Works matching AU Nocentini, Alessio


Results: 122
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    Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment.

    Published in:
    Metabolites (2218-1989), 2020, v. 10, n. 10, p. 412, doi. 10.3390/metabo10100412
    By:
    • Angeli, Andrea;
    • Carta, Fabrizio;
    • Nocentini, Alessio;
    • Winum, Jean-Yves;
    • Zalubovskis, Raivis;
    • Akdemir, Atilla;
    • Onnis, Valentina;
    • Eldehna, Wagdy M.;
    • Capasso, Clemente;
    • Simone, Giuseppina De;
    • Monti, Simona Maria;
    • Carradori, Simone;
    • Donald, William A.;
    • Dedhar, Shoukat;
    • Supuran, Claudiu T.
    Publication type:
    Article
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    Multifaceted Sulfonamide-Derived Thiosemicarbazones: Combining Metal Chelation and Carbonic Anhydrases Inhibition in Anticancer Therapy.

    Published in:
    International Journal of Molecular Sciences, 2025, v. 26, n. 3, p. 1225, doi. 10.3390/ijms26031225
    By:
    • Martínez-Montiel, Mónica;
    • Arrighi, Giulia;
    • Begines, Paloma;
    • González-Bakker, Aday;
    • Puerta, Adrián;
    • Fernandes, Miguel X.;
    • Merino-Montiel, Penélope;
    • Montiel-Smith, Sara;
    • Nocentini, Alessio;
    • Supuran, Claudiu T.;
    • Padrón, José M.;
    • Fernández-Bolaños, José G.;
    • López, Óscar
    Publication type:
    Article
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    Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2284119
    By:
    • Giovannuzzi, Simone;
    • Marapaka, Anil Kumar;
    • Abutaleb, Nader S.;
    • Carta, Fabrizio;
    • Liang, Hsin-Wen;
    • Nocentini, Alessio;
    • Pisano, Luigi;
    • Seleem, Mohamed N.;
    • Flaherty, Daniel P.;
    • Supuran, Claudiu T.
    Publication type:
    Article
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    Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2270180
    By:
    • Romagnoli, Romeo;
    • De Ventura, Tiziano;
    • Manfredini, Stefano;
    • Baldini, Erika;
    • Supuran, Claudiu T.;
    • Nocentini, Alessio;
    • Brancale, Andrea;
    • Bortolozzi, Roberta;
    • Manfreda, Lorenzo;
    • Viola, Giampietro
    Publication type:
    Article
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    Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201407
    By:
    • Badawi, Waleed A.;
    • Rashed, Mahmoud;
    • Nocentini, Alessio;
    • Bonardi, Alessandro;
    • Abd-Alhaseeb, Mohammad M.;
    • Al-Rashood, Sara T.;
    • Veerakanellore, Giri Babu;
    • Majrashi, Taghreed A.;
    • Elkaeed, Eslam B.;
    • Elgendy, Bahaa;
    • Gratteri, Paola;
    • Supuran, Claudiu T.;
    • Eldehna, Wagdy M.;
    • Elagawany, Mohamed
    Publication type:
    Article
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    The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 930, doi. 10.1080/14756366.2022.2053526
    By:
    • Bonardi, Alessandro;
    • Bua, Silvia;
    • Combs, Jacob;
    • Lomelino, Carrie;
    • Andring, Jacob;
    • Osman, Sameh Mohamed;
    • Toti, Alessandra;
    • Di Cesare Mannelli, Lorenzo;
    • Gratteri, Paola;
    • Ghelardini, Carla;
    • McKenna, Robert;
    • Nocentini, Alessio;
    • Supuran, Claudiu T.
    Publication type:
    Article
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    Inhibition studies of bacterial α-carbonic anhydrases with phenols.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 666, doi. 10.1080/14756366.2022.2038592
    By:
    • Giovannuzzi, Simone;
    • Hewitt, Chad S.;
    • Nocentini, Alessio;
    • Capasso, Clemente;
    • Costantino, Gabriele;
    • Flaherty, Daniel P.;
    • Supuran, Claudiu T.
    Publication type:
    Article
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    Discovery of 2,4-thiazolidinedione-tethered coumarins as novel selective inhibitors for carbonic anhydrase IX and XII isoforms.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 531, doi. 10.1080/14756366.2021.2024528
    By:
    • Eldehna, Wagdy M.;
    • Taghour, Mohammed S.;
    • Al-Warhi, Tarfah;
    • Nocentini, Alessio;
    • Elbadawi, Mostafa M.;
    • Mahdy, Hazem A.;
    • Abdelrahman, Mohamed A.;
    • Alotaibi, Ohoud J.;
    • Aljaeed, Nada;
    • Elimam, Diaaeldin M.;
    • Afarinkia, Kamyar;
    • Abdel-Aziz, Hatem A.;
    • Supuran, Claudiu T.
    Publication type:
    Article
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    Coumarins effectively inhibit bacterial a-carbonic anhydrases.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 333, doi. 10.1080/14756366.2021.2012174
    By:
    • Giovannuzzi, Simone;
    • Hewitt, Chad S.;
    • Nocentini, Alessio;
    • Capasso, Clemente;
    • Flaherty, Daniel P.;
    • Supuran, Claudiu T.
    Publication type:
    Article
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    2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 168, doi. 10.1080/14756366.2021.1998026
    By:
    • Fuentes-Aguilar, Alma;
    • Merino-Montiel, Penélope;
    • Montiel-Smith, Sara;
    • Meza-Reyes, Socorro;
    • Vega-Baez, José Luis;
    • Puerta, Adrian;
    • Fernandes, Miguel X.;
    • Padrón, José M.;
    • Petreni, Andrea;
    • Nocentini, Alessio;
    • Supuran, Claudiu T.;
    • López, Oscar;
    • Fernéndez-Bolaños, José G.
    Publication type:
    Article
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