Works by Valente, Sergio


Results: 93
    1

    Cardioprotection Through Pharmacological Activation of Sirtuin 5 in a Murine Model of Acute Myocardial Infarction.

    Published in:
    Drug Design, Development & Therapy, 2025, v. 19, p. 5489, doi. 10.2147/DDDT.S509337
    By:
    • Castiello, Carola;
    • Efentakis, Panagiotis;
    • Nikolaou, Panagiota-Efstathia;
    • Symeonidi, Lydia;
    • Chania, Christina;
    • Barla, Ioanna;
    • Akrani, Ifigeneia;
    • Kostomitsopoulos, Nikolaos;
    • Gikas, Evangelos;
    • Thomaidis, Nikolaos S;
    • Mikros, Emmanuel;
    • Kleinbongard, Petra;
    • Fioravanti, Rossella;
    • Zwergel, Clemens;
    • Valente, Sergio;
    • Mai, Antonello;
    • Andreadou, Ioanna
    Publication type:
    Article
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    Role of SIRT3 in Microgravity Response: A New Player in Muscle Tissue Recovery.

    Published in:
    Cells (2073-4409), 2023, v. 12, n. 5, p. 691, doi. 10.3390/cells12050691
    By:
    • Aventaggiato, Michele;
    • Barreca, Federica;
    • Vitiello, Laura;
    • Vespa, Simone;
    • Valente, Sergio;
    • Rotili, Dante;
    • Mai, Antonello;
    • Lotti, Lavinia Vittoria;
    • Sansone, Luigi;
    • Russo, Matteo A.;
    • Bizzarri, Mariano;
    • Ferretti, Elisabetta;
    • Tafani, Marco
    Publication type:
    Article
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    EZH2 inhibitors: a patent review (2014-2016).

    Published in:
    Expert Opinion on Therapeutic Patents, 2017, v. 27, n. 7, p. 797, doi. 10.1080/13543776.2017.1316976
    By:
    • Stazi, Giulia;
    • Zwergel, Clemens;
    • Mai, Antonello;
    • Valente, Sergio
    Publication type:
    Article
    11

    LSD1 inhibitors: a patent review (2010-2015).

    Published in:
    Expert Opinion on Therapeutic Patents, 2016, v. 26, n. 5, p. 565, doi. 10.1517/13543776.2016.1165209
    By:
    • Stazi, Giulia;
    • Zwergel, Clemens;
    • Valente, Sergio;
    • Mai, Antonello
    Publication type:
    Article
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    Heterocycle-containing tranylcypromine derivatives endowed with high anti-LSDI activity.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 973, doi. 10.1080/14756366.2022.2052869
    By:
    • Fioravanti, Rossella;
    • Rodriguez, Veronica;
    • Caroli, Jonatan;
    • Chianese, Ugo;
    • Benedetti, Rosaria;
    • Di Bello, Elisabetta;
    • Noce, Beatrice;
    • Zwergel, Clemens;
    • Corinti, Davide;
    • Viña, Dolores;
    • Altucci, Lucia;
    • Mattevi, Andrea;
    • Valente, Sergio;
    • Mai, Antonello
    Publication type:
    Article
    17

    Histone deacetylase inhibitors restore IL-10 expression in lipopolysaccharide-induced cell inflammation and reduce IL-1β and IL-6 production in breast silicone implant in C57BL/6J wild-type murine model.

    Published in:
    Autoimmunity, 2016, v. 49, n. 3, p. 155, doi. 10.3109/08916934.2015.1134510
    By:
    • Di Liddo, Rosa;
    • Valente, Sergio;
    • Taurone, Samanta;
    • Zwergel, Clemens;
    • Marrocco, Biagina;
    • Turchetta, Rosaria;
    • Conconi, Maria Teresa;
    • Scarpa, Carlotta;
    • Bertalot, Thomas;
    • Schrenk, Sandra;
    • Mai, Antonello;
    • Artico, Marco
    Publication type:
    Article
    18

    Mechanisms of mesothelial cell response to viral infections: HDAC1-3 inhibition blocks poly(I:C)-induced type I interferon response and modulates the mesenchymal/inflammatory phenotype.

    Published in:
    Frontiers in Cellular & Infection Microbiology, 2024, p. 1, doi. 10.3389/fcimb.2024.1308362
    By:
    • Trionfetti, Flavia;
    • Montaldo, Claudia;
    • Caiello, Ivan;
    • Bontempi, Giulio;
    • Terri, Michela;
    • Tiberi, Marta;
    • Marchant, Vanessa;
    • Domenici, Alessandro;
    • Menè, Paolo;
    • Cordani, Marco;
    • Zwergel, Clemens;
    • Prencipe, Giusi;
    • Ruiz-Ortega, Marta;
    • Valente, Sergio;
    • Mai, Antonello;
    • Tripodi, Marco;
    • Strippoli, Raffaele
    Publication type:
    Article
    19

    Cytoplasmic HDAC4 regulates the membrane repair mechanism in Duchenne muscular dystrophy.

    Published in:
    Journal of Cachexia, Sarcopenia & Muscle, 2022, v. 13, n. 2, p. 1339, doi. 10.1002/jcsm.12891
    By:
    • Renzini, Alessandra;
    • Marroncelli, Nicoletta;
    • Cavioli, Giorgia;
    • Di Francescantonio, Silvia;
    • Forcina, Laura;
    • Lambridis, Alessandro;
    • Di Giorgio, Eros;
    • Valente, Sergio;
    • Mai, Antonello;
    • Brancolini, Claudio;
    • Giampietri, Claudia;
    • Magenta, Alessandra;
    • De Santa, Francesca;
    • Adamo, Sergio;
    • Coletti, Dario;
    • Moresi, Viviana
    Publication type:
    Article
    20

    OPTIMIZED METHOD FOR DNA EXTRACTION AND PCR AMPLIFICATION IN AROEIRA TREE.

    Published in:
    Bioscience Journal, 2023, v. 39, p. 1, doi. 10.14393/BJ-v39n0a2023-62577
    By:
    • SILVA, Jailson do Nascimento;
    • LINHARES, Amanda Camila dos Santos;
    • PALMIERI, Dario Abel;
    • COSTA, Marcones Ferreira;
    • de SÁ, Gisele Holanda;
    • GOMES, Maria Fernanda da Costa;
    • dos SANTOS, Michelli Ferreira;
    • FEITOZA, Lidiane de Lima;
    • VALENTE, Sérgio Emílio dos Santos
    Publication type:
    Article
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    Tree species used in urban forestry in Brazil: a scientometric review.

    Published in:
    Rodriguésia, 2023, v. 74, p. 1, doi. 10.1590/2175-7860202374047
    By:
    • Baldez Vidal-Couto, Daniela;
    • Reis de Brito, Carolina;
    • Medeiros Mascarenhas Andrade, Isis Leite;
    • Freitas Cerqueira, Amanda;
    • Pires Reis, Igor;
    • Valente Tomasini, Sergio Luiz;
    • Carla Dalmolin, Ândrea;
    • Schramm Mielke, Marcelo
    Publication type:
    Article
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    A lima bean core collection based on molecular markers.

    Published in:
    Scientia Agricola, 2020, v. 77, n. 2, p. 1, doi. 10.1590/1678-992X-2018-0140
    By:
    • Ferreira Gomes, Regina Lucia;
    • Ferreira Costa, Marcones;
    • Alves-Pereira, Alessandro;
    • Bajay, Miklos Maximiliano;
    • Gomes Viana, João Paulo;
    • dos Santos Valente, Sérgio Emílio;
    • Celis de Almeida Lopes, Ângela;
    • Zucchi, Maria Imaculada;
    • Baldin Pinheiro, José
    Publication type:
    Article
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    Novel Targeting of DNA Methyltransferase Activity Inhibits Ewing Sarcoma Cell Proliferation and Enhances Tumor Cell Sensitivity to DNA Damaging Drugs by Activating the DNA Damage Response.

    Published in:
    Frontiers in Endocrinology, 2022, v. 13, p. 1, doi. 10.3389/fendo.2022.876602
    By:
    • Cristalli, Camilla;
    • Manara, Maria Cristina;
    • Valente, Sergio;
    • Pellegrini, Evelin;
    • Bavelloni, Alberto;
    • De Feo, Alessandra;
    • Blalock, William;
    • Di Bello, Elisabetta;
    • Piñeyro, David;
    • Merkel, Angelika;
    • Esteller, Manel;
    • Tirado, Oscar M.;
    • Mai, Antonello;
    • Scotlandi, Katia
    Publication type:
    Article
    38

    Novel Quinoline Compounds Active in Cancer Cells through Coupled DNA Methyltransferase Inhibition and Degradation.

    Published in:
    Cancers, 2020, v. 12, n. 2, p. 447, doi. 10.3390/cancers12020447
    By:
    • Zwergel, Clemens;
    • Fioravanti, Rossella;
    • Stazi, Giulia;
    • Sarno, Federica;
    • Battistelli, Cecilia;
    • Romanelli, Annalisa;
    • Nebbioso, Angela;
    • Mendes, Eduarda;
    • Paulo, Alexandra;
    • Strippoli, Raffaele;
    • Tripodi, Marco;
    • Pechalrieu, Dany;
    • Arimondo, Paola B.;
    • De Luca, Teresa;
    • Del Bufalo, Donatella;
    • Trisciuoglio, Daniela;
    • Altucci, Lucia;
    • Valente, Sergio;
    • Mai, Antonello
    Publication type:
    Article
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    HDAC1/2 control mesothelium/ovarian cancer adhesive interactions impacting on Talin-1-α5β1-integrin-mediated actin cytoskeleton and extracellular matrix protein remodeling.

    Published in:
    Journal of Experimental & Clinical Cancer Research (17569966), 2024, v. 43, n. 1, p. 1, doi. 10.1186/s13046-023-02930-8
    By:
    • Terri, Michela;
    • Sandoval, Pilar;
    • Bontempi, Giulio;
    • Montaldo, Claudia;
    • Tomero-Sanz, Henar;
    • de Turris, Valeria;
    • Trionfetti, Flavia;
    • Pascual-Antón, Lucía;
    • Clares-Pedrero, Irene;
    • Battistelli, Cecilia;
    • Valente, Sergio;
    • Zwergel, Clemens;
    • Mai, Antonello;
    • Rosanò, Laura;
    • del Pozo, Miguel Ángel;
    • Sánchez-Álvarez, Miguel;
    • Cabañas, Carlos;
    • Tripodi, Marco;
    • López-Cabrera, Manuel;
    • Strippoli, Raffaele
    Publication type:
    Article
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    Targeting the anti-apoptotic Bcl-2 family proteins: machine learning virtual screening and biological evaluation of new small molecules.

    Published in:
    Theranostics, 2022, v. 12, n. 5, p. 2427, doi. 10.7150/thno.64233
    By:
    • Valentini, Elisabetta;
    • D'Aguanno, Simona;
    • Di Martile, Marta;
    • Montesano, Camilla;
    • Ferraresi, Virginia;
    • Patsilinakos, Alexandros;
    • Sabatino, Manuela;
    • Antonini, Lorenzo;
    • Chiacchiarini, Martina;
    • Valente, Sergio;
    • Mai, Antonello;
    • Colotti, Gianni;
    • Ragno, Rino;
    • Trisciuoglio, Daniela;
    • Del Bufalo, Donatella
    Publication type:
    Article
    47

    Tranylcypromine‐Based LSD1 Inhibitors: Structure‐Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target Modulation.

    Published in:
    ChemMedChem, 2020, v. 15, n. 7, p. 643, doi. 10.1002/cmdc.201900730
    By:
    • Fioravanti, Rossella;
    • Romanelli, Annalisa;
    • Mautone, Nicola;
    • Di Bello, Elisabetta;
    • Rovere, Annarita;
    • Corinti, Davide;
    • Zwergel, Clemens;
    • Valente, Sergio;
    • Rotili, Dante;
    • Botrugno, Oronza A.;
    • Dessanti, Paola;
    • Vultaggio, Stefania;
    • Vianello, Paola;
    • Cappa, Anna;
    • Binda, Claudia;
    • Mattevi, Andrea;
    • Minucci, Saverio;
    • Mercurio, Ciro;
    • Varasi, Mario;
    • Mai, Antonello
    Publication type:
    Article
    48

    Structure-Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase.

    Published in:
    ChemMedChem, 2017, v. 12, n. 16, p. 1359, doi. 10.1002/cmdc.201700040
    By:
    • Madia, Valentina Noemi;
    • Benedetti, Rosaria;
    • Barreca, Maria Letizia;
    • Ngo, Liza;
    • Pescatori, Luca;
    • Messore, Antonella;
    • Pupo, Giovanni;
    • Saccoliti, Francesco;
    • Valente, Sergio;
    • Mai, Antonello;
    • Scipione, Luigi;
    • Zheng, Yujun George;
    • Tintori, Cristina;
    • Botta, Maurizio;
    • Cecchetti, Violetta;
    • Altucci, Lucia;
    • Di Santo, Roberto;
    • Costi, Roberta
    Publication type:
    Article
    49

    Cover Picture: tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells (ChemMedChem 5/2013).

    Published in:
    ChemMedChem, 2013, v. 8, n. 5, p. 673, doi. 10.1002/cmdc.201390015
    By:
    • Valente, Sergio;
    • Trisciuoglio, Daniela;
    • Tardugno, Maria;
    • Benedetti, Rosaria;
    • Labella, Donatella;
    • Secci, Daniela;
    • Mercurio, Ciro;
    • Boggio, Roberto;
    • Tomassi, Stefano;
    • Di Maro, Salvatore;
    • Novellino, Ettore;
    • Altucci, Lucia;
    • Del Bufalo, Donatella;
    • Mai, Antonello;
    • Cosconati, Sandro
    Publication type:
    Article
    50

    tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells.

    Published in:
    ChemMedChem, 2013, v. 8, n. 5, p. 800, doi. 10.1002/cmdc.201300005
    By:
    • Valente, Sergio;
    • Trisciuoglio, Daniela;
    • Tardugno, Maria;
    • Benedetti, Rosaria;
    • Labella, Donatella;
    • Secci, Daniela;
    • Mercurio, Ciro;
    • Boggio, Roberto;
    • Tomassi, Stefano;
    • Di Maro, Salvatore;
    • Novellino, Ettore;
    • Altucci, Lucia;
    • Del Bufalo, Donatella;
    • Mai, Antonello;
    • Cosconati, Sandro
    Publication type:
    Article