Works by Poli, Giulio

Results: 51

A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration.

Published in:

Antioxidants, 2023, v. 12, n. 12, p. 2044, doi. 10.3390/antiox12122044

By:

Berrino, Emanuela;
Carradori, Simone;
Carta, Fabrizio;
Melfi, Francesco;
Gallorini, Marialucia;
Poli, Giulio;
Tuccinardi, Tiziano;
Fernández-Bolaños, José G.;
López, Óscar;
Petzer, Jacobus P.;
Petzer, Anél;
Guglielmi, Paolo;
Secci, Daniela;
Supuran, Claudiu T.

Publication type:

Article

A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by Using a Pharmacophore-based Approach.

Published in:

Molecular Informatics, 2016, v. 35, n. 8/9, p. 434, doi. 10.1002/minf.201501026

By:

Tuccinardi, Tiziano;
Poli, Giulio;
Corchia, Isacco;
Granchi, Carlotta;
Lapillo, Margherita;
Macchia, Marco;
Minutolo, Filippo;
Ortore, Gabriella;
Martinelli, Adriano

Publication type:

Article

An alternative conformation of the N‐terminal loop of human dihydroorotate dehydrogenase drives binding to a potent antiproliferative agent.

Published in:

Acta Crystallographica: Section D, Structural Biology, 2024, v. 80, n. 6, p. 386, doi. 10.1107/S2059798324004066

By:

Alberti, Marta;
Poli, Giulio;
Broggini, Luca;
Sainas, Stefano;
Rizzi, Menico;
Boschi, Donatella;
Ferraris, Davide M.;
Martino, Elena;
Ricagno, Stefano;
Tuccinardi, Tiziano;
Lolli, Marco L.;
Miggiano, Riccardo

Publication type:

Article

Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1 H)-One Scaffold.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 7, p. N.PAG, doi. 10.3390/ph15070768

By:

Ceni, Costanza;
Benko, Michael J.;
Mohamed, Kawthar A.;
Poli, Giulio;
Di Stefano, Miriana;
Tuccinardi, Tiziano;
Digiacomo, Maria;
Valoti, Massimo;
Laprairie, Robert B.;
Macchia, Marco;
Bertini, Simone

Publication type:

Article

New Synthetic Analogues of Natural Polyphenols as Sirtuin 1-Activating Compounds.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 3, p. 339, doi. 10.3390/ph15030339

By:

Bononi, Giulia;
Flori, Lorenzo;
Citi, Valentina;
Acciai, Cecilia;
Nocilla, Viviana;
Martelli, Alma;
Poli, Giulio;
Tuccinardi, Tiziano;
Granchi, Carlotta;
Testai, Lara;
Calderone, Vincenzo;
Minutolo, Filippo

Publication type:

Article

An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present).

Published in:

Expert Opinion on Therapeutic Patents, 2021, v. 31, n. 2, p. 153, doi. 10.1080/13543776.2021.1841166

By:

Bononi, Giulia;
Poli, Giulio;
Rizzolio, Flavio;
Tuccinardi, Tiziano;
Macchia, Marco;
Minutolo, Filippo;
Granchi, Carlotta

Publication type:

Article

Rutin as promising drug for the treatment of Parkinson's disease: an assessment of MAO-B inhibitory potential by docking, molecular dynamics and DFT studies.

Published in:

Molecular Simulation, 2019, v. 45, n. 18, p. 1563, doi. 10.1080/08927022.2019.1662003

By:

Azam, Faizul;
Abodabos, Honiwa Suliman;
Taban, Ismail M.;
Rfieda, Abdalla R.;
Mahmood, Danish;
Anwar, Md Jamir;
Khan, Shamshir;
Sizochenko, Natalia;
Poli, Giulio;
Tuccinardi, Tiziano;
Ali, Hamed I.

Publication type:

Article

Watermelon: setup and validation of an in silico fragment-based approach.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2356179

By:

Di Stefano, Miriana;
Galati, Salvatore;
Piazza, Lisa;
Gado, Francesca;
Granchi, Carlotta;
Macchia, Marco;
Giordano, Antonio;
Tuccinardi, Tiziano;
Poli, Giulio

Publication type:

Article

An in silico toolbox for the prediction of the potential pathogenic effects of missense mutations in the dimeric region of hRPE65.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2022.2162047

By:

Poli, Giulio;
Demontis, Gian Carlo;
Sodi, Andrea;
Saba, Alessandro;
Rizzo, Stanislao;
Macchia, Marco;
Tuccinardi, Tiziano

Publication type:

Article

Predicting potentially pathogenic effects of hRPE65 missense mutations: a computational strategy based on molecular dynamics simulations.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1765, doi. 10.1080/14756366.2022.2090547

By:

Poli, Giulio;
Barravecchia, Ivana;
Demontis, Gian Carlo;
Sodi, Andrea;
Saba, Alessandro;
Rizzo, Stanislao;
Macchia, Marco;
Tuccinardi, Tiziano

Publication type:

Article

New PIN1 inhibitors identified through a pharmacophore-driven, hierarchical consensus docking strategy.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 145, doi. 10.1080/14756366.2021.1979970

By:

Poli, Giulio;
Di Stefano, Miriana;
Estevez, Joan Arias;
Minutolo, Filippo;
Granchi, Carlotta;
Giordano, Antonio;
Parisi, Salvatore;
Mauceri, Matteo;
Canzonieri, Vincenzo;
Macchia, Marco;
Caligiuri, Isabella;
Tuccinardi, Tiziano;
Rizzolio, Flavio

Publication type:

Article

Development of a cheminformatics platform for selectivity analyses of carbonic anhydrase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 365, doi. 10.1080/14756366.2019.1705291

By:

Poli, Giulio;
Galati, Salvatore;
Martinelli, Adriano;
Supuran, Claudiu T.;
Tuccinardi, Tiziano

Publication type:

Article

New insight into structure-activity of furan-based salicylate synthase (MbtI) inhibitors as potential antitubercular agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 823, doi. 10.1080/14756366.2019.1589462

By:

Chiarelli, Laurent R.;
Mori, Matteo;
Beretta, Giangiacomo;
Gelain, Arianna;
Pini, Elena;
Sammartino, Josè Camilla;
Stelitano, Giovanni;
Barlocco, Daniela;
Costantino, Luca;
Lapillo, Margherita;
Poli, Giulio;
Caligiuri, Isabella;
Rizzolio, Flavio;
Bellinzoni, Marco;
Tuccinardi, Tiziano;
Villa, Stefania;
Meneghetti, Fiorella

Publication type:

Article

Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 589, doi. 10.1080/14756366.2019.1571271

By:

Poli, Giulio;
Lapillo, Margherita;
Jha, Vibhu;
Mouawad, Nayla;
Caligiuri, Isabella;
Macchia, Marco;
Minutolo, Filippo;
Rizzolio, Flavio;
Tuccinardi, Tiziano;
Granchi, Carlotta

Publication type:

Article

Binding investigation and preliminary optimisation of the 3-amino-1,2,4-triazin-5(2H)-one core for the development of new Fyn inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 956, doi. 10.1080/14756366.2018.1469017

By:

Poli, Giulio;
Lapillo, Margherita;
Granchi, Carlotta;
Caciolla, Jessica;
Mouawad, Nayla;
Caligiuri, Isabella;
Rizzolio, Flavio;
Langer, Thierry;
Minutolo, Filippo;
Tuccinardi, Tiziano

Publication type:

Article

Development of terphenyl-2-methyloxazol-5(4 H )-one derivatives as selective reversible MAGL inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1240, doi. 10.1080/14756366.2017.1375484

By:

Granchi, Carlotta;
Caligiuri, Isabella;
Bertelli, Eleonora;
Poli, Giulio;
Rizzolio, Flavio;
Macchia, Marco;
Martinelli, Adriano;
Minutolo, Filippo;
Tuccinardi, Tiziano

Publication type:

Article

Identification of a new STAT3 dimerization inhibitor through a pharmacophore-based virtual screening approach.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1011, doi. 10.3109/14756366.2015.1079184

By:

Poli, Giulio;
Gelain, Arianna;
Porta, Federica;
Asai, Akira;
Martinelli, Adriano;
Tuccinardi, Tiziano

Publication type:

Article

Reliability analysis and optimization of the consensus docking approach for the development of virtual screening studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 167, doi. 10.1080/14756366.2016.1193736

By:

Poli, Giulio;
Martinelli, Adriano;
Tuccinardi, Tiziano

Publication type:

Article

Receptor-based virtual screening evaluation for the identification of estrogen receptor β ligands.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 4, p. 662, doi. 10.3109/14756366.2014.959946

By:

Tuccinardi, Tiziano;
Poli, Giulio;
Dell'Agnello, Marco;
Granchi, Carlotta;
Minutolo, Filippo;
Martinelli, Adriano

Publication type:

Article

Identification of Novel Non-Nucleoside Inhibitors of Zika Virus NS5 Protein Targeting MTase Activity.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 4, p. 2437, doi. 10.3390/ijms25042437

By:

Fiorucci, Diego;
Meaccini, Micaela;
Poli, Giulio;
Stincarelli, Maria Alfreda;
Vagaggini, Chiara;
Giannecchini, Simone;
Sutto-Ortiz, Priscila;
Canard, Bruno;
Decroly, Etienne;
Dreassi, Elena;
Brai, Annalaura;
Botta, Maurizio

Publication type:

Article

Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 24, p. 17233, doi. 10.3390/ijms242417233

By:

Galati, Salvatore;
Di Stefano, Miriana;
Bertini, Simone;
Granchi, Carlotta;
Giordano, Antonio;
Gado, Francesca;
Macchia, Marco;
Tuccinardi, Tiziano;
Poli, Giulio

Publication type:

Article

New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 3, p. 2135, doi. 10.3390/ijms24032135

By:

Ferrisi, Rebecca;
Polini, Beatrice;
Ricardi, Caterina;
Gado, Francesca;
Mohamed, Kawthar A.;
Baron, Giovanna;
Faiella, Salvatore;
Poli, Giulio;
Rapposelli, Simona;
Saccomanni, Giuseppe;
Aldini, Giancarlo;
Chiellini, Grazia;
Laprairie, Robert B.;
Manera, Clementina;
Ortore, Gabriella

Publication type:

Article

Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 18, p. N.PAG, doi. 10.3390/ijms231810653

By:

Di Stefano, Miriana;
Galati, Salvatore;
Ortore, Gabriella;
Caligiuri, Isabella;
Rizzolio, Flavio;
Ceni, Costanza;
Bertini, Simone;
Bononi, Giulia;
Granchi, Carlotta;
Macchia, Marco;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

VenomPred: A Machine Learning Based Platform for Molecular Toxicity Predictions.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 4, p. 2105, doi. 10.3390/ijms23042105

By:

Galati, Salvatore;
Di Stefano, Miriana;
Martinelli, Elisa;
Macchia, Marco;
Martinelli, Adriano;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

Novel 8-Substituted Coumarins That Selectively Inhibit Human Carbonic Anhydrase IX and XII.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 5, p. 1208, doi. 10.3390/ijms20051208

By:

Buran, Kerem;
Bua, Silvia;
Poli, Giulio;
Önen Bayram, F. Esra;
Tuccinardi, Tiziano;
T. Supuran, Claudiu

Publication type:

Article

Extensive Reliability Evaluation of Docking-Based Target-Fishing Strategies.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 5, p. 1023, doi. 10.3390/ijms20051023

By:

Lapillo, Margherita;
Tuccinardi, Tiziano;
Martinelli, Adriano;
Macchia, Marco;
Giordano, Antonio;
Poli, Giulio

Publication type:

Article

Three-Dimensional Interactions Analysis of the Anticancer Target c-Src Kinase with Its Inhibitors.

Published in:

Cancers, 2020, v. 12, n. 8, p. 2327, doi. 10.3390/cancers12082327

By:

Jha, Vibhu;
Macchia, Marco;
Tuccinardi, Tiziano;
Poli, Giulio

Publication type:

Article

Aldose Reductase Differential Inhibitors in Green Tea.

Published in:

Biomolecules (2218-273X), 2020, v. 10, n. 7, p. 1003, doi. 10.3390/biom10071003

By:

Balestri, Francesco;
Poli, Giulio;
Pineschi, Carlotta;
Moschini, Roberta;
Cappiello, Mario;
Mura, Umberto;
Tuccinardi, Tiziano;
Del Corso, Antonella

Publication type:

Article

Dissecting the Activity of Catechins as Incomplete Aldose Reductase Differential Inhibitors through Kinetic and Computational Approaches.

Published in:

Biology (2079-7737), 2022, v. 11, n. 9, p. 1324, doi. 10.3390/biology11091324

By:

Balestri, Francesco;
Poli, Giulio;
Piazza, Lucia;
Cappiello, Mario;
Moschini, Roberta;
Signore, Giovanni;
Tuccinardi, Tiziano;
Mura, Umberto;
Del Corso, Antonella

Publication type:

Article

The Extra-Virgin Olive Oil Polyphenols Oleocanthal and Oleacein Counteract Inflammation-Related Gene and miRNA Expression in Adipocytes by Attenuating NF-κB Activation.

Published in:

Nutrients, 2019, v. 11, n. 12, p. 2855, doi. 10.3390/nu11122855

By:

Carpi, Sara;
Scoditti, Egeria;
Massaro, Marika;
Polini, Beatrice;
Manera, Clementina;
Digiacomo, Maria;
Esposito Salsano, Jasmine;
Poli, Giulio;
Tuccinardi, Tiziano;
Doccini, Stefano;
Santorelli, Filippo Maria;
Carluccio, Maria Annunziata;
Macchia, Marco;
Wabitsch, Martin;
De Caterina, Raffaele;
Nieri, Paola

Publication type:

Article

Novel broad spectrum virucidal molecules against enveloped viruses.

Published in:

PLoS ONE, 2018, v. 13, n. 12, p. 1, doi. 10.1371/journal.pone.0208333

By:

Civra, Andrea;
Lembo, David;
Cagno, Valeria;
Tapparel, Caroline;
Tintori, Cristina;
Tiberi, Marika;
Botta, Lorenzo;
Poli, Giulio;
Brai, Annalaura;
Botta, Maurizio;
Cavalli, Roberta

Publication type:

Article

Rhodanine derivatives as potent anti-HIV and anti-HSV microbicides.

Published in:

PLoS ONE, 2018, v. 13, n. 6, p. 1, doi. 10.1371/journal.pone.0198478

By:

Tintori, Cristina;
Iovenitti, Giulia;
Ceresola, Elisa Rita;
Ferrarese, Roberto;
Zamperini, Claudio;
Brai, Annalaura;
Poli, Giulio;
Dreassi, Elena;
Cagno, Valeria;
Lembo, David;
Canducci, Filippo;
Botta, Maurizio

Publication type:

Article

Largazole Analogues as Histone Deacetylase Inhibitors and Anticancer Agents: An Overview of Structure-Activity Relationships.

Published in:

ChemMedChem, 2017, v. 12, n. 23, p. 1917, doi. 10.1002/cmdc.201700563

By:

Poli, Giulio;
Di Fabio, Romano;
Ferrante, Luca;
Summa, Vincenzo;
Botta, Maurizio

Publication type:

Article

Mealworm (Tenebrio molitor): Potential and Challenges to Promote Circular Economy.

Published in:

Animals (2076-2615), 2021, v. 11, n. 9, p. 2568, doi. 10.3390/ani11092568

By:

Moruzzo, Roberta;
Riccioli, Francesco;
Espinosa Diaz, Salomon;
Secci, Chiara;
Poli, Giulio;
Mancini, Simone

Publication type:

Article

Virtual screening identifies a PIN1 inhibitor with possible antiovarian cancer effects.

Published in:

Journal of Cellular Physiology, 2019, v. 234, n. 9, p. 15708, doi. 10.1002/jcp.28224

By:

Russo Spena, Concetta;
De Stefano, Lucia;
Poli, Giulio;
Granchi, Carlotta;
El Boustani, Maguie;
Ecca, Fabrizio;
Grassi, Gabriele;
Grassi, Mario;
Canzonieri, Vincenzo;
Giordano, Antonio;
Tuccinardi, Tiziano;
Caligiuri, Isabella;
Rizzolio, Flavio

Publication type:

Article

KinasePred: A Computational Tool for Small-Molecule Kinase Target Prediction.

Published in:

International Journal of Molecular Sciences, 2025, v. 26, n. 5, p. 2157, doi. 10.3390/ijms26052157

By:

Di Stefano, Miriana;
Piazza, Lisa;
Poles, Clarissa;
Galati, Salvatore;
Granchi, Carlotta;
Giordano, Antonio;
Campisi, Luca;
Macchia, Marco;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

Discovery of a new ATP-citrate lyase (ACLY) inhibitor identified by a pharmacophore-based virtual screening study.

Published in:

Journal of Biomolecular Structure & Dynamics, 2021, v. 39, n. 11, p. 3996, doi. 10.1080/07391102.2020.1773314

By:

Jha, Vibhu;
Galati, Salvatore;
Volpi, Valerio;
Ciccone, Lidia;
Minutolo, Filippo;
Rizzolio, Flavio;
Granchi, Carlotta;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

Anticancer Activity of Euplotin C, Isolated from the Marine Ciliate Euplotes crassus, Against Human Melanoma Cells.

Published in:

Marine Drugs, 2018, v. 16, n. 5, p. 166, doi. 10.3390/md16050166

By:

Carpi, Sara;
Polini, Beatrice;
Alcantara Barata, Gabriela;
Tuccinardi, Tiziano;
Nieri, Paola;
Poli, Giulio;
Fogli, Stefano;
Romanini, Antonella;
Guella, Graziano;
Frontini, Francesco Paolo;
Di Giuseppe, Graziano

Publication type:

Article

Identification of a Non-Retinoid Opsin Ligand Through Pharmacophore-Guided Virtual Screening—A Novel Potential Rhodopsin-Stabilizing Compound.

Published in:

Molecules, 2025, v. 30, n. 11, p. 2328, doi. 10.3390/molecules30112328

By:

Di Stefano, Miriana;
Ghilardi, Maria;
Poles, Clarissa;
Piazza, Lisa;
Demontis, Gian Carlo;
Poli, Giulio;
Tuccinardi, Tiziano;
Macchia, Marco

Publication type:

Article

Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?

Published in:

Molecules, 2022, v. 27, n. 22, p. 7816, doi. 10.3390/molecules27227816

By:

Carradori, Simone;
Fantacuzzi, Marialuigia;
Ammazzalorso, Alessandra;
Angeli, Andrea;
De Filippis, Barbara;
Galati, Salvatore;
Petzer, Anél;
Petzer, Jacobus P.;
Poli, Giulio;
Tuccinardi, Tiziano;
Agamennone, Mariangela;
Supuran, Claudiu T.

Publication type:

Article

Sirtuin 1-Activating Compounds: Discovery of a Class of Thiazole-Based Derivatives.

Published in:

Molecules, 2022, v. 27, n. 19, p. 6535, doi. 10.3390/molecules27196535

By:

Bononi, Giulia;
Citi, Valentina;
Lapillo, Margherita;
Martelli, Alma;
Poli, Giulio;
Tuccinardi, Tiziano;
Granchi, Carlotta;
Testai, Lara;
Calderone, Vincenzo;
Minutolo, Filippo

Publication type:

Article

Identification of Human Dihydroorotate Dehydrogenase Inhibitor by a Pharmacophore-Based Virtual Screening Study.

Published in:

Molecules, 2022, v. 27, n. 12, p. 3660, doi. 10.3390/molecules27123660

By:

Galati, Salvatore;
Sainas, Stefano;
Giorgis, Marta;
Boschi, Donatella;
Lolli, Marco L.;
Ortore, Gabriella;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

Co-Inhibition of P-gp and Hsp90 by an Isatin-Derived Compound Contributes to the Increase of the Chemosensitivity of MCF7/ADR-Resistant Cells to Doxorubicin.

Published in:

Molecules, 2022, v. 27, n. 1, p. 90, doi. 10.3390/molecules27010090

By:

Abdalla, Ashraf N.;
Di Stefano, Miriana;
Poli, Giulio;
Tuccinardi, Tiziano;
Bader, Ammar;
Vassallo, Antonio;
Abdallah, Mohamed E.;
El-Readi, Mahmoud Zaki;
Refaat, Bassem;
Algarni, Alanood S.;
Ahmad, Rizwan;
Alkahtani, Hamad M.;
Abdel-Aziz, Alaa A.-M.;
El-Azab, Adel S.;
Alqathama, Aljawharah

Publication type:

Article

Recent Advances in In Silico Target Fishing.

Published in:

Molecules, 2021, v. 26, n. 17, p. 5124, doi. 10.3390/molecules26175124

By:

Galati, Salvatore;
Di Stefano, Miriana;
Martinelli, Elisa;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

Discovery of Monoacylglycerol Lipase (MAGL) Inhibitors Based on a Pharmacophore-Guided Virtual Screening Study.

Published in:

Molecules, 2021, v. 26, n. 1, p. 78, doi. 10.3390/molecules26010078

By:

Jha, Vibhu;
Biagi, Marzia;
Spinelli, Valeria;
Di Stefano, Miriana;
Macchia, Marco;
Minutolo, Filippo;
Granchi, Carlotta;
Poli, Giulio;
Tuccinardi, Tiziano

Publication type:

Article

Application of MM-PBSA Methods in Virtual Screening.

Published in:

Molecules, 2020, v. 25, n. 8, p. 1971, doi. 10.3390/molecules25081971

By:

Poli, Giulio;
Granchi, Carlotta;
Rizzolio, Flavio;
Tuccinardi, Tiziano;
Costa, Giosuè

Publication type:

Article

Discovery of Novel µ-Opioid Receptor Inverse Agonist from a Combinatorial Library of Tetrapeptides through Structure-Based Virtual Screening.

Published in:

Molecules, 2019, v. 24, n. 21, p. 3872, doi. 10.3390/molecules24213872

By:

Poli, Giulio;
Dimmito, Marilisa Pia;
Mollica, Adriano;
Zengin, Gokhan;
Benyhe, Sandor;
Zador, Ferenc;
Stefanucci, Azzurra

Publication type:

Article

Synthesis and Biological Evaluation of New Glycoconjugated LDH Inhibitors as Anticancer Agents †.

Published in:

Molecules, 2019, v. 24, n. 19, p. 3520, doi. 10.3390/molecules24193520

By:

D'Andrea, Felicia;
Vagelli, Giulia;
Granchi, Carlotta;
Guazzelli, Lorenzo;
Tuccinardi, Tiziano;
Poli, Giulio;
Iacopini, Dalila;
Minutolo, Filippo;
Di Bussolo, Valeria

Publication type:

Article

Design, Synthesis, Docking Studies and Monoamine Oxidase Inhibition of a Small Library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazoles.

Published in:

Molecules, 2019, v. 24, n. 3, p. 484, doi. 10.3390/molecules24030484

By:

Guglielmi, Paolo;
Carradori, Simone;
Poli, Giulio;
Secci, Daniela;
Cirilli, Roberto;
Rotondi, Giulia;
Chimenti, Paola;
Petzer, Anél;
Petzer, Jacobus P.;
McPhee, Derek J.

Publication type:

Article

New Chromane-Based Derivatives as Inhibitors of Mycobacterium tuberculosis Salicylate Synthase (MbtI): Preliminary Biological Evaluation and Molecular Modeling Studies.

Published in:

Molecules, 2018, v. 23, n. 7, p. 1506, doi. 10.3390/molecules23071506

By:

Pini, Elena;
Poli, Giulio;
Tuccinardi, Tiziano;
Chiarelli, Laurent Roberto;
Mori, Matteo;
Gelain, Arianna;
Costantino, Luca;
Villa, Stefania;
Meneghetti, Fiorella;
Barlocco, Daniela

Publication type:

Article