Works by Taliani, Sabrina


Results: 43
    1

    A combined approach of structure‐based virtual screening and NMR to interrupt the PD‐1/PD‐L1 axis: Biphenyl‐benzimidazole containing compounds as novel PD‐L1 inhibitors.

    Published in:
    Archiv der Pharmazie, 2024, v. 357, n. 3, p. 1, doi. 10.1002/ardp.202300583
    By:
    • Donati, Greta;
    • Viviano, Monica;
    • D'Amore, Vincenzo Maria;
    • Cipriano, Alessandra;
    • Diakogiannaki, Isidora;
    • Amato, Jussara;
    • Tomassi, Stefano;
    • Brancaccio, Diego;
    • Russomanno, Pasquale;
    • Di Leva, Francesco Saverio;
    • Arosio, Daniela;
    • Seneci, Pierfausto;
    • Taliani, Sabrina;
    • Magiera‐Mularz, Katarzyna;
    • Musielak, Bogdan;
    • Skalniak, Lukasz;
    • Holak, Tad A.;
    • Castellano, Sabrina;
    • La Pietra, Valeria;
    • Marinelli, Luciana
    Publication type:
    Article
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    Enriching the Arsenal of Pharmacological Tools against MICAL2.

    Published in:
    Molecules, 2021, v. 26, n. 24, p. 7519, doi. 10.3390/molecules26247519
    By:
    • Barravecchia, Ivana;
    • Barresi, Elisabetta;
    • Russo, Camilla;
    • Scebba, Francesca;
    • De Cesari, Chiara;
    • Mignucci, Valerio;
    • De Luca, Davide;
    • Salerno, Silvia;
    • La Pietra, Valeria;
    • Giustiniano, Mariateresa;
    • Pelliccia, Sveva;
    • Brancaccio, Diego;
    • Donati, Greta;
    • Da Settimo, Federico;
    • Taliani, Sabrina;
    • Angeloni, Debora;
    • Marinelli, Luciana
    Publication type:
    Article
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    Apoptosis Therapy in Cancer: The First Single-molecule Co-activating p53 and the Translocator Protein in Glioblastoma.

    Published in:
    Scientific Reports, 2014, p. 1, doi. 10.1038/srep04749
    By:
    • Daniele, Simona;
    • Taliani, Sabrina;
    • Da Pozzo, Eleonora;
    • Giacomelli, Chiara;
    • Costa, Barbara;
    • Trincavelli, Maria Letizia;
    • Rossi, Leonardo;
    • Pietra, Valeria La;
    • Barresi, Elisabetta;
    • Carotenuto, Alfonso;
    • Limatola, Antonio;
    • Lamberti, Anna;
    • Marinelli, Luciana;
    • Novellino, Ettore;
    • Da Settimo, Federico;
    • Martini, Claudia
    Publication type:
    Article
    17

    Derivatives of Benzimidazol-2-ylquinoline and Benzimidazol-2-ylisoquinoline as Selective A<sub>1</sub> Adenosine Receptor Antagonists with Stimulant Activity on Human Colon Motility.

    Published in:
    ChemMedChem, 2011, v. 6, n. 10, p. 1909, doi. 10.1002/cmdc.201100284
    By:
    • Cosimelli, Barbara;
    • Taliani, Sabrina;
    • Greco, Giovanni;
    • Novellino, Ettore;
    • Sala, Annalisa;
    • Severi, Elda;
    • Da Settimo, Federico;
    • La Motta, Concettina;
    • Pugliesi, Isabella;
    • Antonioli, Luca;
    • Fornai, Matteo;
    • Colucci, Rocchina;
    • Blandizzi, Corrado;
    • Daniele, Simona;
    • Trincavelli, Maria Letizia;
    • Martini, Claudia
    Publication type:
    Article
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    A<sub>1</sub> adenosine receptor antagonists, 3-aryl[1,2,4]triazino[4,3- a]benzimidazol-4-(10 H)-ones (ATBIs) and N-alkyl and N-acyl-(7-substituted-2-phenylimidazo[1,2- a][1,3,5]triazin-4-yl)amines (ITAs): Different recognition of bovine and human binding sites

    Published in:
    Drug Development Research, 2004, v. 63, n. 1, p. 1, doi. 10.1002/ddr.10366
    By:
    • Da Settimo, Federico;
    • Primofiore, Giampaolo;
    • Taliani, Sabrina;
    • La Motta, Concettina;
    • Novellino, Ettore;
    • Greco, Giovanni;
    • Lavecchia, Antonio;
    • Cosimelli, Barbara;
    • Iadanza, Manuela;
    • Klotz, Karl-Norbert;
    • Tuscano, Daniela;
    • Trincavelli, Maria Letizia;
    • Martini, Claudia
    Publication type:
    Article
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    Enantiomeric 4-Acylamino-6-alkyloxy-2 Alkylthiopyrimidines As Potential A<sub>3</sub> Adenosine Receptor Antagonists: HPLC Chiral Resolution and Absolute Configuration Assignment by a Full Set of Chiroptical Spectroscopy.

    Published in:
    Chirality, 2016, v. 28, n. 5, p. 434, doi. 10.1002/chir.22599
    By:
    • Rossi, Daniela;
    • Nasti, Rita;
    • Marra, Annamaria;
    • Meneghini, Silvia;
    • Mazzeo, Giuseppe;
    • Longhi, Giovanna;
    • Memo, Maurizio;
    • Cosimelli, Barbara;
    • Greco, Giovanni;
    • Novellino, Ettore;
    • Da Settimo, Federico;
    • Martini, Claudia;
    • Taliani, Sabrina;
    • Abbate, Sergio;
    • Collina, Simona
    Publication type:
    Article
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    18 kDa TSPO targeting drives polarized human microglia towards a protective and restorative neurosteroidome profile.

    Published in:
    Cellular & Molecular Life Sciences, 2025, v. 82, n. 1, p. 1, doi. 10.1007/s00018-024-05544-1
    By:
    • Germelli, Lorenzo;
    • Angeloni, Elisa;
    • Da Pozzo, Eleonora;
    • Tremolanti, Chiara;
    • De Felice, Martina;
    • Giacomelli, Chiara;
    • Marchetti, Laura;
    • Muscatello, Beatrice;
    • Barresi, Elisabetta;
    • Taliani, Sabrina;
    • Da Settimo Passetti, Federico;
    • Trincavelli, Maria Letizia;
    • Martini, Claudia;
    • Costa, Barbara
    Publication type:
    Article
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    Carbonic anhydrase activation profile of indole-based derivatives.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1783, doi. 10.1080/14756366.2021.1959573
    By:
    • Barresi, Elisabetta;
    • Ravichandran, Rahul;
    • Germelli, Lorenzo;
    • Angeli, Andrea;
    • Baglini, Emma;
    • Salerno, Silvia;
    • Marini, Anna Maria;
    • Costa, Barbara;
    • Da Pozzo, Eleonora;
    • Martini, Claudia;
    • Da Settimo, Federico;
    • Supuran, Claudiu;
    • Cosconati, Sandro;
    • Taliani, Sabrina
    Publication type:
    Article
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    Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1874, doi. 10.1080/14756366.2021.1956913
    By:
    • Baglini, Emma;
    • Ravichandran, Rahul;
    • Berrino, Emanuela;
    • Salerno, Silvia;
    • Barresi, Elisabetta;
    • Marini, Anna Maria;
    • Viviano, Monica;
    • Castellano, Sabrina;
    • Da Settimo, Federico;
    • Supuran, Claudiu T.;
    • Cosconati, Sandro;
    • Taliani, Sabrina
    Publication type:
    Article
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    Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1697, doi. 10.1080/14756366.2019.1666836
    By:
    • Milite, Ciro;
    • Amendola, Giorgio;
    • Nocentini, Alessio;
    • Bua, Silvia;
    • Cipriano, Alessandra;
    • Barresi, Elisabetta;
    • Feoli, Alessandra;
    • Novellino, Ettore;
    • Da Settimo, Federico;
    • Supuran, Claudiu T.;
    • Castellano, Sabrina;
    • Cosconati, Sandro;
    • Taliani, Sabrina
    Publication type:
    Article
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    Sex Differences in Blood Accumulation of Neurodegenerative-Related Proteins and Antioxidant Responses to Regular Physical Exercise.

    Published in:
    Journal of Molecular Neuroscience, 2024, v. 74, n. 4, p. 1, doi. 10.1007/s12031-024-02278-4
    By:
    • Chelucci, Elisa;
    • Scarfò, Giorgia;
    • Piccarducci, Rebecca;
    • Rizza, Antonio;
    • Fusi, Jonathan;
    • Epifani, Francesco;
    • Carpi, Sara;
    • Polini, Beatrice;
    • Betti, Laura;
    • Costa, Barbara;
    • Taliani, Sabrina;
    • Cela, Vito;
    • Artini, Paolo;
    • Daniele, Simona;
    • Martini, Claudia;
    • Franzoni, Ferdinando
    Publication type:
    Article
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    TSPO Radioligands for Neuroinflammation: An Overview.

    Published in:
    Molecules, 2024, v. 29, n. 17, p. 4212, doi. 10.3390/molecules29174212
    By:
    • Salerno, Silvia;
    • Viviano, Monica;
    • Baglini, Emma;
    • Poggetti, Valeria;
    • Giorgini, Doralice;
    • Castagnoli, Jacopo;
    • Barresi, Elisabetta;
    • Castellano, Sabrina;
    • Da Settimo, Federico;
    • Taliani, Sabrina
    Publication type:
    Article
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