Works by Tuccinardi, Tiziano

Results: 94

A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration.

Published in:

Antioxidants, 2023, v. 12, n. 12, p. 2044, doi. 10.3390/antiox12122044

By:

Berrino, Emanuela;
Carradori, Simone;
Carta, Fabrizio;
Melfi, Francesco;
Gallorini, Marialucia;
Poli, Giulio;
Tuccinardi, Tiziano;
Fernández-Bolaños, José G.;
López, Óscar;
Petzer, Jacobus P.;
Petzer, Anél;
Guglielmi, Paolo;
Secci, Daniela;
Supuran, Claudiu T.

Publication type:

Article

A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by Using a Pharmacophore-based Approach.

Published in:

Molecular Informatics, 2016, v. 35, n. 8/9, p. 434, doi. 10.1002/minf.201501026

By:

Tuccinardi, Tiziano;
Poli, Giulio;
Corchia, Isacco;
Granchi, Carlotta;
Lapillo, Margherita;
Macchia, Marco;
Minutolo, Filippo;
Ortore, Gabriella;
Martinelli, Adriano

Publication type:

Article

An alternative conformation of the N‐terminal loop of human dihydroorotate dehydrogenase drives binding to a potent antiproliferative agent.

Published in:

Acta Crystallographica: Section D, Structural Biology, 2024, v. 80, n. 6, p. 386, doi. 10.1107/S2059798324004066

By:

Alberti, Marta;
Poli, Giulio;
Broggini, Luca;
Sainas, Stefano;
Rizzi, Menico;
Boschi, Donatella;
Ferraris, Davide M.;
Martino, Elena;
Ricagno, Stefano;
Tuccinardi, Tiziano;
Lolli, Marco L.;
Miggiano, Riccardo

Publication type:

Article

Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1 H)-One Scaffold.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 7, p. N.PAG, doi. 10.3390/ph15070768

By:

Ceni, Costanza;
Benko, Michael J.;
Mohamed, Kawthar A.;
Poli, Giulio;
Di Stefano, Miriana;
Tuccinardi, Tiziano;
Digiacomo, Maria;
Valoti, Massimo;
Laprairie, Robert B.;
Macchia, Marco;
Bertini, Simone

Publication type:

Article

New Synthetic Analogues of Natural Polyphenols as Sirtuin 1-Activating Compounds.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 3, p. 339, doi. 10.3390/ph15030339

By:

Bononi, Giulia;
Flori, Lorenzo;
Citi, Valentina;
Acciai, Cecilia;
Nocilla, Viviana;
Martelli, Alma;
Poli, Giulio;
Tuccinardi, Tiziano;
Granchi, Carlotta;
Testai, Lara;
Calderone, Vincenzo;
Minutolo, Filippo

Publication type:

Article

A patent review of lactate dehydrogenase inhibitors (2014–present).

Published in:

Expert Opinion on Therapeutic Patents, 2024, v. 34, n. 11, p. 1121, doi. 10.1080/13543776.2024.2412575

By:

Bononi, Giulia;
Di Bussolo, Valeria;
Tuccinardi, Tiziano;
Minutolo, Filippo;
Granchi, Carlotta

Publication type:

Article

An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present).

Published in:

Expert Opinion on Therapeutic Patents, 2021, v. 31, n. 2, p. 153, doi. 10.1080/13543776.2021.1841166

By:

Bononi, Giulia;
Poli, Giulio;
Rizzolio, Flavio;
Tuccinardi, Tiziano;
Macchia, Marco;
Minutolo, Filippo;
Granchi, Carlotta

Publication type:

Article

A patent review of Monoacylglycerol Lipase (MAGL) inhibitors (2013-2017).

Published in:

Expert Opinion on Therapeutic Patents, 2017, v. 27, n. 12, p. 1341, doi. 10.1080/13543776.2018.1389899

By:

Granchi, Carlotta;
Caligiuri, Isabella;
Minutolo, Filippo;
Rizzolio, Flavio;
Tuccinardi, Tiziano

Publication type:

Article

Metalloprotease inhibitor profiles of human ADAM8 in vitro and in cell-based assays.

Published in:

Biological Chemistry, 2019, v. 400, n. 6, p. 801, doi. 10.1515/hsz-2018-0396

By:

Schlomann, Uwe;
Dorzweiler, Kristina;
Nuti, Elisa;
Tuccinardi, Tiziano;
Rossello, Armando;
Bartsch, Jörg W.

Publication type:

Article

Rutin as promising drug for the treatment of Parkinson's disease: an assessment of MAO-B inhibitory potential by docking, molecular dynamics and DFT studies.

Published in:

Molecular Simulation, 2019, v. 45, n. 18, p. 1563, doi. 10.1080/08927022.2019.1662003

By:

Azam, Faizul;
Abodabos, Honiwa Suliman;
Taban, Ismail M.;
Rfieda, Abdalla R.;
Mahmood, Danish;
Anwar, Md Jamir;
Khan, Shamshir;
Sizochenko, Natalia;
Poli, Giulio;
Tuccinardi, Tiziano;
Ali, Hamed I.

Publication type:

Article

Watermelon: setup and validation of an in silico fragment-based approach.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2356179

By:

Di Stefano, Miriana;
Galati, Salvatore;
Piazza, Lisa;
Gado, Francesca;
Granchi, Carlotta;
Macchia, Marco;
Giordano, Antonio;
Tuccinardi, Tiziano;
Poli, Giulio

Publication type:

Article

An in silico toolbox for the prediction of the potential pathogenic effects of missense mutations in the dimeric region of hRPE65.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2022.2162047

By:

Poli, Giulio;
Demontis, Gian Carlo;
Sodi, Andrea;
Saba, Alessandro;
Rizzo, Stanislao;
Macchia, Marco;
Tuccinardi, Tiziano

Publication type:

Article

Predicting potentially pathogenic effects of hRPE65 missense mutations: a computational strategy based on molecular dynamics simulations.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1765, doi. 10.1080/14756366.2022.2090547

By:

Poli, Giulio;
Barravecchia, Ivana;
Demontis, Gian Carlo;
Sodi, Andrea;
Saba, Alessandro;
Rizzo, Stanislao;
Macchia, Marco;
Tuccinardi, Tiziano

Publication type:

Article

New PIN1 inhibitors identified through a pharmacophore-driven, hierarchical consensus docking strategy.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 145, doi. 10.1080/14756366.2021.1979970

By:

Poli, Giulio;
Di Stefano, Miriana;
Estevez, Joan Arias;
Minutolo, Filippo;
Granchi, Carlotta;
Giordano, Antonio;
Parisi, Salvatore;
Mauceri, Matteo;
Canzonieri, Vincenzo;
Macchia, Marco;
Caligiuri, Isabella;
Tuccinardi, Tiziano;
Rizzolio, Flavio

Publication type:

Article

Development of a fluorogenic ADAMTS-7 substrate.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 2160, doi. 10.1080/14756366.2021.1983808

By:

Santamaria, Salvatore;
Buemi, Frederic;
Nuti, Elisa;
Cuffaro, Doretta;
De Vita, Elena;
Tuccinardi, Tiziano;
Rossello, Armando;
Howell, Steven;
Mehmood, Shahid;
Snijders, Ambrosius P.;
de Groot, Rens

Publication type:

Article

Development of a cheminformatics platform for selectivity analyses of carbonic anhydrase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 365, doi. 10.1080/14756366.2019.1705291

By:

Poli, Giulio;
Galati, Salvatore;
Martinelli, Adriano;
Supuran, Claudiu T.;
Tuccinardi, Tiziano

Publication type:

Article

New insight into structure-activity of furan-based salicylate synthase (MbtI) inhibitors as potential antitubercular agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 823, doi. 10.1080/14756366.2019.1589462

By:

Chiarelli, Laurent R.;
Mori, Matteo;
Beretta, Giangiacomo;
Gelain, Arianna;
Pini, Elena;
Sammartino, Josè Camilla;
Stelitano, Giovanni;
Barlocco, Daniela;
Costantino, Luca;
Lapillo, Margherita;
Poli, Giulio;
Caligiuri, Isabella;
Rizzolio, Flavio;
Bellinzoni, Marco;
Tuccinardi, Tiziano;
Villa, Stefania;
Meneghetti, Fiorella

Publication type:

Article

Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 589, doi. 10.1080/14756366.2019.1571271

By:

Poli, Giulio;
Lapillo, Margherita;
Jha, Vibhu;
Mouawad, Nayla;
Caligiuri, Isabella;
Macchia, Marco;
Minutolo, Filippo;
Rizzolio, Flavio;
Tuccinardi, Tiziano;
Granchi, Carlotta

Publication type:

Article

Binding investigation and preliminary optimisation of the 3-amino-1,2,4-triazin-5(2H)-one core for the development of new Fyn inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 956, doi. 10.1080/14756366.2018.1469017

By:

Poli, Giulio;
Lapillo, Margherita;
Granchi, Carlotta;
Caciolla, Jessica;
Mouawad, Nayla;
Caligiuri, Isabella;
Rizzolio, Flavio;
Langer, Thierry;
Minutolo, Filippo;
Tuccinardi, Tiziano

Publication type:

Article

Development of terphenyl-2-methyloxazol-5(4 H )-one derivatives as selective reversible MAGL inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1240, doi. 10.1080/14756366.2017.1375484

By:

Granchi, Carlotta;
Caligiuri, Isabella;
Bertelli, Eleonora;
Poli, Giulio;
Rizzolio, Flavio;
Macchia, Marco;
Martinelli, Adriano;
Minutolo, Filippo;
Tuccinardi, Tiziano

Publication type:

Article

Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 920, doi. 10.1080/14756366.2017.1344236

By:

Krasavin, Mikhail;
Korsakov, Mikhail;
Ronzhina, Oksana;
Tuccinardi, Tiziano;
Kalinin, Stanislav;
Tanç, Muhammet;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of carbonic anhydrase isoforms I, II, IX and XII with secondary sulfonamides incorporating benzothiazole scaffolds.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1306, doi. 10.3109/14756366.2015.1128427

By:

Petrou, Anthi;
Geronikaki, Athina;
Terzi, Emine;
Guler, Ozen Ozensoy;
Tuccinardi, Tiziano;
Supuran, Claudiu T.

Publication type:

Article

Identification of a new STAT3 dimerization inhibitor through a pharmacophore-based virtual screening approach.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1011, doi. 10.3109/14756366.2015.1079184

By:

Poli, Giulio;
Gelain, Arianna;
Porta, Federica;
Asai, Akira;
Martinelli, Adriano;
Tuccinardi, Tiziano

Publication type:

Article

Reliability analysis and optimization of the consensus docking approach for the development of virtual screening studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 167, doi. 10.1080/14756366.2016.1193736

By:

Poli, Giulio;
Martinelli, Adriano;
Tuccinardi, Tiziano

Publication type:

Article

4-Aryliden-2-methyloxazol-5(4 H )-one as a new scaffold for selective reversible MAGL inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 1, p. 137, doi. 10.3109/14756366.2015.1010530

By:

Granchi, Carlotta;
Rizzolio, Flavio;
Bordoni, Vittorio;
Caligiuri, Isabella;
Manera, Clementina;
Macchia, Marco;
Minutolo, Filippo;
Martinelli, Adriano;
Giordano, Antonio;
Tuccinardi, Tiziano

Publication type:

Article

Receptor-based virtual screening evaluation for the identification of estrogen receptor β ligands.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 4, p. 662, doi. 10.3109/14756366.2014.959946

By:

Tuccinardi, Tiziano;
Poli, Giulio;
Dell'Agnello, Marco;
Granchi, Carlotta;
Minutolo, Filippo;
Martinelli, Adriano

Publication type:

Article

Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 24, p. 17233, doi. 10.3390/ijms242417233

By:

Galati, Salvatore;
Di Stefano, Miriana;
Bertini, Simone;
Granchi, Carlotta;
Giordano, Antonio;
Gado, Francesca;
Macchia, Marco;
Tuccinardi, Tiziano;
Poli, Giulio

Publication type:

Article

Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 18, p. N.PAG, doi. 10.3390/ijms231810653

By:

Di Stefano, Miriana;
Galati, Salvatore;
Ortore, Gabriella;
Caligiuri, Isabella;
Rizzolio, Flavio;
Ceni, Costanza;
Bertini, Simone;
Bononi, Giulia;
Granchi, Carlotta;
Macchia, Marco;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

VenomPred: A Machine Learning Based Platform for Molecular Toxicity Predictions.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 4, p. 2105, doi. 10.3390/ijms23042105

By:

Galati, Salvatore;
Di Stefano, Miriana;
Martinelli, Elisa;
Macchia, Marco;
Martinelli, Adriano;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

Novel 8-Substituted Coumarins That Selectively Inhibit Human Carbonic Anhydrase IX and XII.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 5, p. 1208, doi. 10.3390/ijms20051208

By:

Buran, Kerem;
Bua, Silvia;
Poli, Giulio;
Önen Bayram, F. Esra;
Tuccinardi, Tiziano;
T. Supuran, Claudiu

Publication type:

Article

Extensive Reliability Evaluation of Docking-Based Target-Fishing Strategies.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 5, p. 1023, doi. 10.3390/ijms20051023

By:

Lapillo, Margherita;
Tuccinardi, Tiziano;
Martinelli, Adriano;
Macchia, Marco;
Giordano, Antonio;
Poli, Giulio

Publication type:

Article

Are Insect-Based Foods Healthy? An Evaluation of the Products Sold in European E-Commerce.

Published in:

Foods, 2025, v. 14, n. 9, p. 1450, doi. 10.3390/foods14091450

By:

Copelotti, Emma;
Fratini, Filippo;
Sforza, Giulia;
Tuccinardi, Tiziano;
Demontis, Gian Carlo;
Mancini, Simone

Publication type:

Article

The TRPA1 channel mediates the analgesic action of dipyrone and pyrazolone derivatives.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 13, p. 3397, doi. 10.1111/bph.13129

By:

Nassini, Romina;
Fusi, Camilla;
Materazzi, Serena;
Coppi, Elisabetta;
Tuccinardi, Tiziano;
Marone, Ilaria M;
De Logu, Francesco;
Preti, Delia;
Tonello, Raquel;
Chiarugi, Alberto;
Patacchini, Riccardo;
Geppetti, Pierangelo;
Benemei, Silvia

Publication type:

Article

The influence of Echinacea purpurea leaf microbiota on chicoric acid level.

Published in:

Scientific Reports, 2019, v. 9, n. 1, p. N.PAG, doi. 10.1038/s41598-019-47329-8

By:

Maggini, Valentina;
De Leo, Marinella;
Granchi, Carlotta;
Tuccinardi, Tiziano;
Mengoni, Alessio;
Gallo, Eugenia Rosaria;
Biffi, Sauro;
Fani, Renato;
Pistelli, Luisa;
Firenzuoli, Fabio;
Bogani, Patrizia

Publication type:

Article

Cancer Extracellular Vesicles: Next-Generation Diagnostic and Drug Delivery Nanotools.

Published in:

Cancers, 2020, v. 12, n. 11, p. 3165, doi. 10.3390/cancers12113165

By:

Palazzolo, Stefano;
Memeo, Lorenzo;
Hadla, Mohamad;
Duzagac, Fahriye;
Steffan, Agostino;
Perin, Tiziana;
Canzonieri, Vincenzo;
Tuccinardi, Tiziano;
Caligiuri, Isabella;
Rizzolio, Flavio

Publication type:

Article

Three-Dimensional Interactions Analysis of the Anticancer Target c-Src Kinase with Its Inhibitors.

Published in:

Cancers, 2020, v. 12, n. 8, p. 2327, doi. 10.3390/cancers12082327

By:

Jha, Vibhu;
Macchia, Marco;
Tuccinardi, Tiziano;
Poli, Giulio

Publication type:

Article

Dual Targeting of the Warburg Effect with a Glucose-Conjugated Lactate Dehydrogenase Inhibitor.

Published in:

ChemBioChem, 2013, v. 14, n. 17, p. 2263, doi. 10.1002/cbic.201300562

By:

Calvaresi, Emilia C.;
Granchi, Carlotta;
Tuccinardi, Tiziano;
Di Bussolo, Valeria;
Huigens, Robert W.;
Lee, Hyang Yeon;
Palchaudhuri, Rahul;
Macchia, Marco;
Martinelli, Adriano;
Minutolo, Filippo;
Hergenrother, Paul J.

Publication type:

Article

Investigating the Binding Mode of an Inhibitor of the MBNL1⋅RNA Complex in Myotonic Dystrophy Type 1 (DM1) Leads to the Unexpected Discovery of a DNA-Selective Binder.

Published in:

ChemBioChem, 2012, v. 13, n. 17, p. 2505, doi. 10.1002/cbic.201200602

By:

Wong, Chun-Ho;
Richardson, Stacie L.;
Ho, Yen-Jun;
Lucas, Alex M. H.;
Tuccinardi, Tiziano;
Baranger, Anne M.;
Zimmerman, Steven C.

Publication type:

Article

Identification of a Possible Endocannabinoid-Mediated Mechanism of Action of Cetylated Fatty Acids.

Published in:

Biomolecules (2218-273X), 2025, v. 15, n. 3, p. 363, doi. 10.3390/biom15030363

By:

Bononi, Giulia;
Granchi, Carlotta;
Tuccinardi, Tiziano;
Minutolo, Filippo

Publication type:

Article

Aldose Reductase Differential Inhibitors in Green Tea.

Published in:

Biomolecules (2218-273X), 2020, v. 10, n. 7, p. 1003, doi. 10.3390/biom10071003

By:

Balestri, Francesco;
Poli, Giulio;
Pineschi, Carlotta;
Moschini, Roberta;
Cappiello, Mario;
Mura, Umberto;
Tuccinardi, Tiziano;
Del Corso, Antonella

Publication type:

Article

Dissecting the Activity of Catechins as Incomplete Aldose Reductase Differential Inhibitors through Kinetic and Computational Approaches.

Published in:

Biology (2079-7737), 2022, v. 11, n. 9, p. 1324, doi. 10.3390/biology11091324

By:

Balestri, Francesco;
Poli, Giulio;
Piazza, Lucia;
Cappiello, Mario;
Moschini, Roberta;
Signore, Giovanni;
Tuccinardi, Tiziano;
Mura, Umberto;
Del Corso, Antonella

Publication type:

Article

Steroidal and non-steroidal third-generation aromatase inhibitors induce pain-like symptoms via TRPA1.

Published in:

Nature Communications, 2014, v. 5, n. 12, p. 5736, doi. 10.1038/ncomms6736

By:

Fusi, Camilla;
Materazzi, Serena;
Benemei, Silvia;
Coppi, Elisabetta;
Trevisan, Gabriela;
Marone, Ilaria M.;
Minocci, Daiana;
De Logu, Francesco;
Tuccinardi, Tiziano;
Di Tommaso, Maria Rosaria;
Susini, Tommaso;
Moneti, Gloriano;
Pieraccini, Giuseppe;
Geppetti, Pierangelo;
Nassini, Romina

Publication type:

Article

The Extra-Virgin Olive Oil Polyphenols Oleocanthal and Oleacein Counteract Inflammation-Related Gene and miRNA Expression in Adipocytes by Attenuating NF-κB Activation.

Published in:

Nutrients, 2019, v. 11, n. 12, p. 2855, doi. 10.3390/nu11122855

By:

Carpi, Sara;
Scoditti, Egeria;
Massaro, Marika;
Polini, Beatrice;
Manera, Clementina;
Digiacomo, Maria;
Esposito Salsano, Jasmine;
Poli, Giulio;
Tuccinardi, Tiziano;
Doccini, Stefano;
Santorelli, Filippo Maria;
Carluccio, Maria Annunziata;
Macchia, Marco;
Wabitsch, Martin;
De Caterina, Raffaele;
Nieri, Paola

Publication type:

Article

Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1752, doi. 10.1002/cmdc.201600140

By:

Granchi, Carlotta;
Lapillo, Margherita;
Spena, Concetta Russo;
Rizzolio, Flavio;
Tuccinardi, Tiziano;
Martin, Teresa A.;
Carlson, Kathryn E.;
Katzenellenbogen, John A.;
Minutolo, Filippo

Publication type:

Article

Salicylketoximes That Target Glucose Transporter 1 Restrict Energy Supply to Lung Cancer Cells.

Published in:

ChemMedChem, 2015, v. 10, n. 11, p. 1892, doi. 10.1002/cmdc.201500320

By:

Granchi, Carlotta;
Qian, Yanrong;
Lee, Hyang Yeon;
Paterni, Ilaria;
Pasero, Carolina;
Iegre, Jessica;
Carlson, Kathryn E.;
Tuccinardi, Tiziano;
Chen, Xiaozhuo;
Katzenellenbogen, John A.;
Hergenrother, Paul J.;
Minutolo, Filippo

Publication type:

Article

A Virtual Screening Study of the 18 kDa Translocator Protein using Pharmacophore Models Combined with 3D-QSAR Studies.

Published in:

ChemMedChem, 2009, v. 4, n. 10, p. 1686, doi. 10.1002/cmdc.200900254

By:

Tuccinardi, Tiziano;
Taliani, Sabrina;
Bellandi, Marusca;
Da Settimo, Federico;
Da Pozzo, Eleonora;
Martini, Claudia;
Martinelli, Adriano

Publication type:

Article

Substituted Pyrazolo[3,4- b]pyridines as Potent A<sub>1</sub> Adenosine Antagonists: Synthesis, Biological Evaluation, and Development of an A<sub>1</sub> Bovine Receptor Model.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 898, doi. 10.1002/cmdc.200700355

By:

Tuccinardi, Tiziano;
Schenone, Silvia;
Bondavalli, Francesco;
Brullo, Chiara;
Bruno, Olga;
Mosti, Luisa;
Zizzari, Alessandra Tania;
Tintori, Cristina;
Manetti, Fabrizio;
Ciampi, Osele;
Trincavelli, Maria Letizia;
Martini, Claudia;
Martinelli, Adriano;
Botta, Maurizio

Publication type:

Article

Synthesis of Stable Analogues of Geranylgeranyl Diphosphate Possessing a ( Z, E, E)-Geranylgeranyl Side Chain, Docking Analysis, and Biological Assays for Prenyl Protein Transferase Inhibition.

Published in:

ChemMedChem, 2006, v. 1, n. 2, p. 218, doi. 10.1002/cmdc.200500010

By:

Minutolo, Filippo;
Bertini, Simone;
Betti, Laura;
Danesi, Romano;
Gervasi, Gianbattista;
Giannaccini, Gino;
Martinelli, Adriano;
Papini, Anna Maria;
Peroni, Elisa;
Placanica, Giorgio;
Rapposelli, Simona;
Tuccinardi, Tiziano;
Macchia, Marco

Publication type:

Article

Stereoselectivity of Aldose Reductase in the Reduction of Glutathionyl-Hydroxynonanal Adduct.

Published in:

Antioxidants, 2019, v. 8, n. 10, p. 502, doi. 10.3390/antiox8100502

By:

Balestri, Francesco;
Barracco, Vito;
Renzone, Giovanni;
Tuccinardi, Tiziano;
Pomelli, Christian Silvio;
Cappiello, Mario;
Lessi, Marco;
Rotondo, Rossella;
Bellina, Fabio;
Scaloni, Andrea;
Mura, Umberto;
Del Corso, Antonella;
Moschini, Roberta

Publication type:

Article

Former Foodstuff Products in Tenebrio Molitor Rearing: Effects on Growth, Chemical Composition, Microbiological Load, and Antioxidant Status.

Published in:

Animals (2076-2615), 2019, v. 9, n. 8, p. 484, doi. 10.3390/ani9080484

By:

Mancini, Simone;
Fratini, Filippo;
Turchi, Barbara;
Mattioli, Simona;
Dal Bosco, Alessandro;
Tuccinardi, Tiziano;
Nozic, Sanjin;
Paci, Gisella

Publication type:

Article