Karl W.;
De Kimpe, Norbert

Publication type:

Article

The Effect of a Novel Serine Protease Inhibitor on Inflammation and Intestinal Permeability in a Murine Colitis Transfer Model.

Published in:

Frontiers in Pharmacology, 2021, v. 12, p. 1, doi. 10.3389/fphar.2021.682065

By:

Van Spaendonk, Hanne;
Ceuleers, Hannah;
Smet, Annemieke;
Berg, Maya;
Joossens, Jurgen;
Van der Veken, Pieter;
Francque, Sven M.;
Lambeir, Anne-Marie;
De Man, Joris G.;
De Meester, Ingrid;
Augustyns, Koen;
De Winter, Benedicte Y.

Publication type:

Article

Efforts towards an On‐Target Version of the Groebke–Blackburn–Bienaymé (GBB) Reaction for Discovery of Druglike Urokinase (uPA) Inhibitors.

Published in:

Chemistry - A European Journal, 2019, v. 25, n. 53, p. 12380, doi. 10.1002/chem.201901917

By:

Gladysz, Rafaela;
Vrijdag, Johannes;
Van Rompaey, Dries;
Lambeir, Anne‐Marie;
Augustyns, Koen;
De Winter, Hans;
Van der Veken, Pieter

Publication type:

Article

Development of a Novel Chemical Probe for the Selective Enrichment of Phosphorylated Serine- and Threonine-Containing Peptides.

Published in:

ChemBioChem, 2005, v. 6, n. 12, p. 2271, doi. 10.1002/cbic.200500209

By:

Pieter van der Veken;
Eef H. C. Dirksen;
Eelco Ruijter;
Ronald C. Elgersma;
Albert J. R. Heck;
Dirk T. S. Rijkers;
Monique Slijper;
Rob M. J. Liskamp

Publication type:

Article

Blockade of fibroblast activation protein in combination with radiation treatment in murine models of pancreatic adenocarcinoma.

Published in:

PLoS ONE, 2019, v. 14, n. 2, p. 1, doi. 10.1371/journal.pone.0211117

By:

Gunderson, Andrew J.;
Yamazaki, Tomoko;
McCarty, Kayla;
Phillips, Michaela;
Alice, Alejandro;
Bambina, Shelly;
Zebertavage, Lauren;
Friedman, David;
Cottam, Benjamin;
Newell, Pippa;
Gough, Michael J.;
Crittenden, Marka R.;
Van der Veken, Pieter;
Young, Kristina H.

Publication type:

Article

Substrate Activity Screening (SAS) and Related Approaches in Medicinal Chemistry.

Published in:

ChemMedChem, 2016, v. 11, n. 5, p. 467, doi. 10.1002/cmdc.201500569

By:

Gladysz, Rafaela;
Lambeir, Anne‐Marie;
Joossens, Jurgen;
Augustyns, Koen;
Van der Veken, Pieter

Publication type:

Article

Synthesis of Bicyclic N-Arylmethyl-Substituted Iminoribitol Derivatives as Selective Nucleoside Hydrolase Inhibitors.

Published in:

ChemMedChem, 2009, v. 4, n. 2, p. 249, doi. 10.1002/cmdc.200800231

By:

Berg, Maya;
Bal, Gunther;
Goeminne, Annelies;
Van der Veken, Pieter;
Versées, Wim;
Steyaert, Jan;
Haemers, Achiel;
Augustyns, Koen

Publication type:

Article

3-methyl-1,2,3-butanetricarboxylic acid: An atmospheric tracer for terpene secondary organic aerosol.

Published in:

Geophysical Research Letters, 2007, v. 34, n. 24, p. n/a, doi. 10.1029/2007GL031338

By:

Szmigielski, Rafal;
Surratt, Jason D.;
Gómez-González, Yadian;
Van der Veken, Pieter;
Kourtchev, Ivan;
Vermeylen, Reinhilde;
Blockhuys, Frank;
Jaoui, Mohammed;
Kleindienst, Tadeusz E.;
Lewandowski, Michael;
Offenberg, John H.;
Edney, Edward O.;
Seinfeld, John H.;
Maenhaut, Willy;
Claeys, Magda

Publication type:

Article

Multi-slice computed tomography with N1177 identifies ruptured atherosclerotic plaques in rabbits.

Published in:

Basic Research in Cardiology, 2010, v. 105, n. 1, p. 51, doi. 10.1007/s00395-009-0052-0

By:

Van Herck, Jozef Leo;
De Meyer, Guido R. Y.;
Martinet, Wim;
Salgado, Rodrigo A.;
Shivalkar, Bharati;
De Mondt, Roel;
Van De Ven, Helene;
Ludwig, Annick;
Van Der Veken, Pieter;
Van Vaeck, Luc;
Bult, Hidde;
Herman, Arnold G.;
Vrints, Christiaan J.

Publication type:

Article

Spatiotemporal expression and inhibition of prolyl oligopeptidase contradict its involvement in key pathologic mechanisms of kainic acid–induced temporal lobe epilepsy in rats.

Published in:

Epilepsia Open, 2019, v. 4, n. 1, p. 92, doi. 10.1002/epi4.12293

By:

Ali, Idrish;
Van Eetveldt, Annemie;
Van Elzen, Roos;
Kalathil Raju, Tom;
Van Der Veken, Pieter;
Lambeir, Anne‐Marie;
Dedeurwaerdere, Stefanie

Publication type:

Article

The effect of pharmacological inhibition of Serine Proteases on neuronal networks in vitro.

Published in:

PeerJ, 2019, p. 1, doi. 10.7717/peerj.6796

By:

De Vijver, Sebastiaan Van;
Missault, Stephan;
Van Soom, Jeroen;
Van Der Veken, Pieter;
Augustyns, Koen;
Joossens, Jurgen;
Dedeurwaerdere, Stefanie;
Giugliano, Michele

Publication type:

Article

In Vivo Amyloid-β Imaging in the APPPS1-21 Transgenic Mouse Model with a 89Zr-Labeled Monoclonal Antibody.

Published in:

Frontiers in Aging Neuroscience, 2016, p. 1, doi. 10.3389/fnagi.2016.00067

By:

Waldron, Ann-Marie;
Fissers, Jens;
Van Eetveldt, Annemie;
Van Broeck, Bianca;
Mercken, Marc;
Pemberton, Darrel J.;
Van Der Veken, Pieter;
Augustyns, Koen;
Joossens, Jurgen;
Stroobants, Sigrid;
Dedeurwaerdere, Stefanie;
Wyffels, Leonie;
Staelens, Steven

Publication type:

Article

Novel Generation of FAP Inhibitor-Based Homodimers for Improved Application in Radiotheranostics.

Published in:

Cancers, 2023, v. 15, n. 6, p. 1889, doi. 10.3390/cancers15061889

By:

Martin, Marcel;
Ballal, Sanjana;
Yadav, Madhav Prasad;
Bal, Chandrasekhar;
Van Rymenant, Yentl;
De Loose, Joni;
Verhulst, Emile;
De Meester, Ingrid;
Van Der Veken, Pieter;
Roesch, Frank

Publication type:

Article

Novel drug discovery strategies for atherosclerosis that target necrosis and necroptosis.

Published in:

Expert Opinion on Drug Discovery, 2018, v. 13, n. 6, p. 477, doi. 10.1080/17460441.2018.1457644

By:

Coornaert, Isabelle;
Hofmans, Sam;
Devisscher, Lars;
Augustyns, Koen;
Van Der Veken, Pieter;
De Meyer, Guido R.Y.;
Martinet, Wim

Publication type:

Article

A novel serine protease inhibitor as potential treatment for dry eye syndrome and ocular inflammation.

Published in:

Scientific Reports, 2020, v. 10, n. 1, p. N.PAG, doi. 10.1038/s41598-020-74159-w

By:

Joossen, Cedric;
Baán, Adrienn;
Moreno-Cinos, Carlos;
Joossens, Jurgen;
Cools, Nathalie;
Lanckacker, Ellen;
Moons, Lieve;
Lemmens, Kim;
Lambeir, Anne-Marie;
Fransen, Erik;
Delputte, Peter;
Caljon, Guy;
Van Der Veken, Pieter;
Maes, Louis;
De Meester, Ingrid;
Kiekens, Filip;
Augustyns, Koen;
Cos, Paul

Publication type:

Article

Circulating Stromal Cell-Derived Factor 1α Levels in Heart Failure: A Matter of Proper Sampling.

Published in:

PLoS ONE, 2015, v. 10, n. 10, p. 1, doi. 10.1371/journal.pone.0141408

By:

Baerts, Lesley;
Waumans, Yannick;
Brandt, Inger;
Jungraithmayr, Wolfgang;
Van der Veken, Pieter;
Vanderheyden, Marc;
De Meester, Ingrid

Publication type:

Article

An Essential Signal Peptide Peptidase Identified in an RNAi Screen of Serine Peptidases of Trypanosoma brucei.

Published in:

PLoS ONE, 2015, v. 10, n. 3, p. 1, doi. 10.1371/journal.pone.0123241

By:

Moss, Catherine X.;
Brown, Elaine;
Hamilton, Alana;
Van der Veken, Pieter;
Augustyns, Koen;
Mottram, Jeremy C.

Publication type:

Article

Schistosomicidal and molluscicidal activities of aminoalkylamino substituted neo- and norneocryptolepine derivatives

Published in:

Pharmaceutical Biology, 2012, v. 50, n. 2, p. 134, doi. 10.3109/13880209.2011.578278

By:

El Bardicy, Samia;
El Sayed, Ibrahim;
Yousif, Fouad;
Van der Veken, Pieter;
Haemers, Achiel;
Augustyns, Koen;
Pieters, Luc

Publication type:

Article

An Interdisciplinary Approach Provides Insights into the Pronounced Selectivity of Compound 42 for DPP9.

Published in:

ChemMedChem, 2025, v. 20, n. 5, p. 1, doi. 10.1002/cmdc.202400700

By:

Beyens, Olivier;
Corthaut, Sam;
Lambeir, Anne‐Marie;
Van Der Veken, Pieter;
Sterckx, Yann G.‐J.;
De Meester, Ingrid;
De Winter, Hans

Publication type:

Article

Vildagliptin‐Derived Dipeptidyl Peptidase 9 (DPP9) Inhibitors: Identification of a DPP8/9‐Specific Lead.

Published in:

ChemMedChem, 2022, v. 17, n. 15, p. 1, doi. 10.1002/cmdc.202200097

By:

Benramdane, Siham;
De Loose, Joni;
Beyens, Olivier;
Van Rymenant, Yentl;
Vliegen, Gwendolyn;
Augustyns, Koen;
De Winter, Hans;
De Meester, Ingrid;
Van der Veken, Pieter

Publication type:

Article

In Vitro Evaluation of the Squaramide-Conjugated Fibroblast Activation Protein Inhibitor-Based Agents AAZTA 5.SA.FAPi and DOTA.SA.FAPi.

Published in:

Molecules, 2021, v. 26, n. 12, p. 3482, doi. 10.3390/molecules26123482

By:

Moon, Euy Sung;
Van Rymenant, Yentl;
Battan, Sandeep;
De Loose, Joni;
Bracke, An;
Van der Veken, Pieter;
De Meester, Ingrid;
Rösch, Frank

Publication type:

Article

Resistance and cross-resistance profile of the diaryltriazine NNRTI and candidate microbicide UAMC01398.

Published in:

2016

By:

Ariën, Kevin K.;
Venkatraj, Muthusamy;
Michiels, Johan;
Joossens, Jurgen;
Vereecken, Katleen;
Van der Veken, Pieter;
Heeres, Jan;
De Winter, Hans;
Heyndrickx, Leo;
Augustyns, Koen;
Vanham, Guido

Publication type:

journal article

Diaryltriazine non-nucleoside reverse transcriptase inhibitors are potent candidates for pre-exposure prophylaxis in the prevention of sexual HIV transmission.

Published in:

Journal of Antimicrobial Chemotherapy (JAC), 2013, v. 68, n. 9, p. 2038, doi. 10.1093/jac/dkt166

By:

Ariën, Kevin K.;
Venkatraj, Muthusamy;
Michiels, Johan;
Joossens, Jurgen;
Vereecken, Katleen;
Van der Veken, Pieter;
Abdellati, Saïd;
Cuylaerts, Vicky;
Crucitti, Tania;
Heyndrickx, Leo;
Heeres, Jan;
Augustyns, Koen;
Lewi, Paul J.;
Vanham, Guido

Publication type:

Article

Works by Van Der Veken, Pieter

Dipeptidyl Peptidase 9 in Human Leukocytes: Novel Inhibitors Induce Caspase‐1‐ and Gasdermin‐Dependent Cell Death.

Repositioning the Substrate Activity Screening (SAS) Approach as a Fragment-Based Method for Identification of Weak Binders.

The Dipeptidyl Peptidases 4, 8, and 9 in Mouse Monocytes and Macrophages: DPP8/9 Inhibition Attenuates M1 Macrophage Activation in Mice.

Mass spectrometric characterization of organosulfates related to secondary organic aerosol from isoprene.

Targeting fibroblast activation protein (FAP): next generation PET radiotracers using squaramide coupled bifunctional DOTA and DATA5m chelators.

ATG4B Inhibitor UAMC-2526 Potentiates the Chemotherapeutic Effect of Gemcitabine in a Panc02 Mouse Model of Pancreatic Ductal Adenocarcinoma.

Expression and spatial heterogeneity of dipeptidyl peptidases in endothelial cells of conduct vessels and capillaries.

Evaluation of [<sup>18</sup>F]BR420 and [<sup>18</sup>F]BR351 as radiotracers for MMP-9 imaging in colorectal cancer.

Selective Glucocorticoid Receptor Properties of GSK866 Analogs with Cysteine Reactive Warheads.

Design and Synthesis of 1,3-Diarylpyrazoles and Investigation of Their Cytotoxicity and Antiparasitic Profile.

Prolyl Carboxypeptidase Mediates the C-Terminal Cleavage of (Pyr)-Apelin-13 in Human Umbilical Vein and Aortic Endothelial Cells.

Molecular Imaging of Apoptosis: The Case of Caspase-3 Radiotracers.

ClpP Protease, a Promising Antimicrobial Target.

Synthesis and Evaluation of a Zr-89-Labeled Monoclonal Antibody for Immuno-PET Imaging of Amyloid-β Deposition in the Brain.

Development of caspase-3-selective activity-based probes for PET imaging of apoptosis.

Newly developed serine protease inhibitors decrease visceral hypersensitivity in a post-inflammatory rat model for irritable bowel syndrome.

Synthesis of γ,δ-Aziridino α-Amino Acid Derivatives and their Stereoselective Ring Transformation to 2-(Aminomethyl)-1-aminocyclopropanecarboxylic Acid Derivatives.

The Effect of a Novel Serine Protease Inhibitor on Inflammation and Intestinal Permeability in a Murine Colitis Transfer Model.

Efforts towards an On‐Target Version of the Groebke–Blackburn–Bienaymé (GBB) Reaction for Discovery of Druglike Urokinase (uPA) Inhibitors.

Development of a Novel Chemical Probe for the Selective Enrichment of Phosphorylated Serine- and Threonine-Containing Peptides.

Blockade of fibroblast activation protein in combination with radiation treatment in murine models of pancreatic adenocarcinoma.

Substrate Activity Screening (SAS) and Related Approaches in Medicinal Chemistry.

Synthesis of Bicyclic N-Arylmethyl-Substituted Iminoribitol Derivatives as Selective Nucleoside Hydrolase Inhibitors.

3-methyl-1,2,3-butanetricarboxylic acid: An atmospheric tracer for terpene secondary organic aerosol.

Multi-slice computed tomography with N1177 identifies ruptured atherosclerotic plaques in rabbits.

Spatiotemporal expression and inhibition of prolyl oligopeptidase contradict its involvement in key pathologic mechanisms of kainic acid–induced temporal lobe epilepsy in rats.

The effect of pharmacological inhibition of Serine Proteases on neuronal networks in vitro.

In Vivo Amyloid-β Imaging in the APPPS1-21 Transgenic Mouse Model with a <sup>89</sup>Zr-Labeled Monoclonal Antibody.

Novel Generation of FAP Inhibitor-Based Homodimers for Improved Application in Radiotheranostics.

Novel drug discovery strategies for atherosclerosis that target necrosis and necroptosis.

A novel serine protease inhibitor as potential treatment for dry eye syndrome and ocular inflammation.

Circulating Stromal Cell-Derived Factor 1α Levels in Heart Failure: A Matter of Proper Sampling.

An Essential Signal Peptide Peptidase Identified in an RNAi Screen of Serine Peptidases of Trypanosoma brucei.

Schistosomicidal and molluscicidal activities of aminoalkylamino substituted neo- and norneocryptolepine derivatives

An Interdisciplinary Approach Provides Insights into the Pronounced Selectivity of Compound 42 for DPP9.

Vildagliptin‐Derived Dipeptidyl Peptidase 9 (DPP9) Inhibitors: Identification of a DPP8/9‐Specific Lead.

In Vitro Evaluation of the Squaramide-Conjugated Fibroblast Activation Protein Inhibitor-Based Agents AAZTA 5.SA.FAPi and DOTA.SA.FAPi.

Resistance and cross-resistance profile of the diaryltriazine NNRTI and candidate microbicide UAMC01398.

Diaryltriazine non-nucleoside reverse transcriptase inhibitors are potent candidates for pre-exposure prophylaxis in the prevention of sexual HIV transmission.