Works matching AU Schirmeister, Tanja
Results: 94
Next Generation of Fluorometric Protease Assays: 7‐Nitrobenz‐2‐oxa‐1,3‐diazol‐4‐yl‐amides (NBD‐Amides) as Class‐Spanning Protease Substrates.
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- Chemistry - A European Journal, 2023, v. 29, n. 50, p. 1, doi. 10.1002/chem.202301855
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- Article
Two Tags in One Probe: Combining Fluorescence‐ and Biotin‐based Detection of the Trypanosomal Cysteine Protease Rhodesain.
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- Chemistry - A European Journal, 2022, v. 28, n. 62, p. 1, doi. 10.1002/chem.202201636
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- Article
Synthesis and biological evaluation of novel peptidomimetics as rhodesain inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1184, doi. 10.3109/14756366.2015.1108972
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- Article
Identification of a potential allosteric site of Golgi α-mannosidase II using computer-aided drug design.
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- PLoS ONE, 2019, v. 14, n. 5, p. 1, doi. 10.1371/journal.pone.0216132
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- Article
Protocol for Rational Design of Covalently Interacting Inhibitors.
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- ChemPhysChem, 2014, v. 15, n. 15, p. 3226, doi. 10.1002/cphc.201402542
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- Article
Thiirancarboxamides as Inhibitors of Papain.
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- Archiv der Pharmazie, 2004, v. 337, n. 2, p. 90, doi. 10.1002/ardp.200300820
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- Article
β-Lactam Derivatives as Enzyme Inhibitors: 1-Peptidyl Derivatives of 4-Phenylazetidin-2-one as Inhibitors of Elastase and Papain.
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- Archiv der Pharmazie, 2000, v. 333, n. 8, p. 243, doi. 10.1002/1521-4184(20008)333:8<243::AID-ARDP243>3.0.CO;2-O
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- Article
Aziridine-2,3-dicarboxylic Acid Derivatives as Inhibitors of Papain.
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- Archiv der Pharmazie, 1996, v. 329, n. 5, p. 239, doi. 10.1002/ardp.19963290504
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- Article
Bacteria from the Amycolatopsis genus associated with a toxic bird secrete protective secondary metabolites.
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- Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-52316-3
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- Article
BANΔIT: B'‐Factor Analysis for Drug Design and Structural Biology.
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- Molecular Informatics, 2021, v. 40, n. 1, p. 1, doi. 10.1002/minf.202000144
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- Article
Screening of Protease Inhibitors as Antiplasmodial Agents. Part I: Aziridines and Epoxides.
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- ChemMedChem, 2007, v. 2, n. 8, p. 1214, doi. 10.1002/cmdc.200700070
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- Article
The Importance of the Active Site Histidine for the Activity of Epoxide- or Aziridine-Based Inhibitors of Cysteine Proteases.
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- ChemMedChem, 2007, v. 2, n. 1, p. 120, doi. 10.1002/cmdc.200600159
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- Article
Aziridide-Based Inhibitors of Cathepsin L: Synthesis, Inhibition Activity, and Docking Studies.
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- ChemMedChem, 2006, v. 1, n. 10, p. 1126, doi. 10.1002/cmdc.200600106
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- Article
Rational Design of Aziridine-Containing Cysteine Protease Inhibitors with Improved Potency: Studies on Inhibition Mechanism.
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- ChemMedChem, 2006, v. 1, n. 9, p. 1021, doi. 10.1002/cmdc.200600081
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- Article
The Significance of Ionic Bonding in Sulfur Dioxide: Bond Orders from X-ray Diffraction Data.
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- Angewandte Chemie International Edition, 2012, v. 51, n. 27, p. 6776, doi. 10.1002/anie.201200745
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- Article
Cis autocatalytic cleavage of glycine‐linked Zika virus NS2B‐NS3 protease constructs.
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- FEBS Letters, 2019, v. 593, n. 16, p. 2204, doi. 10.1002/1873-3468.13507
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- Article
Evaluation of curcumin irreversibility.
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- 2020
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- Letter
Eliciting callus culture for production of hepatoprotective flavonoids and phenolics from Sequoia sempervirens (D. Don Endl).
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- Natural Product Research, 2020, v. 34, n. 21, p. 3125, doi. 10.1080/14786419.2019.1607334
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- Article
Drug combination studies of curcumin and genistein against rhodesain of Trypanosoma brucei rhodesiense.
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- Natural Product Research, 2019, v. 33, n. 24, p. 3577, doi. 10.1080/14786419.2018.1483927
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- Article
Novel Opportunities for Cathepsin S Inhibitors in Cancer Immunotherapy by Nanocarrier-Mediated Delivery.
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- Cells (2073-4409), 2020, v. 9, n. 9, p. 2021, doi. 10.3390/cells9092021
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- Article
Novel bioreactor internals for the cultivation of spore‐forming fungi in pellet form.
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- Engineering in Life Sciences, 2022, v. 22, n. 7, p. 474, doi. 10.1002/elsc.202100094
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- Article
Applicability of a single‐use bioreactor compared to a glass bioreactor for the fermentation of filamentous fungi and evaluation of the reproducibility of growth in pellet form.
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- Engineering in Life Sciences, 2021, v. 21, n. 5, p. 324, doi. 10.1002/elsc.202000069
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- Article
Comparison of the separation of aziridine isomers applying heptakis(2,3-di-O-methyl-6-sulfato)β-CD and heptakis(2,3-di-O-acetyl-6-sulfato)β-CD in aqueous and nonaqueous systems.
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- Electrophoresis, 2005, v. 26, n. 20, p. 3897, doi. 10.1002/elps.200500176
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- Article
Peptidyl nitroalkene inhibitors of main protease rationalized by computational and crystallographic investigations as antivirals against SARS-CoV-2.
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- Communications Chemistry, 2024, v. 7, n. 1, p. 1, doi. 10.1038/s42004-024-01104-7
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- Article
Discovery of benzimidazole‐based Leishmania mexicana cysteine protease CPB2.8ΔCTE inhibitors as potential therapeutics for leishmaniasis.
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- Chemical Biology & Drug Design, 2018, v. 92, n. 3, p. 1585, doi. 10.1111/cbdd.13326
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- Article
Ensemble‐based ADME–Tox profiling and virtual screening for the discovery of new inhibitors of the <italic>Leishmania mexicana</italic> cysteine protease CPB2.8ΔCTE.
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- Chemical Biology & Drug Design, 2018, v. 91, n. 2, p. 597, doi. 10.1111/cbdd.13124
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- Article
Fly versus man: evolutionary impairment of nucleolar targeting affects the degradome of Drosophila's Taspase1.
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- FASEB Journal, 2015, v. 29, n. 5, p. 1973, doi. 10.1096/fj.14-262451
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- Article
Natural Product Repertoire of the Genus Amphimedon.
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- Marine Drugs, 2019, v. 17, n. 1, p. 19, doi. 10.3390/md17010019
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- Article
Cytotoxicity of Endoperoxides from the Caribbean Sponge Plakortis halichondrioides towards Sensitive and Multidrug-Resistant Leukemia Cells: Acids vs. Esters Activity Evaluation.
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- Marine Drugs, 2017, v. 15, n. 3, p. 63, doi. 10.3390/md15030063
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- Article
Identification of Plakortide E from the Caribbean Sponge Plakortis halichondroides as a Trypanocidal Protease Inhibitor using Bioactivity-Guided Fractionation.
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- Marine Drugs, 2014, v. 12, n. 9, p. 2614, doi. 10.3390/md12052614
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- Article
Identification of Plakortide E from the Caribbean Sponge Plakortis halichondroides as a Trypanocidal Protease Inhibitor using Bioactivity-Guided Fractionation.
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- Marine Drugs, 2014, v. 12, n. 5, p. 2614, doi. 10.3390/md12052614
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- Article
Antioxidant and Anti-Protease Activities of Diazepinomicin from the Sponge-Associated Micromonospora Strain RV115.
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- Marine Drugs, 2012, v. 10, n. 10, p. 2208, doi. 10.3390/md10102208
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- Article
New Tetromycin Derivatives with Anti-Trypanosomal and Protease Inhibitory Activities.
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- Marine Drugs, 2011, v. 9, n. 10, p. 1682, doi. 10.3390/md9101682
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- Article
Identification of novel small-molecular inhibitors of Staphylococcus aureus sortase A using hybrid virtual screening.
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- Journal of Antibiotics, 2022, v. 75, n. 6, p. 321, doi. 10.1038/s41429-022-00524-8
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- Article
Inhibition of cysteine proteases by peptides containing aziridine-2,3-dicarboxylic acid building blocks.
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- Biopolymers, 1999, v. 51, n. 1, p. 87, doi. 10.1002/(SICI)1097-0282(1999)51:1<87::AID-BIP10>3.0.CO;2-Z
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- Article
Peptidomimetic inhibitors of TMPRSS2 block SARS-CoV-2 infection in cell culture.
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- Communications Biology, 2022, v. 5, n. 1, p. 1, doi. 10.1038/s42003-022-03613-4
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- Article
Cathepsin B in Antigen-Presenting Cells Controls Mediators of the Th1 Immune Response during Leishmania major Infection.
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- PLoS Neglected Tropical Diseases, 2014, v. 8, n. 9, p. 1, doi. 10.1371/journal.pntd.0003194
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- Article
Cathepsin B in Antigen-Presenting Cells Controls Mediators of the Th1 Immune Response during Leishmania major Infection.
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- PLoS Neglected Tropical Diseases, 2014, v. 8, n. 9, p. 1, doi. 10.1371/journal.pntd.0003194
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- Article
Subnanomolar Cathepsin S Inhibitors with High Selectivity: Optimizing Covalent Reversible α‐Fluorovinylsulfones and α‐Sulfonates as Potential Immunomodulators in Cancer.
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- ChemMedChem, 2023, v. 18, n. 15, p. 1, doi. 10.1002/cmdc.202300160
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- Article
Front Cover: Structure‐Activity Relationships of Benzamides and Isoindolines Designed as SARS‐CoV Protease Inhibitors Effective against SARS‐CoV‐2 (2/2021)
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- ChemMedChem, 2021, v. 16, n. 2, p. 301, doi. 10.1002/cmdc.202000987
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- Article
Structure-Activity Relationships of Benzamides and Isoindolines Designed as SARS-CoV Protease Inhibitors Effective against SARS-CoV-2.
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- ChemMedChem, 2021, v. 16, n. 2, p. 340, doi. 10.1002/cmdc.202000548
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- Article
Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment.
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- ChemMedChem, 2020, v. 15, n. 16, p. 1552, doi. 10.1002/cmdc.202000360
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- Article
Development of Novel Benzodiazepine‐Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense.
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- ChemMedChem, 2020, v. 15, n. 11, p. 995, doi. 10.1002/cmdc.202000158
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- Article
Asymmetric Disulfanylbenzamides as Irreversible and Selective Inhibitors of Staphylococcus aureus Sortase A.
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- ChemMedChem, 2020, v. 15, n. 10, p. 839, doi. 10.1002/cmdc.201900687
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- Article
Inhibition of the Cysteine Protease Human Cathepsin L by Triazine Nitriles: Amide⋅⋅⋅Heteroarene π-Stacking Interactions and Chalcogen Bonding in the S3 Pocket.
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- ChemMedChem, 2017, v. 12, n. 3, p. 257, doi. 10.1002/cmdc.201600563
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- Article
Fluorine Scan of Inhibitors of the Cysteine Protease Human Cathepsin L: Dipolar and Quadrupolar Effects in the π-Stacking of Fluorinated Phenyl Rings on Peptide Amide Bonds.
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- ChemMedChem, 2016, v. 11, n. 10, p. 1042, doi. 10.1002/cmdc.201600132
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- Article
Dipeptidyl Enoates As Potent Rhodesain Inhibitors That Display a Dual Mode of Action.
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- ChemMedChem, 2015, v. 10, n. 9, p. 1484, doi. 10.1002/cmdc.201500204
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- Article
Development of Novel Selective Peptidomimetics Containing a Boronic Acid Moiety, Targeting the 20S Proteasome as Anticancer Agents.
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- ChemMedChem, 2014, v. 9, n. 8, p. 1801, doi. 10.1002/cmdc.201402075
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- Article
Synthesis and Biological Evaluation of Papain-Family Cathepsin L-Like Cysteine Protease Inhibitors Containing a 1,4-Benzodiazepine Scaffold as Antiprotozoal Agents.
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- ChemMedChem, 2014, v. 9, n. 8, p. 1817, doi. 10.1002/cmdc.201402079
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- Article
Development of Rhodesain Inhibitors with a 3-Bromoisoxazoline Warhead.
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- ChemMedChem, 2013, v. 8, n. 12, p. 2070, doi. 10.1002/cmdc.201300390
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- Article