Works by Tramontano, Enzo


Results: 83
    1
    2
    3
    4
    5
    6
    7
    8
    9
    10

    Targeting SARS-CoV-2 nsp13 Helicase and Assessment of Druggability Pockets: Identification of Two Potent Inhibitors by a Multi-Site In Silico Drug Repurposing Approach.

    Published in:
    Molecules, 2022, v. 27, n. 21, p. 7522, doi. 10.3390/molecules27217522
    By:
    • Romeo, Isabella;
    • Ambrosio, Francesca Alessandra;
    • Costa, Giosuè;
    • Corona, Angela;
    • Alkhatib, Mohammad;
    • Salpini, Romina;
    • Lemme, Saverio;
    • Vergni, Davide;
    • Svicher, Valentina;
    • Santoro, Maria Mercedes;
    • Tramontano, Enzo;
    • Ceccherini-Silberstein, Francesca;
    • Artese, Anna;
    • Alcaro, Stefano
    Publication type:
    Article
    11
    12
    13
    14
    15
    16
    17
    18
    19
    20

    Natural Product Kuwanon-L Inhibits HIV-1 Replication through Multiple Target Binding.

    Published in:
    ChemBioChem, 2017, v. 18, n. 4, p. 374, doi. 10.1002/cbic.201600592
    By:
    • Martini, Riccardo;
    • Esposito, Francesca;
    • Corona, Angela;
    • Ferrarese, Roberto;
    • Ceresola, Elisa Rita;
    • Visconti, Laura;
    • Tintori, Cristina;
    • Barbieri, Alessandro;
    • Calcaterra, Andrea;
    • Iovine, Valentina;
    • Canducci, Filippo;
    • Tramontano, Enzo;
    • Botta, Maurizio
    Publication type:
    Article
    21
    22
    23
    24

    The antipsychotic drug lurasidone inhibits coronaviruses by affecting multiple targets.

    Published in:
    Frontiers in Cellular & Infection Microbiology, 2024, p. 1, doi. 10.3389/fcimb.2024.1487604
    By:
    • Baroni, Sara;
    • Carletti, Tea;
    • Donalisio, Manuela;
    • Arduino, Irene;
    • Cazzaniga, Irene;
    • Giorgino, Toni;
    • Esposito, Francesca;
    • Porta, Alessia;
    • Diomede, Luisa;
    • De Luigi, Ada;
    • Gobbi, Marco;
    • Lembo, David;
    • Marcello, Alessandro;
    • Tramontano, Enzo;
    • Milani, Mario;
    • Mastrangelo, Eloise
    Publication type:
    Article
    25
    26
    27

    Cytopathic SARS-CoV-2 screening on VERO-E6 cells in a large-scale repurposing effort.

    Published in:
    Scientific Data, 2022, v. 9, n. 1, p. 1, doi. 10.1038/s41597-022-01532-x
    By:
    • Zaliani, Andrea;
    • Vangeel, Laura;
    • Reinshagen, Jeanette;
    • Iaconis, Daniela;
    • Kuzikov, Maria;
    • Keminer, Oliver;
    • Wolf, Markus;
    • Ellinger, Bernhard;
    • Esposito, Francesca;
    • Corona, Angela;
    • Tramontano, Enzo;
    • Manelfi, Candida;
    • Herzog, Katja;
    • Jochmans, Dirk;
    • De Jonghe, Steven;
    • Chiu, Winston;
    • Francken, Thibault;
    • Schepers, Joost;
    • Collard, Caroline;
    • Abbasi, Kayvan
    Publication type:
    Article
    28
    29

    Development and Identification of a Novel Anti-HIV-1 Peptide Derived by Modification of the N-Terminal Domain of HIV-1 Integrase.

    Published in:
    Frontiers in Microbiology, 2016, p. 1, doi. 10.3389/fmicb.2016.00845
    By:
    • Sala, Marina;
    • Spensiero, Antonia;
    • Esposito, Francesca;
    • Scala, Maria C.;
    • Vernieri, Ermelinda;
    • Bertamino, Alessia;
    • Manfra, Michele;
    • Carotenuto, Alfonso;
    • Grieco, Paolo;
    • Novellino, Ettore;
    • Cadeddu, Marta;
    • Tramontano, Enzo;
    • Schols, Dominique;
    • Campiglia, Pietro;
    • Gomez-Monterrey, Isabel M.
    Publication type:
    Article
    30
    31
    32

    Cover Picture: Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors (ChemMedChem 16/2016).

    Published in:
    ChemMedChem, 2016, v. 11, n. 16, p. 1669, doi. 10.1002/cmdc.201600392
    By:
    • Corona, Angela;
    • Desantis, Jenny;
    • Massari, Serena;
    • Distinto, Simona;
    • Masaoka, Takashi;
    • Sabatini, Stefano;
    • Esposito, Francesca;
    • Manfroni, Giuseppe;
    • Maccioni, Elias;
    • Cecchetti, Violetta;
    • Pannecouque, Christophe;
    • Le Grice, Stuart F. J.;
    • Tramontano, Enzo;
    • Tabarrini, Oriana
    Publication type:
    Article
    33

    Design, Synthesis, and Biological Evaluation of 1,3-Diarylpropenones as Dual Inhibitors of HIV-1 Reverse Transcriptase.

    Published in:
    ChemMedChem, 2014, v. 9, n. 8, p. 1869, doi. 10.1002/cmdc.201402015
    By:
    • Meleddu, Rita;
    • Cannas, Valeria;
    • Distinto, Simona;
    • Sarais, Giorgia;
    • Del Vecchio, Claudia;
    • Esposito, Francesca;
    • Bianco, Giulia;
    • Corona, Angela;
    • Cottiglia, Filippo;
    • Alcaro, Stefano;
    • Parolin, Cristina;
    • Artese, Anna;
    • Scalise, Daniela;
    • Fresta, Massimo;
    • Arridu, Antonella;
    • Ortuso, Francesco;
    • Maccioni, Elias;
    • Tramontano, Enzo
    Publication type:
    Article
    34

    Biological Activities of Aerial Parts Extracts of Euphorbia characias.

    Published in:
    BioMed Research International, 2016, v. 2016, p. 1, doi. 10.1155/2016/1538703
    By:
    • Pisano, Maria Barbara;
    • Cosentino, Sofia;
    • Viale, Silvia;
    • Spanò, Delia;
    • Corona, Angela;
    • Esposito, Francesca;
    • Tramontano, Enzo;
    • Montoro, Paola;
    • Tuberoso, Carlo Ignazio Giovanni;
    • Medda, Rosaria;
    • Pintus, Francesca
    Publication type:
    Article
    35
    36
    37
    38
    39
    40
    41
    42
    43
    44

    Cognitive Impairment and Risk of Depressive Episodes from a Bipolar Spectrum Perspective: A Case-Control Study in Older Adults during the COVID-19 Lockdown.

    Published in:
    Psychiatry International, 2024, v. 5, n. 3, p. 482, doi. 10.3390/psychiatryint5030034
    By:
    • Primavera, Diego;
    • Bert, Fabrizio;
    • Romano, Ferdinando;
    • La Torre, Giuseppe;
    • Gonzalez, Cesar Ivan Aviles;
    • Perra, Alessandra;
    • Fragoso-Castilla, Pedro José;
    • Guerra Muñoz, Martha Esther;
    • Tramontano, Enzo;
    • Machado, Sergio;
    • Nardi, Antonio Egidio;
    • Sancassiani, Federica;
    • Carta, Mauro Giovanni
    Publication type:
    Article
    45
    46
    47
    48
    49
    50

    The Stability of Social and Behavioral Rhythms and Unexpected Low Rate of Relevant Depressive Symptoms in Old Adults during the COVID-19 Pandemic.

    Published in:
    Journal of Clinical Medicine, 2024, v. 13, n. 7, p. 2005, doi. 10.3390/jcm13072005
    By:
    • Sancassiani, Federica;
    • Cossu, Giulia;
    • Cantone, Elisa;
    • Romano, Ferdinando;
    • Perra, Alessandra;
    • Urban, Antonio;
    • Pinna, Samantha;
    • Del Giacco, Stefano;
    • Littera, Roberto;
    • Firinu, Davide;
    • Chessa, Luchino;
    • Tramontano, Enzo;
    • Nardi, Antonio Egidio;
    • Carta, Mauro Giovanni
    Publication type:
    Article