Works by Nocentini, Alessio

Results: 122

Exploration of Aromatic Hydrazides as Inhibitors of Human Carbonic Anhydrases.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 4, p. 1, doi. 10.1002/ardp.202400963

By:

Menendez, German Benito;
Giovannuzzi, Simone;
Bonardi, Alessandro;
Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Exploring aliphatic sulfonamides as multiclass inhibitors of the carbonic anhydrases from the pathogen bacterium Vibrio cholerae.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 1, p. 1, doi. 10.1002/ardp.202400814

By:

Paoletti, Niccolò;
Giovannuzzi, Simone;
Bonardi, Alessandro;
De Luca, Viviana;
Capasso, Clemente;
Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

1,5‐Benzodiazepines as a platform for the design of carbonic anhydrase inhibitors.

Published in:

Archiv der Pharmazie, 2022, v. 355, n. 3, p. 1, doi. 10.1002/ardp.202100405

By:

Ismail, Chiraz;
Nocentini, Alessio;
Supuran, Claudiu T.;
Winum, Jean‐Yves;
Gharbi, Rafik

Publication type:

Article

Novel benzenesulfonamide‐bearing pyrazoles and 1,2,4‐thiadiazoles as selective carbonic anhydrase inhibitors.

Published in:

Archiv der Pharmazie, 2022, v. 355, n. 1, p. 1, doi. 10.1002/ardp.202100241

By:

Kumar, Rajiv;
Kumar, Amit;
Ram, Sita;
Angeli, Andrea;
Bonardi, Alessandro;
Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.;
Sharma, Pawan K.

Publication type:

Article

Drug Screening in Human Cells by NMR Spectroscopy Allows the Early Assessment of Drug Potency.

Published in:

Angewandte Chemie International Edition, 2020, v. 59, n. 16, p. 6535, doi. 10.1002/anie.201913436

By:

Luchinat, Enrico;
Barbieri, Letizia;
Cremonini, Matteo;
Nocentini, Alessio;
Supuran, Claudiu T.;
Banci, Lucia

Publication type:

Article

Design and Comparative Evaluation of the Anticonvulsant Profile, Carbonic-Anhydrate Inhibition and Teratogenicity of Novel Carbamate Derivatives of Branched Aliphatic Carboxylic Acids with 4-Aminobenzensulfonamide.

Published in:

Neurochemical Research, 2017, v. 42, n. 7, p. 1972, doi. 10.1007/s11064-017-2216-x

By:

Bibi, David;
Mawasi, Hafiz;
Nocentini, Alessio;
Supuran, Claudiu;
Wlodarczyk, Bogdan;
Finnell, Richard;
Bialer, Meir

Publication type:

Article

Selective carbonic anhydrase IX and XII inhibitors based around a functionalized coumarin scaffold.

Published in:

Drug Development Research, 2023, v. 84, n. 4, p. 681, doi. 10.1002/ddr.22049

By:

Huwaimel, Bader I.;
Jonnalagadda, Sravan K.;
Jonnalagadda, Shirisha;
Kumari, Shikha;
Nocentini, Alessio;
Supuran, Claudiu T.;
Trippier, Paul C.

Publication type:

Article

Carbonic Anhydrase Inhibition Activities of Schiff's Bases Based on Quinazoline-Linked Benzenesulfonamide.

Published in:

Molecules, 2022, v. 27, n. 22, p. 7703, doi. 10.3390/molecules27227703

By:

El-Azab, Adel S.;
Abdel-Aziz, Alaa A.-M.;
Ghabbour, Hazem A.;
Bua, Silvia;
Nocentini, Alessio;
Alkahtani, Hamad M.;
Alsaif, Nawaf A.;
Al-Agamy, Mohamed H. M.;
Supuran, Claudiu T.

Publication type:

Article

Continued Structural Exploration of Sulfocoumarin as Selective Inhibitor of Tumor-Associated Human Carbonic Anhydrases IX and XII.

Published in:

Molecules, 2022, v. 27, n. 13, p. 4076, doi. 10.3390/molecules27134076

By:

Giovannuzzi, Simone;
Capasso, Clemente;
Nocentini, Alessio;
Supuran, Claudiu T.

Publication type:

Article

The Glitazone Class of Drugs as Carbonic Anhydrase Inhibitors—A Spin-Off Discovery from Fragment Screening.

Published in:

Molecules, 2021, v. 26, n. 10, p. 3010, doi. 10.3390/molecules26103010

By:

Mueller, Sarah L.;
Chrysanthopoulos, Panagiotis K.;
Halili, Maria A.;
Hepburn, Caryn;
Nebl, Tom;
Supuran, Claudiu T.;
Nocentini, Alessio;
Peat, Thomas S.;
Poulsen, Sally-Ann;
Alfonso-Prieto, Mercedes

Publication type:

Article

Anion Inhibition Studies of the Beta-Carbonic Anhydrase from Escherichia coli.

Published in:

Molecules, 2020, v. 25, n. 11, p. 2564, doi. 10.3390/molecules25112564

By:

Del Prete, Sonia;
De Luca, Viviana;
Nocentini, Alessio;
Scaloni, Andrea;
Mastrolorenzo, Margaret D.;
Supuran, Claudiu T.;
Capasso, Clemente;
Muñoz-Torrero, Diego

Publication type:

Article

Hypoxia-Activated Prodrug Derivatives of Carbonic Anhydrase Inhibitors in Benzenesulfonamide Series: Synthesis and Biological Evaluation.

Published in:

Molecules, 2020, v. 25, n. 10, p. 2347, doi. 10.3390/molecules25102347

By:

Anduran, Emilie;
Aspatwar, Ashok;
Parvathaneni, Nanda-Kumar;
Suylen, Dennis;
Bua, Silvia;
Nocentini, Alessio;
Parkkila, Seppo;
Supuran, Claudiu T.;
Dubois, Ludwig;
Lambin, Philippe;
Winum, Jean-Yves;
Carta, Fabrizio;
Angeli, Andrea

Publication type:

Article

Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation.

Published in:

Molecules, 2019, v. 24, n. 19, p. 3580, doi. 10.3390/molecules24193580

By:

Kartsev, Victor;
Geronikaki, Athina;
Bua, Silvia;
Nocentini, Alessio;
Petrou, Anthi;
Lichitsky, Boris;
Frasinyuk, Mykhaylo;
Leitans, Janis;
Kazaks, Andris;
Tars, Kaspars;
Supuran, Claudiu T.

Publication type:

Article

Use of Innovative (Micro)Extraction Techniques to Characterise Harpagophytum procumbens Root and its Commercial Food Supplements.

Published in:

Phytochemical Analysis, 2018, v. 29, n. 3, p. 233, doi. 10.1002/pca.2737

By:

Diuzheva, Alina;
Carradori, Simone;
Andruch, Vasil;
Locatelli, Marcello;
De Luca, Elisa;
Tiecco, Matteo;
Germani, Raimondo;
Menghini, Luigi;
Nocentini, Alessio;
Gratteri, Paola;
Campestre, Cristina

Publication type:

Article

Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors.

Published in:

ChemMedChem, 2020, v. 15, n. 21, p. 2052, doi. 10.1002/cmdc.202000500

By:

Clima, Lilia;
Craciun, Bogdan Florin;
Angeli, Andrea;
Petreni, Andrea;
Bonardi, Alessandro;
Nocentini, Alessio;
Carta, Fabrizio;
Gratteri, Paola;
Pinteala, Mariana;
Supuran, Claudiu T.

Publication type:

Article

Natural Polyphenols Selectively Inhibit β‐Carbonic Anhydrase from the Dandruff‐Producing Fungus <italic>Malassezia globosa</italic>: Activity and Modeling Studies.

Published in:

ChemMedChem, 2018, v. 13, n. 8, p. 816, doi. 10.1002/cmdc.201800015

By:

Nocentini, Alessio;
Bua, Silvia;
Del Prete, Sonia;
Heravi, Yeganeh Entezari;
Saboury, Ali A.;
Karioti, Anastasia;
Bilia, Anna Rita;
Capasso, Clemente;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Discovery of novel drugs for Chagas disease: is carbonic anhydrase a target for antiprotozoal drugs?

Published in:

Expert Opinion on Drug Discovery, 2022, v. 17, n. 10, p. 1147, doi. 10.1080/17460441.2022.2117295

By:

Beatriz Vermelho, Alane;
Rodrigues, Giseli Capaci;
Nocentini, Alessio;
Mansoldo, Felipe R. P.;
Supuran, Claudiu T.

Publication type:

Article

Advances in the discovery of novel agents for the treatment of glaucoma.

Published in:

Expert Opinion on Drug Discovery, 2021, v. 16, n. 10, p. 1209, doi. 10.1080/17460441.2021.1922384

By:

Mincione, Francesco;
Nocentini, Alessio;
Supuran, Claudiu T.

Publication type:

Article

Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery.

Published in:

Expert Opinion on Drug Discovery, 2019, v. 14, n. 11, p. 1175, doi. 10.1080/17460441.2019.1651289

By:

Nocentini, Alessio;
Supuran, Claudiu T.

Publication type:

Article

Native mass spectrometry of human carbonic anhydrase I and its inhibitor complexes.

Published in:

Journal of Biological Inorganic Chemistry (JBIC), 2020, v. 25, n. 7, p. 979, doi. 10.1007/s00775-020-01818-8

By:

Zoppi, Carlotta;
Nocentini, Alessio;
Supuran, Claudiu T.;
Pratesi, Alessandro;
Messori, Luigi

Publication type:

Article

Synthesis, Crystal Structure, Inhibitory Activity and Molecular Docking of Coumarins/Sulfonamides Containing Triazolyl Pyridine Moiety as Potent Selective Carbonic Anhydrase IX and XII Inhibitors.

Published in:

Crystals (2073-4352), 2021, v. 11, n. 9, p. 1076, doi. 10.3390/cryst11091076

By:

Aimene, Yassine;
Eychenne, Romain;
Rodriguez, Frédéric;
Mallet-Ladeira, Sonia;
Saffon-Merceron, Nathalie;
Winum, Jean-Yves;
Nocentini, Alessio;
Supuran, Claudiu T.;
Benoist, Eric;
Seridi, Achour

Publication type:

Article

Carbonic Anhydrase Inhibitors Featuring a Porphyrin Scaffold: Synthesis, Optical and Biological Properties.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 21, p. 1, doi. 10.1002/ejoc.202101538

By:

Merabti, Amina;
Roger, Maxime;
Nguyen, Christophe;
Nocentini, Alessio;
Gerbier, Philippe;
Richeter, Sébastien;
Gary‐Bobo, Magali;
Supuran, Claudiu T.;
Clément, Sébastien;
Winum, Jean‐Yves

Publication type:

Article

Multifaceted Sulfonamide-Derived Thiosemicarbazones: Combining Metal Chelation and Carbonic Anhydrases Inhibition in Anticancer Therapy.

Published in:

International Journal of Molecular Sciences, 2025, v. 26, n. 3, p. 1225, doi. 10.3390/ijms26031225

By:

Martínez-Montiel, Mónica;
Arrighi, Giulia;
Begines, Paloma;
González-Bakker, Aday;
Puerta, Adrián;
Fernandes, Miguel X.;
Merino-Montiel, Penélope;
Montiel-Smith, Sara;
Nocentini, Alessio;
Supuran, Claudiu T.;
Padrón, José M.;
Fernández-Bolaños, José G.;
López, Óscar

Publication type:

Article

Hydrogen Sulfide-Releasing Carbonic Anhydrase Inhibitors Effectively Suppress Cancer Cell Growth.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 18, p. 10006, doi. 10.3390/ijms251810006

By:

Bonardi, Alessandro;
Nocentini, Alessio;
de Luca, Viviana;
Capasso, Clemente;
Elkaeed, Eslam B.;
Eldehna, Wagdy M.;
Supuran, Claudiu T.

Publication type:

Article

Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 5, p. 2584, doi. 10.3390/ijms25052584

By:

Bua, Silvia;
Bonardi, Alessandro;
Mük, Georgiana Ramona;
Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Leveraging SARS-CoV-2 Main Protease (M pro) for COVID-19 Mitigation with Selenium-Based Inhibitors.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 2, p. 971, doi. 10.3390/ijms25020971

By:

De Luca, Viviana;
Angeli, Andrea;
Nocentini, Alessio;
Gratteri, Paola;
Pratesi, Silvia;
Tanini, Damiano;
Carginale, Vincenzo;
Capperucci, Antonella;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 11, p. 9401, doi. 10.3390/ijms24119401

By:

Martínez-Montiel, Mónica;
Romero-Hernández, Laura L.;
Giovannuzzi, Simone;
Begines, Paloma;
Puerta, Adrián;
Ahuja-Casarín, Ana I.;
Fernandes, Miguel X.;
Merino-Montiel, Penélope;
Montiel-Smith, Sara;
Nocentini, Alessio;
Padrón, José M.;
Supuran, Claudiu T.;
Fernández-Bolaños, José G.;
López, Óscar

Publication type:

Article

Squaramide-Tethered Sulfonamides and Coumarins: Synthesis, Inhibition of Tumor-Associated CAs IX and XII and Docking Simulations.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 14, p. 7685, doi. 10.3390/ijms23147685

By:

Arrighi, Giulia;
Puerta, Adrián;
Petrini, Andrea;
Hicke, Francisco J.;
Nocentini, Alessio;
Fernandes, Miguel X.;
Padrón, José M.;
Supuran, Claudiu T.;
Fernández-Bolaños, José G.;
López, Óscar

Publication type:

Article

Aromatic Sulfonamides including a Sulfonic Acid Tail: New Membrane Impermeant Carbonic Anhydrase Inhibitors for Targeting Selectively the Cancer-Associated Isoforms.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 1, p. 461, doi. 10.3390/ijms23010461

By:

Giovannuzzi, Simone;
D'Ambrosio, Mario;
Luceri, Cristina;
Osman, Sameh Mohamed;
Pallecchi, Marco;
Bartolucci, Gianluca;
Nocentini, Alessio;
Supuran, Claudiu T.

Publication type:

Article

Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 21, p. 11583, doi. 10.3390/ijms222111583

By:

Grande, Rossella;
Carradori, Simone;
Puca, Valentina;
Vitale, Irene;
Angeli, Andrea;
Nocentini, Alessio;
Bonardi, Alessandro;
Gratteri, Paola;
Lanuti, Paola;
Bologna, Giuseppina;
Simeone, Pasquale;
Capasso, Clemente;
De Luca, Viviana;
Supuran, Claudiu T.

Publication type:

Article

Development of Novel Quinoline-Based Sulfonamides as Selective Cancer-Associated Carbonic Anhydrase Isoform IX Inhibitors.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 20, p. 11119, doi. 10.3390/ijms222011119

By:

Shaldam, Moataz;
Nocentini, Alessio;
Elsayed, Zainab M.;
Ibrahim, Tamer M.;
Salem, Rofaida;
El-Domany, Ramadan A.;
Capasso, Clemente;
Supuran, Claudiu T.;
Eldehna, Wagdy M.

Publication type:

Article

Role of Carbonic Anhydrase in Cerebral Ischemia and Carbonic Anhydrase Inhibitors as Putative Protective Agents.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 9, p. 5029, doi. 10.3390/ijms22095029

By:

Bulli, Irene;
Dettori, Ilaria;
Coppi, Elisabetta;
Cherchi, Federica;
Venturini, Martina;
Di Cesare Mannelli, Lorenzo;
Ghelardini, Carla;
Nocentini, Alessio;
Supuran, Claudiu T.;
Pugliese, Anna Maria;
Pedata, Felicita;
Battino, Maurizio

Publication type:

Article

Synthesis and Enantioselective Pharmacokinetic/Pharmacodynamic Analysis of New CNS-Active Sulfamoylphenyl Carbamate Derivatives.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 7, p. 3361, doi. 10.3390/ijms22073361

By:

Odi, Reem;
Bibi, David;
Shusterman, Bella;
Erenburg, Natalia;
Shaul, Chanan;
Supuran, Claudiu T.;
Nocentini, Alessio;
Bialer, Meir;
Czuczwar, Stanislaw Jerzy

Publication type:

Article

Effect of Sulfonamides and Their Structurally Related Derivatives on the Activity of ι -Carbonic Anhydrase from Burkholderia territorii.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 2, p. 571, doi. 10.3390/ijms22020571

By:

De Luca, Viviana;
Petreni, Andrea;
Nocentini, Alessio;
Scaloni, Andrea;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

The Effect of Substituted Benzene-Sulfonamides and Clinically Licensed Drugs on the Catalytic Activity of CynT2, a Carbonic Anhydrase Crucial for Escherichia coli Life Cycle.

Published in:

International Journal of Molecular Sciences, 2020, v. 21, n. 11, p. 4175, doi. 10.3390/ijms21114175

By:

Del Prete, Sonia;
De Luca, Viviana;
Bua, Silvia;
Nocentini, Alessio;
Carginale, Vincenzo;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Aryl-4,5-dihydro-1H-pyrazole-1-carboxamide Derivatives Bearing a Sulfonamide Moiety Show Single-digit Nanomolar-to-Subnanomolar Inhibition Constants against the Tumor-associated Human Carbonic Anhydrases IX and XII.

Published in:

International Journal of Molecular Sciences, 2020, v. 21, n. 7, p. 2621, doi. 10.3390/ijms21072621

By:

Hargunani, Priya;
Tadge, Nikhil;
Ceruso, Mariangela;
Leitans, Janis;
Kazaks, Andris;
Tars, Kaspars;
Gratteri, Paola;
Supuran, Claudiu T.;
Nocentini, Alessio;
Toraskar, Mrunmayee P.

Publication type:

Article

A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 19, p. 4724, doi. 10.3390/ijms20194724

By:

Provensi, Gustavo;
Carta, Fabrizio;
Nocentini, Alessio;
Supuran, Claudiu T.;
Casamenti, Fiorella;
Passani, M. Beatrice;
Fossati, Silvia

Publication type:

Article

Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 10, p. 2484, doi. 10.3390/ijms20102484

By:

Abdelrahman, Mohamed A.;
Eldehna, Wagdy M.;
Nocentini, Alessio;
Bua, Silvia;
Al-Rashood, Sara T.;
Hassan, Ghada S.;
Bonardi, Alessandro;
Almehizia, Abdulrahman A.;
Alkahtani, Hamad M.;
Alharbi, Amal;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

β3-Adrenoreceptor Activity Limits Apigenin Efficacy in Ewing Sarcoma Cells: A Dual Approach to Prevent Cell Survival.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 9, p. 2149, doi. 10.3390/ijms20092149

By:

Pasha, Amada;
Vignoli, Marina;
Subbiani, Angela;
Nocentini, Alessio;
Selleri, Silvia;
Gratteri, Paola;
Dabraio, Annalisa;
Casini, Tommaso;
Filippi, Luca;
Fotzi, Ilaria;
Favre, Claudio;
Calvani, Maura

Publication type:

Article

Drug Screening in Human Cells by NMR Spectroscopy Allows the Early Assessment of Drug Potency.

Published in:

Angewandte Chemie, 2020, v. 132, n. 16, p. 6597, doi. 10.1002/ange.201913436

By:

Luchinat, Enrico;
Barbieri, Letizia;
Cremonini, Matteo;
Nocentini, Alessio;
Supuran, Claudiu T.;
Banci, Lucia

Publication type:

Article

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 10, p. 412, doi. 10.3390/metabo10100412

By:

Angeli, Andrea;
Carta, Fabrizio;
Nocentini, Alessio;
Winum, Jean-Yves;
Zalubovskis, Raivis;
Akdemir, Atilla;
Onnis, Valentina;
Eldehna, Wagdy M.;
Capasso, Clemente;
Simone, Giuseppina De;
Monti, Simona Maria;
Carradori, Simone;
Donald, William A.;
Dedhar, Shoukat;
Supuran, Claudiu T.

Publication type:

Article

Determination of intracellular protein–ligand binding affinity by competition binding in‐cell NMR.

Published in:

Acta Crystallographica: Section D, Structural Biology, 2021, v. 77, n. 10, p. 1270, doi. 10.1107/S2059798321009037

By:

Luchinat, Enrico;
Barbieri, Letizia;
Cremonini, Matteo;
Pennestri, Matteo;
Nocentini, Alessio;
Supuran, Claudiu T.;
Banci, Lucia

Publication type:

Article

Structural and biochemical characterization of novel carbonic anhydrases from Phaeodactylum tricornutum.

Published in:

Acta Crystallographica: Section D, Structural Biology, 2020, v. 76, n. 7, p. 676, doi. 10.1107/S2059798320007202

By:

Jin, Shengyang;
Vullo, Daniela;
Bua, Silvia;
Nocentini, Alessio;
Supuran, Claudiu T.;
Gao, Yong-gui

Publication type:

Article

Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII.

Published in:

Pharmaceuticals (14248247), 2023, v. 16, n. 2, p. 188, doi. 10.3390/ph16020188

By:

Ialongo, Davide;
Messore, Antonella;
Madia, Valentina Noemi;
Tudino, Valeria;
Nocentini, Alessio;
Gratteri, Paola;
Giovannuzzi, Simone;
Supuran, Claudiu T.;
Nicolai, Alice;
Scarpa, Susanna;
Taurone, Samanta;
Camarda, Michele;
Artico, Marco;
Papa, Veronica;
Saccoliti, Francesco;
Scipione, Luigi;
Di Santo, Roberto;
Costi, Roberta

Publication type:

Article

Calixarenes Incorporating Sulfonamide Moieties: Versatile Ligands for Carbonic Anhydrases Inhibition.

Published in:

Chemistry - A European Journal, 2022, v. 28, n. 6, p. 1, doi. 10.1002/chem.202103527

By:

Sbravati, Davide;
Bonardi, Alessandro;
Bua, Silvia;
Angeli, Andrea;
Ferraroni, Marta;
Nocentini, Alessio;
Casnati, Alessandro;
Gratteri, Paola;
Sansone, Francesco;
Supuran, Claudiu T.

Publication type:

Article

Phosphorus versus Sulfur: Discovery of Benzenephosphonamidates as Versatile Sulfonamide‐Mimic Chemotypes Acting as Carbonic Anhydrase Inhibitors.

Published in:

Chemistry - A European Journal, 2019, v. 25, n. 5, p. 1188, doi. 10.1002/chem.201805039

By:

Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies.

Published in:

Chemistry - A European Journal, 2018, v. 24, n. 31, p. 7840, doi. 10.1002/chem.201800941

By:

Nocentini, Alessio;
Carta, Fabrizio;
Tanc, Muhammet;
Selleri, Silvia;
Supuran, Claudiu T.;
Bazzicalupi, Carla;
Gratteri, Paola

Publication type:

Article

Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2284119

By:

Giovannuzzi, Simone;
Marapaka, Anil Kumar;
Abutaleb, Nader S.;
Carta, Fabrizio;
Liang, Hsin-Wen;
Nocentini, Alessio;
Pisano, Luigi;
Seleem, Mohamed N.;
Flaherty, Daniel P.;
Supuran, Claudiu T.

Publication type:

Article

Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2270180

By:

Romagnoli, Romeo;
De Ventura, Tiziano;
Manfredini, Stefano;
Baldini, Erika;
Supuran, Claudiu T.;
Nocentini, Alessio;
Brancale, Andrea;
Bortolozzi, Roberta;
Manfreda, Lorenzo;
Viola, Giampietro

Publication type:

Article

Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2249267

By:

Balašova, Anastasija;
Pustenko, Aleksandrs;
Nocentini, Alessio;
Vullo, Daniela;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article