Works matching AU Musilek, Kamil


Results: 134
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    Development of versatile and potent monoquaternary reactivators of acetylcholinesterase.

    Published in:
    Archives of Toxicology, 2021, v. 95, n. 3, p. 985, doi. 10.1007/s00204-021-02981-w
    By:
    • Gorecki, Lukas;
    • Hepnarova, Vendula;
    • Karasova, Jana Zdarova;
    • Hrabinova, Martina;
    • Courageux, Charlotte;
    • Dias, José;
    • Kucera, Tomas;
    • Kobrlova, Tereza;
    • Muckova, Lubica;
    • Prchal, Lukas;
    • Malinak, David;
    • Jun, Daniel;
    • Musilek, Kamil;
    • Worek, Franz;
    • Nachon, Florian;
    • Soukup, Ondrej;
    • Korabecny, Jan
    Publication type:
    Article
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    Takrin a jeho deriváty v terapii Alzheimerovy choroby.

    Published in:
    Czech & Slovak Pharmacy / Česká a Slovenská Farmacie, 2012, v. 61, n. 5, p. 210
    By:
    • Korábeãný, Jan;
    • Špilovská, Katarína;
    • Benek, Ondřiej;
    • Musílek, Kamil;
    • Soukup, Ondřiej;
    • Kuča, Kamil
    Publication type:
    Article
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    Methylacridinium and its Cholinergic Properties.

    Published in:
    Neurotoxicity Research, 2009, v. 16, n. 4, p. 372, doi. 10.1007/s12640-009-9071-8
    By:
    • Soukup, Ondrej;
    • Proska, Jan;
    • Binder, Jiri;
    • Karasova, Jana Zdarova;
    • Tobin, Gunnar;
    • Jun, Daniel;
    • Marek, Jan;
    • Musílek, Kamil;
    • Fusek, Josef;
    • Kuca, Kamil
    Publication type:
    Article
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    Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 410, doi. 10.1080/14756366.2020.1871336
    By:
    • Oleksak, Patrik;
    • Psotka, Miroslav;
    • Vancurova, Marketa;
    • Sapega, Olena;
    • Bieblova, Jana;
    • Reinis, Milan;
    • Rysanek, David;
    • Mikyskova, Romana;
    • Chalupova, Katarina;
    • Malinak, David;
    • Svobodova, Jana;
    • Andrys, Rudolf;
    • Rehulkova, Helena;
    • Skopek, Vojtech;
    • Ngoc Lam, Pham;
    • Bartek, Jiri;
    • Hodny, Zdenek;
    • Musilek, Kamil
    Publication type:
    Article
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    Pyridinium-2-carbaldoximes with quinolinium carboxamide moiety are simultaneous reactivators of acetylcholinesterase and butyrylcholinesterase inhibited by nerve agent surrogates.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 437, doi. 10.1080/14756366.2020.1869954
    By:
    • Lee, Hyun Myung;
    • Andrys, Rudolf;
    • Jonczyk, Jakub;
    • Kim, Kyuneun;
    • Vishakantegowda, Avinash G.;
    • Malinak, David;
    • Skarka, Adam;
    • Schmidt, Monika;
    • Vaskova, Michaela;
    • Latka, Kamil;
    • Bajda, Marek;
    • Jung, Young-Sik;
    • Malawska, Barbara;
    • Musilek, Kamil
    Publication type:
    Article
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    Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 478, doi. 10.1080/14756366.2019.1710501
    By:
    • Malinak, David;
    • Dolezal, Rafael;
    • Hepnarova, Vendula;
    • Hozova, Miroslava;
    • Andrys, Rudolf;
    • Bzonek, Petr;
    • Racakova, Veronika;
    • Korabecny, Jan;
    • Gorecki, Lukas;
    • Mezeiova, Eva;
    • Psotka, Miroslav;
    • Jun, Daniel;
    • Kuca, Kamil;
    • Musilek, Kamil
    Publication type:
    Article
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    Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer's disease therapy.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 479, doi. 10.1080/14756366.2018.1545766
    By:
    • Pachón-Angona, Irene;
    • Refouvelet, Bernard;
    • Andrýs, Rudolf;
    • Martin, Helène;
    • Luzet, Vincent;
    • Iriepa, Isabel;
    • Moraleda, Ignacio;
    • Diez-Iriepa, Daniel;
    • Oset-Gasque, María-Jesús;
    • Marco-Contelles, José;
    • Musilek, Kamil;
    • Ismaili, Lhassane
    Publication type:
    Article
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    Acetylcholinesterase Inhibition of Diversely Functionalized Quinolinones for Alzheimer's Disease Therapy.

    Published in:
    International Journal of Molecular Sciences, 2020, v. 21, n. 11, p. 3913, doi. 10.3390/ijms21113913
    By:
    • Bautista-Aguilera, Óscar M.;
    • Ismaili, Lhassane;
    • Chioua, Mourad;
    • Andrys, Rudolf;
    • Schmidt, Monika;
    • Bzonek, Petr;
    • Martínez-Grau, María Ángeles;
    • Beadle, Christopher D.;
    • Vetman, Tatiana;
    • López-Muñoz, Francisco;
    • Iriepa, Isabel;
    • Refouvelet, Bernard;
    • Musilek, Kamil;
    • Marco-Contelles, José
    Publication type:
    Article
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    Benzothiazolyl Ureas are Low Micromolar and Uncompetitive Inhibitors of 17β-HSD10 with Implications to Alzheimer's Disease Treatment.

    Published in:
    International Journal of Molecular Sciences, 2020, v. 21, n. 6, p. 2059, doi. 10.3390/ijms21062059
    By:
    • Schmidt, Monika;
    • Benek, Ondrej;
    • Vinklarova, Lucie;
    • Hrabinova, Martina;
    • Zemanova, Lucie;
    • Chribek, Matej;
    • Kralova, Vendula;
    • Hroch, Lukas;
    • Dolezal, Rafael;
    • Lycka, Antonin;
    • Prchal, Lukas;
    • Jun, Daniel;
    • Aitken, Laura;
    • Gunn-Moore, Frank;
    • Kuca, Kamil;
    • Musilek, Kamil
    Publication type:
    Article
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