Found: 17
Select item for more details and to access through your institution.
The deuterated pyrazoloquinolinone targeting a6 subunit-containing GABAA receptor as novel candidate for inhibition of trigeminovascular system activation: implication for migraine therapy.
- Published in:
- Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1451634
- By:
- Publication type:
- Article
Assessing the synergistic effects of morphine and MP‐III‐024 co‐administration: enhanced antinociception with reduced side effects.
- Published in:
- FASEB Journal, 2022, v. 36, p. N.PAG, doi. 10.1096/fasebj.2022.36.S1.R5946
- By:
- Publication type:
- Article
Supra‐additive effects of morphine and the α2/3 preferring GABA<sub>A</sub> receptor ligand MP‐III‐024 on mechanical hyperalgesia and thermal nociception.
- Published in:
- FASEB Journal, 2021, v. 35, p. N.PAG, doi. 10.1096/fasebj.2021.35.S1.03252
- By:
- Publication type:
- Article
An alpha 5‐GABA<sub>A</sub> receptor positive allosteric modulator attenuates social and cognitive deficits without changing dopamine system hyperactivity in rats exposed to valproic acid in utero.
- Published in:
- Autism Research: Official Journal of the International Society for Autism Research, 2024, v. 17, n. 8, p. 1534, doi. 10.1002/aur.3178
- By:
- Publication type:
- Article
Postweaning positive modulation of α5GABAA receptors improves autism‐like features in prenatal valproate rat model in a sex‐specific manner.
- Published in:
- Autism Research: Official Journal of the International Society for Autism Research, 2022, v. 15, n. 5, p. 806, doi. 10.1002/aur.2699
- By:
- Publication type:
- Article
α5-GABAA Receptor Modulation Reverses Behavioral and Neurophysiological Correlates of Psychosis in Rats with Ventral Hippocampal Alzheimer's Disease-like Pathology.
- Published in:
- International Journal of Molecular Sciences, 2023, v. 24, n. 14, p. 11788, doi. 10.3390/ijms241411788
- By:
- Publication type:
- Article
GL-II-73, a Positive Allosteric Modulator of α5GABA A Receptors, Reverses Dopamine System Dysfunction Associated with Pilocarpine-Induced Temporal Lobe Epilepsy.
- Published in:
- International Journal of Molecular Sciences, 2023, v. 24, n. 14, p. 11588, doi. 10.3390/ijms241411588
- By:
- Publication type:
- Article
Extrasynaptic Localization Is Essential for a5GABAA Receptor Modulation of Dopamine System Function.
- Published in:
- eNeuro, 2024, v. 11, n. 3, p. 1, doi. 10.1523/ENEURO.0344-23.2023
- By:
- Publication type:
- Article
Therapeutic effects of KRM-II-81, positive allosteric modulator for α2/3 subunit containing GABA<sub>A</sub> receptors, in a mouse model of Dravet syndrome.
- Published in:
- Frontiers in Pharmacology, 2023, p. 1, doi. 10.3389/fphar.2023.1273633
- By:
- Publication type:
- Article
Comparative anticonvulsant activity of the GABAkine KRM‐II‐81 and a deuterated analog.
- Published in:
- Drug Development Research, 2023, v. 84, n. 3, p. 527, doi. 10.1002/ddr.22042
- By:
- Publication type:
- Article
Preformulation and development of preliminary nanoemulsion carrier for patent protected compound GL-II-73.
- Published in:
- Macedonian Pharmaceutical Bulletin / Makedonsko Farmacevtski Bilten, 2023, v. 69, p. 53, doi. 10.33320/maced.pharm.bull.2023.69.03.026
- By:
- Publication type:
- Article
Effects of α5 GABA<sub>A</sub> receptor modulation on social interaction, memory, and neuroinflammation in a mouse model of Alzheimer's disease.
- Published in:
- CNS Neuroscience & Therapeutics, 2022, v. 28, n. 11, p. 1767, doi. 10.1111/cns.13914
- By:
- Publication type:
- Article
Metabolism, pharmacokinetics, and anticonvulsant activity of a deuterated analog of the α2/3‐selective GABAkine KRM‐II‐81.
- Published in:
- Biopharmaceutics & Drug Disposition, 2022, v. 43, n. 2, p. 66, doi. 10.1002/bdd.2313
- By:
- Publication type:
- Article
GABA-A Alpha 2/3 but Not Alpha 1 Receptor Subunit Ligand Inhibits Harmaline and Pimozide-Induced Tremor in Rats.
- Published in:
- Biomolecules (2218-273X), 2023, v. 13, n. 2, p. 197, doi. 10.3390/biom13020197
- By:
- Publication type:
- Article
Synthesis and Receptor Binding Studies of α5 GABA A R Selective Novel Imidazodiazepines Targeted for Psychiatric and Cognitive Disorders.
- Published in:
- Molecules, 2023, v. 28, n. 12, p. 4771, doi. 10.3390/molecules28124771
- By:
- Publication type:
- Article
Synergistic antihyperalgesic and antinociceptive effects of morphine and methyl 8-ethynyl-6-(pyridin-2-yl)-4H-benzo[f]imidazo[1,5-a][1,4]diazepine-3-carboxylate (MP-III-024): a positive allosteric modulator at α2GABAA and α3GABAA receptors.
- Published in:
- Psychopharmacology, 2021, v. 238, n. 6, p. 1585, doi. 10.1007/s00213-021-05791-1
- By:
- Publication type:
- Article
Improvement of Cognitive Functions And Neurotrophic Effects through by Α5‐GABAA Receptor Positive Allosteric Modulation in Animal Models of Risk for Alzheimer's Disease.
- Published in:
- Alzheimer's & Dementia: The Journal of the Alzheimer's Association, 2023, v. 19, n. 21, p. 1, doi. 10.1002/alz.074419
- By:
- Publication type:
- Article