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Works by Nudelman, Abraham

Results: 34

1

Formaldehyde-releasing prodrugs specifically affect cancer cells by depletion of intracellular glutathione and augmentation of reactive oxygen species.

Published in:

Cancer Chemotherapy & Pharmacology, 2008, v. 62, n. 3, p. 471, doi. 10.1007/s00280-007-0627-0

By:

Levovich, Inesa;
Nudelman, Abraham;
Berkovitch, Gili;
Swift, Lonnie P.;
Cutts, Suzanne M.;
Phillips, Don R.;
Rephaeli, Ada

Publication type:

Article

2

The cardio-protecting agent and topoisomerase II catalytic inhibitor sobuzoxane enhances doxorubicin-DNA adduct mediated cytotoxicity.

Published in:

Cancer Chemotherapy & Pharmacology, 2008, v. 61, n. 5, p. 739, doi. 10.1007/s00280-007-0528-2

By:

Swift, Lonnie P.;
Cutts, Suzanne M.;
Nudelman, Abraham;
Levovich, Inessa;
Rephaeli, Ada;
Phillips, Don R.

Publication type:

Article

3

Aryl chain analogues of the biotin vitamers as potential herbicides. Part 3.

Published in:

Pest Management Science, 2007, v. 63, n. 10, p. 974, doi. 10.1002/ps.1427

By:

Ashkenazi, Tali;
Pinkert, Dalia;
Nudelman, Ayelet;
Widberg, Ayala;
Wexler, Barry;
Wittenbach, Vernon;
Flint, Dennis;
Nudelman, Abraham

Publication type:

Article

4

Inhibitors of biotin biosynthesis as potential herbicides: Part 2.

Published in:

Pest Management Science, 2005, v. 61, n. 10, p. 1024, doi. 10.1002/ps.1075

By:

Ashkenazi, Tali;
Widberg, Ayala;
Nudelman, Abraham;
Wittenbach, Vernon;
Flint, Dennis

Publication type:

Article

5

Department of Chemistry, Bar-Ilan University (BIU).

Published in:

Israel Journal of Chemistry, 2014, v. 54, n. 10, p. 1488, doi. 10.1002/ijch.201410010

By:

Albeck, Ammon;
Chill, Jordan H.;
Fischer, Bilha;
Mastai, Yitzhak;
Nudelman, Abraham;
Wilson‐Gordon, Arlene D.

Publication type:

Article

6

Studies in Sugar Chemistry VII<sup>1)</sup>. Glucuronides of Podophyllum Derivatives.

Published in:

Archiv der Pharmazie, 1997, v. 330, n. 9/10, p. 285, doi. 10.1002/ardp.19973300904

By:

Nudelman, Abraham;
Ruse, Margaretta;
Gottlieb, Hugo E.;
Fairchild, Craig

Publication type:

Article

7

'Vinylogs' and 'Acetylenylogs' of β-Adrenergic Agents.

Published in:

Archiv der Pharmazie, 1996, v. 329, n. 3, p. 125, doi. 10.1002/ardp.19963290304

By:

Nudelman, Abraham;
Binnes, Yitschak;
Shmueli-Broide, Naomi;
Odessa, Yael;
Hieble, J. Paul;
Sulpizio, Anthony C.

Publication type:

Article

8

Hypoxic Radiosensitizers: Substituted Styryl Derivatives.

Published in:

Archiv der Pharmazie, 1994, v. 327, n. 10, p. 619, doi. 10.1002/ardp.19943271004

By:

Nudelman, Abraham;
Falb, Eliezer;
Odesa, Yael;
Shmueli-Broide, Naomi

Publication type:

Article

9

Approaches to Mutual Prodrugs: Calcium - β-Blockers Wege zu mehrfach wirksamen Vorstufen von Ca-Antagonisten/β-Blockern.

Published in:

Archiv der Pharmazie, 1993, v. 326, n. 11, p. 907, doi. 10.1002/ardp.19933261112

By:

Nudelman, Abraham;
Kelner, Rachel

Publication type:

Article

10

Multifunctional 5-aminolevulinic acid prodrugs activating diverse cell-death pathways.

Published in:

Investigational New Drugs, 2012, v. 30, n. 3, p. 1028, doi. 10.1007/s10637-011-9669-6

By:

Berkovitch-Luria, Gili;
Weitman, Michal;
Nudelman, Abraham;
Rephaeli, Ada;
Malik, Zvi

Publication type:

Article

11

The histone deacetylase inhibitor butyroyloxymethyl diethylphosphate (AN-7) protects normal cells against toxicity of anticancer agents while augmenting their anticancer activity.

Published in:

Investigational New Drugs, 2012, v. 30, n. 1, p. 130, doi. 10.1007/s10637-010-9542-z

By:

Tarasenko, Nataly;
Kessler-Icekson, Gania;
Boer, Pnina;
Inbal, Aida;
Schlesinger, Hadassa;
Phillips, Don;
Cutts, Suzanne;
Nudelman, Abraham;
Rephaeli, Ada

Publication type:

Article

12

The selectivty and anti-metastatic activity of oral bioavailable butyric acid prodrugs.

Published in:

Investigational New Drugs, 2006, v. 24, n. 5, p. 383, doi. 10.1007/s10637-006-6213-1

By:

Ada Rephaeli;
Michal Entin-Meer;
Dikla Angel;
Nataly Tarasenko;
Tal Gruss-Fischer;
Irena Bruachman;
Don Phillips;
Suzanne Cutts;
Daphne Haas-Kogan;
Abraham Nudelman

Publication type:

Article

13

Histone deacetylase inhibitors: the anticancer, antimetastatic and antiangiogenic activities of AN-7 are superior to those of the clinically tested AN-9 (Pivanex).

Published in:

Clinical & Experimental Metastasis, 2008, v. 25, n. 7, p. 703, doi. 10.1007/s10585-008-9179-x

By:

Tarasenko, Nataly;
Nudelman, Abraham;
Tarasenko, Igor;
Entin-Meer, Michal;
Hass-Kogan, Daphne;
Inbal, Aida;
Rephaeli, Ada

Publication type:

Article

14

Comparison of the tissue distribution and metabolism of AN1284, a potent anti-inflammatory agent, after subcutaneous and oral administration in mice.

Published in:

Naunyn-Schmiedeberg's Archives of Pharmacology, 2021, v. 394, n. 10, p. 2077, doi. 10.1007/s00210-021-02125-y

By:

Weitman, Michal;
Bejar, Corina;
Melamed, Michal;
Weill, Tehilla;
Yanovsky, Inessa;
Zeeli, Shani;
Nudelman, Abraham;
Weinstock, Marta

Publication type:

Article

15

In vivo and in vitro antitumor activity of butyroyloxymethyl-diethyl phosphate (AN-7), a histone deacetylase inhibitor, in human prostate cancer.

Published in:

International Journal of Cancer, 2005, v. 116, n. 2, p. 226, doi. 10.1002/ijc.21030

By:

Rephaeli, Ada;
Blank-Porat, Diana;
Tarasenko, Nataly;
Entin-Meer, Michal;
Levovich, Inesa;
Cutts, Suzanne M.;
Phillips, Don R.;
Malik, Zvi;
Nudelman, Abraham

Publication type:

Article

16

The Power and Potential of Doxorubicin-DNA Adducts.

Published in:

IUBMB Life, 2005, v. 57, n. 2, p. 73, doi. 10.1080/15216540500079093

By:

Cutts, Suzanne;
Nudelman, Abraham;
Rephaeli, Ada;
Phillips, Don R.

Publication type:

Article

17

A Convenient Synthesis of Chiral Oxazolidin-2-Ones and Thiazolidin-2-Ones and an Improved Preparation of Triphosgene.

Published in:

Synthetic Communications, 1993, v. 23, n. 20, p. 2839, doi. 10.1080/00397919308012605

By:

Falb, Eliezer;
Nudelman, Abraham;
Hassner, Alfred

Publication type:

Article

18

An evaluation of the interaction of pixantrone with formaldehyde-releasing drugs in cancer cells.

Published in:

Cancer Chemotherapy & Pharmacology, 2022, v. 89, n. 6, p. 773, doi. 10.1007/s00280-022-04435-1

By:

Mansour, Oula C.;
Nudelman, Abraham;
Rephaeli, Ada;
Phillips, Don R.;
Cutts, Suzanne M.;
Evison, Benny J.

Publication type:

Article

19

The hydroxyl epimer of doxorubicin controls the rate of formation of cytotoxic anthracycline-DNA adducts.

Published in:

Cancer Chemotherapy & Pharmacology, 2013, v. 71, n. 3, p. 809, doi. 10.1007/s00280-012-2049-x

By:

Forrest, Robert;
Swift, Lonnie;
Evison, Benny;
Rephaeli, Ada;
Nudelman, Abraham;
Phillips, Don;
Cutts, Suzanne

Publication type:

Article

20

Adrenergic Agents, II<sup>1)</sup>: 1-Aryl-N<sup>2</sup>-alkyl-ethanediamines as Isosters of Adrenergic Arylethanolamines.

Published in:

Archiv der Pharmazie, 1990, v. 323, n. 4, p. 229, doi. 10.1002/ardp.19903230410

By:

Berger, Sarah;
Nudelman, Abraham

Publication type:

Article

21

Comparison of the anticancer properties of a novel valproic acid prodrug to leading histone deacetylase inhibitors.

Published in:

Journal of Cellular Biochemistry, 2018, v. 119, n. 4, p. 3417, doi. 10.1002/jcb.26512

By:

Tarasenko, Nataly;
Chekroun‐Setti, Hanna;
Nudelman, Abraham;
Rephaeli, Ada

Publication type:

Article

22

Prodrugs of butyric acid from bench to bedside: Synthetic design, mechanisms of action, and clinical applications.

Published in:

Drug Development Research, 2000, v. 50, n. 3/4, p. 379, doi. 10.1002/1098-2299(200007/08)50:3/4<379::AID-DDR20>3.0.CO;2-8

By:

Rephaeli, Ada;
Zhuk, Regina;
Nudelman, Abraham

Publication type:

Article

23

Comparison between the effect of butyric acid and its prodrug pivaloyloxymethylbutyrate on histones hyperacetylation in an HL-60 leukemic cell line.

Published in:

International Journal of Cancer, 1994, v. 56, n. 6, p. 906, doi. 10.1002/ijc.2910560625

By:

Aviram, Adina;
Zimrah, Yael;
Shaklai, Mali;
Nudelman, Abraham;
Rephaeli, Ada

Publication type:

Article

24

Derivatives of butyric acid as potential anti-neoplastic agents.

Published in:

International Journal of Cancer, 1991, v. 49, n. 1, p. 66, doi. 10.1002/ijc.2910490113

By:

Rephaeli, Ada;
Rabizadeh, Ester;
Aviram, Adina;
Shaklai, Mati;
Ruse, Margaretta;
Nudelman, Abraham

Publication type:

Article

25

Effect of Histone Deacetylase Inhibitor, Butyroyloxymethyl-Diethyl Phosphate (AN-7), on Corneal Neovascularization in a Mouse Model.

Published in:

2017

By:

Schaap-Fogler, Michal;
Bahar, Irit;
Rephaeli, Ada;
Dahbash, Mor;
Nudelman, Abraham;
Livny, Eitan;
Barliya, Tilda;
Nisgav, Yael;
Livnat, Tami

Publication type:

journal article

26

Valproic Acid Prodrug Affects Selective Markers, Augments Doxorubicin Anticancer Activity and Attenuates Its Toxicity in a Murine Model of Aggressive Breast Cancer.

Published in:

Pharmaceuticals (14248247), 2021, v. 14, n. 12, p. 1244, doi. 10.3390/ph14121244

By:

Tarasenko, Nataly;
Wilner, Harel Josef;
Nudelman, Abraham;
Kessler-Icekson, Gania;
Rephaeli, Ada

Publication type:

Article

27

The Therapeutic Potential of AN-7, a Novel Histone Deacetylase Inhibitor, for Treatment of Mycosis Fungoides/Sezary Syndrome Alone or with Doxorubicin.

Published in:

PLoS ONE, 2016, v. 11, n. 1, p. 1, doi. 10.1371/journal.pone.0146115

By:

Moyal, Lilach;
Feldbaum, Nataly;
Goldfeiz, Neta;
Rephaeli, Ada;
Nudelman, Abraham;
Weitman, Michal;
Tarasenko, Nataly;
Gorovitz, Batia;
Maron, Leah;
Yehezkel, Shiran;
Amitay-Laish, Iris;
Lubin, Ido;
Hodak, Emmilia

Publication type:

Article

28

Disparate Impact of Butyroyloxymethyl Diethylphosphate (AN-7), a Histone Deacetylase Inhibitor, and Doxorubicin in Mice Bearing a Mammary Tumor.

Published in:

PLoS ONE, 2012, v. 7, n. 2, p. 1, doi. 10.1371/journal.pone.0031393

By:

Tarasenko, Nataly;
Cutts, Suzanne M.;
Phillips, Don R.;
Inbal, Aida;
Nudelman, Abraham;
Kessler-Icekson, Gania;
Rephaeli, Ada

Publication type:

Article

29

Synthesis and preliminary biological evaluation of gabactyzine, a benactyzine-GABA mutual prodrug, as an organophosphate antidote.

Published in:

Scientific Reports, 2022, v. 12, n. 1, p. 1, doi. 10.1038/s41598-022-23141-9

By:

Weitman, Michal;
Eisenkraft, Arik;
TaShma, Zeev;
Makarovsky, Igor;
Last, David;
Daniels, Dianne;
Guez, David;
Shneor, Ran;
Mardor, Yael;
Nudelman, Abraham;
Krivoy, Amir

Publication type:

Article

30

Acetyl Bromide-Alcohols as Convenient Reaction Systems for: a) Removal of N - tert -Boc, N -Cbz And N -Ac Protective Groups, b) Esterifications and Transesterifications, c) Debenzylation of Aryl-O-Benzyl Ethers.

Published in:

Synthetic Communications, 1999, v. 29, n. 8, p. 1405, doi. 10.1080/00397919908086117

By:

And, Anat Lesk;
Nudelman, Abraham

Publication type:

Article

31

Acetyl Chloride-Methanol as a Convenient Reagent for: A) Quantitative Formation of Amine Hydrochlorides B) Carboxylate Ester Formation C) Mild Removal of N-t-Boc-Protective Group.

Published in:

Synthetic Communications, 1998, v. 28, n. 3, p. 471, doi. 10.1080/00397919808005101

By:

Nudelman, Ayelet;
Bechor, Yosi;
Falb, Eliezer;
Fischer, Bilha;
Wexler, Barry A.;
Nudelman, Abraham

Publication type:

Article

32

AN-7, a butyric acid prodrug, sensitizes cutaneous T-cell lymphoma cell lines to doxorubicin via inhibition of DNA double strand breaks repair.

Published in:

Investigational New Drugs, 2018, v. 36, n. 1, p. 1, doi. 10.1007/s10637-017-0500-x

By:

Moyal, Lilach;
Goldfeiz, Neta;
Gorovitz, Batia;
Rephaeli, Ada;
Tal, Efrat;
Tarasenko, Nataly;
Nudelman, Abraham;
Ziv, Yael;
Hodak, Emmilia

Publication type:

Article

33

Effects of histone deacetylase inhibitory prodrugs on epigenetic changes and DNA damage response in tumor and heart of glioblastoma xenograft.

Published in:

Investigational New Drugs, 2017, v. 35, n. 4, p. 412, doi. 10.1007/s10637-017-0448-x

By:

Tarasenko, Nataly;
Nudelman, Abraham;
Rozic, Gabriela;
Cutts, Suzanne;
Rephaeli, Ada

Publication type:

Article

34

Mode of interaction between butyroyloxymethyl-diethyl phosphate (AN-7) and doxorubicin in MCF-7 and resistant MCF-7/Dx cell lines.

Published in:

Journal of Cancer Research & Clinical Oncology, 2006, v. 132, n. 10, p. 673, doi. 10.1007/s00432-006-0116-6

By:

Engel, Dikla;
Nudelman, Abraham;
Levovich, Inesa;
Gruss-Fischer, Tal;
Entin-Meer, Michal;
Phillips, Don;
Cutts, Suzanne;
Rephaeli, Ada

Publication type:

Article