Works by Scheuermann, Jörg

Results: 42

RGD Cyclopeptide Equipped with a Lysine‐Engaging Salicylaldehyde Showing Enhanced Integrin Affinity and Cell Detachment Potency.

Published in:

Chemistry - A European Journal, 2023, v. 29, n. 19, p. 1, doi. 10.1002/chem.202203768

By:

Sacco, Giovanni;
Arosio, Daniela;
Paolillo, Mayra;
Gloger, Andreas;
Scheuermann, Jörg;
Pignataro, Luca;
Belvisi, Laura;
Dal Corso, Alberto;
Gennari, Cesare

Publication type:

Article

Cover Feature: Affinity Selections of DNA‐Encoded Chemical Libraries on Carbonic Anhydrase IX‐Expressing Tumor Cells Reveal a Dependence on Ligand Valence (Chem. Eur. J. 35/2021).

Published in:

Chemistry - A European Journal, 2021, v. 27, n. 35, p. 8888, doi. 10.1002/chem.202101855

By:

Oehler, Sebastian;
Catalano, Marco;
Scapozza, Ilario;
Bigatti, Martina;
Bassi, Gabriele;
Favalli, Nicholas;
Mortensen, Michael R.;
Samain, Florent;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Affinity Selections of DNA‐Encoded Chemical Libraries on Carbonic Anhydrase IX‐Expressing Tumor Cells Reveal a Dependence on Ligand Valence.

Published in:

Chemistry - A European Journal, 2021, v. 27, n. 35, p. 8985, doi. 10.1002/chem.202100816

By:

Oehler, Sebastian;
Catalano, Marco;
Scapozza, Ilario;
Bigatti, Martina;
Bassi, Gabriele;
Favalli, Nicholas;
Mortensen, Michael R.;
Samain, Florent;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

A DNA‐Encoded Chemical Library Based on Peptide Macrocycles.

Published in:

Chemistry - A European Journal, 2021, v. 27, n. 24, p. 7160, doi. 10.1002/chem.202005423

By:

Onda, Yuichi;
Bassi, Gabriele;
Elsayed, Abdullah;
Ulrich, Franziska;
Oehler, Sebastian;
Plais, Louise;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Identification of Structure-Activity Relationships from Screening a Structurally Compact DNA-Encoded Chemical Library.

Published in:

Angewandte Chemie, 2015, v. 127, n. 13, p. 3999, doi. 10.1002/ange.201410736

By:

Franzini, Raphael M.;
Ekblad, Torun;
Zhong, Nan;
Wichert, Moreno;
Decurtins, Willy;
Nauer, Angela;
Zimmermann, Mauro;
Samain, Florent;
Scheuermann, Jörg;
Brown, Peter J.;
Hall, Jonathan;
Gräslund, Susanne;
Schüler, Herwig;
Neri, Dario

Publication type:

Article

Entwicklung zielgerichteter niedermolekularer zytotoxischer Wirkstoffverbindungen mit DNA-codierten chemischen Bibliotheken.

Published in:

Angewandte Chemie, 2013, v. 125, n. 5, p. 1424, doi. 10.1002/ange.201204631

By:

Krall, Nikolaus;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

A Traceless Vascular-Targeting Antibody-Drug Conjugate for Cancer Therapy.

Published in:

Angewandte Chemie, 2012, v. 124, n. 4, p. 965, doi. 10.1002/ange.201106527

By:

Bernardes, Gonçalo J. L.;
Casi, Giulio;
Trüssel, Sabrina;
Hartmann, Isabelle;
Schwager, Kathrin;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

A Portable Albumin Binder from a DNA-Encoded Chemical Library.

Published in:

Angewandte Chemie International Edition, 2008, v. 47, n. 17, p. 3196, doi. 10.1002/anie.200704936

By:

Dumelin, Christoph E.;
Trüssel, Sabrina;
Buller, Fabian;
Trachsel, Eveline;
Bootz, Frank;
Zhang, Yixin;
Mannocci, Luca;
Beck, Susanne C.;
Drumea-Mirancea, Mihaela;
Seeliger, Mathias W.;
Baltes, Christof;
Müggler, Thomas;
Kranz, Felicitas;
Rudin, Markus;
Melkko, Samu;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Isolation of High-Affinity Trypsin Inhibitors from a DNA-Encoded Chemical Library.

Published in:

Angewandte Chemie International Edition, 2007, v. 46, n. 25, p. 4671, doi. 10.1002/anie.200700654

By:

Melkko, Samu;
Zhang, Yixin;
Dumelin, Christoph E.;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

A Specific and Covalent JNK-1 Ligand Selected from an Encoded Self-Assembling Chemical Library.

Published in:

Chemistry - A European Journal, 2017, v. 23, n. 34, p. 8152, doi. 10.1002/chem.201701644

By:

Zimmermann, Gunther;
Rieder, Ulrike;
Bajic, Davor;
Vanetti, Sara;
Chaikuad, Apirat;
Knapp, Stefan;
Scheuermann, Jörg;
Mattarella, Martin;
Neri, Dario

Publication type:

Article

Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker.

Published in:

Frontiers in Pharmacology, 2023, p. 1, doi. 10.3389/fphar.2023.1320524

By:

Lopez, Lydia Bisbal;
Ravazza, Domenico;
Bocci, Matilde;
Zana, Aureliano;
Principi, Lucrezia;
Plaza, Sheila Dakhel;
Galbiati, Andrea;
Gilardoni, Ettore;
Scheuermann, Jörg;
Neri, Dario;
Pignataro, Luca;
Gennari, Cesare;
Cazzamalli, Samuele;
Dal Corso, Alberto

Publication type:

Article

Discovery of Small-Molecule Interleukin-2 Inhibitors from a DNA-Encoded Chemical Library.

Published in:

Chemistry - A European Journal, 2012, v. 18, n. 25, p. 7729, doi. 10.1002/chem.201200952

By:

Leimbacher, Markus;
Zhang, Yixin;
Mannocci, Luca;
Stravs, Michael;
Geppert, Tim;
Scheuermann, Jörg;
Schneider, Gisbert;
Neri, Dario

Publication type:

Article

Discovery and investigation of lead compounds as binders to the Extra-Domain B of the angiogenesis marker, fibronectin.

Published in:

Drug Development Research, 2003, v. 58, n. 3, p. 268, doi. 10.1002/ddr.10161

By:

Scheuermann, Jörg;
Volonterio, Alessandro;
Zerbe, Oliver;
Zanda, Matteo;
Neri, Dario

Publication type:

Article

Encoded self-assembling chemical libraries.

Published in:

Nature Biotechnology, 2004, v. 22, n. 5, p. 568, doi. 10.1038/nbt961

By:

Melkko, Samu;
Scheuermann, Jörg;
Dumelin, Christoph E.;
Neri, Dario

Publication type:

Article

A Single‐Stranded DNA‐Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks.

Published in:

Advanced Science, 2020, v. 7, n. 22, p. 1, doi. 10.1002/advs.202001970

By:

Bassi, Gabriele;
Favalli, Nicholas;
Vuk, Miriam;
Catalano, Marco;
Martinelli, Adriano;
Trenner, Anika;
Porro, Antonio;
Yang, Su;
Tham, Chuin Lean;
Moroglu, Mustafa;
Yue, Wyatt W.;
Conway, Stuart J.;
Vogt, Peter K.;
Sartori, Alessandro A.;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Flexibility-tuning of dual-display DNA-encoded chemical libraries facilitates cyclic peptide ligand discovery.

Published in:

Nature Communications, 2025, v. 16, n. 1, p. 1, doi. 10.1038/s41467-025-58507-w

By:

Petrov, Dimitar;
Plais, Louise;
Schira, Kristina;
Cai, Junyu;
Keller, Michelle;
Lessing, Alice;
Bassi, Gabriele;
Cazzamalli, Samuele;
Neri, Dario;
Gloger, Andreas;
Scheuermann, Jörg

Publication type:

Article

Impact of DNA-Encoded Chemical Library Technology on Drug Discovery.

Published in:

Chimia, 2022, v. 76, n. 5, p. 388, doi. 10.2533/chimia.2022.388

By:

Keller, Michelle;
Schira, Kristina;
Scheuermann, Jörg

Publication type:

Article

DNA‐encoded chemical libraries – achievements and remaining challenges.

Published in:

FEBS Letters, 2018, v. 592, n. 12, p. 2168, doi. 10.1002/1873-3468.13068

By:

Favalli, Nicholas;
Bassi, Gabriele;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Automated and enhanced extraction of a small molecule-drug conjugate using an enzyme-inhibitor interaction based SPME tool followed by direct analysis by ESI-MS.

Published in:

Analytical & Bioanalytical Chemistry, 2019, v. 411, n. 28, p. 7387, doi. 10.1007/s00216-019-02165-7

By:

Ghiasikhou, Sahar;
Cazzamalli, Samuele;
Scheuermann, Jörg;
Neri, Dario;
Zenobi, Renato

Publication type:

Article

Affinity Enhancement of Protein Ligands by Reversible Covalent Modification of Neighboring Lysine Residues.

Published in:

Angewandte Chemie, 2018, v. 130, n. 52, p. 17424, doi. 10.1002/ange.201811650

By:

Dal Corso, Alberto;
Catalano, Marco;
Schmid, Anja;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Ligand-Based Vascular Targeting of Disease.

Published in:

ChemMedChem, 2007, v. 2, n. 1, p. 22, doi. 10.1002/cmdc.200600181

By:

Rybak, Jascha-N.;
Trachsel, Eveline;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Affinity Enhancement of Protein Ligands by Reversible Covalent Modification of Neighboring Lysine Residues.

Published in:

Angewandte Chemie International Edition, 2018, v. 57, n. 52, p. 17178, doi. 10.1002/anie.201811650

By:

Dal Corso, Alberto;
Catalano, Marco;
Schmid, Anja;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Integration von internen Qualitäts-, Sicherheits- und Umweltschutz-Audits in Pharmaunternehmen.

Published in:

Pharmazeutische Industrie (Pharmind), 2005, v. 67, n. 11, p. 1277

By:

Mocha, Denise;
Scheuermann, Hans-Jörg;
Skuballa, Birgit;
Ottnad, Michael;
Wozniewski, Thomas;
Müller, Rainer Helmut

Publication type:

Article

Integration von internen Qualitäts-, Sicherheits- und Umweltschutz-Audits in Pharmaunternehmen.

Published in:

Pharmazeutische Industrie (Pharmind), 2005, v. 67, n. 10, p. 1148

By:

Mocha, Denise;
Scheuermann, Hans-Jörg;
Skuballa, Birgit;
Ottnad, Michael;
Wozniewski, Thomas;
Müller, Rainer Helmut

Publication type:

Article

Intergration von internen Qualitäts-, Sicherheits- und Umweltschutz-Audits in Pharmaunternehmen.

Published in:

Pharmazeutische Industrie (Pharmind), 2005, v. 67, n. 9, p. 1023

By:

Mocha, Denise;
Scheuermann, Hans-Jörg;
Skulballa, Birgit;
Ottnad, Michael;
Wozniewski, Thomas;
Müller, Rainer Helmut

Publication type:

Article

Einblick in die Organisation von Managementsystemen im Bereich der Produktion chemisch-pharmazeutischer Unternehmen in Deutschland.

Published in:

Pharmazeutische Industrie (Pharmind), 2004, v. 66, n. 8, p. 948

By:

Rank, Franziska;
Scheuermann, Hans-Jörg;
Wozniewski, Thomas;
Müller, Rainer Helmut

Publication type:

Article

Automated screening for small organic ligands using DNA-encoded chemical libraries.

Published in:

Nature Protocols, 2016, v. 11, n. 4, p. 764, doi. 10.1038/nprot.2016.039

By:

Decurtins, Willy;
Wichert, Moreno;
Franzini, Raphael M;
Buller, Fabian;
Stravs, Michael A;
Zhang, Yixin;
Neri, Dario;
Scheuermann, Jörg

Publication type:

Article

Quantitative Assessment of Affinity Selection Performance by Using DNA‐Encoded Chemical Libraries.

Published in:

ChemBioChem, 2019, v. 20, n. 7, p. 955, doi. 10.1002/cbic.201800766

By:

Sannino, Alessandro;
Gabriele, Elena;
Bigatti, Martina;
Mulatto, Sara;
Piazzi, Jacopo;
Scheuermann, Jörg;
Neri, Dario;
Donckele, Etienne J.;
Samain, Florent

Publication type:

Article

Back Cover: Quantitative PCR is a Valuable Tool to Monitor the Performance of DNA-Encoded Chemical Library Selections (ChemBioChem 9/2017).

Published in:

ChemBioChem, 2017, v. 18, n. 9, p. 880, doi. 10.1002/cbic.201700181

By:

Li, Yizhou;
Zimmermann, Gunther;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Hit-Validation Methodologies for Ligands Isolated from DNA-Encoded Chemical Libraries.

Published in:

ChemBioChem, 2017, v. 18, n. 9, p. 853, doi. 10.1002/cbic.201600637

By:

Zimmermann, Gunther;
Li, Yizhou;
Rieder, Ulrike;
Mattarella, Martin;
Neri, Dario;
Scheuermann, Jörg

Publication type:

Article

Quantitative PCR is a Valuable Tool to Monitor the Performance of DNA-Encoded Chemical Library Selections.

Published in:

ChemBioChem, 2017, v. 18, n. 9, p. 848, doi. 10.1002/cbic.201600626

By:

Li, Yizhou;
Zimmermann, Gunther;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

DNA-Encoded Chemical Libraries: A Tool for Drug Discovery and for Chemical Biology.

Published in:

ChemBioChem, 2010, v. 11, n. 7, p. 931, doi. 10.1002/cbic.201000066

By:

Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Screening of Three Transition Metal‐Mediated Reactions Compatible with DNA‐Encoded Chemical Libraries.

Published in:

Helvetica Chimica Acta, 2019, v. 102, n. 4, p. N.PAG, doi. 10.1002/hlca.201900033

By:

Favalli, Nicholas;
Bassi, Gabriele;
Zanetti, Tania;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

Dual-display of small molecules enables the discovery of ligand pairs and facilitates affinity maturation.

Published in:

Nature Chemistry, 2015, v. 7, n. 3, p. 241, doi. 10.1038/nchem.2158

By:

Wichert, Moreno;
Krall, Nikolaus;
Decurtins, Willy;
Franzini, Raphael M.;
Pretto, Francesca;
Schneider, Petra;
Neri, Dario;
Scheuermann, Jörg

Publication type:

Article

Isolation of a Natural Killer Group 2D Small‐Molecule Ligand from DNA‐Encoded Chemical Libraries.

Published in:

ChemMedChem, 2022, v. 17, n. 21, p. 1, doi. 10.1002/cmdc.202200350

By:

Dakhel, Sheila;
Galbiati, Andrea;
Migliorini, Francesca;
Comacchio, Claudia;
Oehler, Sebastian;
Prati, Luca;
Scheuermann, Jörg;
Cazzamalli, Samuele;
Neri, Dario;
Bassi, Gabriele;
Favalli, Nicholas

Publication type:

Article

Selective Fragments for the CREBBP Bromodomain Identified from an Encoded Self‐assembly Chemical Library.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1752, doi. 10.1002/cmdc.202000528

By:

Catalano, Marco;
Moroglu, Mustafa;
Balbi, Petra;
Mazzieri, Federica;
Clayton, James;
Andrews, Katrina H.;
Bigatti, Martina;
Scheuermann, Jörg;
Conway, Stuart J.;
Neri, Dario

Publication type:

Article

Cover Feature: A DNA‐Encoded Library of Chemical Compounds Based on Common Scaffolding Structures Reveals the Impact of Ligand Geometry on Protein Recognition (ChemMedChem 13/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 13, p. 1261, doi. 10.1002/cmdc.201800416

By:

Favalli, Nicholas;
Biendl, Stefan;
Hartmann, Marco;
Piazzi, Jacopo;
Sladojevich, Filippo;
Gräslund, Susanne;
Brown, Peter J.;
Näreoja, Katja;
Schüler, Herwig;
Scheuermann, Jörg;
Franzini, Raphael;
Neri, Dario

Publication type:

Article

A DNA‐Encoded Library of Chemical Compounds Based on Common Scaffolding Structures Reveals the Impact of Ligand Geometry on Protein Recognition.

Published in:

ChemMedChem, 2018, v. 13, n. 13, p. 1303, doi. 10.1002/cmdc.201800193

By:

Favalli, Nicholas;
Biendl, Stefan;
Hartmann, Marco;
Piazzi, Jacopo;
Sladojevich, Filippo;
Gräslund, Susanne;
Brown, Peter J.;
Näreoja, Katja;
Schüler, Herwig;
Scheuermann, Jörg;
Franzini, Raphael;
Neri, Dario

Publication type:

Article

Impact of a Central Scaffold on the Binding Affinity of Fragment Pairs Isolated from DNA-Encoded Self-Assembling Chemical Libraries.

Published in:

ChemMedChem, 2017, v. 12, n. 21, p. 1748, doi. 10.1002/cmdc.201700569

By:

Bigatti, Martina;
Dal Corso, Alberto;
Vanetti, Sara;
Cazzamalli, Samuele;
Rieder, Ulrike;
Scheuermann, Jörg;
Neri, Dario;
Sladojevich, Filippo

Publication type:

Article

Identification of Structure-Activity Relationships from Screening a Structurally Compact DNA-Encoded Chemical Library.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 13, p. 3927, doi. 10.1002/anie.201410736

By:

Franzini, Raphael M.;
Ekblad, Torun;
Zhong, Nan;
Wichert, Moreno;
Decurtins, Willy;
Nauer, Angela;
Zimmermann, Mauro;
Samain, Florent;
Scheuermann, Jörg;
Brown, Peter J.;
Hall, Jonathan;
Gräslund, Susanne;
Schüler, Herwig;
Neri, Dario

Publication type:

Article

Small Targeted Cytotoxics: Current State and Promises from DNA-Encoded Chemical Libraries.

Published in:

Angewandte Chemie International Edition, 2013, v. 52, n. 5, p. 1384, doi. 10.1002/anie.201204631

By:

Krall, Nikolaus;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article

A Traceless Vascular-Targeting Antibody-Drug Conjugate for Cancer Therapy.

Published in:

Angewandte Chemie International Edition, 2012, v. 51, n. 4, p. 941, doi. 10.1002/anie.201106527

By:

Bernardes, Gonçalo J. L.;
Casi, Giulio;
Trüssel, Sabrina;
Hartmann, Isabelle;
Schwager, Kathrin;
Scheuermann, Jörg;
Neri, Dario

Publication type:

Article