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Azaindoles as Zinc-Binding Small-Molecule Inhibitors of the JAMM Protease CSN5.
Published in:
Angewandte Chemie, 2017, v. 129, n. 5, p. 1314, doi. 10.1002/ange.201608672
By:
- Altmann, Eva;
- Erbel, Paul;
- Renatus, Martin;
- Schaefer, Michael;
- Schlierf, Anita;
- Druet, Adelaide;
- Kieffer, Laurence;
- Sorge, Mickael;
- Pfister, Keith;
- Hassiepen, Ulrich;
- Jones, Matthew;
- Ruedisser, Simon;
- Ostermeier, Daniela;
- Martoglio, Bruno;
- Jefferson, Anne B.;
- Quancard, Jean
Publication type:
Article
Azaindoles as Zinc-Binding Small-Molecule Inhibitors of the JAMM Protease CSN5.
Published in:
Angewandte Chemie International Edition, 2017, v. 56, n. 5, p. 1294, doi. 10.1002/anie.201608672
By:
- Altmann, Eva;
- Erbel, Paul;
- Renatus, Martin;
- Schaefer, Michael;
- Schlierf, Anita;
- Druet, Adelaide;
- Kieffer, Laurence;
- Sorge, Mickael;
- Pfister, Keith;
- Hassiepen, Ulrich;
- Jones, Matthew;
- Ruedisser, Simon;
- Ostermeier, Daniela;
- Martoglio, Bruno;
- Jefferson, Anne B.;
- Quancard, Jean
Publication type:
Article
The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit Generation.
Published in:
ChemMedChem, 2023, v. 18, n. 9, p. 1, doi. 10.1002/cmdc.202300002
By:
- Quancard, Jean;
- Vulpetti, Anna;
- Bach, Anders;
- Cox, Brian;
- Guéret, Stéphanie M.;
- Hartung, Ingo V.;
- Koolman, Hannes F.;
- Laufer, Stefan;
- Messinger, Josef;
- Sbardella, Gianluca;
- Craft, Russell
Publication type:
Article
The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Phenotypic Drug Discovery.
Published in:
ChemMedChem, 2021, v. 16, n. 11, p. 1736, doi. 10.1002/cmdc.202100041
By:
- Quancard, Jean;
- Bach, Anders;
- Cox, Brian;
- Craft, Russell;
- Finsinger, Dirk;
- Guéret, Stéphanie M.;
- Hartung, Ingo V.;
- Laufer, Stefan;
- Messinger, Josef;
- Sbardella, Gianluca;
- Koolman, Hannes F.
Publication type:
Article
The European Federation for Medicinal Chemistry (EFMC) Best Practice Initiative: Validating Chemical Probes.
Published in:
ChemMedChem, 2020, v. 15, n. 24, p. 2388, doi. 10.1002/cmdc.202000597
By:
- Quancard, Jean;
- Cox, Brian;
- Finsinger, Dirk;
- Guéret, Stéphanie M.;
- Hartung, Ingo V.;
- Koolman, Hannes F.;
- Messinger, Josef;
- Sbardella, Gianluca;
- Laufer, Stefan
Publication type:
Article
Pharmacological Inhibition of MALT1 Protease Leads to a Progressive IPEX-Like Pathology.
Published in:
Frontiers in Immunology, 2020, v. 11, p. 1, doi. 10.3389/fimmu.2020.00745
By:
- Martin, Kea;
- Junker, Ursula;
- Tritto, Elaine;
- Sutter, Esther;
- Rubic-Schneider, Tina;
- Morgan, Hannah;
- Niwa, Satoru;
- Li, Jianping;
- Schlapbach, Achim;
- Walker, Dana;
- Bigaud, Marc;
- Beerli, Christian;
- Littlewood-Evans, Amanda;
- Rudolph, Bettina;
- Laisney, Marc;
- Ledieu, David;
- Beltz, Karen;
- Quancard, Jean;
- Bornancin, Frédéric;
- Zamurovic Ribrioux, Natasa
Publication type:
Article
Stabilizing Inactive Conformations of MALT1 as an Effective Approach to Inhibit Its Protease Activity.
Published in:
Advanced Therapeutics, 2020, v. 3, n. 9, p. 1, doi. 10.1002/adtp.202000078
By:
- Hughes, Nicola;
- Erbel, Paul;
- Bornancin, Frédéric;
- Wiesmann, Christian;
- Schiering, Nikolaus;
- Villard, Frédéric;
- Decock, Arnaud;
- Rubi, Bertran;
- Melkko, Samu;
- Spanka, Carsten;
- Buschmann, Nicole;
- Pissot‐Soldermann, Carole;
- Simic, Oliver;
- Beerli, René;
- Sorge, Mickael;
- Tintelnot‐Blomley, Marina;
- Beltz, Karen;
- Régnier, Catherine H.;
- Quancard, Jean;
- Schlapbach, Achim
Publication type:
Article
Targeted inhibition of the COP9 signalosome for treatment of cancer.
Published in:
Nature Communications, 2016, v. 7, n. 10, p. 13166, doi. 10.1038/ncomms13166
By:
- Schlierf, Anita;
- Altmann, Eva;
- Quancard, Jean;
- Jefferson, Anne B.;
- Assenberg, René;
- Renatus, Martin;
- Jones, Matthew;
- Hassiepen, Ulrich;
- Schaefer, Michael;
- Kiffe, Michael;
- Weiss, Andreas;
- Wiesmann, Christian;
- Sedrani, Richard;
- Eder, Jörg;
- Martoglio, Bruno
Publication type:
Article
Pathophysiological Consequences of a Break in S1P1-Dependent Homeostasis of Vascular Permeability Revealed by S1P1 Competitive Antagonism.
Published in:
PLoS ONE, 2016, v. 11, n. 12, p. 1, doi. 10.1371/journal.pone.0168252
By:
- Bigaud, Marc;
- Dincer, Zuhal;
- Bollbuck, Birgit;
- Dawson, Janet;
- Beckmann, Nicolau;
- Beerli, Christian;
- Fishli-Cavelti, Gina;
- Nahler, Michaela;
- Angst, Daniela;
- Janser, Philipp;
- Otto, Heike;
- Rosner, Elisabeth;
- Hersperger, Rene;
- Bruns, Christian;
- Quancard, Jean
Publication type:
Article
Requirement of Mucosa‐Associated Lymphoid Tissue Lymphoma Translocation Protein 1 Protease Activity for Fcγ Receptor–Induced Arthritis, but Not Fcγ Receptor–Mediated Platelet Elimination, in Mice.
Published in:
Arthritis & Rheumatology, 2020, v. 72, n. 6, p. 919, doi. 10.1002/art.41204
By:
- Martin, Kea;
- Touil, Ratiba;
- Cvijetic, Grozdan;
- Israel, Laura;
- Kolb, Yeter;
- Sarret, Sophie;
- Valeaux, Stéphanie;
- Degl'Innocenti, Elena;
- Le Meur, Thomas;
- Caesar, Nadja;
- Bardet, Maureen;
- Beerli, Christian;
- Zerwes, Hans‐Guenter;
- Kovarik, Jiri;
- Beltz, Karen;
- Schlapbach, Achim;
- Quancard, Jean;
- Régnier, Catherine H.;
- Bigaud, Marc;
- Junt, Tobias
Publication type:
Article
The T‐cell fingerprint of MALT1 paracaspase revealed by selective inhibition.
Published in:
Immunology & Cell Biology, 2018, v. 96, n. 1, p. 81, doi. 10.1111/imcb.1018
By:
- Bardet, Maureen;
- Unterreiner, Adeline;
- Malinverni, Claire;
- Lafossas, Frédérique;
- Vedrine, Corinne;
- Boesch, Danielle;
- Kolb, Yeter;
- Kaiser, Daniel;
- Glück, Anton;
- Schneider, Martin A.;
- Katopodis, Andreas;
- Renatus, Martin;
- Simic, Oliver;
- Schlapbach, Achim;
- Quancard, Jean;
- Régnier, Catherine H.;
- Bold, Guido;
- Pissot‐Soldermann, Carole;
- Carballido, José M.;
- Kovarik, Jiri
Publication type:
Article
A lead discovery strategy driven by a comprehensive analysis of proteases in the peptide substrate space.
Published in:
Protein Science: A Publication of the Protein Society, 2010, v. 19, n. 11, p. 2096, doi. 10.1002/pro.490
By:
- Sukuru, Sai Chetan K.;
- Nigsch, Florian;
- Quancard, Jean;
- Renatus, Martin;
- Chopra, Rajiv;
- Brooijmans, Natasja;
- Mikhailov, Dmitri;
- Deng, Zhan;
- Cornett, Allen;
- Jenkins, Jeremy L.;
- Hommel, Ulrich;
- Davies, John W.;
- Glick, Meir
Publication type:
Article
Inside Cover: Prolinoamino Acids as Tools to Build Bifunctionalized, Stable β-Turns in Water (ChemBioChem 1/2010).
Published in:
ChemBioChem, 2010, v. 11, n. 1, p. 2, doi. 10.1002/cbic.200990091
By:
- Mothes, Céline;
- Larregola, Maud;
- Quancard, Jean;
- Goasdoué, Nicole;
- Lavielle, Solange;
- Chassaing, Gérard;
- Lequin, Olivier;
- Karoyan, Philippe
Publication type:
Article
Prolinoamino Acids as Tools to Build Bifunctionalized, Stable β-Turns in Water.
Published in:
ChemBioChem, 2010, v. 11, n. 1, p. 55, doi. 10.1002/cbic.200900572
By:
- Mothes, Céline;
- Larregola, Maud;
- Quancard, Jean;
- Goasdoué, Nicole;
- Lavielle, Solange;
- Chassaing, Gérard;
- Lequin, Olivier;
- Karoyan, Philippe
Publication type:
Article

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