Works by Meyer-Almes, Franz-Josef
Results: 32
The cis-state of an azobenzene photoswitch is stabilized through specific interactions with a protein surface.
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- Journal of Molecular Recognition, 2015, v. 28, n. 3, p. 201, doi. 10.1002/jmr.2415
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- Article
Thermodynamics of ligand binding to histone deacetylase like amidohydrolase from Bordetella/Alcaligenes.
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- Journal of Molecular Recognition, 2014, v. 27, n. 3, p. 160, doi. 10.1002/jmr.2345
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- Article
Substrate specificity and function of acetylpolyamine amidohydrolases from Pseudomonas aeruginosa.
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- BMC Biochemistry, 2016, v. 17, p. 1, doi. 10.1186/s12858-016-0063-z
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- Article
3‐Chloro‐5‐Substituted‐1,2,4‐Thiadiazoles (TDZs) as Selective and Efficient Protein Thiol Modifiers.
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- ChemBioChem, 2022, v. 23, n. 21, p. 1, doi. 10.1002/cbic.202200417
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- Article
Assessment of Tractable Cysteines for Covalent Targeting by Screening Covalent Fragments.
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- ChemBioChem, 2021, v. 22, n. 4, p. 743, doi. 10.1002/cbic.202000700
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- Article
Design and synthesis of peptides as stabilizers of histone deacetylase 4.
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- Journal of Peptide Science, 2024, v. 30, n. 9, p. 1, doi. 10.1002/psc.3603
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- Article
Kinetically selective and potent inhibitors of HDAC8.
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- Biological Chemistry, 2019, v. 400, n. 6, p. 733, doi. 10.1515/hsz-2018-0363
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- Article
Azobenzene switch with a long-lived cis-state to photocontrol the enzyme activity of a histone deacetylase-like amidohydrolase.
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- Biological Chemistry, 2014, v. 395, n. 4, p. 401, doi. 10.1515/hsz-2013-0246
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- Article
HDAC4 Inhibitors with Cyclic Linker and Non‐hydroxamate Zinc Binding Group: Design, Synthesis, HDAC Screening and in vitro Cytotoxicity evaluation.
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- ChemistrySelect, 2021, v. 6, n. 26, p. 6748, doi. 10.1002/slct.202102061
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- Article
Discrimination between conformational selection and induced fit protein-ligand binding using Integrated Global Fit analysis.
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- European Biophysics Journal, 2016, v. 45, n. 3, p. 245, doi. 10.1007/s00249-015-1090-1
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- Article
Determination of the binding mechanism of histone deacetylase inhibitors.
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- Chemical Biology & Drug Design, 2019, v. 93, n. 6, p. 1214, doi. 10.1111/cbdd.13449
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- Article
Impact of binding mechanism on selective inhibition of histone deacetylase isoforms.
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- Chemical Biology & Drug Design, 2017, v. 90, n. 6, p. 1215, doi. 10.1111/cbdd.13041
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- Article
Class IIa HDACs repressive activities on MEF2-depedent transcription are associated with poor prognosis of ER<sup>+</sup> breast tumors.
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- FASEB Journal, 2013, v. 27, n. 3, p. 942, doi. 10.1096/fj.12-209346
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- Article
Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine‐2,5‐dione Hybrids as Potential Antitumor Agents.
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- ChemMedChem, 2020, v. 15, n. 19, p. 1813, doi. 10.1002/cmdc.202000458
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- Article
Potent and Selective Non-hydroxamate Histone Deacetylase 8 Inhibitors.
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- ChemMedChem, 2016, v. 11, n. 23, p. 2598, doi. 10.1002/cmdc.201600528
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- Article
Highly Ligand Efficient and Selective N-2-(Thioethyl)picolinamide Histone Deacetylase Inhibitors Inspired by the Natural Product Psammaplin A.
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- ChemMedChem, 2013, v. 8, n. 1, p. 149, doi. 10.1002/cmdc.201200450
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- Article
Rapid Determination of Kinetic Constants for Slow-Binding Inhibitors and Inactivators of Human Histone Deacetylase 8.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 11, p. 5593, doi. 10.3390/ijms25115593
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- Article
Design, Synthesis, and Biological Evaluation of Novel Quinazolin-4(3H)-One-Based Histone Deacetylase 6 (HDAC6) Inhibitors for Anticancer Activity.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 13, p. 11044, doi. 10.3390/ijms241311044
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- Article
Methionine 274 Is Not the Determining Factor for Selective Inhibition of Histone Deacetylase 8 (HDAC8) by L-Shaped Inhibitors.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 19, p. 11775, doi. 10.3390/ijms231911775
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- Article
Significance of Five-Membered Heterocycles in Human Histone Deacetylase Inhibitors.
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- Molecules, 2023, v. 28, n. 15, p. 5686, doi. 10.3390/molecules28155686
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- Article
Non-Hydroxamate Zinc-Binding Groups as Warheads for Histone Deacetylases.
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- Molecules, 2021, v. 26, n. 17, p. 5151, doi. 10.3390/molecules26175151
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- Article
Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 10, p. 1032, doi. 10.3390/ph14101032
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- Article
A fluorescence lifetime-based binding assay for acetylpolyamine amidohydrolases from Pseudomonas aeruginosa using a [1,3]dioxolo[4,5- f][1,3]benzodioxole (DBD) ligand probe.
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- Analytical & Bioanalytical Chemistry, 2014, v. 406, n. 20, p. 4889, doi. 10.1007/s00216-014-7886-5
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- Article
Compact, cost-efficient microfluidics-based stopped-flow device.
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- Analytical & Bioanalytical Chemistry, 2011, v. 399, n. 3, p. 1117, doi. 10.1007/s00216-010-4446-5
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- Article
Switching the Switch: Ligand Induced Disulfide Formation in HDAC8.
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- Chemistry - A European Journal, 2020, v. 26, n. 58, p. 13249, doi. 10.1002/chem.202001712
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- Article
Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX.
- Published in:
- eLife, 2024, p. 1, doi. 10.7554/eLife.101401
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- Article
Transcriptomic and genomic studies classify NKL54 as a histone deacetylase inhibitor with indirect influence on MEF2-dependent transcription.
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- Nucleic Acids Research, 2022, v. 50, n. 5, p. 2566, doi. 10.1093/nar/gkac081
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- Article
Inhibitor-mediated stabilization of the conformational structure of a histone deacetylase-like amidohydrolase.
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- FEBS Journal, 2007, v. 274, n. 14, p. 3578, doi. 10.1111/j.1742-4658.2007.05887.x
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- Article
A Fluorescence-Lifetime-Based Binding Assay for Class IIa Histone Deacetylases.
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- Chemistry - A European Journal, 2017, v. 23, n. 13, p. 3107, doi. 10.1002/chem.201605140
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- Article
Novel fluorescence based receptor binding assay method for receptors lacking ligand conjugates with preserved affinity: Study on estrogen receptor α.
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- Biopolymers, 2003, v. 72, n. 4, p. 256, doi. 10.1002/bip.10402
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- Article
The Proapoptotic Influenza A Virus Protein PB1-F2 Forms a Nonselective Ion Channel.
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- PLoS ONE, 2010, v. 5, n. 6, p. 1, doi. 10.1371/journal.pone.0011112
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- Article
The catalytic domain of free or ligand bound histone deacetylase 4 occurs in solution predominantly in closed conformation.
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- Protein Science: A Publication of the Protein Society, 2024, v. 33, n. 3, p. 1, doi. 10.1002/pro.4917
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- Article