Works matching AU Nada, Hossam
Results: 19
Identification of 1H-purine-2,6-dione derivative as a potential SARS-CoV-2 main protease inhibitor: molecular docking, dynamic simulations, and energy calculations.
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- PeerJ, 2022, p. 1, doi. 10.7717/peerj.14120
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- Article
4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological studies.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 994, doi. 10.1080/14756366.2022.2055553
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- Article
Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 629, doi. 10.1080/14756366.2018.1446432
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- Article
Cantharidin-Based Verbenone Derivatives as a Novel Insecticide against Plutella xylostella : Design, Synthesis, Insecticidal Activity Evaluation, and 3D QSAR Study.
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- Biomolecules (2218-273X), 2023, v. 13, n. 8, p. 1272, doi. 10.3390/biom13081272
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- Article
Development of New Meridianin/Leucettine-Derived Hybrid Small Molecules as Nanomolar Multi-Kinase Inhibitors with Antitumor Activity.
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- Biomedicines, 2021, v. 9, n. 9, p. 1131, doi. 10.3390/biomedicines9091131
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- Article
New insights into protein–protein interaction modulators in drug discovery and therapeutic advance.
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- Signal Transduction & Targeted Therapy, 2024, v. 9, n. 1, p. 1, doi. 10.1038/s41392-024-02036-3
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- Article
Natural products as IL‐6 inhibitors for inflammatory diseases: Synthetic and SAR perspective.
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- Medicinal Research Reviews, 2024, v. 44, n. 4, p. 1683, doi. 10.1002/med.22022
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- Article
Small Molecule c-KIT Inhibitors for the Treatment of Gastrointestinal Stromal Tumors: A Review on Synthesis, Design Strategies, and Structure–Activity Relationship (SAR).
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- International Journal of Molecular Sciences, 2023, v. 24, n. 11, p. 9450, doi. 10.3390/ijms24119450
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- Article
Identification of Novel and Potent Indole-Based Benzenesulfonamides as Selective Human Carbonic Anhydrase II Inhibitors: Design, Synthesis, In Vitro, and In Silico Studies.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 5, p. 2540, doi. 10.3390/ijms23052540
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- Article
The Journey of DDR1 and DDR2 Kinase Inhibitors as Rising Stars in the Fight Against Cancer.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 12, p. 6535, doi. 10.3390/ijms22126535
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- Article
Integration of Hybridization Strategies in Pyridine–Urea Scaffolds for Novel Anticancer Agents: Design, Synthesis, and Mechanistic Insights.
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- Molecules, 2023, v. 28, n. 13, p. 4952, doi. 10.3390/molecules28134952
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- Article
Structure Activity Relationship of Key Heterocyclic Anti-Angiogenic Leads of Promising Potential in the Fight against Cancer.
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- Molecules, 2021, v. 26, n. 3, p. 553, doi. 10.3390/molecules26030553
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- Article
Melatonin Analogues Potently Inhibit MAO-B and Protect PC12 Cells against Oxidative Stress.
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- Antioxidants, 2021, v. 10, n. 10, p. 1604, doi. 10.3390/antiox10101604
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- Article
Small Molecules in Parkinson's Disease Therapy: From Dopamine Pathways to New Emerging Targets.
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- Pharmaceuticals (14248247), 2024, v. 17, n. 12, p. 1688, doi. 10.3390/ph17121688
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- Article
Design, Synthesis and Biological Evaluation of Novel MDH Inhibitors Targeting Tumor Microenvironment.
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- Pharmaceuticals (14248247), 2023, v. 16, n. 5, p. 683, doi. 10.3390/ph16050683
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- Article
Hit Identification of a Novel Quinazoline Sulfonamide as a Promising EphB3 Inhibitor: Design, Virtual Combinatorial Library, Synthesis, Biological Evaluation, and Docking Simulation Studies.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 12, p. 1247, doi. 10.3390/ph14121247
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- Article
Chalcone‐based benzenesulfonamides as potent and selective inhibitors for human carbonic anhydrase II: Design, synthesis, in vitro, and in silico studies.
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- Archiv der Pharmazie, 2024, v. 357, n. 11, p. 1, doi. 10.1002/ardp.202400069
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- Article
A novel indole derivative, 2‐{3‐[1‐(benzylsulfonyl)piperidin‐4‐yl]‐2‐methyl‐1H‐indol‐1‐yl}‐1‐(pyrrolidin‐1‐yl)ethenone, suppresses hedgehog signaling and drug‐resistant tumor growth
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- Archiv der Pharmazie, 2024, v. 357, n. 10, p. 1, doi. 10.1002/ardp.202400218
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- Article
Discovery and optimization of natural-based nanomolar c-Kit inhibitors via in silico and in vitro studies.
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- Journal of Biomolecular Structure & Dynamics, 2023, v. 41, n. 21, p. 11904, doi. 10.1080/07391102.2022.2164061
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- Article