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Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold †.
- Published in:
- Molecules, 2024, v. 29, n. 14, p. 3290, doi. 10.3390/molecules29143290
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- Article
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 5, p. 2584, doi. 10.3390/ijms25052584
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- Article
Leveraging SARS-CoV-2 Main Protease (M pro) for COVID-19 Mitigation with Selenium-Based Inhibitors.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 2, p. 971, doi. 10.3390/ijms25020971
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- Article
Selective carbonic anhydrase IX and XII inhibitors based around a functionalized coumarin scaffold.
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- Drug Development Research, 2023, v. 84, n. 4, p. 681, doi. 10.1002/ddr.22049
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- Article
Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 11, p. 9401, doi. 10.3390/ijms24119401
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- Article
Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII.
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- Pharmaceuticals (14248247), 2023, v. 16, n. 2, p. 188, doi. 10.3390/ph16020188
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Carbonic Anhydrase Inhibitors as Novel Antibacterials in the Era of Antibiotic Resistance: Where Are We Now?
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- Antibiotics (2079-6382), 2023, v. 12, n. 1, p. 142, doi. 10.3390/antibiotics12010142
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- Article
Carbonic Anhydrase Inhibition Activities of Schiff's Bases Based on Quinazoline-Linked Benzenesulfonamide.
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- Molecules, 2022, v. 27, n. 22, p. 7703, doi. 10.3390/molecules27227703
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- Article
Biochemical and Biophysical Characterization of Carbonic Anhydrase VI from Human Milk and Saliva.
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- Protein Journal, 2022, v. 41, n. 4/5, p. 489, doi. 10.1007/s10930-022-10070-9
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- Article
Squaramide-Tethered Sulfonamides and Coumarins: Synthesis, Inhibition of Tumor-Associated CAs IX and XII and Docking Simulations.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 14, p. 7685, doi. 10.3390/ijms23147685
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- Article
Continued Structural Exploration of Sulfocoumarin as Selective Inhibitor of Tumor-Associated Human Carbonic Anhydrases IX and XII.
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- Molecules, 2022, v. 27, n. 13, p. 4076, doi. 10.3390/molecules27134076
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- Article
Carbonic Anhydrase Inhibitors Featuring a Porphyrin Scaffold: Synthesis, Optical and Biological Properties.
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- European Journal of Organic Chemistry, 2022, v. 2022, n. 21, p. 1, doi. 10.1002/ejoc.202101538
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- Article
1,5‐Benzodiazepines as a platform for the design of carbonic anhydrase inhibitors.
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- Archiv der Pharmazie, 2022, v. 355, n. 3, p. 1, doi. 10.1002/ardp.202100405
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- Article
Calixarenes Incorporating Sulfonamide Moieties: Versatile Ligands for Carbonic Anhydrases Inhibition.
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- Chemistry - A European Journal, 2022, v. 28, n. 6, p. 1, doi. 10.1002/chem.202103527
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- Article
Novel benzenesulfonamide‐bearing pyrazoles and 1,2,4‐thiadiazoles as selective carbonic anhydrase inhibitors.
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- Archiv der Pharmazie, 2022, v. 355, n. 1, p. 1, doi. 10.1002/ardp.202100241
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- Article
Aromatic Sulfonamides including a Sulfonic Acid Tail: New Membrane Impermeant Carbonic Anhydrase Inhibitors for Targeting Selectively the Cancer-Associated Isoforms.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 1, p. 461, doi. 10.3390/ijms23010461
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- Article
Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 21, p. 11583, doi. 10.3390/ijms222111583
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- Article
Development of Novel Quinoline-Based Sulfonamides as Selective Cancer-Associated Carbonic Anhydrase Isoform IX Inhibitors.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 20, p. 11119, doi. 10.3390/ijms222011119
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- Article
Determination of intracellular protein–ligand binding affinity by competition binding in‐cell NMR.
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- Acta Crystallographica: Section D, Structural Biology, 2021, v. 77, n. 10, p. 1270, doi. 10.1107/S2059798321009037
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- Article
Carbonic Anhydrase IV Selective Inhibitors Counteract the Development of Colitis-Associated Visceral Pain in Rats.
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- Cells (2073-4409), 2021, v. 10, n. 10, p. 2540, doi. 10.3390/cells10102540
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Synthesis, Crystal Structure, Inhibitory Activity and Molecular Docking of Coumarins/Sulfonamides Containing Triazolyl Pyridine Moiety as Potent Selective Carbonic Anhydrase IX and XII Inhibitors.
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- Crystals (2073-4352), 2021, v. 11, n. 9, p. 1076, doi. 10.3390/cryst11091076
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- Article
The Glitazone Class of Drugs as Carbonic Anhydrase Inhibitors—A Spin-Off Discovery from Fragment Screening.
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- Molecules, 2021, v. 26, n. 10, p. 3010, doi. 10.3390/molecules26103010
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- Article
Role of Carbonic Anhydrase in Cerebral Ischemia and Carbonic Anhydrase Inhibitors as Putative Protective Agents.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 9, p. 5029, doi. 10.3390/ijms22095029
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- Article
Synthesis and Enantioselective Pharmacokinetic/Pharmacodynamic Analysis of New CNS-Active Sulfamoylphenyl Carbamate Derivatives.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 7, p. 3361, doi. 10.3390/ijms22073361
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- Article
Effect of Sulfonamides and Their Structurally Related Derivatives on the Activity of ι -Carbonic Anhydrase from Burkholderia territorii.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 2, p. 571, doi. 10.3390/ijms22020571
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Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors.
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- ChemMedChem, 2020, v. 15, n. 21, p. 2052, doi. 10.1002/cmdc.202000500
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Native mass spectrometry of human carbonic anhydrase I and its inhibitor complexes.
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- Journal of Biological Inorganic Chemistry (JBIC), 2020, v. 25, n. 7, p. 979, doi. 10.1007/s00775-020-01818-8
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- Article
Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment.
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- Metabolites (2218-1989), 2020, v. 10, n. 10, p. 412, doi. 10.3390/metabo10100412
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Structural and biochemical characterization of novel carbonic anhydrases from Phaeodactylum tricornutum.
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- Acta Crystallographica: Section D, Structural Biology, 2020, v. 76, n. 7, p. 676, doi. 10.1107/S2059798320007202
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- Article
The Effect of Substituted Benzene-Sulfonamides and Clinically Licensed Drugs on the Catalytic Activity of CynT2, a Carbonic Anhydrase Crucial for Escherichia coli Life Cycle.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 11, p. 4175, doi. 10.3390/ijms21114175
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Anion Inhibition Studies of the Beta-Carbonic Anhydrase from Escherichia coli.
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- Molecules, 2020, v. 25, n. 11, p. 2564, doi. 10.3390/molecules25112564
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- Article
Hypoxia-Activated Prodrug Derivatives of Carbonic Anhydrase Inhibitors in Benzenesulfonamide Series: Synthesis and Biological Evaluation.
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- Molecules, 2020, v. 25, n. 10, p. 2347, doi. 10.3390/molecules25102347
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- Article
Drug Screening in Human Cells by NMR Spectroscopy Allows the Early Assessment of Drug Potency.
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- Angewandte Chemie, 2020, v. 132, n. 16, p. 6597, doi. 10.1002/ange.201913436
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- Article
Drug Screening in Human Cells by NMR Spectroscopy Allows the Early Assessment of Drug Potency.
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- Angewandte Chemie International Edition, 2020, v. 59, n. 16, p. 6535, doi. 10.1002/anie.201913436
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- Article
Aryl-4,5-dihydro-1H-pyrazole-1-carboxamide Derivatives Bearing a Sulfonamide Moiety Show Single-digit Nanomolar-to-Subnanomolar Inhibition Constants against the Tumor-associated Human Carbonic Anhydrases IX and XII.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 7, p. 2621, doi. 10.3390/ijms21072621
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A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease.
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- International Journal of Molecular Sciences, 2019, v. 20, n. 19, p. 4724, doi. 10.3390/ijms20194724
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- Article
Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation.
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- Molecules, 2019, v. 24, n. 19, p. 3580, doi. 10.3390/molecules24193580
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- Article
Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights.
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- International Journal of Molecular Sciences, 2019, v. 20, n. 10, p. 2484, doi. 10.3390/ijms20102484
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- Article
β3-Adrenoreceptor Activity Limits Apigenin Efficacy in Ewing Sarcoma Cells: A Dual Approach to Prevent Cell Survival.
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- International Journal of Molecular Sciences, 2019, v. 20, n. 9, p. 2149, doi. 10.3390/ijms20092149
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- Article
Phosphorus versus Sulfur: Discovery of Benzenephosphonamidates as Versatile Sulfonamide‐Mimic Chemotypes Acting as Carbonic Anhydrase Inhibitors.
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- Chemistry - A European Journal, 2019, v. 25, n. 5, p. 1188, doi. 10.1002/chem.201805039
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- Article
Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies.
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- Chemistry - A European Journal, 2018, v. 24, n. 31, p. 7840, doi. 10.1002/chem.201800941
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Use of Innovative (Micro)Extraction Techniques to Characterise Harpagophytum procumbens Root and its Commercial Food Supplements.
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- Phytochemical Analysis, 2018, v. 29, n. 3, p. 233, doi. 10.1002/pca.2737
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- Article
Natural Polyphenols Selectively Inhibit β‐Carbonic Anhydrase from the Dandruff‐Producing Fungus <italic>Malassezia globosa</italic>: Activity and Modeling Studies.
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- ChemMedChem, 2018, v. 13, n. 8, p. 816, doi. 10.1002/cmdc.201800015
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Design and Comparative Evaluation of the Anticonvulsant Profile, Carbonic-Anhydrate Inhibition and Teratogenicity of Novel Carbamate Derivatives of Branched Aliphatic Carboxylic Acids with 4-Aminobenzensulfonamide.
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- Neurochemical Research, 2017, v. 42, n. 7, p. 1972, doi. 10.1007/s11064-017-2216-x
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Solution and Solid-State Analysis of Binding of 13-Substituted Berberine Analogues to Human Telomeric G-quadruplexes.
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- Chemistry - An Asian Journal, 2016, v. 11, n. 7, p. 1107, doi. 10.1002/asia.201600116
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- Article