Works by Passarella, Daniele


Results: 75
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    Automated fluorine-18 radiolabeling via an alkyne–azide cycloaddition reaction on a dual peptide-functionalized liposome surface for in vivo PET imaging.

    Published in:
    Frontiers in Pharmacology, 2025, p. 1, doi. 10.3389/fphar.2025.1566257
    By:
    • Iannone, Marco;
    • Kravicz, Marcelo;
    • Rainone, Paolo;
    • Antoniou, Antonia I.;
    • Stucchi, Stefano;
    • Valtorta, Silvia;
    • Amenta, Arianna;
    • Turolla, Elia Anna;
    • Pellegrino, Sara;
    • Passarella, Daniele;
    • Vino, Elisa;
    • Todde, Sergio;
    • Re, Francesca;
    • Seneci, Pierfausto;
    • Moresco, Rosa Maria
    Publication type:
    Article
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    Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule Dynamics.

    Published in:
    Chemistry - A European Journal, 2023, v. 29, n. 5, p. 1, doi. 10.1002/chem.202203431
    By:
    • Boiarska, Zlata;
    • Pérez‐Peña, Helena;
    • Abel, Anne‐Catherine;
    • Marzullo, Paola;
    • Álvarez‐Bernad, Beatriz;
    • Bonato, Francesca;
    • Santini, Benedetta;
    • Horvath, Dragos;
    • Lucena‐Agell, Daniel;
    • Vasile, Francesca;
    • Sironi, Maurizio;
    • Díaz, J. Fernando;
    • Prota, Andrea E.;
    • Pieraccini, Stefano;
    • Passarella, Daniele
    Publication type:
    Article
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    Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule Dynamics.

    Published in:
    Chemistry - A European Journal, 2023, v. 29, n. 5, p. 1, doi. 10.1002/chem.202203431
    By:
    • Boiarska, Zlata;
    • Pérez‐Peña, Helena;
    • Abel, Anne‐Catherine;
    • Marzullo, Paola;
    • Álvarez‐Bernad, Beatriz;
    • Bonato, Francesca;
    • Santini, Benedetta;
    • Horvath, Dragos;
    • Lucena‐Agell, Daniel;
    • Vasile, Francesca;
    • Sironi, Maurizio;
    • Díaz, J. Fernando;
    • Prota, Andrea E.;
    • Pieraccini, Stefano;
    • Passarella, Daniele
    Publication type:
    Article
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    Front Cover: Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule Dynamics (Chem. Eur. J. 5/2023).

    Published in:
    Chemistry - A European Journal, 2023, v. 29, n. 5, p. 1, doi. 10.1002/chem.202300067
    By:
    • Boiarska, Zlata;
    • Pérez‐Peña, Helena;
    • Abel, Anne‐Catherine;
    • Marzullo, Paola;
    • Álvarez‐Bernad, Beatriz;
    • Bonato, Francesca;
    • Santini, Benedetta;
    • Horvath, Dragos;
    • Lucena‐Agell, Daniel;
    • Vasile, Francesca;
    • Sironi, Maurizio;
    • Díaz, J. Fernando;
    • Prota, Andrea E.;
    • Pieraccini, Stefano;
    • Passarella, Daniele
    Publication type:
    Article
    6

    Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule Dynamics.

    Published in:
    Chemistry - A European Journal, 2023, v. 29, n. 5, p. 1, doi. 10.1002/chem.202203431
    By:
    • Boiarska, Zlata;
    • Pérez‐Peña, Helena;
    • Abel, Anne‐Catherine;
    • Marzullo, Paola;
    • Álvarez‐Bernad, Beatriz;
    • Bonato, Francesca;
    • Santini, Benedetta;
    • Horvath, Dragos;
    • Lucena‐Agell, Daniel;
    • Vasile, Francesca;
    • Sironi, Maurizio;
    • Díaz, J. Fernando;
    • Prota, Andrea E.;
    • Pieraccini, Stefano;
    • Passarella, Daniele
    Publication type:
    Article
    7

    Quantitative live cell imaging of a tauopathy model enables the identification of a polypharmacological drug candidate that restores physiological microtubule interaction.

    Published in:
    Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-45851-6
    By:
    • Pinzi, Luca;
    • Conze, Christian;
    • Bisi, Nicolo;
    • Torre, Gabriele Dalla;
    • Soliman, Ahmed;
    • Monteiro-Abreu, Nanci;
    • Trushina, Nataliya I.;
    • Krusenbaum, Andrea;
    • Dolouei, Maryam Khodaei;
    • Hellwig, Andrea;
    • Christodoulou, Michael S.;
    • Passarella, Daniele;
    • Bakota, Lidia;
    • Rastelli, Giulio;
    • Brandt, Roland
    Publication type:
    Article
    8

    Quantitative live cell imaging of a tauopathy model enables the identification of a polypharmacological drug candidate that restores physiological microtubule interaction.

    Published in:
    Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-45851-6
    By:
    • Pinzi, Luca;
    • Conze, Christian;
    • Bisi, Nicolo;
    • Torre, Gabriele Dalla;
    • Soliman, Ahmed;
    • Monteiro-Abreu, Nanci;
    • Trushina, Nataliya I.;
    • Krusenbaum, Andrea;
    • Dolouei, Maryam Khodaei;
    • Hellwig, Andrea;
    • Christodoulou, Michael S.;
    • Passarella, Daniele;
    • Bakota, Lidia;
    • Rastelli, Giulio;
    • Brandt, Roland
    Publication type:
    Article
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    Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 M pro.

    Published in:
    Molecules, 2023, v. 28, n. 2, p. 514, doi. 10.3390/molecules28020514
    By:
    • Citarella, Andrea;
    • Moi, Davide;
    • Pedrini, Martina;
    • Pérez-Peña, Helena;
    • Pieraccini, Stefano;
    • Stagno, Claudio;
    • Micale, Nicola;
    • Schirmeister, Tanja;
    • Sibille, Giulia;
    • Gribaudo, Giorgio;
    • Silvani, Alessandra;
    • Passarella, Daniele;
    • Giannini, Clelia
    Publication type:
    Article
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    Synthesis and Biological Evaluation of Migrastatin Macrotriazoles.

    Published in:
    European Journal of Organic Chemistry, 2017, v. 2017, n. 1, p. 60, doi. 10.1002/ejoc.201600988
    By:
    • Gabba, Adele;
    • Robakiewicz, Stefania;
    • Taciak, Bartłomiej;
    • Ulewicz, Katarzyna;
    • Broggini, Gianluigi;
    • Rastelli, Giulio;
    • Krol, Magadalena;
    • Murphy, Paul V.;
    • Passarella, Daniele
    Publication type:
    Article
    23

    Synthesis of Pironetin-Dumetorine Hybrids as Tubulin Binders.

    Published in:
    European Journal of Organic Chemistry, 2016, v. 2016, n. 11, p. 2029, doi. 10.1002/ejoc.201600130
    By:
    • Marucci, Cristina;
    • Christodoulou, Michael S.;
    • Pieraccini, Stefano;
    • Sironi, Maurizio;
    • Dapiaggi, Federico;
    • Cartelli, Daniele;
    • Calogero, Alessandra M.;
    • Cappelletti, Graziella;
    • Vilanova, Concepción;
    • Gazzola, Silvia;
    • Broggini, Gianluigi;
    • Passarella, Daniele
    Publication type:
    Article
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    Structure–Activity Relationships of Hexahydrocyclopenta[c]quinoline Derivatives as Allosteric Inhibitors of CDK2 and EGFR.

    Published in:
    ChemMedChem, 2018, v. 13, n. 24, p. 2627, doi. 10.1002/cmdc.201800687
    By:
    • Carlino, Luca;
    • Christodoulou, Michael S.;
    • Restelli, Valentina;
    • Caporuscio, Fabiana;
    • Foschi, Francesca;
    • Semrau, Marta S.;
    • Costanzi, Elisa;
    • Tinivella, Annachiara;
    • Pinzi, Luca;
    • Lo Presti, Leonardo;
    • Battistutta, Roberto;
    • Storici, Paola;
    • Broggini, Massimo;
    • Passarella, Daniele;
    • Rastelli, Giulio
    Publication type:
    Article
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    Total Synthesis of (−)‐Cannabidiol‐C<sub>4</sub>.

    Published in:
    European Journal of Organic Chemistry, 2022, v. 2022, n. 22, p. 1, doi. 10.1002/ejoc.202200392
    By:
    • Marzullo, Paola;
    • Maiocchi, Alice;
    • Paladino, Giuseppe;
    • Ciriello, Umberto;
    • Lo Presti, Leonardo;
    • Passarella, Daniele
    Publication type:
    Article
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    Probing an Allosteric Pocket of CDK2 with Small Molecules.

    Published in:
    ChemMedChem, 2017, v. 12, n. 1, p. 33, doi. 10.1002/cmdc.201600474
    By:
    • Christodoulou, Michael S.;
    • Caporuscio, Fabiana;
    • Restelli, Valentina;
    • Carlino, Luca;
    • Cannazza, Giuseppe;
    • Costanzi, Elisa;
    • Citti, Cinzia;
    • Lo Presti, Leonardo;
    • Pisani, Pasquale;
    • Battistutta, Roberto;
    • Broggini, Massimo;
    • Passarella, Daniele;
    • Rastelli, Giulio
    Publication type:
    Article
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    Camptothecin-7-yl-methanthiole: Semisynthesis and Biological Evaluation.

    Published in:
    ChemMedChem, 2012, v. 7, n. 12, p. 2134, doi. 10.1002/cmdc.201200322
    By:
    • Christodoulou, Michael S.;
    • Zunino, Franco;
    • Zuco, Valentina;
    • Borrelli, Stella;
    • Comi, Daniela;
    • Fontana, Gabriele;
    • Martinelli, Marisa;
    • Lorens, James B.;
    • Evensen, Lasse;
    • Sironi, Maurizio;
    • Pieraccini, Stefano;
    • Dalla Via, Lisa;
    • Gia, Ornella Maria;
    • Passarella, Daniele
    Publication type:
    Article
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    Self-Assembly Nanoparticles of Natural Bioactive Abietane Diterpenes.

    Published in:
    International Journal of Molecular Sciences, 2021, v. 22, n. 19, p. 10210, doi. 10.3390/ijms221910210
    By:
    • Ntungwe, Epole;
    • Domínguez-Martín, Eva María;
    • Bangay, Gabrielle;
    • Garcia, Catarina;
    • Guerreiro, Iris;
    • Colombo, Eleonora;
    • Saraiva, Lucilia;
    • Díaz-Lanza, Ana María;
    • Rosatella, Andreia;
    • Alves, Marta M.;
    • Reis, Catarina Pinto;
    • Passarella, Daniele;
    • Rijo, Patricia
    Publication type:
    Article
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    Embelin as Lead Compound for New Neuroserpin Polymerization Inhibitors.

    Published in:
    Life (2075-1729), 2020, v. 10, n. 7, p. 111, doi. 10.3390/life10070111
    By:
    • Visentin, Cristina;
    • Musso, Loana;
    • Broggini, Luca;
    • Bonato, Francesca;
    • Russo, Rosaria;
    • Moriconi, Claudia;
    • Bolognesi, Martino;
    • Miranda, Elena;
    • Dallavalle, Sabrina;
    • Passarella, Daniele;
    • Ricagno, Stefano
    Publication type:
    Article
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