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Synthetically accessible de novo design using reaction vectors: Application to PARP1 inhibitors**.
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- Molecular Informatics, 2024, v. 43, n. 4, p. 1, doi. 10.1002/minf.202300183
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- Article
Privileged Scaffolds for Potent and Specific Inhibitors of Mono-ADP-Ribosylating PARPs.
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- Molecules, 2023, v. 28, n. 15, p. 5849, doi. 10.3390/molecules28155849
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- Article
From Serendipity to Rational Identification of the 5,6,7,8-Tetrahydrobenzo[4,5]thieno[2,3- d ]pyrimidin-4(3 H)-one Core as a New Chemotype of AKT1 Inhibitors for Acute Myeloid Leukemia.
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- Pharmaceutics, 2022, v. 14, n. 11, p. 2295, doi. 10.3390/pharmaceutics14112295
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- Article
From Quinoline to Quinazoline‐Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search.
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- ChemMedChem, 2021, v. 16, n. 19, p. 3044, doi. 10.1002/cmdc.202100282
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- Article
Bis-3-Chloropiperidines Targeting TAR RNA as A Novel Strategy to Impair the HIV-1 Nucleocapsid Protein.
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- Molecules, 2021, v. 26, n. 7, p. 1874, doi. 10.3390/molecules26071874
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- Article
Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 19, p. 7037, doi. 10.3390/ijms21197037
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- Article
3,7-Dihydroxytropolones Inhibit Initiation of Hepatitis B Virus Minus-Strand DNA Synthesis.
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- Molecules, 2020, v. 25, n. 19, p. 4434, doi. 10.3390/molecules25194434
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- Article
1,2,4-Triazolo[1,5-a]pyrimidines as a Novel Class of Inhibitors of the HIV-1 Reverse Transcriptase-Associated Ribonuclease H Activity.
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- Molecules, 2020, v. 25, n. 5, p. 1183, doi. 10.3390/molecules25051183
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- Article
Cover Picture: Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues (ChemMedChem 16/2017).
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- ChemMedChem, 2017, v. 12, n. 16, p. 1224, doi. 10.1002/cmdc.201700470
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- Article
Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues.
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- ChemMedChem, 2017, v. 12, n. 16, p. 1293, doi. 10.1002/cmdc.201700286
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- Article
Cover Picture: Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors (ChemMedChem 16/2016).
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- ChemMedChem, 2016, v. 11, n. 16, p. 1669, doi. 10.1002/cmdc.201600392
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- Article
Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors.
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- ChemMedChem, 2016, v. 11, n. 16, p. 1709, doi. 10.1002/cmdc.201600015
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- Article
The Pyrazolobenzothiazine Core as a New Chemotype of p38 Alpha Mitogen-Activated Protein Kinase Inhibitors.
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- Chemical Biology & Drug Design, 2015, v. 86, n. 4, p. 531, doi. 10.1111/cbdd.12516
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- Article
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity.
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- ChemMedChem, 2013, v. 8, n. 12, p. 1941, doi. 10.1002/cmdc.201300287
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- Article
Design, Synthesis, and Evaluation of WC5 Analogues as Inhibitors of Human Cytomegalovirus Immediate-Early 2 Protein, a Promising Target for Anti-HCMV Treatment.
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- ChemMedChem, 2013, v. 8, n. 8, p. 1403, doi. 10.1002/cmdc.201300106
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- Article
6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis.
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- Chemical Biology & Drug Design, 2012, v. 80, n. 5, p. 781, doi. 10.1111/cbdd.12022
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- Article
Structural Investigation of the Naphthyridone Scaffold: Identification of a 1,6-Naphthyridone Derivative with Potent and Selective Anti-HIV Activity.
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- ChemMedChem, 2011, v. 6, n. 7, p. 1249, doi. 10.1002/cmdc.201100073
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- Article
N-Benzoyl-N-methylsulfonylanthranilates: unexpected cyclization reaction to 4-alkoxy-2,1-benzothiazines.
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- ARKIVOC: Online Journal of Organic Chemistry, 2011, p. 165
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- Article
Inside Cover: Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives (ChemMedChem 11/2010).
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- ChemMedChem, 2010, v. 5, n. 11, p. 1798, doi. 10.1002/cmdc.201090050
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- Article
Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives.
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- ChemMedChem, 2010, v. 5, n. 11, p. 1880, doi. 10.1002/cmdc.201000267
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- Article
2-Phenylquinolones as Inhibitors of the HIV-1 Tat-TAR Interaction.
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- ChemMedChem, 2009, v. 4, n. 6, p. 935, doi. 10.1002/cmdc.200800437
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- Article
Cell-dependent interference of a series of new 6-aminoquinolone derivatives with viral (HIV/CMV) transactivation.
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- Journal of Antimicrobial Chemotherapy (JAC), 2005, v. 56, n. 5, p. 847, doi. 10.1093/jac/dki328
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- Article
8-Methyl-7-substituted-1,6-naphthyridine-3-carboxylic acids as New 6-desfluoroquinolone antibacterials.
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- Journal of Heterocyclic Chemistry, 1999, v. 36, n. 4, p. 953, doi. 10.1002/jhet.5570360422
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- Article
4 H-1-benzothiopyran-4-one-3-carboxylic acids and 3,4-dihydro-2 H-isothiazolo[5,4- b.
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- Journal of Heterocyclic Chemistry, 1993, v. 30, n. 4, p. 1143, doi. 10.1002/jhet.5570300455
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- Article
1,4-Benzothiazine-2-carboxylic acid 1-oxides as analogues of antibacterial quinolones.
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- Journal of Heterocyclic Chemistry, 1992, v. 29, n. 2, p. 375, doi. 10.1002/jhet.5570290215
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- Article