Works matching AU Siwek, Agata

Results: 75

Computational studies of the cyclization of thiosemicarbazides.

Published in:

Journal of Physical Organic Chemistry, 2007, v. 20, n. 7, p. 463, doi. 10.1002/poc.1179

By:

Siwek, Agata;
Paneth, Piotr

Publication type:

Article

The antidepressant-like activity of chiral xanthone derivatives may be mediated by 5-HT1A receptor and β-arrestin signalling.

Published in:

Journal of Psychopharmacology, 2020, v. 34, n. 12, p. 1431, doi. 10.1177/0269881120959605

By:

Sałaciak, Kinga;
Głuch-Lutwin, Monika;
Siwek, Agata;
Szafarz, Małgorzata;
Kazek, Grzegorz;
Bednarski, Marek;
Nowiński, Leszek;
Mitchell, Emma;
Jastrzębska-Więsek, Magdalena;
Partyka, Anna;
Wesołowska, Anna;
Kołaczkowski, Marcin;
Szkaradek, Natalia;
Marona, Henryk;
Sapa, Jacek;
Pytka, Karolina

Publication type:

Article

Lack of NMDA–AMPA interaction in antidepressant-like effect of CGP 37849, an antagonist of NMDA receptor, in the forced swim test.

Published in:

Journal of Neural Transmission, 2008, v. 115, n. 11, p. 1519, doi. 10.1007/s00702-008-0128-2

By:

Dybała, Małgorzata;
Siwek, Agata;
Poleszak, Ewa;
Pilc, Andrzej;
Nowak, Gabriel

Publication type:

Article

Synthetic route to isotopically labelled-oxamate.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2011, v. 54, n. 6, p. 344, doi. 10.1002/jlcr.1876

By:

Siwek, Agata;
Trotsko, Nazar;
Wujec, Monika;
Kamiński, Rafał;
Paneth, Piotr

Publication type:

Article

Anti-inflammatory effects of new human histamine H3 receptor ligands with flavonoid structure on BV-2 neuroinflammation.

Published in:

Inflammation Research, 2023, v. 72, n. 2, p. 181, doi. 10.1007/s00011-022-01658-z

By:

Honkisz-Orzechowska, Ewelina;
Popiołek-Barczyk, Katarzyna;
Linart, Zuzanna;
Filipek-Gorzała, Jadwiga;
Rudnicka, Anna;
Siwek, Agata;
Werner, Tobias;
Stark, Holger;
Chwastek, Jakub;
Starowicz, Katarzyna;
Kieć-Kononowicz, Katarzyna;
Łażewska, Dorota

Publication type:

Article

Reproductive and fetal toxicity studies of histamine H3 receptor antagonist DL76 used in mice to prevent maximal electroshock-induced seizure.

Published in:

Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1364353

By:

Bastaki, Salim M.;
Abdulrazzaq, Yousef M.;
Zidan, Marwan Abdelrahim;
Shafiullah, Mohamed;
Alaryani, Saif Ghdayer;
Alnuaimi, Fatima Awad;
Adeghate, Ernest;
Mohsin, Sahar;
Akour, Amal;
Siwek, Agata;
Łażewska, Dorota;
Kieć-Kononowicz, Katarzyna;
Sadek, Bassem

Publication type:

Article

Chemically Homogenous Compounds with Antagonistic Properties at All α1-Adrenoceptor Subtypes but not β1-Adrenoceptor Attenuate Adrenaline-Induced Arrhythmia in Rats.

Published in:

Frontiers in Pharmacology, 2016, p. 1, doi. 10.3389/fphar.2016.00229

By:

Pytka, Karolina;
Lustyk, Klaudia;
Żmudzka, Elżbieta;
Kotańska, Magdalena;
Siwek, Agata;
Zygmunt, Małgorzata;
Dziedziczak, Agnieszka;
Śniecikowska, Joanna;
Olczyk, Adrian;
Gałuszka, Adam;
Śmieja, Jarosław;
Waszkielewicz, Anna M.;
Marona, Henryk;
Filipek, Barbara;
Sapa, Jacek;
Mogilski, Szczepan;
Akar, Fadi G.;
Heijman, Jordi;
Baartscheer, Antonius

Publication type:

Article

Characteristics of metabolic stability and the cell permeability of 2‐pyrimidinyl‐piperazinyl‐alkyl derivatives of 1H‐imidazo[2,1‐f]purine‐2,4(3H,8H)‐dione with antidepressant‐ and anxiolytic‐like activities

Published in:

Chemical Biology & Drug Design, 2019, v. 93, n. 4, p. 511, doi. 10.1111/cbdd.13442

By:

Zagórska, Agnieszka;
Partyka, Anna;
Bucki, Adam;
Kołaczkowski, Marcin;
Jastrzębska‐Więsek, Magdalena;
Czopek, Anna;
Siwek, Agata;
Głuch‐Lutwin, Monika;
Bednarski, Marek;
Bajda, Marek;
Jończyk, Jakub;
Piska, Kamil;
Koczurkiewicz, Paulina;
Wesołowska, Anna;
Pawłowski, Maciej

Publication type:

Article

Design, synthesis, and anticonvulsant activity of some derivatives of xanthone with aminoalkanol moieties.

Published in:

Chemical Biology & Drug Design, 2017, v. 89, n. 3, p. 339, doi. 10.1111/cbdd.12842

By:

Waszkielewicz, Anna M.;
Słoczyńska, Karolina;
Pękala, Elżbieta;
Żmudzki, Paweł;
Siwek, Agata;
Gryboś, Anna;
Marona, Henryk

Publication type:

Article

Synthesis, Antidepressant Evaluation and Docking Studies of Long-Chain Alkylnitroquipazines as Serotonin Transporter Inhibitors.

Published in:

Chemical Biology & Drug Design, 2013, v. 81, n. 6, p. 695, doi. 10.1111/cbdd.12116

By:

Gabrielsen, Mari;
Wołosewicz, Karol;
Zawadzka, Anna;
Kossakowski, Jerzy;
Nowak, Gabriel;
Wolak, Małgorzata;
Stachowicz, Katarzyna;
Siwek, Agata;
Ravna, Aina W.;
Kufareva, Irina;
Kozerski, Lech;
Bednarek, Elżbieta;
Sitkowski, Jerzy;
Bocian, Wojciech;
Abagyan, Ruben;
Bojarski, Andrzej J.;
Sylte, Ingebrigt;
Chilmonczyk, Zdzisław

Publication type:

Article

Multifunctional, Fluorene‐Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease.

Published in:

Angewandte Chemie International Edition, 2025, v. 64, n. 6, p. 1, doi. 10.1002/anie.202420510

By:

Panek, Dawid;
Pasieka, Anna;
Jończyk, Jakub;
Gawlińska, Milena;
Zaręba, Paula;
Siwek, Agata;
Wolak, Małgorzata;
Mordyl, Barbara;
Głuch‐Lutwin, Monika;
Latacz, Gniewomir;
Brazzolotto, Xavier;
Chantegreil, Fabien;
Nachon, Florian;
Zdarova Karasova, Jana;
Pejchal, Jaroslav;
Mzik, Martin;
Sestak, Vit;
Prchal, Lukas;
Odvarkova, Jitka;
Soukup, Ondrej

Publication type:

Article

Cytotoxic effect and molecular docking of 4-ethoxycarbonylmethyl-1-(piperidin-4-ylcarbonyl)-thiosemicarbazide-a novel topoisomerase II inhibitor.

Published in:

Journal of Molecular Modeling, 2013, v. 19, n. 3, p. 1319, doi. 10.1007/s00894-012-1679-6

By:

Siwek, Agata;
Stączek, Paweł;
Wujec, Monika;
Bielawski, Krzysztof;
Bielawska, Anna;
Paneth, Piotr

Publication type:

Article

Antifungal effect of 4-arylthiosemicarbazides against Candida species. Search for molecular basis of antifungal activity of thiosemicarbazide derivatives.

Published in:

Journal of Molecular Modeling, 2012, v. 18, n. 9, p. 4159, doi. 10.1007/s00894-012-1420-5

By:

Siwek, Agata;
Stefańska, Joanna;
Dzitko, Katarzyna;
Ruszczak, Artur

Publication type:

Article

Problems with molecular mechanics implementations on the example of 4-benzoyl-1-(4-methyl-imidazol-5-yl)-carbonylthiosemicarbazide.

Published in:

Journal of Molecular Modeling, 2012, v. 18, n. 3, p. 843, doi. 10.1007/s00894-011-1117-1

By:

Siwek, Agata;
Świderek, Katarzyna;
Jankowski, Stefan

Publication type:

Article

Biological and docking studies of topoisomerase IV inhibition by thiosemicarbazides.

Published in:

Journal of Molecular Modeling, 2011, v. 17, n. 9, p. 2297, doi. 10.1007/s00894-010-0889-z

By:

Siwek, Agata;
Stączek, Paweł;
Wujec, Monika;
Stefańska, Joanna;
Kosikowska, Urszula;
Malm, Anna;
Jankowski, Stefan;
Paneth, Piotr

Publication type:

Article

Ionic liquids as surfactants in micellar liquid chromatography.

Published in:

Journal of Separation Science, 2013, v. 36, n. 9/10, p. 1530, doi. 10.1002/jssc.201201059

By:

Flieger, Jolanta;
Siwek, Agata;
Pizoń, Magdalena;
Czajkowska‐Żelazko, Anna

Publication type:

Article

Usefulness of chaotropic salt additive in RP- HPLC of organic nonionized compounds.

Published in:

Journal of Separation Science, 2013, v. 36, n. 3, p. 469, doi. 10.1002/jssc.201200798

By:

Flieger, Jolanta;
Siwek, Agata;
Pizoń, Magdalena

Publication type:

Article

Synthesis and antimicrobial evaluation of new 1-{[4-(4-Halogenophenyl)-4 H-1,2,4- triazol-3-yl]sulfanyl}acetyl-4-substituted thiosemicarbazides and products of their cyclization.

Published in:

Heteroatom Chemistry, 2012, v. 23, n. 1, p. 117, doi. 10.1002/hc.20758

By:

Trotsko, Nazar;
Król, Jakub;
Siwek, Agata;
Wujec, Monika;
Kosikowska, Urszula;
Malm, Anna

Publication type:

Article

Study of direction of cyclization of 1-azolil-4-aryl/alkyl-thiosemicarbazides.

Published in:

Heteroatom Chemistry, 2010, v. 21, n. 7, p. 521, doi. 10.1002/hc.20643

By:

Siwek, Agata;
Wujec, Monika;
Dobosz, Maria;
Wawrzycka-Gorczyca, Irena

Publication type:

Article

Structure-activity relationship of s-triazoles and thiadiazoles as analgesics.

Published in:

Heteroatom Chemistry, 2010, v. 21, n. 4, p. 256, doi. 10.1002/hc.20605

By:

Siwek, Agata;
Wujec, Monika;
Plech, Tomasz;
Kuśmierz, Edyta;
Jagiełło-Wójtowicz, Ewa;
Chodkowska, Anna

Publication type:

Article

Synthesis and in vitro antibacterial evaluation of 1-substituted-4-ethoxycarbonylmethylthiosemicarbazides and products of their dehydrocyclization.

Published in:

Heteroatom Chemistry, 2010, v. 21, n. 3, p. 131, doi. 10.1002/hc.20597

By:

Siwek, Agata;
Stefańska, Joanna;
Wawrzycka-Gorczyca, Irena;
Wujec, Monika

Publication type:

Article

Synthesis and theoretical characterization of some new 4-substituted-1,3-diphenyl-5-thioxo-4,5-dihydro-1 H-1,2,4-triazoles with potential pharmacological activity.

Published in:

Heteroatom Chemistry, 2008, v. 19, n. 7, p. 713, doi. 10.1002/hc.20499

By:

Siwek, Agata;
Wujec, Monika;
Dobosz, Maria;
Paneth, Piotr

Publication type:

Article

Thiol-thione tautomeric forms recognition on the example of 4-[3-(2-methyl-furan-3-yl)-5-thioxo-1,2,4-triazolin-4-yl]acetic acid.

Published in:

Heteroatom Chemistry, 2008, v. 19, n. 4, p. 337, doi. 10.1002/hc.20433

By:

Siwek, Agata;
Wujec, Monika;
Wawrzycka-Gorczyca, Irena;
Dobosz, Maria;
Paneth, Piotr

Publication type:

Article

Design, Synthesis and Anticonvulsant Activity of New Phenoxyalkyl, Phenoxyethoxyethyl and Phenoxyacetyl Derivatives of Aminoalkanols.

Published in:

ChemistrySelect, 2022, v. 7, n. 19, p. 1, doi. 10.1002/slct.202201233

By:

Pańczyk‐Straszak, Katarzyna;
Rapacz, Anna;
Marona, Henryk;
Żelaszczyk, Dorota;
Karczewska, Elżbieta;
Zając, Martyna;
Skiba‐Kurek, Iwona;
Siwek, Agata;
Waszkielewicz, Anna

Publication type:

Article

Synthesis and biological evaluation of N-arylpiperazine derivatives of 4,4-dimethylisoquinoline-1,3(2H,4H)-dione as potential antiplatelet agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 536, doi. 10.1080/14756366.2018.1437155

By:

Marcinkowska, Monika;
Kotańska, Magdalena;
Zagórska, Agnieszka;
Śniecikowska, Joanna;
Kubacka, Monika;
Siwek, Agata;
Bucki, Adam;
Pawłowski, Maciej;
Bednarski, Marek;
Sapa, Jacek;
Starek, Małgorzata;
Dąbrowska, Monika;
Kołaczkowski, Marcin

Publication type:

Article

Synthesis and biological evaluation of 2-fluoro and 3-trifluoromethyl-phenyl-piperazinylalkyl derivatives of 1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione as potential antidepressant agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 10, doi. 10.1080/14756366.2016.1198902

By:

Zagórska, Agnieszka;
Bucki, Adam;
Kołaczkowski, Marcin;
Siwek, Agata;
Głuch-Lutwin, Monika;
Starowicz, Gabriela;
Kazek, Grzegorz;
Partyka, Anna;
Wesołowska, Anna;
Słoczyńska, Karolina;
Pękala, Elżbieta;
Pawłowski, Maciej

Publication type:

Article

Synthesis and biological evaluation of 2-fluoro and 3-trifluoromethyl-phenyl-piperazinylalkyl derivatives of 1 H -imidazo[2,1- f ]purine-2,4(3 H ,8 H )-dione as potential antidepressant agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 10, doi. 10.1080/14756366.2016.1198902

By:

Zagórska, Agnieszka;
Bucki, Adam;
Kołaczkowski, Marcin;
Siwek, Agata;
Głuch-Lutwin, Monika;
Starowicz, Gabriela;
Kazek, Grzegorz;
Partyka, Anna;
Wesołowska, Anna;
Słoczyńska, Karolina;
Pękala, Elżbieta;
Pawłowski, Maciej

Publication type:

Article

Cytotoxicity and topoisomerase I/II inhibition activity of novel 4-aryl/alkyl-1-(piperidin-4-yl)-carbonylthiosemicarbazides and 4-benzoylthiosemicarbazides.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 2, p. 243, doi. 10.3109/14756366.2013.768987

By:

Siwek, Agata;
Bielawska, Anna;
Maciorkowska, Elzbieta;
Lepiarczyk, Monika;
Bielawski, Krzysztof;
Trotsko, Nazar;
Wujec, Monika

Publication type:

Article

Antidepressant-like activity of magnesium in the chronic mild stress model in rats: alterations in the NMDA receptor subunits.

Published in:

International Journal of Neuropsychopharmacology, 2014, v. 17, n. 3, p. 393, doi. 10.1017/S1461145713001089

By:

Pochwat, Bartlomiej;
Szewczyk, Bernadeta;
Sowa-Kucma, Magdalena;
Siwek, Agata;
Doboszewska, Urszula;
Piekoszewski, Wojciech;
Gruca, Piotr;
Papp, Mariusz;
Nowak, Gabriel

Publication type:

Article

Multifunctional, Fluorene‐Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease.

Published in:

Angewandte Chemie, 2025, v. 137, n. 6, p. 1, doi. 10.1002/ange.202420510

By:

Panek, Dawid;
Pasieka, Anna;
Jończyk, Jakub;
Gawlińska, Milena;
Zaręba, Paula;
Siwek, Agata;
Wolak, Małgorzata;
Mordyl, Barbara;
Głuch‐Lutwin, Monika;
Latacz, Gniewomir;
Brazzolotto, Xavier;
Chantegreil, Fabien;
Nachon, Florian;
Zdarova Karasova, Jana;
Pejchal, Jaroslav;
Mzik, Martin;
Sestak, Vit;
Prchal, Lukas;
Odvarkova, Jitka;
Soukup, Ondrej

Publication type:

Article

Potential of nafimidone derivatives against co‐morbidities of epilepsy: In vitro, in vivo, and in silico investigations.

Published in:

Drug Development Research, 2022, v. 83, n. 1, p. 184, doi. 10.1002/ddr.21858

By:

Sari, Suat;
Barut, Burak;
Marcinkowska, Monika;
Sabuncuoğlu, Suna;
Avci, Ahmet;
Koçak Aslan, Ebru;
Özel, Arzu;
Siwek, Agata

Publication type:

Article

Xanthine–Dopamine Hybrid Molecules as Multitarget Drugs with Potential for the Treatment of Neurodegenerative Diseases.

Published in:

Biomolecules (2218-273X), 2023, v. 13, n. 7, p. 1079, doi. 10.3390/biom13071079

By:

Załuski, Michał;
Karcz, Tadeusz;
Drabczyńska, Anna;
Vielmuth, Christin;
Olejarz-Maciej, Agnieszka;
Głuch-Lutwin, Monika;
Mordyl, Barbara;
Siwek, Agata;
Satała, Grzegorz;
Müller, Christa E.;
Kieć-Kononowicz, Katarzyna

Publication type:

Article

Analysis of Density Changes of Selected Brain Receptors After a 14-Day Supply of Chromium(III) and Evaluation of Chromium(III) Affinity to Selected Receptors and Transporters.

Published in:

Biological Trace Element Research, 2020, v. 196, n. 2, p. 359, doi. 10.1007/s12011-019-01924-y

By:

Piotrowska, Anna;
Siwek, Agata;
Wolak, Małgorzata;
Nowak, Gabriel

Publication type:

Article

The Possibilities of Using Chromium Salts as an Agent Supporting Treatment of Polycystic Ovary Syndrome.

Published in:

Biological Trace Element Research, 2019, v. 192, n. 2, p. 91, doi. 10.1007/s12011-019-1654-5

By:

Piotrowska, Anna;
Pilch, Wanda;
Czerwińska-Ledwig, Olga;
Zuziak, Roxana;
Siwek, Agata;
Wolak, Małgorzata;
Nowak, Gabriel

Publication type:

Article

Anti‐Alzheimer's multitarget‐directed ligands with serotonin 5‐HT6 antagonist, butyrylcholinesterase inhibitory, and antioxidant activity.

Published in:

Archiv der Pharmazie, 2019, v. 352, n. 7, p. N.PAG, doi. 10.1002/ardp.201900041

By:

Marcinkowska, Monika;
Bucki, Adam;
Panek, Dawid;
Siwek, Agata;
Fajkis, Nikola;
Bednarski, Marek;
Zygmunt, Małgorzata;
Godyń, Justyna;
Del Rio Valdivieso, Alvaro;
Kotańska, Magdalena;
Kołaczkowski, Marcin;
Więckowska, Anna

Publication type:

Article

Aminoalkyl Derivatives of 8-Alkoxypurine-2,6-diones: Multifunctional 5-HT1A/5-HT7 Receptor Ligands and PDE Inhibitors with Antidepressant Activity.

Published in:

Archiv der Pharmazie, 2016, v. 349, n. 12, p. 889, doi. 10.1002/ardp.201600260

By:

Chłoń ‐ Rzepa, Grażyna;
Zagórska, Agnieszka;
Żmudzki, Paweł;
Bucki, Adam;
Kołaczkowski, Marcin;
Partyka, Anna;
Wesołowska, Anna;
Kazek, Grzegorz;
Głuch ‐ Lutwin, Monika;
Siwek, Agata;
Starowicz, Gabriela;
Pawłowski, Maciej

Publication type:

Article

Structure-5-HT/D2 Receptor Affinity Relationship in a New Group of 1-Arylpiperazynylalkyl Derivatives of 8-Dialkylamino-3,7-dimethyl-1 H-purine-2,6(3 H,7 H)-dione.

Published in:

Archiv der Pharmazie, 2016, v. 349, n. 10, p. 774, doi. 10.1002/ardp.201600162

By:

Żmudzki, Paweł;
Satała, Grzegorz;
Chłoń ‐ Rzepa, Grażyna;
Bojarski, Andrzej J.;
Kazek, Grzegorz;
Siwek, Agata;
Gryboś, Anna;
Głuch ‐ Lutwin, Monika;
Wesołowska, Anna;
Pawłowski, Maciej

Publication type:

Article

Synthesis and Pharmacological Activity of a New Series of 1-(1 H-Indol-4-yloxy)-3-(2-(2-methoxyphenoxy)ethylamino)propan-2-ol Analogs.

Published in:

Archiv der Pharmazie, 2016, v. 349, n. 3, p. 211, doi. 10.1002/ardp.201500234

By:

Bednarski, Marek;
Otto, Monika;
Dudek, Magdalena;
Kołaczkowski, Marcin;
Bucki, Adam;
Siwek, Agata;
Groszek, Grażyna;
Maziarz, Elżbieta;
Wilk, Piotr;
Sapa, Jacek

Publication type:

Article

Antiarrhythmic and α-Adrenoceptor Antagonistic Properties of Novel Arylpiperazine Derivatives of Pyrrolidin-2-one.

Published in:

Archiv der Pharmazie, 2015, v. 348, n. 12, p. 861, doi. 10.1002/ardp.201500180

By:

Zaręba, Paula;
Dudek, Magdalena;
Lustyk, Klaudia;
Siwek, Agata;
Starowicz, Gabriela;
Bednarski, Marek;
Nowiński, Leszek;
Zygmunt, Małgorzata;
Sapa, Jacek;
Malawska, Barbara;
Kulig, Katarzyna

Publication type:

Article

Synthesis and Pharmacological Evaluation of Novel Tricyclic[2,1- f]theophylline Derivatives.

Published in:

Archiv der Pharmazie, 2013, v. 346, n. 11, p. 832, doi. 10.1002/ardp.201300257

By:

Zagórska, Agnieszka;
Pawłowski, Maciej;
Siwek, Agata;
Kazek, Grzegorz;
Partyka, Anna;
Wróbel, Dagmara;
Jastrzębska ‐ Więsek, Magdalena;
Wesołowska, Anna

Publication type:

Article

Novel Mannich Bases, 5-Arylimidazolidine-2,4-dione Derivatives with Dual 5-HT1A Receptor and Serotonin Transporter Affinity.

Published in:

Archiv der Pharmazie, 2013, v. 346, n. 2, p. 98, doi. 10.1002/ardp.201200378

By:

Czopek, Anna;
Kołaczkowski, Marcin;
Bucki, Adam;
Byrtus, Hanna;
Pawłowski, Maciej;
Siwek, Agata;
Bojarski, Andrzej J.;
Bednarski, Marek;
Wróbel, Dagmara;
Wesołowska, Anna

Publication type:

Article

Novel 1-(1-Arylimiazolin-2-Yl)-3-Arylalkilurea Derivatives with Modulatory Activity on Opioid MOP Receptors.

Published in:

Molecules, 2024, v. 29, n. 3, p. 571, doi. 10.3390/molecules29030571

By:

Straszak, Dominik;
Woźniak, Sylwia;
Siwek, Agata;
Głuch-Lutwin, Monika;
Kołaczkowski, Marcin;
Pietrzak, Aldona;
Drop, Bartłomiej;
Matosiuk, Dariusz

Publication type:

Article

Modulation of the MOP Receptor (μ Opioid Receptor) by Imidazo[1,2- a ]imidazole-5,6-Diones: In Search of the Elucidation of the Mechanism of Action.

Published in:

Molecules, 2022, v. 27, n. 9, p. 2930, doi. 10.3390/molecules27092930

By:

Straszak, Dominik;
Siwek, Agata;
Głuch-Lutwin, Monika;
Mordyl, Barbara;
Kołaczkowski, Marcin;
Pietrzak, Aldona;
Rahnama-Hezavah, Mansur;
Drop, Bartłomiej;
Matosiuk, Dariusz

Publication type:

Article

The Structural Determinants for α 1 -Adrenergic/Serotonin Receptors Activity among Phenylpiperazine-Hydantoin Derivatives.

Published in:

Molecules, 2021, v. 26, n. 22, p. 7025, doi. 10.3390/molecules26227025

By:

Kucwaj-Brysz, Katarzyna;
Dela, Anna;
Podlewska, Sabina;
Bednarski, Marek;
Siwek, Agata;
Satała, Grzegorz;
Czarnota, Kinga;
Handzlik, Jadwiga;
Kieć-Kononowicz, Katarzyna

Publication type:

Article

Design, Sustainable Synthesis and Biological Evaluation of a Novel Dual α2A/5-HT7 Receptor Antagonist with Antidepressant-Like Properties.

Published in:

Molecules, 2021, v. 26, n. 13, p. 3828, doi. 10.3390/molecules26133828

By:

Canale, Vittorio;
Kotańska, Magdalena;
Dziubina, Anna;
Stefaniak, Matylda;
Siwek, Agata;
Starowicz, Gabriela;
Marciniec, Krzysztof;
Kasza, Patryk;
Satała, Grzegorz;
Duszyńska, Beata;
Bantreil, Xavier;
Lamaty, Frédéric;
Bednarski, Marek;
Sapa, Jacek;
Zajdel, Paweł

Publication type:

Article

Impact of N-Alkylamino Substituents on Serotonin Receptor (5-HTR) Affinity and Phosphodiesterase 10A (PDE10A) Inhibition of Isoindole-1,3-dione Derivatives.

Published in:

Molecules, 2020, v. 25, n. 17, p. 3868, doi. 10.3390/molecules25173868

By:

Czopek, Anna;
Partyka, Anna;
Bucki, Adam;
Pawłowski, Maciej;
Kołaczkowski, Marcin;
Siwek, Agata;
Głuch-Lutwin, Monika;
Koczurkiewicz, Paulina;
Pękala, Elżbieta;
Jaromin, Anna;
Tyliszczak, Bożena;
Wesołowska, Anna;
Zagórska, Agnieszka;
Jampilek, Josef

Publication type:

Article

Antiarrhythmic activity in occlusion-reperfusion model of 1-(1H-indol-4-yloxy)-3-{[2-(2-methoxyphenoxy)ethyl]amino} propan-2-ol and its enantiomers.

Published in:

Clinical & Experimental Pharmacology & Physiology, 2016, v. 43, n. 1, p. 81, doi. 10.1111/1440-1681.12491

By:

Bednarski, Marek;
Otto, Monika;
Dudek, Magdalena;
Siwek, Agata;
Zygmunt, Małgorzata;
Knutelska, Joanna;
Nowiński, Leszek;
Groszek, Grażyna;
Sapa, Jacek

Publication type:

Article

Synthesis, structure and investigations of tuberculosis inhibition activities of new 4-methyl-1-substituted-1 H-1,2,4-triazole-5(4 H)-thione.

Published in:

Journal of Heterocyclic Chemistry, 2008, v. 45, n. 6, p. 1893, doi. 10.1002/jhet.5570450655

By:

Wujec, Monika;
Siwek, Agata;
Swatko-Ossor, Marta;
Mazur, Liliana;
Rzaczynska, Zofia

Publication type:

Article

Study on the effect of EMD386088, a 5-HT receptor partial agonist, in enhancing the anti-immobility action of some antidepressants in rats.

Published in:

Naunyn-Schmiedeberg's Archives of Pharmacology, 2018, v. 391, n. 1, p. 37, doi. 10.1007/s00210-017-1431-y

By:

Jastrzębska-Więsek, Magdalena;
Siwek, Agata;
Partyka, Anna;
Kołaczkowski, Marcin;
Walczak, Maria;
Smolik, Magdalena;
Latacz, Gniewomir;
Kieć-Kononowicz, Katarzyna;
Wesołowska, Anna

Publication type:

Article

Study of a mechanism responsible for potential antidepressant activity of EMD 386088, a 5-HT partial agonist in rats.

Published in:

Naunyn-Schmiedeberg's Archives of Pharmacology, 2016, v. 389, n. 8, p. 839, doi. 10.1007/s00210-016-1245-3

By:

Jastrzębska-Więsek, Magdalena;
Siwek, Agata;
Partyka, Anna;
Antkiewicz-Michaluk, Lucyna;
Michaluk, Jerzy;
Romańska, Irena;
Kołaczkowski, Marcin;
Wesołowska, Anna

Publication type:

Article