Works by Previti, Santo

Results: 16

Synthesis and Combination Studies of Novel Dipeptide Nitriles with Curcumin for a Potent Synergistic Action Against Rhodesain, Cysteine Protease of Trypanosoma brucei rhodesiense.

Published in:

Pharmaceuticals (14248247), 2025, v. 18, n. 6, p. 847, doi. 10.3390/ph18060847

By:

Di Chio, Carla;
Starvaggi, Josè;
Previti, Santo;
De Luca, Fabiola;
Natale, Benito;
Cosconati, Sandro;
Schirmeister, Tanja;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Article

Evaluation of curcumin irreversibility.

Published in:

2020

By:

Ettari, Roberta;
Previti, Santo;
Maiorana, Santina;
Allegra, Alessandro;
Schirmeister, Tanja;
Grasso, Silvana;
Zappalà, Maria

Publication type:

Letter

Drug combination studies of curcumin and genistein against rhodesain of Trypanosoma brucei rhodesiense.

Published in:

Natural Product Research, 2019, v. 33, n. 24, p. 3577, doi. 10.1080/14786419.2018.1483927

By:

Ettari, Roberta;
Previti, Santo;
Maiorana, Santina;
Allegra, Alessandro;
Schirmeister, Tanja;
Grasso, Silvana;
Zappalà, Maria

Publication type:

Article

Opening the amino acid toolbox for peptide‐based NTS2‐selective ligands as promising lead compounds for pain management.

Published in:

Journal of Peptide Science, 2023, v. 29, n. 6, p. 1, doi. 10.1002/psc.3471

By:

Previti, Santo;
Desgagné, Michael;
Tourwé, Dirk;
Cavelier, Florine;
Sarret, Philippe;
Ballet, Steven

Publication type:

Article

Drug combination studies of PS-1 and quercetin against rhodesain of Trypanosoma brucei rhodesiense.

Published in:

Natural Product Research, 2022, v. 36, n. 16, p. 4282, doi. 10.1080/14786419.2021.1978993

By:

Di Chio, Carla;
Previti, Santo;
De Luca, Fabiola;
Allegra, Alessandro;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Article

Synthesis and biological evaluation of novel peptidomimetics as rhodesain inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1184, doi. 10.3109/14756366.2015.1108972

By:

Ettari, Roberta;
Previti, Santo;
Cosconati, Sandro;
Kesselring, Jochen;
Schirmeister, Tanja;
Grasso, Silvana;
Zappalà, Maria

Publication type:

Article

Drug Combination Studies of Isoquinolinone AM12 with Curcumin or Quercetin: A New Combination Strategy to Synergistically Inhibit 20S Proteasome.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 19, p. 10708, doi. 10.3390/ijms251910708

By:

Di Chio, Carla;
Previti, Santo;
Starvaggi, Josè;
De Luca, Fabiola;
Calabrò, Maria Luisa;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Article

Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 8, p. 4410, doi. 10.3390/ijms25084410

By:

Di Chio, Carla;
Starvaggi, Josè;
Totaro, Noemi;
Previti, Santo;
Natale, Benito;
Cosconati, Sandro;
Bogacz, Marta;
Schirmeister, Tanja;
Legac, Jenny;
Rosenthal, Philip J.;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Article

The Inhibition of NS2B/NS3 Protease: A New Therapeutic Opportunity to Treat Dengue and Zika Virus Infection.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 8, p. 4376, doi. 10.3390/ijms25084376

By:

Starvaggi, Josè;
Previti, Santo;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Article

Dipeptide Nitrile CD34 with Curcumin: A New Improved Combination Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 10, p. 8477, doi. 10.3390/ijms24108477

By:

Di Chio, Carla;
Previti, Santo;
Totaro, Noemi;
De Luca, Fabiola;
Allegra, Alessandro;
Schirmeister, Tanja;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Article

Monoclonal Antibodies: The Greatest Resource to Treat Multiple Myeloma.

Published in:

2023

By:

De Luca, Fabiola;
Allegra, Alessandro;
Di Chio, Carla;
Previti, Santo;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Literature Review

Drug Combination Studies of the Dipeptide Nitrile CD24 with Curcumin: A New Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 22, p. 14470, doi. 10.3390/ijms232214470

By:

Di Chio, Carla;
Previti, Santo;
De Luca, Fabiola;
Bogacz, Marta;
Zimmer, Collin;
Wagner, Annika;
Schirmeister, Tanja;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Article

Development of Novel Benzodiazepine‐Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense.

Published in:

ChemMedChem, 2020, v. 15, n. 11, p. 995, doi. 10.1002/cmdc.202000158

By:

Di Chio, Carla;
Previti, Santo;
Amendola, Giorgio;
Cosconati, Sandro;
Schirmeister, Tanja;
Zappalà, Maria;
Ettari, Roberta

Publication type:

Article

Design and Synthesis of <sup>68</sup>Ga‐Labeled Peptide‐Based Heterodimers for Dual Targeting of NTS<sub>1</sub> and GRPR.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400843

By:

Bodin, Sacha;
Previti, Santo;
Jestin, Emmanuelle;
Rémond, Emmanuelle;
Vimont, Delphine;
Lamare, Frédéric;
Ait‐Arsa, Imade;
Hindié, Elif;
Cavelier, Florine;
Morgat, Clément

Publication type:

Article

Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1552, doi. 10.1002/cmdc.202000360

By:

Maiorana, Santina;
Ettari, Roberta;
Previti, Santo;
Amendola, Giorgio;
Wagner, Annika;
Cosconati, Sandro;
Hellmich, Ute A.;
Schirmeister, Tanja;
Zappalà, Maria

Publication type:

Article

Development of Reduced Peptide Bond Pseudopeptide Michael Acceptors for the Treatment of Human African Trypanosomiasis.

Published in:

Molecules, 2022, v. 27, n. 12, p. 3765, doi. 10.3390/molecules27123765

By:

Previti, Santo;
Ettari, Roberta;
Di Chio, Carla;
Ravichandran, Rahul;
Bogacz, Marta;
Hellmich, Ute A.;
Schirmeister, Tanja;
Cosconati, Sandro;
Zappalà, Maria

Publication type:

Article