Works by Nicolas Gouault

Results: 17

Synthesis and Potential Anti-Inflammatory Activity of Some Tetrahydrophthalazinones.
Published in:
Journal of Enzyme Inhibition & Medicinal Chemistry, 2004, v. 19, n. 6, p. 475, doi. 10.1080/14756360412331280536
By:
- Gouault, Nicolas;
- Pinel, Benoit;
- Cupif, Jean-Francois;
- Depince, Alexandra;
- Martin-Chouly, Corinne A. E.;
- Belleguic, Chantal;
- David, Michele
Publication type:
Article
Structural and molecular bases to IRE1 activity modulation.
Published in:
Biochemical Journal, 2021, v. 478, n. 15, p. 2953, doi. 10.1042/BCJ20200919
By:
- Langlais, Timothy;
- Pelizzari-Raymundo, Diana;
- Mahdizadeh, Sayyed Jalil;
- Gouault, Nicolas;
- Carreaux, Francois;
- Chevet, Eric;
- Eriksson, Leif A.;
- Guillory, Xavier
Publication type:
Article
Solid-phase synthesis and evaluation of libraries of substituted 4,5-dihydropyridazinones as vasodilator agents.
Published in:
Journal of Pharmacy & Pharmacology, 2004, v. 56, n. 8, p. 1029
By:
- Nicolas Gouault;
- Corinne A.E. Martin-Chouly;
- Claire Lugnier;
- Jean-François Cupif;
- Amaury Tonnelier;
- Frédéric Feger;
- Vincent Lagente;
- Michèle David
Publication type:
Article
Designed mono- and di-covalent inhibitors trap modeled functional motions for Trypanosoma cruzi proline racemase in crystallography.
Published in:
PLoS Neglected Tropical Diseases, 2018, v. 12, n. 10, p. 1, doi. 10.1371/journal.pntd.0006853
By:
- Amaral, Patricia de Aguiar;
- Autheman, Delphine;
- de Melo, Guilherme Dias;
- Gouault, Nicolas;
- Cupif, Jean-François;
- Goyard, Sophie;
- Dutra, Patricia;
- Coatnoan, Nicolas;
- Cosson, Alain;
- Monet, Damien;
- Saul, Frederick;
- Haouz, Ahmed;
- Uriac, Philippe;
- Blondel, Arnaud;
- Minoprio, Paola
Publication type:
Article
One‐Pot Double Cyclizations Involving an Aza‐Prins Process.
Published in:
European Journal of Organic Chemistry, 2024, v. 27, n. 39, p. 1, doi. 10.1002/ejoc.202400617
By:
- Gouault, Nicolas;
- Roydor, Maxence;
- Renault, Jacques;
- Banik, Swarnayu;
- Subba Reddy, B. V.;
- Lalli, Claudia
Publication type:
Article
Three different approaches to C-H bond functionalization in the synthesis of antitumor alkaloids rhazinilam, rhazinal and rhazinicine.
Published in:
ARKIVOC: Online Journal of Organic Chemistry, 2010, p. 247
By:
- Le Floc'h, Delphine;
- Gouault, Nicolas;
- David, Michèle;
- van de Weghe, Pierre
Publication type:
Article
Irreversible inhibitors of the proline racemase unveil innovative mechanism of action as antibacterial agents against Clostridioides difficile.
Published in:
Chemical Biology & Drug Design, 2022, v. 99, n. 4, p. 513, doi. 10.1111/cbdd.14005
By:
- Gateau, Cécile;
- Melo, Guilherme D.;
- Uriac, Philippe;
- Tasseau, Olivier;
- Renault, Jacques;
- Blondel, Arnaud;
- Gouault, Nicolas;
- Barbut, Frédéric;
- Minoprio, Paola
Publication type:
Article
Synthesis of Novel Cyclic Nitrones with gem‐Difluoroalkyl Side Chains Through Cascade Reactions.
Published in:
European Journal of Organic Chemistry, 2020, v. 2020, n. 35, p. 5741, doi. 10.1002/ejoc.202000972
By:
- Soulieman, Ali;
- Ibrahim, Rima;
- Barakat, Zeinab;
- Gouault, Nicolas;
- Roisnel, Thierry;
- Boustie, Joel;
- Grée, René;
- Hachem, Ali
Publication type:
Article
Structure Activity Relationship Studies around DB18 , a Potent and Selective Inhibitor of CLK Kinases.
Published in:
Molecules, 2022, v. 27, n. 19, p. 6149, doi. 10.3390/molecules27196149
By:
- Brahmaiah, Dabbugoddu;
- Bhavani, Anagani Kanaka Durga;
- Aparna, Pasula;
- Kumar, Nangunoori Sampath;
- Solhi, Hélène;
- Le Guevel, Rémy;
- Baratte, Blandine;
- Robert, Thomas;
- Ruchaud, Sandrine;
- Bach, Stéphane;
- Jadav, Surender Singh;
- Reddy, Chada Raji;
- Mosset, Paul;
- Gouault, Nicolas;
- Levoin, Nicolas;
- Grée, René
Publication type:
Article
Isolation and Structure Identification of Novel Brominated Diketopiperazines from Nocardia ignorata--A Lichen-Associated Actinobacterium.
Published in:
Molecules, 2017, v. 22, n. 3, p. 371, doi. 10.3390/molecules22030371
By:
- Noël, Alba;
- Ferron, Solenn;
- Rouaud, Isabelle;
- Gouault, Nicolas;
- Hurvois, Jean-Pierre;
- Tomasi, Sophie
Publication type:
Article
On the Formation of a Protic Ionic Liquid in Nature.
Published in:
Angewandte Chemie, 2014, v. 126, n. 44, p. 11956, doi. 10.1002/ange.201404402
By:
- Chen, Li;
- Mullen, Genevieve E.;
- Le Roch, Myriam;
- Cassity, Cody G.;
- Gouault, Nicolas;
- Fadamiro, Henry Y.;
- Barletta, Robert E.;
- O'Brien, Richard A.;
- Sykora, Richard E.;
- Stenson, Alexandra C.;
- West, Kevin N.;
- Horne, Howard E.;
- Hendrich, Jeffrey M.;
- Xiang, Kang Rui;
- Davis, James H.
Publication type:
Article
Aza‐Prins Cyclization on Ketones to Access Piperidines with Tetrasubstituted Carbon Stereocenters.
Published in:
Advanced Synthesis & Catalysis, 2024, v. 366, n. 1, p. 31, doi. 10.1002/adsc.202301116
By:
- Bergounioux, Alexandre;
- Lhotellier, Romane;
- Roisnel, Thierry;
- Gouault, Nicolas;
- Argouarch, Gilles;
- Lalli, Claudia
Publication type:
Article
Combined Approaches for Drug Design Points the Way to Novel Proline Racemase Inhibitor Candidates to Fight Chagas’ Disease.
Published in:
PLoS ONE, 2013, v. 8, n. 4, p. 1, doi. 10.1371/journal.pone.0060955
By:
- Berneman, Armand;
- Montout, Lory;
- Goyard, Sophie;
- Chamond, Nathalie;
- Cosson, Alain;
- d’Archivio, Simon;
- Gouault, Nicolas;
- Uriac, Philippe;
- Blondel, Arnaud;
- Minoprio, Paola
Publication type:
Article
Reactivity of N-Boc-Protected Amino-Ynones in the Presence of Zinc Chloride: Formation of Acetylenic Cyclic Imines and Their Palladium Complexes.
Published in:
European Journal of Organic Chemistry, 2015, v. 2015, n. 22, p. 4868, doi. 10.1002/ejoc.201500569
By:
- Vu, Huy‐Dinh;
- Renault, Jacques;
- Roisnel, Thierry;
- Robert, Clémence;
- Jéhan, Philippe;
- Gouault, Nicolas;
- Uriac, Philippe
Publication type:
Article
Methanesulfonic Acid Mediated Cyclization and Meyer-Schuster Rearrangement of γ-Amino-ynones: Access to Enantiopure Pyrrolidine Exocyclic Vinylogous Amides.
Published in:
European Journal of Organic Chemistry, 2014, v. 2014, n. 21, p. 4506, doi. 10.1002/ejoc.201402336
By:
- Vu, Huy‐Dinh;
- Renault, Jacques;
- Roisnel, Thierry;
- Gouault, Nicolas;
- Uriac, Philippe
Publication type:
Article
From Aspartic Acid to Dihydropyridone-2-carboxylates: Access to Enantiopure 6-Substituted 4-Oxo- and 4-Hydroxypipecolic Acid Derivatives.
Published in:
European Journal of Organic Chemistry, 2013, v. 2013, n. 29, p. 6677, doi. 10.1002/ejoc.201300812
By:
- Vu, Huy‐Dinh;
- Renault, Jacques;
- Toupet, Loïc;
- Uriac, Philippe;
- Gouault, Nicolas
Publication type:
Article
On the Formation of a Protic Ionic Liquid in Nature.
Published in:
Angewandte Chemie International Edition, 2014, v. 53, n. 44, p. 11762, doi. 10.1002/anie.201404402
By:
- Chen, Li;
- Mullen, Genevieve E.;
- Le Roch, Myriam;
- Cassity, Cody G.;
- Gouault, Nicolas;
- Fadamiro, Henry Y.;
- Barletta, Robert E.;
- O'Brien, Richard A.;
- Sykora, Richard E.;
- Stenson, Alexandra C.;
- West, Kevin N.;
- Horne, Howard E.;
- Hendrich, Jeffrey M.;
- Xiang, Kang Rui;
- Davis, James H.
Publication type:
Article