Works by Murarka, Sandip


Results: 23
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    Identification of pyrazolopyridazinones as PDEδ inhibitors.

    Published in:
    Nature Communications, 2016, v. 7, n. 4, p. 11360, doi. 10.1038/ncomms11360
    By:
    • Papke, Björn;
    • Murarka, Sandip;
    • Vogel, Holger A;
    • Martín-Gago, Pablo;
    • Kovacevic, Marija;
    • Truxius, Dina C;
    • Fansa, Eyad K;
    • Ismail, Shehab;
    • Zimmermann, Gunther;
    • Heinelt, Kaatje;
    • Schultz-Fademrecht, Carsten;
    • Al Saabi, Alaa;
    • Baumann, Matthias;
    • Nussbaumer, Peter;
    • Wittinghofer, Alfred;
    • Waldmann, Herbert;
    • Bastiaens, Philippe I.H.
    Publication type:
    Article
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    A PDE6δ-KRas Inhibitor Chemotype with up to Seven H-Bonds and Picomolar Affinity that Prevents Efficient Inhibitor Release by Arl2.

    Published in:
    Angewandte Chemie International Edition, 2017, v. 56, n. 9, p. 2423, doi. 10.1002/anie.201610957
    By:
    • Martín‐Gago, Pablo;
    • Fansa, Eyad K.;
    • Klein, Christian H.;
    • Murarka, Sandip;
    • Janning, Petra;
    • Schürmann, Marc;
    • Metz , Malte;
    • Ismail, Shehab;
    • Schultz‐Fademrecht, Carsten;
    • Baumann, Matthias;
    • Bastiaens, Philippe I. H.;
    • Wittinghofer, Alfred;
    • Waldmann, Herbert
    Publication type:
    Article
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