Works by Norman, Derek D.

Results: 9

E2F7 drives autotaxin/Enpp2 transcription via chromosome looping: Repression by p53 in murine but not in human carcinomas.

Published in:

FASEB Journal, 2023, v. 37, n. 7, p. 1, doi. 10.1096/fj.202300838R

By:

Lin, Kuan‐Hung;
Lee, Sue Chin;
Dacheux, Mélanie A.;
Norman, Derek D.;
Balogh, Andrea;
Bavaria, Mitul;
Lee, Hsinyu;
Tigyi, Gabor

Publication type:

Article

Targeting the hydrophobic pocket of autotaxin with virtual screening of inhibitors identifies a common aromatic sulfonamide structural motif.

Published in:

FEBS Journal, 2014, v. 281, n. 4, p. 1017, doi. 10.1111/febs.12674

By:

Fells, James I.;
Lee, Sue Chin;
Norman, Derek D.;
Tsukahara, Ryoko;
Kirby, Jason R.;
Nelson, Sandra;
Seibel, William;
Papoian, Ruben;
Patil, Renukadevi;
Miller, Duane D.;
Parrill, Abby L.;
Pham, Truc‐Chi;
Baker, Daniel L.;
Bittman, Robert;
Tigyi, Gabor

Publication type:

Article

Osteoclast‐Derived Autotaxin, a Distinguishing Factor for Inflammatory Bone Loss.

Published in:

Arthritis & Rheumatology, 2019, v. 71, n. 11, p. 1801, doi. 10.1002/art.41005

By:

Flammier, Sacha;
Peyruchaud, Olivier;
Bourguillault, Fanny;
Duboeuf, François;
Davignon, Jean‐Luc;
Norman, Derek D.;
Isaac, Sylvie;
Marotte, Hubert;
Tigyi, Gabor;
Machuca‐Gayet, Irma;
Coury, Fabienne

Publication type:

Article

Regulation of Tumor Immunity by Lysophosphatidic Acid.

Published in:

Cancers, 2020, v. 12, n. 5, p. 1202, doi. 10.3390/cancers12051202

By:

Lee, Sue Chin;
Dacheux, Mélanie A.;
Norman, Derek D.;
Balázs, Louisa;
Torres, Raul M.;
Augelli-Szafran, Corinne E.;
Tigyi, Gábor J.

Publication type:

Article

Prometastatic Effect of ATX Derived from Alveolar Type II Pneumocytes and B16-F10 Melanoma Cells.

Published in:

Cancers, 2022, v. 14, n. 6, p. 1586, doi. 10.3390/cancers14061586

By:

Dacheux, Mélanie A.;
Lee, Sue Chin;
Shin, Yoojin;
Norman, Derek D.;
Lin, Kuan-Hung;
E, Shuyu;
Yue, Junming;
Benyó, Zoltán;
Tigyi, Gábor J.

Publication type:

Article

Functional modulation of lysophosphatidic acid type 2 G‐protein coupled receptor facilitates alveolar bone formation.

Published in:

Journal of Cellular Physiology, 2024, v. 239, n. 1, p. 112, doi. 10.1002/jcp.31148

By:

Kim, Tae‐Young;
Kim, Anna;
Aryal, Yam Prasad;
Sung, Shijin;
Pokharel, Elina;
Neupane, Sanjiv;
Choi, So‐Young;
Ha, Jung‐Hong;
Jung, Jae‐Kwang;
Yamamoto, Hitoshi;
An, Chang‐Hyeon;
Suh, Jo‐Young;
Sohn, Wern‐Joo;
Lee, Youngkyun;
Jang, Il‐Ho;
Norman, Derek D.;
Tigyi, Gabor J.;
An, Seo‐Young;
Kim, Jae‐Young

Publication type:

Article

Structure-Based Discovery of MolPort-137: A Novel Autotaxin Inhibitor That Improves Paclitaxel Efficacy.

Published in:

International Journal of Molecular Sciences, 2025, v. 26, n. 2, p. 597, doi. 10.3390/ijms26020597

By:

Rai, Prateek;
Clark, Christopher J.;
Kardam, Vandana;
Womack, Carl B.;
Thammathong, Joshua;
Norman, Derek D.;
Tigyi, Gábor J.;
Bicker, Kevin;
Weissmiller, April M.;
Dubey, Kshatresh Dutta;
Banerjee, Souvik

Publication type:

Article

Novel Autotaxin Inhibitor ATX-1d Significantly Enhances Potency of Paclitaxel—An In Silico and In Vitro Study.

Published in:

Molecules, 2024, v. 29, n. 18, p. 4285, doi. 10.3390/molecules29184285

By:

Rai, Prateek;
Clark, Christopher J.;
Womack, Carl B.;
Dearing, Curtis;
Thammathong, Joshua;
Norman, Derek D.;
Tigyi, Gábor J.;
Sen, Subhabrata;
Bicker, Kevin;
Weissmiller, April M.;
Banerjee, Souvik

Publication type:

Article

Designing Dual Inhibitors of Autotaxin-LPAR GPCR Axis.

Published in:

Molecules, 2022, v. 27, n. 17, p. 5487, doi. 10.3390/molecules27175487

By:

Banerjee, Souvik;
Lee, Suechin;
Norman, Derek D.;
Tigyi, Gabor J.

Publication type:

Article