Works by Nicolas Gouault

Results: 17

Solid-phase synthesis and evaluation of libraries of substituted 4,5-dihydropyridazinones as vasodilator agents.

Published in:

Journal of Pharmacy & Pharmacology, 2004, v. 56, n. 8, p. 1029

By:

Nicolas Gouault;
Corinne A.E. Martin-Chouly;
Claire Lugnier;
Jean-François Cupif;
Amaury Tonnelier;
Frédéric Feger;
Vincent Lagente;
Michèle David

Publication type:

Article

Aza‐Prins Cyclization on Ketones to Access Piperidines with Tetrasubstituted Carbon Stereocenters.

Published in:

Advanced Synthesis & Catalysis, 2024, v. 366, n. 1, p. 31, doi. 10.1002/adsc.202301116

By:

Bergounioux, Alexandre;
Lhotellier, Romane;
Roisnel, Thierry;
Gouault, Nicolas;
Argouarch, Gilles;
Lalli, Claudia

Publication type:

Article

Structure Activity Relationship Studies around DB18 , a Potent and Selective Inhibitor of CLK Kinases.

Published in:

Molecules, 2022, v. 27, n. 19, p. 6149, doi. 10.3390/molecules27196149

By:

Brahmaiah, Dabbugoddu;
Bhavani, Anagani Kanaka Durga;
Aparna, Pasula;
Kumar, Nangunoori Sampath;
Solhi, Hélène;
Le Guevel, Rémy;
Baratte, Blandine;
Robert, Thomas;
Ruchaud, Sandrine;
Bach, Stéphane;
Jadav, Surender Singh;
Reddy, Chada Raji;
Mosset, Paul;
Gouault, Nicolas;
Levoin, Nicolas;
Grée, René

Publication type:

Article

Isolation and Structure Identification of Novel Brominated Diketopiperazines from Nocardia ignorata--A Lichen-Associated Actinobacterium.

Published in:

Molecules, 2017, v. 22, n. 3, p. 371, doi. 10.3390/molecules22030371

By:

Noël, Alba;
Ferron, Solenn;
Rouaud, Isabelle;
Gouault, Nicolas;
Hurvois, Jean-Pierre;
Tomasi, Sophie

Publication type:

Article

Reactivity of N-Boc-Protected Amino-Ynones in the Presence of Zinc Chloride: Formation of Acetylenic Cyclic Imines and Their Palladium Complexes.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 22, p. 4868, doi. 10.1002/ejoc.201500569

By:

Vu, Huy‐Dinh;
Renault, Jacques;
Roisnel, Thierry;
Robert, Clémence;
Jéhan, Philippe;
Gouault, Nicolas;
Uriac, Philippe

Publication type:

Article

Methanesulfonic Acid Mediated Cyclization and Meyer-Schuster Rearrangement of γ-Amino-ynones: Access to Enantiopure Pyrrolidine Exocyclic Vinylogous Amides.

Published in:

European Journal of Organic Chemistry, 2014, v. 2014, n. 21, p. 4506, doi. 10.1002/ejoc.201402336

By:

Vu, Huy‐Dinh;
Renault, Jacques;
Roisnel, Thierry;
Gouault, Nicolas;
Uriac, Philippe

Publication type:

Article

From Aspartic Acid to Dihydropyridone-2-carboxylates: Access to Enantiopure 6-Substituted 4-Oxo- and 4-Hydroxypipecolic Acid Derivatives.

Published in:

European Journal of Organic Chemistry, 2013, v. 2013, n. 29, p. 6677, doi. 10.1002/ejoc.201300812

By:

Vu, Huy‐Dinh;
Renault, Jacques;
Toupet, Loïc;
Uriac, Philippe;
Gouault, Nicolas

Publication type:

Article

On the Formation of a Protic Ionic Liquid in Nature.

Published in:

Angewandte Chemie International Edition, 2014, v. 53, n. 44, p. 11762, doi. 10.1002/anie.201404402

By:

Chen, Li;
Mullen, Genevieve E.;
Le Roch, Myriam;
Cassity, Cody G.;
Gouault, Nicolas;
Fadamiro, Henry Y.;
Barletta, Robert E.;
O'Brien, Richard A.;
Sykora, Richard E.;
Stenson, Alexandra C.;
West, Kevin N.;
Horne, Howard E.;
Hendrich, Jeffrey M.;
Xiang, Kang Rui;
Davis, James H.

Publication type:

Article

Irreversible inhibitors of the proline racemase unveil innovative mechanism of action as antibacterial agents against Clostridioides difficile.

Published in:

Chemical Biology & Drug Design, 2022, v. 99, n. 4, p. 513, doi. 10.1111/cbdd.14005

By:

Gateau, Cécile;
Melo, Guilherme D.;
Uriac, Philippe;
Tasseau, Olivier;
Renault, Jacques;
Blondel, Arnaud;
Gouault, Nicolas;
Barbut, Frédéric;
Minoprio, Paola

Publication type:

Article

One‐Pot Double Cyclizations Involving an Aza‐Prins Process.

Published in:

European Journal of Organic Chemistry, 2024, v. 27, n. 39, p. 1, doi. 10.1002/ejoc.202400617

By:

Gouault, Nicolas;
Roydor, Maxence;
Renault, Jacques;
Banik, Swarnayu;
Subba Reddy, B. V.;
Lalli, Claudia

Publication type:

Article

Synthesis of Novel Cyclic Nitrones with gem‐Difluoroalkyl Side Chains Through Cascade Reactions.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 35, p. 5741, doi. 10.1002/ejoc.202000972

By:

Soulieman, Ali;
Ibrahim, Rima;
Barakat, Zeinab;
Gouault, Nicolas;
Roisnel, Thierry;
Boustie, Joel;
Grée, René;
Hachem, Ali

Publication type:

Article

On the Formation of a Protic Ionic Liquid in Nature.

Published in:

Angewandte Chemie, 2014, v. 126, n. 44, p. 11956, doi. 10.1002/ange.201404402

By:

Chen, Li;
Mullen, Genevieve E.;
Le Roch, Myriam;
Cassity, Cody G.;
Gouault, Nicolas;
Fadamiro, Henry Y.;
Barletta, Robert E.;
O'Brien, Richard A.;
Sykora, Richard E.;
Stenson, Alexandra C.;
West, Kevin N.;
Horne, Howard E.;
Hendrich, Jeffrey M.;
Xiang, Kang Rui;
Davis, James H.

Publication type:

Article

Structural and molecular bases to IRE1 activity modulation.

Published in:

Biochemical Journal, 2021, v. 478, n. 15, p. 2953, doi. 10.1042/BCJ20200919

By:

Langlais, Timothy;
Pelizzari-Raymundo, Diana;
Mahdizadeh, Sayyed Jalil;
Gouault, Nicolas;
Carreaux, Francois;
Chevet, Eric;
Eriksson, Leif A.;
Guillory, Xavier

Publication type:

Article

Combined Approaches for Drug Design Points the Way to Novel Proline Racemase Inhibitor Candidates to Fight Chagas’ Disease.

Published in:

PLoS ONE, 2013, v. 8, n. 4, p. 1, doi. 10.1371/journal.pone.0060955

By:

Berneman, Armand;
Montout, Lory;
Goyard, Sophie;
Chamond, Nathalie;
Cosson, Alain;
d’Archivio, Simon;
Gouault, Nicolas;
Uriac, Philippe;
Blondel, Arnaud;
Minoprio, Paola

Publication type:

Article

Synthesis and Potential Anti-Inflammatory Activity of Some Tetrahydrophthalazinones.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2004, v. 19, n. 6, p. 475, doi. 10.1080/14756360412331280536

By:

Gouault, Nicolas;
Pinel, Benoit;
Cupif, Jean-Francois;
Depince, Alexandra;
Martin-Chouly, Corinne A. E.;
Belleguic, Chantal;
David, Michele

Publication type:

Article

Designed mono- and di-covalent inhibitors trap modeled functional motions for Trypanosoma cruzi proline racemase in crystallography.

Published in:

PLoS Neglected Tropical Diseases, 2018, v. 12, n. 10, p. 1, doi. 10.1371/journal.pntd.0006853

By:

Amaral, Patricia de Aguiar;
Autheman, Delphine;
de Melo, Guilherme Dias;
Gouault, Nicolas;
Cupif, Jean-François;
Goyard, Sophie;
Dutra, Patricia;
Coatnoan, Nicolas;
Cosson, Alain;
Monet, Damien;
Saul, Frederick;
Haouz, Ahmed;
Uriac, Philippe;
Blondel, Arnaud;
Minoprio, Paola

Publication type:

Article

Three different approaches to C-H bond functionalization in the synthesis of antitumor alkaloids rhazinilam, rhazinal and rhazinicine.

Published in:

ARKIVOC: Online Journal of Organic Chemistry, 2010, p. 247

By:

Le Floc'h, Delphine;
Gouault, Nicolas;
David, Michèle;
van de Weghe, Pierre

Publication type:

Article