Works by Valette, Héric

Results: 33

Synthesis and preliminary evaluation of a carbon-11-labelled agonist of the α7 nicotinic acetylcholine receptor.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2001, v. 44, n. 11, p. 785, doi. 10.1002/jlcr.504

By:

Dolle, Frédéric;
Valette, Héric;
Hinnen, Françoise;
Vaufrey, Françoise;
Demphel, Stéphane;
Coulon, Christine;
Ottaviani, Michéle;
Bottlaender, Michel;
Crouzel, Christian

Publication type:

Article

Highly efficient synthesis of [11C]S12968 and [11C]S12967, for the in vivo imaging of the cardiac calcium channels using PET.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2001, v. 44, n. 7, p. 481, doi. 10.1002/jlcr.476

By:

Dolle, Frédéric;
Valette, Héric;
Hinnen, Françoise;
Demphel, Stéphane;
Bramoulle, Yann;
Peglion, Jean-Louis;
Crouzel, Christian

Publication type:

Article

Highly efficient synthesis of [11C]Me-QNB, a selective radioligand for the quantification of the cardiac muscarinic receptors using PET.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2001, v. 44, n. 5, p. 337, doi. 10.1002/jlcr.460

By:

Dolle, Frédéric;
Hinnen, Françoise;
Vaufrey, Françoise;
Demphel, Stéphane;
Bramoulle, Yann;
Fournier, Denis;
Ponchant, Michel;
Valette, Héric;
Crouzel, Christian

Publication type:

Article

Highly efficient synthesis of [11C]PE2I, a selective radioligand for the quantification of the dopamine transporter using PET.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2000, v. 43, n. 10, p. 997, doi. 10.1002/1099-1344(200009)43:10<997::AID-JLCR385>3.0.CO;2-#

By:

Dolle, Frédéric;
Bottlaender, Michel;
Demphel, Stéphane;
Emond, Patrick;
Fuseau, Chantal;
Coulon, Christine;
Ottaviani, Michele;
Valette, Héric;
Loc'h, Christian;
Halldin, Christer;
Mauclaire, Laurent;
Guilloteau, Denis;
Maziere, Bernard;
Crouzel, Christian

Publication type:

Article

Synthesis of 2-[18F]fluoro-3-[2(S)-2-azetidinylmethoxy]pyridine, a highly potent radioligand for in vivo imaging central nicotinic acetylcholine receptors.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1998, v. 41, n. 5, p. 451, doi. 10.1002/(SICI)1099-1344(199805)41:5<451::AID-JLCR111>3.0.CO;2-R

By:

Dolle, Frédéric;
Valette, Héric;
Bottlaender, Michel;
Hinnen, Françoise;
Vaufrey, Françoise;
Guenther, Ilonka;
Crouzel, Christian

Publication type:

Article

Synthesis and 11C-labelling of two selective high affinity nicotinic cholinergic agonists for evaluation as radioligands for PET studies.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1996, v. 38, n. 12, p. 1099, doi. 10.1002/(SICI)1099-1344(199612)38:12<1099::AID-JLCR934>3.0.CO;2-G

By:

Dolle, Frédéric;
Dolci, Lilian;
Valette, Héric;
Bottlaender, Michel;
Fournier, Denis;
Fuseau, Chantal;
Vaufrey, Françoise;
Crouzel, Christian

Publication type:

Article

Transport of Selected PET Radiotracers by Human P-Glycoprotein (ABCB1) and Breast Cancer Resistance Protein (ABCG2): An In Vitro Screening.

Published in:

Journal of Nuclear Medicine, 2011, v. 52, n. 3, p. 415, doi. 10.2967/jnumed.110.079608

By:

Tournier, Nicolas;
Valette, Héric;
Peyronneau, Marie-Anne;
Saba, Wadad;
Goutal, Sébastien;
Kuhnast, Bertrand;
Dollé, Frédéric;
Scherrmann, Jean-Michel;
Cisternino, Salvatore;
Bottlaender, Michel

Publication type:

Article

In Vivo Imaging of Human Cerebral Nicotinic Acetylcholine Receptors with 2-18F-Fluoro-A-85380 and PET.

Published in:

Journal of Nuclear Medicine, 2005, v. 46, n. 2, p. 240

By:

Gallezot, Jean-Dominique;
Bottlaender, Michel;
Grégoire, Marie-Claude;
Roumenov, Dimitri;
Deverre, Jean-Robert;
Coulon, Christine;
Ottaviani, Michèle;
Dollé, Frédéric;
Syrota, André;
Valette, Héric

Publication type:

Article

Biodistribution and Radiation Dosimetry of 18F-Fluoro-A-85380 in Healthy Volunteers.

Published in:

Journal of Nuclear Medicine, 2003, v. 44, n. 4, p. 596

By:

Bottlaender, Michel;
Valette, Héric;
Roumenov, Dimitri;
Dollé, Frédéric;
Coulon, Christine;
Ottaviani, Michèle;
Hinnen, Françoise;
Ricard, Marcel

Publication type:

Article

In Vivo Quantification of Myocardial Dihydropyridine Binding Sites: A PET Study in Dogs.

Published in:

Journal of Nuclear Medicine, 2002, v. 43, n. 9, p. 1227

By:

Valette, Héric;
Dollé, Frédéric;
Guenther, Ilonka;
Fuseau, Chantal;
Coulon, Christine;
Hinnen, Françoise;
Péglion, Jean-Louis;
Crouzel, Christian

Publication type:

Article

Myocardial Kinetics of the 11C-Labeled Enantiomers of the Ca2+ Channel Inhibitor S11568: An In Vivo Study.

Published in:

Journal of Nuclear Medicine, 2001, v. 42, n. 6, p. 932

By:

Valette, Héric;
Dollé, Frédéric;
Guenther, Ilonka;
Hinnen, Françoise;
Fuseau, Chantal;
Coulon, Christine;
Péglion, Jean-Louis;
Crouzel, Christian

Publication type:

Article

[18F]ZW-104, a new radioligand for imaging α2-α3-α4/β2 central nicotinic acetylcholine receptors: Evaluation in mutant mice.

Published in:

Synapse, 2010, v. 64, n. 7, p. 570, doi. 10.1002/syn.20776

By:

Saba, Wadad;
Valette, Héric;
Granon, Sylvie;
Xiao, Yingxian;
Kellar, Kenneth J.;
Dollé, Frédéric;
Bottlaender, Michel

Publication type:

Article

[11C]SL25.1188, a new reversible radioligand to study the monoamine oxidase type B with PET: Preclinical characterisation in nonhuman primate.

Published in:

Synapse, 2010, v. 64, n. 1, p. 61, doi. 10.1002/syn.20703

By:

Saba, Wadad;
Valette, Héric;
Peyronneau, Marie-Anne;
Bramoullé, Yann;
Coulon, Christine;
Curet, Olivier;
George, Pascal;
Dollé, Frédéric;
Bottlaender, Michel

Publication type:

Article

[18F]FPhEP and [18F]F2PhEP, two new epibatidine-based radioligands: Evaluation for imaging nicotinic acetylcholine receptors in baboon brain.

Published in:

Synapse, 2007, v. 61, n. 9, p. 764, doi. 10.1002/syn.20426

By:

Valette, Héric;
Dollé, Frédéric;
Saba, Wadad;
Roger, Gaelle;
Hinnen, Françoise;
Coulon, Christine;
Ottaviani, Michele;
Syrota, André;
Bottlaender, Michel

Publication type:

Article

[11C]LBT-999: A suitable radioligand for investigation of extra-striatal dopamine transporter with PET.

Published in:

Synapse, 2007, v. 61, n. 1, p. 17, doi. 10.1002/syn.20337

By:

Saba, Wadad;
Valette, Héric;
Schöllhorn-Peyronneau, Marie-Anne;
Coulon, Christine;
Ottaviani, Michele;
Chalon, Sylvie;
Dolle, Frédéric;
Emond, Patrick;
Halldin, Christer;
Helfenbein, Julie;
Madelmont, Jean-Claude;
Deloye, Jean-Bernard;
Guilloteau, Denis;
Bottlaender, Michel

Publication type:

Article

Acute effects of physostigmine and galantamine on the binding of [18F]fluoro-A-85380: A PET study in monkeys.

Published in:

Synapse, 2005, v. 56, n. 4, p. 217, doi. 10.1002/syn.20145

By:

Valette, Héric;
Bottlaender, Michel;
Dollé, Frédéric;
Coulon, Christine;
Ottaviani, Michèle;
Syrota, André

Publication type:

Article

Anesthesia affects the disposition of [18F]fluoro-A-85380: A PET study in monkeys.

Published in:

Synapse, 2002, v. 44, n. 1, p. 58, doi. 10.1002/syn.10047

By:

Valette, Héric;
Bottlaender, Michel;
Coulon, Christine;
Ottaviani, Michèle;
Syrota, André

Publication type:

Article

Radiosynthesis of 2- exo-(2′-[18F]Fluoro-3′-(4-fluorophenyl)-pyridin-5′-yl)-7-azabicyclo[2.2.1]heptane ([18F]F2PhEP), a potent epibatidine-based radioligand for nicotinic acetylcholine receptor PET imaging

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2006, v. 49, n. 6, p. 489, doi. 10.1002/jlcr.1063

By:

Roger, Gaëlle;
Hinnen, Françoise;
Valette, Héric;
Saba, Wadad;
Bottlaender, Michel;
Dollé, Frédéric

Publication type:

Article

Radiosynthesis and in vivo evaluation of [11C]Ro-647312: a novel NR1/2B subtype selective NMDA receptor radioligand.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2004, v. 47, n. 13, p. 911, doi. 10.1002/jlcr.877

By:

Dollé, Frédéric;
Valette, Héric;
Demphel, Stéphane;
Coulon, Christine;
Ottaviani, Michelle;
Bottlaender, Michel;
Kassiou, Michael

Publication type:

Article

Influence of P-Glycoprotein Inhibition or Deficiency at the Blood-Brain Barrier on F-2-Fluoro-2-Deoxy- d-glucose (F-FDG) Brain Kinetics.

Published in:

AAPS Journal, 2015, v. 17, n. 3, p. 652, doi. 10.1208/s12248-015-9739-3

By:

Tournier, Nicolas;
Saba, Wadad;
Goutal, Sébastien;
Gervais, Philippe;
Valette, Héric;
Scherrmann, Jean-Michel;
Bottlaender, Michel;
Cisternino, Salvatore

Publication type:

Article

Effects of Selected OATP and/or ABC Transporter Inhibitors on the Brain and Whole-Body Distribution of Glyburide.

Published in:

AAPS Journal, 2013, v. 15, n. 4, p. 1082, doi. 10.1208/s12248-013-9514-2

By:

Tournier, Nicolas;
Saba, Wadad;
Cisternino, Salvatore;
Peyronneau, Marie-Anne;
Damont, Annelaure;
Goutal, Sébastien;
Dubois, Albertine;
Dollé, Frédéric;
Scherrmann, Jean-Michel;
Valette, Héric;
Kuhnast, Bertrand;
Bottlaender, Michel

Publication type:

Article

Discrepancies in the P-glycoprotein-Mediated Transport of F-MPPF: A Pharmacokinetic Study in Mice and Non-human Primates.

Published in:

Pharmaceutical Research, 2012, v. 29, n. 9, p. 2468, doi. 10.1007/s11095-012-0776-7

By:

Tournier, Nicolas;
Cisternino, Salvatore;
Peyronneau, Marie-Anne;
Goutal, Sébastien;
Dolle, Frédéric;
Scherrmann, Jean-Michel;
Bottlaender, Michel;
Saba, Wadad;
Valette, Héric

Publication type:

Article

Differential influence of propofol and isoflurane anesthesia in a non-human primate on the brain kinetics and binding of [18F] DPA-714, a positron emission tomography imaging marker of glial activation.

Published in:

European Journal of Neuroscience, 2015, v. 42, n. 1, p. 1738, doi. 10.1111/ejn.12946

By:

Saba, Wadad;
Goutal, Sébastien;
Kuhnast, Bertrand;
Dollé, Frédéric;
Auvity, Sylvain;
Fontyn, Yoan;
Cayla, Jérôme;
Peyronneau, Marie‐Anne;
Valette, Héric;
Tournier, Nicolas

Publication type:

Article

Imaging Central Nicotinic Acetylcholine Receptors in Baboons with [18F]Fluoro-A-85380.

Published in:

Journal of Nuclear Medicine, 1999, v. 40, n. 8, p. 1374

By:

Valette, Héric;
Bottlaender, Michel;
Dollé, Frédéric;
Guenther, Ilonka;
Fuseau, Chantal;
Coulon, Christine;
Ottaviani, Michele;
Crouzel, Christian

Publication type:

Article

Down-Regulation of Cardiac Muscarinic Receptors Induced by Di-Isopropylfluorophosphate.

Published in:

Journal of Nuclear Medicine, 1997, v. 38, n. 9, p. 1430

By:

Valette, Héric;
Syrota, André;
Fuseau, Chantal

Publication type:

Article

Late Sympathetic Reinnervation and Normalization of Canine Myocardial Beta-Adrenergic Receptor Density Following Denervation.

Published in:

Journal of Nuclear Medicine, 1995, v. 36, n. 9, p. 1726

By:

Valette, Héric;
Syrota, André;
Deleuze, Philippe;
Crouzel, Christian;
Delforge, Jacques;
Fuseau, Chantal;
Loisance, Daniel

Publication type:

Article

Canine Myocardial Beta-Adrenergic, Muscarinic Receptor Densities After Denervation: A PET Study.

Published in:

Journal of Nuclear Medicine, 1995, v. 36, n. 1, p. 140

By:

Valette, Héric;
Deleuze, Philippe;
Syrota, André;
Delforge, Jacques;
Crouzel, Christian;
Fuseau, Chantai;
Loisance, Daniel

Publication type:

Article

Bromine-76-Metabromobenzylguanidine : A PET Radiotracer for Mapping Sympathetic Nerves of the Heart.

Published in:

Journal of Nuclear Medicine, 1993, v. 34, n. 10, p. 1739

By:

Valette, Héric;
Loc'h, Christian;
Mardon, Karine;
Bendriem, Bernard;
Merlet, Pascal;
Fuseau, Chantal;
Sabry, Sana;
Raffel, David;
Mazière, Bernard;
Syrota, André

Publication type:

Article

Prognostic Value of Cardiac Metaiodobenzylguanidine Imaging in Patients with Heart Failure.

Published in:

Journal of Nuclear Medicine, 1992, v. 33, n. 4, p. 471

By:

Merlet, Pascal;
Valette, Héric;
Dubois-Randé, Jean-Luc;
Moyse, Dominique;
Duboc, Denis;
Dove, Patrick;
Bourguignon, Michel Henri;
Benvenuti, Christophe;
Duval, Anne Marie;
Agostini, Denis;
Loisance, Daniel;
Castaigne, Alain;
Syrota, André

Publication type:

Article

Improved Detection of Anterior Left Ventricular Aneurysm with Multiharmonic Fourier Analysis.

Published in:

Journal of Nuclear Medicine, 1990, v. 31, n. 8, p. 1303

By:

Valette, Héric B.;
Bourguignon, Michel H.;
Merlet, Pascal;
Grégoire, Marie-Claude;
Le Guludec, Dominique;
Pascal, Odile;
Briandet, Philippe;
Syrota, André

Publication type:

Article

In vivo quantification of monoamine oxidase A in baboon brain: a PET study using [11C]befloxatone and the multi-injection approach.

Published in:

Journal of Cerebral Blood Flow & Metabolism, 2010, v. 30, n. 4, p. 792, doi. 10.1038/jcbfm.2009.242

By:

Bottlaender, Michel;
Valette, Héric;
Delforge, Jacques;
Saba, Wadad;
Guenther, Ilonka;
Curet, Olivier;
George, Pascal;
Dollé, Frédéric;
Grégoire, Marie-Claude

Publication type:

Article

Decrease of nicotinic receptors in the nigrostriatal system in Parkinson's disease.

Published in:

Journal of Cerebral Blood Flow & Metabolism, 2009, v. 29, n. 9, p. 1601, doi. 10.1038/jcbfm.2009.74

By:

Kas, Aurélie;
Bottlaender, Michel;
Gallezot, Jean Dominique;
Vidailhet, Marie;
Villafane, Gabriel;
Grégoire, Marie Claude;
Coulon, Christine;
Valette, Héric;
Dollé, Frédéric;
Ribeiro, Maria-Joao;
Hantraye, Philippe;
Remy, Philippe

Publication type:

Article

Quantification of cerebral nicotinic acetylcholine receptors by PET using 2-[18F]fluoro-A-85380 and the multiinjection approach.

Published in:

Journal of Cerebral Blood Flow & Metabolism, 2008, v. 28, n. 1, p. 172, doi. 10.1038/sj.jcbfm.9600505

By:

Gallezot, Jean-Dominique;
Bottlaender, Michel A.;
Delforge, Jacques;
Valette, Héric;
Saba, Wadad;
Dolle, Frédéric;
Coulon, Christine M.;
Ottaviani, Michèle P;
Hinnen, Françoise;
Syrota, André;
Grégoire, Marie-Claude

Publication type:

Article

Works by Valette, Héric

Synthesis and preliminary evaluation of a carbon-11-labelled agonist of the α7 nicotinic acetylcholine receptor.

Highly efficient synthesis of [<sup>11</sup>C]S12968 and [<sup>11</sup>C]S12967, for the in vivo imaging of the cardiac calcium channels using PET.

Highly efficient synthesis of [<sup>11</sup>C]Me-QNB, a selective radioligand for the quantification of the cardiac muscarinic receptors using PET.

Highly efficient synthesis of [<sup>11</sup>C]PE2I, a selective radioligand for the quantification of the dopamine transporter using PET.

Synthesis of 2-[<sup>18</sup>F]fluoro-3-[2(S)-2-azetidinylmethoxy]pyridine, a highly potent radioligand for in vivo imaging central nicotinic acetylcholine receptors.

Synthesis and <sup>11</sup>C-labelling of two selective high affinity nicotinic cholinergic agonists for evaluation as radioligands for PET studies.

Transport of Selected PET Radiotracers by Human P-Glycoprotein (ABCB1) and Breast Cancer Resistance Protein (ABCG2): An In Vitro Screening.

In Vivo Imaging of Human Cerebral Nicotinic Acetylcholine Receptors with 2-<sup>18</sup>F-Fluoro-A-85380 and PET.

Biodistribution and Radiation Dosimetry of <sup>18</sup>F-Fluoro-A-85380 in Healthy Volunteers.

In Vivo Quantification of Myocardial Dihydropyridine Binding Sites: A PET Study in Dogs.

Myocardial Kinetics of the<sup> 11</sup>C-Labeled Enantiomers of the Ca<sup>2+</sup> Channel Inhibitor S11568: An In Vivo Study.

[<sup>18</sup>F]ZW-104, a new radioligand for imaging α2-α3-α4/β2 central nicotinic acetylcholine receptors: Evaluation in mutant mice.

[<sup>11</sup>C]SL25.1188, a new reversible radioligand to study the monoamine oxidase type B with PET: Preclinical characterisation in nonhuman primate.

[<sup>18</sup>F]FPhEP and [<sup>18</sup>F]F<sub>2</sub>PhEP, two new epibatidine-based radioligands: Evaluation for imaging nicotinic acetylcholine receptors in baboon brain.

[<sup>11</sup>C]LBT-999: A suitable radioligand for investigation of extra-striatal dopamine transporter with PET.

Acute effects of physostigmine and galantamine on the binding of [<sup>18</sup>F]fluoro-A-85380: A PET study in monkeys.

Anesthesia affects the disposition of [<sup>18</sup>F]fluoro-A-85380: A PET study in monkeys.

Radiosynthesis of 2- exo-(2′-[<sup>18</sup>F]Fluoro-3′-(4-fluorophenyl)-pyridin-5′-yl)-7-azabicyclo[2.2.1]heptane ([<sup>18</sup>F]F<sub>2</sub>PhEP), a potent epibatidine-based radioligand for nicotinic acetylcholine receptor PET imaging

Radiosynthesis and in vivo evaluation of [<sup>11</sup>C]Ro-647312: a novel NR1/2B subtype selective NMDA receptor radioligand.

Influence of P-Glycoprotein Inhibition or Deficiency at the Blood-Brain Barrier on F-2-Fluoro-2-Deoxy- d-glucose (F-FDG) Brain Kinetics.

Effects of Selected OATP and/or ABC Transporter Inhibitors on the Brain and Whole-Body Distribution of Glyburide.

Discrepancies in the P-glycoprotein-Mediated Transport of F-MPPF: A Pharmacokinetic Study in Mice and Non-human Primates.

Differential influence of propofol and isoflurane anesthesia in a non-human primate on the brain kinetics and binding of [<sup>18</sup>F] DPA-714, a positron emission tomography imaging marker of glial activation.

Imaging Central Nicotinic Acetylcholine Receptors in Baboons with [<sup>18</sup>F]Fluoro-A-85380.

Down-Regulation of Cardiac Muscarinic Receptors Induced by Di-Isopropylfluorophosphate.

Late Sympathetic Reinnervation and Normalization of Canine Myocardial Beta-Adrenergic Receptor Density Following Denervation.

Canine Myocardial Beta-Adrenergic, Muscarinic Receptor Densities After Denervation: A PET Study.

Bromine-76-Metabromobenzylguanidine : A PET Radiotracer for Mapping Sympathetic Nerves of the Heart.

Prognostic Value of Cardiac Metaiodobenzylguanidine Imaging in Patients with Heart Failure.

Improved Detection of Anterior Left Ventricular Aneurysm with Multiharmonic Fourier Analysis.

In vivo quantification of monoamine oxidase A in baboon brain: a PET study using [<sup>11</sup>C]befloxatone and the multi-injection approach.

Decrease of nicotinic receptors in the nigrostriatal system in Parkinson's disease.

Quantification of cerebral nicotinic acetylcholine receptors by PET using 2-[<sup>18</sup>F]fluoro-A-85380 and the multiinjection approach.