Works by Porcal, Williams

Results: 19

Garbage in, garbage out: how reliable training data improved a virtual screening approach against SARS-CoV-2 MPro.

Published in:

Frontiers in Pharmacology, 2023, p. 1, doi. 10.3389/fphar.2023.1193282

By:

Ruatta, Santiago M.;
Prada Gori, Denis N.;
Fló Díaz, Martín;
Lorenzelli, Franca;
Perelmuter, Karen;
Alberca, Lucas N.;
Bellera, Carolina L.;
Medeiros, Andrea;
López, Gloria V.;
Ingold, Mariana;
Porcal, Williams;
Dibello, Estefanía;
Ihnatenko, Irina;
Kunick, Conrad;
Incerti, Marcelo;
Luzardo, Martín;
Colobbio, Maximiliano;
Carlos Ramos, Juan;
Manta, Eduardo;
Minini, Lucía

Publication type:

Article

Biological Assessment of a 18F-Labeled Sulforhodamine 101 in a Mouse Model of Alzheimer's Disease as a Potential Astrocytosis Marker.

Published in:

Frontiers in Neuroscience, 2019, p. 1, doi. 10.3389/fnins.2019.00734

By:

Kreimerman, Ingrid;
Reyes, Ana Laura;
Paolino, Andrea;
Pardo, Tania;
Porcal, Williams;
Ibarra, Manuel;
Oliver, Patricia;
Savio, Eduardo;
Engler, Henry

Publication type:

Article

Microwave-Assisted Solid-Phase Synthesis of a 1,2-Disubstituted Benzimidazole Library by Using a Phosphonium Linker.

Published in:

Journal of Heterocyclic Chemistry, 2013, v. 50, n. 3, p. 720, doi. 10.1002/jhet.1619

By:

Ríos, Natalia;
Chavarría, Cecilia;
Gil, Carmen;
Porcal, Williams

Publication type:

Article

Benzo[1, 2- c]1, 2, 5-oxadiazole N-Oxide Derivatives as Potential Antitrypanosomal Drugs. Structure-Activity Relationships. Part II.

Published in:

Archiv der Pharmazie, 2002, v. 335, n. 1, p. 15, doi. 10.1002/1521-4184(200201)335:1<15::AID-ARDP15>3.0.CO;2-8

By:

Aguirre, Gabriela;
Cerecetto, Hugo;
Di Maio, Rossanna;
González, Mercedes;
Porcal, Williams;
Seoane, Gustavo;
Ortega, Miguel A.;
Aldana, Ignacio;
Monge, Antonio;
Denicola, Ana

Publication type:

Article

Greener Synthesis of Antiproliferative Furoxans via Multicomponent Reactions.

Published in:

Molecules, 2022, v. 27, n. 6, p. 1756, doi. 10.3390/molecules27061756

By:

Ingold, Mariana;
de la Sovera, Victoria;
Dapueto, Rosina;
Hernández, Paola;
Porcal, Williams;
López, Gloria V.

Publication type:

Article

Evaluation of chromosomal aberrations induced by 188Re-dendrimer nanosystem on B16f1 melanoma cells.

Published in:

International Journal of Radiation Biology, 2018, v. 94, n. 7, p. 664, doi. 10.1080/09553002.2018.1478161

By:

Tassano, Marcos;
Oddone, Natalia;
Fernández, Marcelo;
Porcal, Williams;
García, María Fernanda;
Martínez-López, Wilner;
Benech, Juan Claudio;
Cabral, Pablo

Publication type:

Article

A Focused Library of NO‐Donor Compounds with Potent Antiproliferative Activity Based on Green Multicomponent Reactions.

Published in:

ChemMedChem, 2019, v. 14, n. 18, p. 1669, doi. 10.1002/cmdc.201900385

By:

Ingold, Mariana;
Colella, Lucía;
Hernández, Paola;
Batthyány, Carlos;
Tejedor, David;
Puerta, Adrián;
García‐Tellado, Fernando;
Padrón, José M.;
Porcal, Williams;
López, Gloria. V.

Publication type:

Article

Cell uptake mechanisms of PAMAM G4-FITC dendrimer in human myometrial cells.

Published in:

Journal of Nanoparticle Research, 2013, v. 15, n. 7, p. 1, doi. 10.1007/s11051-013-1776-1

By:

Oddone, Natalia;
Zambrana, Ana;
Tassano, Marcos;
Porcal, Williams;
Cabral, Pablo;
Benech, Juan

Publication type:

Article

Front Cover: Synthetic Study of 5‐Hydroxymethylfurfural in Groebke‐Blackburn‐Bienaymé Reaction (Eur. J. Org. Chem. 10/2022).

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 10, p. 1, doi. 10.1002/ejoc.202200219

By:

de la Sovera, Victoria;
López, Gloria V.;
Porcal, Williams

Publication type:

Article

Synthetic Study of 5‐Hydroxymethylfurfural in Groebke‐Blackburn‐Bienaymé Reaction.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 10, p. 1, doi. 10.1002/ejoc.202101369

By:

de la Sovera, Victoria;
López, Gloria V.;
Porcal, Williams

Publication type:

Article

Renewable carbon resource from biomass: building molecular architectures from furanic platforms.

Published in:

Pure & Applied Chemistry, 2024, v. 96, n. 9, p. 1271, doi. 10.1515/pac-2024-0230

By:

López, Gloria V.;
Porcal, Williams

Publication type:

Article

Sensitivity of Haemonchus contortus to anthelmintics using different in vitro screening assays: a comparative study.

Published in:

Parasites & Vectors, 2022, v. 15, n. 1, p. 1, doi. 10.1186/s13071-022-05253-3

By:

Munguía, Beatriz;
Saldaña, Jenny;
Nieves, Magdalena;
Melian, María Elisa;
Ferrer, Manuela;
Teixeira, Ramiro;
Porcal, Williams;
Manta, Eduardo;
Domínguez, Laura

Publication type:

Article

Structural relationships in the solid state of the anti-chagas agent ( E)-phenylethenylbenzofuroxan.

Published in:

Molecular Diversity, 2010, v. 14, n. 4, p. 643, doi. 10.1007/s11030-009-9202-4

By:

Martins, Felipe;
Ayala, Alejandro;
Porcal, Williams;
Cerecetto, Hugo;
González, Mercedes;
Ellena, Javier

Publication type:

Article

Fully-automated radiosynthesis of the amyloid tracer [11C] PiB via direct [11C]CO2 fixation-reduction.

Published in:

EJNMMI Radiopharmacy & Chemistry, 2019, v. 4, n. 1, p. N.PAG, doi. 10.1186/s41181-019-0065-4

By:

Buccino, Pablo;
Savio, Eduardo;
Porcal, Williams

Publication type:

Article

An efficient preparation of labelling precursor of [C]L-deprenyl-D and automated radiosynthesis.

Published in:

EJNMMI Radiopharmacy & Chemistry, 2017, v. 2, n. 1, p. 1, doi. 10.1186/s41181-017-0029-5

By:

Zirbesegger, Kevin;
Buccino, Pablo;
Kreimerman, Ingrid;
Engler, Henry;
Porcal, Williams;
Savio, Eduardo

Publication type:

Article

Identification of Thioredoxin Glutathione Reductase Inhibitors That Kill Cestode and Trematode Parasites.

Published in:

PLoS ONE, 2012, v. 7, n. 4, p. 1, doi. 10.1371/journal.pone.0035033

By:

Ross, Fabiana;
Hernández, Paola;
Porcal, Williams;
López, Gloria V.;
Cerecetto, Hugo;
lez, Mercedes Gonzá;
Basika, Tatiana;
Carmona, Carlos;
Martín Fló;
Maggioli, Gabriela;
Bonilla, Mariana;
Gladyshev, Vadim N.;
Boiani, Mariana;
Salinas, Gustavo

Publication type:

Article

Identification of 2-(4-N,N-Dimethylaminophenyl)-5-methyl-1-phenethyl-1H-benzimidazole targeting HIV-1 CA capsid protein and inhibiting HIV-1 replication in cellulo.

Published in:

BMC Pharmacology & Toxicology, 2022, v. 23, n. 1, p. 1, doi. 10.1186/s40360-022-00581-7

By:

Alvarez, Guzmán;
van Pul, Lisa;
Robert, Xavier;
Artía, Zoraima;
van Nuenen, Ad C.;
Long, Mathieu;
Sierra, Natalia;
Porcal, Williams;
Kootstra, Neeltje A.;
Guillon, Christophe

Publication type:

Article

Labeling and Biological Evaluation of 99mTc-HYNIC-Trastuzumab as a Potential Radiopharmaceutical for In Vivo Evaluation of HER2 Expression in Breast Cancer.

Published in:

World Journal of Nuclear Medicine, 2013, v. 12, n. 1, p. 27, doi. 10.4103/1450-1147.113953

By:

Calzada, Victoria;
Garcia, Fernanda;
Fernández, Marcelo;
Porcal, Williams;
Quinn, Thomas;
Alonso, Omar;
Gambini, Juan Pablo;
Cabral, Pablo

Publication type:

Article

99mTc Stearyl 6-(benzylidenehydrazinyl) nicotinamide Liposomes as Tumor Permeability Evaluation Tracer.

Published in:

AAPS PharmSciTech, 2021, v. 22, n. 3, p. 1, doi. 10.1208/s12249-021-01984-1

By:

Cabrera, Mirel;
Lecot, Nicole;
Fernández, Marcelo;
Gambini, J. P.;
Porcal, Williams;
Cabral, Pablo

Publication type:

Article

Works by Porcal, Williams

Garbage in, garbage out: how reliable training data improved a virtual screening approach against SARS-CoV-2 MPro.

Biological Assessment of a <sup>18</sup>F-Labeled Sulforhodamine 101 in a Mouse Model of Alzheimer's Disease as a Potential Astrocytosis Marker.

Microwave-Assisted Solid-Phase Synthesis of a 1,2-Disubstituted Benzimidazole Library by Using a Phosphonium Linker.

Benzo[1, 2- c]1, 2, 5-oxadiazole N-Oxide Derivatives as Potential Antitrypanosomal Drugs. Structure-Activity Relationships. Part II.

Greener Synthesis of Antiproliferative Furoxans via Multicomponent Reactions.

Evaluation of chromosomal aberrations induced by <sup>188</sup>Re-dendrimer nanosystem on B16f1 melanoma cells.

A Focused Library of NO‐Donor Compounds with Potent Antiproliferative Activity Based on Green Multicomponent Reactions.

Cell uptake mechanisms of PAMAM G4-FITC dendrimer in human myometrial cells.

Front Cover: Synthetic Study of 5‐Hydroxymethylfurfural in Groebke‐Blackburn‐Bienaymé Reaction (Eur. J. Org. Chem. 10/2022).

Synthetic Study of 5‐Hydroxymethylfurfural in Groebke‐Blackburn‐Bienaymé Reaction.

Renewable carbon resource from biomass: building molecular architectures from furanic platforms.

Sensitivity of Haemonchus contortus to anthelmintics using different in vitro screening assays: a comparative study.

Structural relationships in the solid state of the anti-chagas agent ( E)-phenylethenylbenzofuroxan.

Fully-automated radiosynthesis of the amyloid tracer [<sup>11</sup>C] PiB via direct [<sup>11</sup>C]CO<sub>2</sub> fixation-reduction.

An efficient preparation of labelling precursor of [C]L-deprenyl-D and automated radiosynthesis.

Identification of Thioredoxin Glutathione Reductase Inhibitors That Kill Cestode and Trematode Parasites.

Identification of 2-(4-N,N-Dimethylaminophenyl)-5-methyl-1-phenethyl-1H-benzimidazole targeting HIV-1 CA capsid protein and inhibiting HIV-1 replication in cellulo.

Labeling and Biological Evaluation of <sup>99m</sup>Tc-HYNIC-Trastuzumab as a Potential Radiopharmaceutical for In Vivo Evaluation of HER2 Expression in Breast Cancer.

99mTc Stearyl 6-(benzylidenehydrazinyl) nicotinamide Liposomes as Tumor Permeability Evaluation Tracer.