Works matching AU Rogers, Catherine M.

Results: 15
    1

    LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor.

    Published in:
    Angewandte Chemie, 2015, v. 127, n. 21, p. 6315, doi. 10.1002/ange.201501394
    By:
    • Clark, Peter G. K.;
    • Vieira, Lucas C. C.;
    • Tallant, Cynthia;
    • Fedorov, Oleg;
    • Singleton, Dean C.;
    • Rogers, Catherine M.;
    • Monteiro, Octovia P.;
    • Bennett, James M.;
    • Baronio, Roberta;
    • Müller, Susanne;
    • Daniels, Danette L.;
    • Méndez, Jacqui;
    • Knapp, Stefan;
    • Brennan, Paul E.;
    • Dixon, Darren J.
    Publication type:
    Article
    2

    A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction.

    Published in:
    Angewandte Chemie, 2014, v. 126, n. 24, p. 6240, doi. 10.1002/ange.201402750
    By:
    • Rooney, Timothy P. C.;
    • Filippakopoulos, Panagis;
    • Fedorov, Oleg;
    • Picaud, Sarah;
    • Cortopassi, Wilian A.;
    • Hay, Duncan A.;
    • Martin, Sarah;
    • Tumber, Anthony;
    • Rogers, Catherine M.;
    • Philpott, Martin;
    • Wang, Minghua;
    • Thompson, Amber L.;
    • Heightman, Tom D.;
    • Pryde, David C.;
    • Cook, Andrew;
    • Paton, Robert S.;
    • Müller, Susanne;
    • Knapp, Stefan;
    • Brennan, Paul E.;
    • Conway, Stuart J.
    Publication type:
    Article
    3

    Phenomics‐Based Discovery of Novel Orthosteric Choline Kinase Inhibitors.

    Published in:
    Angewandte Chemie International Edition, 2025, v. 64, n. 7, p. 1, doi. 10.1002/anie.202420149
    By:
    • Bauer, Ludwig G.;
    • Ward, Jennifer A.;
    • Díaz‐Sáez, Laura;
    • Sundström, Yvonne;
    • Tolvanen, Tuomas;
    • Alarcón Barrera, Juan Carlos;
    • Kostidis, Sarantos;
    • Rogers, Catherine M.;
    • Panagakou, Ioanna;
    • Singh, Usha;
    • Rothweiler, Elisabeth M.;
    • Gonzalez Orta, Alejandro;
    • Kaniskan, H. Ümit;
    • Hu, Jianping;
    • Jin, Jian;
    • Sievers, Sonja;
    • Waldmann, Herbert;
    • Giera, Martin;
    • Sundström, Michael;
    • Berg, Louise
    Publication type:
    Article
    4
    5

    Phänomik‐basierte Entdeckung neuer orthosterischer Cholinkinase Inhibitoren.

    Published in:
    Angewandte Chemie, 2025, v. 137, n. 7, p. 1, doi. 10.1002/ange.202420149
    By:
    • Bauer, Ludwig G.;
    • Ward, Jennifer A.;
    • Díaz‐Sáez, Laura;
    • Sundström, Yvonne;
    • Tolvanen, Tuomas;
    • Alarcón Barrera, Juan Carlos;
    • Kostidis, Sarantos;
    • Rogers, Catherine M.;
    • Panagakou, Ioanna;
    • Singh, Usha;
    • Rothweiler, Elisabeth M.;
    • Gonzalez Orta, Alejandro;
    • Kaniskan, H. Ümit;
    • Hu, Jianping;
    • Jin, Jian;
    • Sievers, Sonja;
    • Waldmann, Herbert;
    • Giera, Martin;
    • Sundström, Michael;
    • Berg, Louise
    Publication type:
    Article
    6

    Design, Synthesis and Characterization of Covalent KDM5 Inhibitors.

    Published in:
    Angewandte Chemie, 2019, v. 131, n. 2, p. 525, doi. 10.1002/ange.201810179
    By:
    • Vazquez‐Rodriguez, Saleta;
    • Wright, Miranda;
    • Rogers, Catherine M.;
    • Cribbs, Adam P.;
    • Velupillai, Srikannathasan;
    • Philpott, Martin;
    • Lee, Henry;
    • Dunford, James E.;
    • Huber, Kilian V. M.;
    • Robers, Matthew B.;
    • Vasta, James D.;
    • Thezenas, Marie‐Laetitia;
    • Bonham, Sarah;
    • Kessler, Benedikt;
    • Bennett, James;
    • Fedorov, Oleg;
    • Raynaud, Florence;
    • Donovan, Adam;
    • Blagg, Julian;
    • Bavetsias, Vassilios
    Publication type:
    Article
    7

    Discovery of a PCAF Bromodomain Chemical Probe.

    Published in:
    Angewandte Chemie, 2017, v. 129, n. 3, p. 845, doi. 10.1002/ange.201610816
    By:
    • Moustakim, Moses;
    • Clark, Peter G. K.;
    • Trulli, Laura;
    • Fuentes de Arriba, Angel L.;
    • Ehebauer, Matthias T.;
    • Chaikuad, Apirat;
    • Murphy, Emma J.;
    • Mendez ‐ Johnson, Jacqui;
    • Daniels, Danette;
    • Hou, Chun ‐ Feng D.;
    • Lin, Yu ‐ Hui;
    • Walker, John R.;
    • Hui, Raymond;
    • Yang, Hongbing;
    • Dorrell, Lucy;
    • Rogers, Catherine M.;
    • Monteiro, Octovia P.;
    • Fedorov, Oleg;
    • Huber, Kilian V. M.;
    • Knapp, Stefan
    Publication type:
    Article
    8

    Rücktitelbild: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. 3/2017).

    Published in:
    Angewandte Chemie, 2017, v. 129, n. 3, p. 928, doi. 10.1002/ange.201612063
    By:
    • Moustakim, Moses;
    • Clark, Peter G. K.;
    • Trulli, Laura;
    • Fuentes de Arriba, Angel L.;
    • Ehebauer, Matthias T.;
    • Chaikuad, Apirat;
    • Murphy, Emma J.;
    • Mendez ‐ Johnson, Jacqui;
    • Daniels, Danette;
    • Hou, Chun ‐ Feng D.;
    • Lin, Yu ‐ Hui;
    • Walker, John R.;
    • Hui, Raymond;
    • Yang, Hongbing;
    • Dorrell, Lucy;
    • Rogers, Catherine M.;
    • Monteiro, Octovia P.;
    • Fedorov, Oleg;
    • Huber, Kilian V. M.;
    • Knapp, Stefan
    Publication type:
    Article
    9

    Design, Synthesis and Characterization of Covalent KDM5 Inhibitors.

    Published in:
    Angewandte Chemie International Edition, 2019, v. 58, n. 2, p. 515, doi. 10.1002/anie.201810179
    By:
    • Vazquez‐Rodriguez, Saleta;
    • Wright, Miranda;
    • Rogers, Catherine M.;
    • Cribbs, Adam P.;
    • Velupillai, Srikannathasan;
    • Philpott, Martin;
    • Lee, Henry;
    • Dunford, James E.;
    • Huber, Kilian V. M.;
    • Robers, Matthew B.;
    • Vasta, James D.;
    • Thezenas, Marie‐Laetitia;
    • Bonham, Sarah;
    • Kessler, Benedikt;
    • Bennett, James;
    • Fedorov, Oleg;
    • Raynaud, Florence;
    • Donovan, Adam;
    • Blagg, Julian;
    • Bavetsias, Vassilios
    Publication type:
    Article
    10

    Discovery of an MLLT1/3 YEATS Domain Chemical Probe.

    Published in:
    Angewandte Chemie International Edition, 2018, v. 57, n. 50, p. 16302, doi. 10.1002/anie.201810617
    By:
    • Moustakim, Moses;
    • Christott, Thomas;
    • Monteiro, Octovia P.;
    • Bennett, James;
    • Giroud, Charline;
    • Ward, Jennifer;
    • Rogers, Catherine M.;
    • Smith, Paul;
    • Panagakou, Ioanna;
    • Díaz‐Sáez, Laura;
    • Felce, Suet Ling;
    • Gamble, Vicki;
    • Gileadi, Carina;
    • Halidi, Nadia;
    • Heidenreich, David;
    • Chaikuad, Apirat;
    • Knapp, Stefan;
    • Huber, Kilian V. M.;
    • Farnie, Gillian;
    • Heer, Jag
    Publication type:
    Article
    11

    Discovery of a PCAF Bromodomain Chemical Probe.

    Published in:
    Angewandte Chemie International Edition, 2017, v. 56, n. 3, p. 827, doi. 10.1002/anie.201610816
    By:
    • Moustakim, Moses;
    • Clark, Peter G. K.;
    • Trulli, Laura;
    • Fuentes de Arriba, Angel L.;
    • Ehebauer, Matthias T.;
    • Chaikuad, Apirat;
    • Murphy, Emma J.;
    • Mendez-Johnson, Jacqui;
    • Daniels, Danette;
    • Hou, Chun-Feng D.;
    • Lin, Yu-Hui;
    • Walker, John R.;
    • Hui, Raymond;
    • Yang, Hongbing;
    • Dorrell, Lucy;
    • Rogers, Catherine M.;
    • Monteiro, Octovia P.;
    • Fedorov, Oleg;
    • Huber, Kilian V. M.;
    • Knapp, Stefan
    Publication type:
    Article
    12

    Back Cover: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. Int. Ed. 3/2017).

    Published in:
    Angewandte Chemie International Edition, 2017, v. 56, n. 3, p. 908, doi. 10.1002/anie.201612063
    By:
    • Moustakim, Moses;
    • Clark, Peter G. K.;
    • Trulli, Laura;
    • Fuentes de Arriba, Angel L.;
    • Ehebauer, Matthias T.;
    • Chaikuad, Apirat;
    • Murphy, Emma J.;
    • Mendez-Johnson, Jacqui;
    • Daniels, Danette;
    • Hou, Chun-Feng D.;
    • Lin, Yu-Hui;
    • Walker, John R.;
    • Hui, Raymond;
    • Yang, Hongbing;
    • Dorrell, Lucy;
    • Rogers, Catherine M.;
    • Monteiro, Octovia P.;
    • Fedorov, Oleg;
    • Huber, Kilian V. M.;
    • Knapp, Stefan
    Publication type:
    Article
    13

    Engineering an in-vitro model of rodent cartilage.

    Published in:
    Journal of Pharmacy & Pharmacology, 2012, v. 64, n. 6, p. 821, doi. 10.1111/j.2042-7158.2012.01491.x
    By:
    • Rogers, Catherine M.;
    • Woolley, Terry S.;
    • Cruwys, Simon C.;
    • Buttery, Lee D.K.;
    • Rose, Felicity R.A.J.;
    • Shakesheff, Kevin M.
    Publication type:
    Article
    14

    LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor.

    Published in:
    Angewandte Chemie International Edition, 2015, v. 54, n. 21, p. 6217, doi. 10.1002/anie.201501394
    By:
    • Clark, Peter G. K.;
    • Vieira, Lucas C. C.;
    • Dixon, Darren J.;
    • Tallant, Cynthia;
    • Fedorov, Oleg;
    • Singleton, Dean C.;
    • Rogers, Catherine M.;
    • Monteiro, Octovia P.;
    • Bennett, James M.;
    • Baronio, Roberta;
    • Müller, Susanne;
    • Knapp, Stefan;
    • Brennan, Paul E.;
    • Daniels, Danette L.;
    • Méndez, Jacqui
    Publication type:
    Article
    15

    A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction.

    Published in:
    Angewandte Chemie International Edition, 2014, v. 53, n. 24, p. 6126, doi. 10.1002/anie.201402750
    By:
    • Rooney, Timothy P. C.;
    • Filippakopoulos, Panagis;
    • Fedorov, Oleg;
    • Picaud, Sarah;
    • Cortopassi, Wilian A.;
    • Hay, Duncan A.;
    • Martin, Sarah;
    • Tumber, Anthony;
    • Rogers, Catherine M.;
    • Philpott, Martin;
    • Wang, Minghua;
    • Thompson, Amber L.;
    • Heightman, Tom D.;
    • Pryde, David C.;
    • Cook, Andrew;
    • Paton, Robert S.;
    • Müller, Susanne;
    • Knapp, Stefan;
    • Brennan, Paul E.;
    • Conway, Stuart J.
    Publication type:
    Article