Works by Scozzafava, Andrea

Results: 79

Plasmonic Particles that Hit Hypoxic Cells.

Published in:

Advanced Functional Materials, 2015, v. 25, n. 2, p. 316, doi. 10.1002/adfm.201402118

By:

Ratto, Fulvio;
Witort, Ewa;
Tatini, Francesca;
Centi, Sonia;
Lazzeri, Lorenza;
Carta, Fabrizio;
Lulli, Matteo;
Vullo, Daniela;
Fusi, Franco;
Supuran, Claudiu T.;
Scozzafava, Andrea;
Capaccioli, Sergio;
Pini, Roberto

Publication type:

Article

Efficient polycyclic aromatic hydrocarbons dihydroxylation in direct micellar systems.

Published in:

Biotechnology & Bioengineering, 2001, v. 74, n. 3, p. 240, doi. 10.1002/bit.1113

By:

Randazzo, Demetrio;
Berti, Debora;
Briganti, Fabrizio;
Baglioni, Piero;
Scozzafava, Andrea;
Di Gennaro, Patrizia;
Galli, Enrica;
Bestetti, Giuseppina

Publication type:

Article

Enzymatic decolorization of spent textile dyeing baths composed by mixtures of synthetic dyes and additives.

Published in:

Applied Microbiology & Biotechnology, 2012, v. 96, n. 2, p. 395, doi. 10.1007/s00253-011-3809-y

By:

Ciullini, Ilaria;
Gullotto, Antonella;
Tilli, Silvia;
Sannia, Giovanni;
Basosi, Riccardo;
Scozzafava, Andrea;
Briganti, Fabrizio

Publication type:

Article

Treatment of NSAPs-rich petrochemical wastewaters using a two-stage combined process of fungi and activated sludge.

Published in:

Environmental Technology, 2021, v. 42, n. 24, p. 3783, doi. 10.1080/09593330.2020.1752814

By:

Palli, Laura;
Tilli, Silvia;
Gregorio, Simona Di;
Scozzafava, Andrea;
Gori, Riccardo

Publication type:

Article

CARBONIC ANHYDRASE INHIBITORS. Part 871 INHIBITION OF CARBONIC ANHYDRASE ISOZYMES I, II AND IV WITH ARSINOLIPIDS.

Published in:

Main Group Metal Chemistry, 1999, v. 22, n. 12, p. 693

By:

Ioannou, Panayiotis V.;
Kordalis, Nick L.;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

CARBONIC ANHYDRASE INHIBITORS. Part 591 INHIBITION OF CARBONIC ANHYDRASE ISOZYMES I, II AND IV WITH ARSANILIC ACID DERIVATIVES.

Published in:

Main Group Metal Chemistry, 1998, v. 21, n. 6, p. 357

By:

Scozzafava, Andrea;
Briganti, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

CARBONIC ANHYDRASE INHIBITORS. Part 501 INTERACTION OF ISOZYMES I AND II OF CARBONIC ANHYDRASE WITH Ge(IV) AND Sb(III) DERIVATIVES.

Published in:

Main Group Metal Chemistry, 1997, v. 20, n. 10, p. 641

By:

Rivière-Baudet, Monique;
Supuran, Claudiu T.;
Scozzafava, Andrea;
Briganti, Fabrizio;
Baz, Fatima El;
Maarouf, Zhara Ben;
Rivière, Pierre

Publication type:

Article

COMPLEXES WITH BIOLOGICALLY ACTIVE LIGANDS. Part 81 SYNTHESIS AND CARBONIC ANHYDRASE INHIBITORY ACTIVITY OF 5-BENZOYLAMIDO- AND 5-(3-NITROBENZOYLAMIDO)-1,3,4-THIADIAZOLE-2-SULFONAMIDE AND THEIR METAL COMPLEXES.

Published in:

Main Group Metal Chemistry, 1997, v. 20, n. 3, p. 151

By:

Jitianu, Andrei;
Ilies, Marc A.;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

INHIBITION OF CARBONIC ANHYDRASE ISOZYMES I AND II WITH THIOPHOSPHORYLIC COMPOUNDS CONTAINING 4-CARBOXYBENZENE-SULFONAMIDO MOIETIES.

Published in:

Main Group Metal Chemistry, 1996, v. 19, n. 8, p. 503

By:

Scozzafava, Andrea;
Briganti, Fabrizio;
Supuran, Claudiu T.;
Fenesan, loan;
Popescu, Rodica;
Muresan, Viorica;
Farcas, Sorin

Publication type:

Article

Carbonic anhydrase IX from cancer-associated fibroblasts drives epithelial-mesenchymal transition in prostate carcinoma cells.

Published in:

Cell Cycle, 2013, v. 12, n. 11, p. 1791, doi. 10.4161/cc.24902

By:

Fiaschi, Tania;
Giannoni, Elisa;
Taddei, Maria Letizia;
Cirri, Paolo;
Marini, Alberto;
Pintus, Gianfranco;
Nativi, Cristina;
Richichi, Barbara;
Scozzafava, Andrea;
Carta, Fabrizio;
Torre, Eugenio;
Supuran, Claudiu T.;
Chiarugi, Paola

Publication type:

Article

Polymetallic macromolecules are potential contrast agents of improved efficiency.

Published in:

Magnetic Resonance in Medicine, 1994, v. 31, n. 1, p. 58, doi. 10.1002/mrm.1910310109

By:

Cavagna, Frederich;
Luchinat, Claudio;
Scozzafava, Andrea;
Xia, Zhicheng

Publication type:

Article

Thiophosphorylic and Phosophorylic Arylsulfon-Amides as Carbonic Anhidrase Inhibitors.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 1999, v. 147, n. 1, p. 85, doi. 10.1080/10426509908053523

By:

Claudiu, T. Supuran;
Andrea, Scozzafava;
Briganti, Fabrizio;
Ioan, Fenesan;
Rodica, Popescu;
Viorica, Muresan

Publication type:

Article

The salicylate 1,2-dioxygenase as a model for a conventional gentisate 1,2-dioxygenase: crystal structures of the G106A mutant and its adducts with gentisate and salicylate.

Published in:

FEBS Journal, 2013, v. 280, n. 7, p. 1643, doi. 10.1111/febs.12173

By:

Ferraroni, Marta;
Matera, Irene;
Bürger, Sibylle;
Reichert, Sabrina;
Steimer, Lenz;
Scozzafava, Andrea;
Stolz, Andreas;
Briganti, Fabrizio

Publication type:

Article

Dioxygen, an unexpected carbonic anhydrase ligand.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 999, doi. 10.1080/14756366.2018.1475371

By:

Ferraroni, Marta;
Gaspari, Roberto;
Scozzafava, Andrea;
Cavalli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Sulphonamide inhibition studies of the β-carbonic anhydrase from the bacterial pathogen Clostridium perfringens.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 31, doi. 10.1080/14756366.2017.1388233

By:

Vullo, Daniela;
Kumar, R. Siva Sai;
Scozzafava, Andrea;
Ferry, James G.;
Supuran, Claudiu T.

Publication type:

Article

Rosmarinic acid inhibits some metabolic enzymes including glutathione S -transferase, lactoperoxidase, acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase isoenzymes.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1698, doi. 10.3109/14756366.2015.1135914

By:

Gülçin, İlhami;
Scozzafava, Andrea;
Supuran, Claudiu T.;
Koksal, Zeynep;
Turkan, Fikret;
Çetinkaya, Songül;
Bingöl, Zeynebe;
Huyut, Zübeyir;
Alwasel, Saleh H.

Publication type:

Article

The effect of caffeic acid phenethyl ester (CAPE) on metabolic enzymes including acetylcholinesterase, butyrylcholinesterase, glutathione S-transferase, lactoperoxidase, and carbonic anhydrase isoenzymes I, II, IX, and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1095, doi. 10.3109/14756366.2015.1094470

By:

Gülçin, İlhami;
Scozzafava, Andrea;
Supuran, Claudiu T.;
Akıncıoğlu, Hulya;
Koksal, Zeynep;
Turkan, Fikret;
Alwasel, Saleh

Publication type:

Article

Synthesis and inhibition potency of novel ureido benzenesulfonamides incorporating GABA as tumor-associated carbonic anhydrase IX and XII inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 2, p. 205, doi. 10.3109/14756366.2015.1014477

By:

Ceruso, Mariangela;
Antel, Sabrina;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β -carbonic anhydrase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 1, p. 132, doi. 10.3109/14756366.2015.1010529

By:

Bozdag, Murat;
Carta, Fabrizio;
Vullo, Daniela;
Isik, Semra;
AlOthman, Zeid;
Osman, Sameh M.;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

The impact of hydroquinone on acetylcholine esterase and certain human carbonic anhydrase isoenzymes (hCA I, II, IX, and XII).

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 941, doi. 10.3109/14756366.2014.999236

By:

Scozzafava, Andrea;
Kalın, Pınar;
Supuran, Claudiu T.;
Gülçin, İlhami;
Alwasel, Saleh H.

Publication type:

Article

Carbonic anhydrase inhibitors: guaiacol and catechol derivatives effectively inhibit certain human carbonic anhydrase isoenzymes (hCA I, II, IX and XII).

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 4, p. 586, doi. 10.3109/14756366.2014.956310

By:

Scozzafava, Andrea;
Passaponti, Maurizio;
Supuran, Claudiu T.;
Gülçin, İlhami

Publication type:

Article

Peptidomimetics as protein arginine deiminase 4 (PAD4) inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 3, p. 466, doi. 10.3109/14756366.2014.947976

By:

Trabocchi, Andrea;
Pala, Nicolino;
Krimmelbein, Ilga;
Menchi, Gloria;
Guarna, Antonio;
Sechi, Mario;
Dreker, Tobias;
Scozzafava, Andrea;
Supuran, Claudiu T.;
Carta, Fabrizio

Publication type:

Article

Dipotassium-trioxohydroxytetrafluorotriborate, K2[B3O3F4OH], is a potent inhibitor of human carbonic anhydrases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 2, p. 341, doi. 10.3109/14756366.2014.918610

By:

Vullo, Daniela;
Milos, Mladen;
Galic, Borivoj;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Sulfonamides incorporating fluorine and 1,3,5-triazine moieties are effective inhibitors of three β-class carbonic anhydrases from Mycobacterium tuberculosis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 5, p. 686, doi. 10.3109/14756366.2013.842233

By:

Ceruso, Mariangela;
Vullo, Daniela;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Biochemical characterization of the γ-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis, PgiCA.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 4, p. 532, doi. 10.3109/14756366.2013.822371

By:

Del Prete, Sonia;
De Luca, Viviana;
Vullo, Daniela;
Scozzafava, Andrea;
Carginale, Vincenzo;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Biochemical properties of a new α-carbonic anhydrase from the human pathogenic bacterium, Vibrio cholerae.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 1, p. 23, doi. 10.3109/14756366.2012.747197

By:

Del Prete, Sonia;
De Luca, Viviana;
Scozzafava, Andrea;
Carginale, Vincenzo;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Cloning, polymorphism, and inhibition of beta-carbonic anhydrase of Helicobacter pylori.

Published in:

2008

By:

Morishita S;
Nishimori I;
Minakuchi T;
Onishi S;
Takeuchi H;
Sugiura T;
Vullo D;
Scozzafava A;
Supuran CT;
Morishita, Saori;
Nishimori, Isao;
Minakuchi, Tomoko;
Onishi, Saburo;
Takeuchi, Hiroaki;
Sugiura, Tetsuro;
Vullo, Daniela;
Scozzafava, Andrea;
Supuran, Claudiu T

Publication type:

journal article

Cloning, polymorphism, and inhibition of β-carbonic anhydrase of Helicobacter pylori.

Published in:

Journal of Gastroenterology, 2008, v. 43, n. 11, p. 849, doi. 10.1007/s00535-008-2240-3

By:

Morishita, Saori;
Nishimori, Isao;
Minakuchi, Tomoko;
Onishi, Saburo;
Takeuchi, Hiroaki;
Sugiura, Tetsuro;
Vullo, Daniela;
Scozzafava, Andrea;
Supuran, Claudiu

Publication type:

Article

Hypoxia activates the capacity of tumor-associated carbonic anhydrase IX to acidify extracellular pH

Published in:

FEBS Letters, 2004, v. 577, n. 3, p. 439, doi. 10.1016/j.febslet.2004.10.043

By:

Švastová, Eliška;
Hulíková, Alǽbeta;
Rafajová, Monika;
Zat'ovičová, Miriam;
Gibadulinová, Adriana;
Casini, Angela;
Cecchi, Alessandro;
Scozzafava, Andrea;
Supuran, Claudiu T.;
Pastorek, Jaromír;
Pastoreková, Silvia

Publication type:

Article

Crystal structure of human carbonic anhydrase XIII and its complex with the inhibitor acetazolamide.

Published in:

Proteins, 2009, v. 74, n. 1, p. 164, doi. 10.1002/prot.22144

By:

Di Fiore, Anna;
Monti, Simona Maria;
Hilvo, Mika;
Parkkila, Seppo;
Romano, Vincenza;
Scaloni, Andrea;
Pedone, Carlo;
Scozzafava, Andrea;
Supuran, Claudiu T.;
De Simone, Giuseppina

Publication type:

Article

Carbonic Anhydrase Inhibitors: Design of Membrane-Impermeant Copper(II) Complexes of DTPA-, DOTA-, and TETA-Tailed Sulfonamides Targeting the Tumor-Associated Transmembrane Isoform IX.

Published in:

ChemMedChem, 2008, v. 3, n. 11, p. 1780, doi. 10.1002/cmdc.200800267

By:

Rami, Marouan;
Cecchi, Alessandro;
Montero, Jean-Louis;
Innocenti, Alessio;
Vullo, Daniela;
Scozzafava, Andrea;
Winum, Jean-Yves;
Supuran, Claudiu T.

Publication type:

Article

Carbonic Anhydrase Inhibitors: Binding of Indanesulfonamides to the Human Isoform II.

Published in:

ChemMedChem, 2008, v. 3, n. 3, p. 473, doi. 10.1002/cmdc.200700274

By:

D'Ambrosio, Katia;
Masereel, Bernard;
Thiry, Anne;
Scozzafava, Andrea;
Supuran, Claudiu T.;
De Simone, Giuseppina

Publication type:

Article

Characterization of the first beta-class carbonicanhydrase from an arthropod (Drosophilamelanogaster) and phylogenetic analysis ofbeta-class carbonic anhydrases in invertebrates.

Published in:

BMC Biochemistry, 2010, v. 11, p. 28, doi. 10.1186/1471-2091-11-28

By:

Syrjänen, Leo;
Tolvanen, Martti;
Hilvo, Mika;
Olatubosun, Ayodeji;
Innocenti, Alessio;
Scozzafava, Andrea;
Leppiniemi, Jenni;
Niederhauser, Barbara;
Hytönen, Vesa P.;
Gorr, Thomas A.;
Parkkila, Seppo;
Supuran, Claudiu T.

Publication type:

Article

Evaluation of an FIA Operated Amperometric Bacterial Biosensor, Based on Pseudomonas Putida F1 for the Detection of Benzene, Toluene, Ethylbenzene, and Xylenes (BTEX).

Published in:

Analytical Letters, 2005, v. 38, n. 10, p. 1531, doi. 10.1081/AL-200065793

By:

Rasinger, JosefD.;
Marrazza, Giovanna;
Briganti, Fabrizio;
Scozzafava, Andrea;
Mascini, Marco;
Turner, A.P. F.

Publication type:

Article

Which Carbonic Anhydrases are Targeted by the Antiepileptic Sulfonamides and Sulfamates?

Published in:

2009

By:

De Simone, Giuseppina;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Letter

Carbonic anhydrase IX: A new druggable target for the design of antitumor agents.

Published in:

Medicinal Research Reviews, 2008, v. 28, n. 3, p. 445, doi. 10.1002/med.20112

By:

Winum, Jean-Yves;
Rami, Marouan;
Scozzafava, Andrea;
Montero, Jean-Louis;
Supuran, Claudiu

Publication type:

Article

Therapeutic potential of sulfamides as enzyme inhibitors.

Published in:

Medicinal Research Reviews, 2006, v. 26, n. 6, p. 767, doi. 10.1002/med.20068

By:

Winum, Jean-Yves;
Scozzafava, Andrea;
Montero, Jean-Louis;
Supuran, Claudiu T.

Publication type:

Article

Sulfamates and their therapeutic potential.

Published in:

Medicinal Research Reviews, 2005, v. 25, n. 2, p. 186, doi. 10.1002/med.20021

By:

Winum, Jean-Yves;
Scozzafava, Andrea;
Montero, Jean-Louis;
Supuran, Claudiu T.

Publication type:

Article

Protease inhibitors of the sulfonamide type: Anticancer, antiinflammatory, and antiviral agents.

Published in:

Medicinal Research Reviews, 2003, v. 23, n. 5, p. 535, doi. 10.1002/med.10047

By:

Claudiu T. Supuran;
Angela Casini;
Andrea Scozzafava

Publication type:

Article

Carbonic anhydrase inhibitors.

Published in:

Medicinal Research Reviews, 2003, v. 23, n. 2, p. 146, doi. 10.1002/med.10025

By:

Supuran, Claudiu T.;
Scozzafava, Andrea;
Casini, Angela

Publication type:

Article

Bacterial protease inhibitors.

Published in:

Medicinal Research Reviews, 2002, v. 22, n. 4, p. 329, doi. 10.1002/med.10007

By:

Supuran, Claudiu T.;
Scozzafava, Andrea;
Clare, Brian W.

Publication type:

Article

Secondary/tertiary benzenesulfonamides with inhibitory action against the cytosolic human carbonic anhydrase isoforms I and II.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2013, v. 28, n. 2, p. 294, doi. 10.3109/14756366.2012.658788

By:

Alp, Cemalettin;
Maresca, Alfonso;
Alp, Nurdan Alcan;
Gültekin, Mehmet Serdar;
Ekinci, Deniz;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of the β-class carbonic anhydrases from Mycobacterium tuberculosis with carboxylic acids.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2013, v. 28, n. 2, p. 392, doi. 10.3109/14756366.2011.650168

By:

Maresca, Alfonso;
Vullo, Daniela;
Scozzafava, Andrea;
Manole, Gheorghe;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of the alpha- and beta-carbonic anhydrases from the gastric pathogen Helycobacter pylori with anions.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2013, v. 28, n. 2, p. 388, doi. 10.3109/14756366.2011.649268

By:

Maresca, Alfonso;
Vullo, Daniela;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Dihalogenated sulfanilamides and benzolamides are effective inhibitors of the three β-class carbonic anhydrases from Mycobacterium tuberculosis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2013, v. 28, n. 2, p. 384, doi. 10.3109/14756366.2011.645539

By:

Maresca, Alfonso;
Scozzafava, Andrea;
Vullo, Daniela;
Supuran, Claudiu T.

Publication type:

Article

Carbonic anhydrase inhibitors. Biphenylsulfonamides with inhibitory action towards the transmembrane, tumor-associated isozymes IX possess cytotoxic activity against human colon, lung and breast cancer cell lines.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2009, v. 24, n. 2, p. 499, doi. 10.1080/14756360802218441

By:

Morsy, Salwa M. I.;
Badawi, Abdelfattah M.;
Cecchi, Alessandro;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

QSAR studies for the inhibition of the transmembrane carbonic anhydrase isozyme XIV with sulfonamides using PRECLAV software.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2009, v. 24, n. 2, p. 337, doi. 10.1080/14756360802187489

By:

Singh, Shalini;
Khadikar, Padmakar V.;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Carbonic anhydrase inhibitors. Cloning, characterization and inhibition studies of the cytosolic isozyme III with anions.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2009, v. 24, n. 1, p. 70, doi. 10.1080/14756360801907143

By:

Nishimori, Isao;
Minakuchi, Tomoko;
Onishi, Saburo;
Vullo, Daniela;
Cecchi, Alessandro;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Carbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II and IX with some 1,3,4-oxadiazole- and 1,2,4-triazole-thiols.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2008, v. 23, n. 1, p. 101, doi. 10.1080/14756360701342417

By:

Almajan, Gabriela Laura;
Barbuceanu, Stefania-Felicia;
innocenti, Alessio;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Carbonic anhydrase inhibitors. Selective inhibition of human tumor-associated isozymes IX and XII and cytosolic isozymes I and II with some substituted-2-mercapto-benzenesulfonamides.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2006, v. 21, n. 5, p. 563, doi. 10.1080/14756360600648146

By:

Saczewski, Franciszek;
Innocenti, Alessio;
Brzozowski, Zdzisław;
Sławiński, Jarosław;
Pomarnacka, Elżbieta;
Kornicka, Anita;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article