Katalytische Synthesen N-heterocyclischer Inone und Indione durch In-situ-Aktivierung von Carbonsäuren mit Oxalylchlorid.
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- Angewandte Chemie, 2011, v. 123, n. 44, p. 10632, doi. 10.1002/ange.201103296
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Works matching AU Merkul, Eugen
Results: 18
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Dreikomponentensynthese von Indionen durch eine Glyoxylierungs-Stephens-Castro-Kupplungs-Sequenz.
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- Angewandte Chemie, 2011, v. 123, n. 13, p. 3023, doi. 10.1002/ange.201007194
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- Article
3
One-Pot Synthesis of Camalexins and 3,3′-Biindoles by the Masuda Borylation-Suzuki Arylation (MBSA) Sequence.
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- European Journal of Organic Chemistry, 2013, v. 2013, n. 21, p. 4564, doi. 10.1002/ejoc.201300133
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- Article
4
Concise Syntheses of Meridianins by Carbonylative Alkynylation and a Four-Component Pyrimidine SynthesisThis work was supported by the Deutsche Forschungsgemeinschaft (Graduiertenkolleg 850), by the Fonds der Chemischen Industrie, and by the Dr.-Otto-Röhm Gedächtnisstiftung. We thank Dr. Dieter Dorsch, Merck KGaA, Darmstadt, for providing screening data of the meridianins and derivatives in kinase inhibition assays, BASF AG for the generous donation of chemicals, and Michaela Schmitt for experimental assistance.
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- Angewandte Chemie International Edition, 2005, v. 44, n. 42, p. 6951, doi. 10.1002/anie.200501703
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5
Consecutive One-Pot Sonogashira-Glaser Coupling Sequence - Direct Preparation of Symmetrical Diynes by Sequential Pd/Cu Catalysis.
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- European Journal of Organic Chemistry, 2011, v. 2011, n. 2, p. 238, doi. 10.1002/ejoc.201001472
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- Article
6
One-Pot Three-Component Synthesis of 3-Halofurans and 3-Chloro-4-iodofurans.
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- European Journal of Organic Chemistry, 2006, v. 2006, n. 13, p. 2991, doi. 10.1002/ejoc.200600225
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- Article
7
Preclinical targeting of liver fibrosis with a <sup>89</sup>Zr-labeled Fibrobody® directed against platelet derived growth factor receptor-β.
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- European Journal of Nuclear Medicine & Molecular Imaging, 2024, v. 51, n. 12, p. 3545, doi. 10.1007/s00259-024-06785-9
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- Article
8
In Vivo Characterization of Platinum(II)-Based Linker Technology for the Development of Antibody--Drug Conjugates: Taking Advantage of Dual Labeling with <sup>195m</sup>Pt and <sup>89</sup>Zr.
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- Journal of Nuclear Medicine, 2018, v. 59, n. 7, p. 1146, doi. 10.2967/jnumed.117.206672
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- Article
9
Consecutive Three-Component Synthesis of Ynones by Decarbonylative Sonogashira Coupling.
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- Chemistry - A European Journal, 2009, v. 15, n. 20, p. 5006, doi. 10.1002/chem.200900119
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- Article
10
First platinum(II)-based metal-organic linker technology (Lx®) for a plug-and-play development of antibody-drug conjugates (ADCs).
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- Expert Opinion on Drug Delivery, 2019, v. 16, n. 8, p. 783, doi. 10.1080/17425247.2019.1645118
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- Article
11
Titelbild: An Efficient Conjugation Approach for Coupling Drugs to Native Antibodies via the Pt<sup>II</sup> Linker Lx for Improved Manufacturability of Antibody–Drug Conjugates (Angew. Chem. 6/2021).
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- Angewandte Chemie, 2021, v. 133, n. 6, p. 2741, doi. 10.1002/ange.202016966
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- Article
12
An Efficient Conjugation Approach for Coupling Drugs to Native Antibodies via the Pt<sup>II</sup> Linker Lx for Improved Manufacturability of Antibody–Drug Conjugates.
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- Angewandte Chemie, 2021, v. 133, n. 6, p. 3045, doi. 10.1002/ange.202011593
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- Article
13
Cover Picture: An Efficient Conjugation Approach for Coupling Drugs to Native Antibodies via the Pt<sup>II</sup> Linker Lx for Improved Manufacturability of Antibody–Drug Conjugates (Angew. Chem. Int. Ed. 6/2021).
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- Angewandte Chemie International Edition, 2021, v. 60, n. 6, p. 2709, doi. 10.1002/anie.202016966
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- Article
14
An Efficient Conjugation Approach for Coupling Drugs to Native Antibodies via the Pt<sup>II</sup> Linker Lx for Improved Manufacturability of Antibody–Drug Conjugates.
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- Angewandte Chemie International Edition, 2021, v. 60, n. 6, p. 3008, doi. 10.1002/anie.202011593
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- Publication type:
- Article
15
Consecutive Three-Component Synthesis of 3-(Hetero)Aryl-1H-pyrazoles with Propynal Diethylacetal as a Three-Carbon Building Block.
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- Molecules, 2011, v. 16, n. 11, p. 9340, doi. 10.3390/molecules16119340
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- Article
16
Kurze Meridianin-Synthesen durch carbonylierende Alkinylierung; eine Vierkomponenten-Pyrimidin-Synthese.
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- Angewandte Chemie, 2005, v. 117, n. 42, p. 7112, doi. 10.1002/ange.200501703
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- Publication type:
- Article
17
Catalytic Syntheses of N-Heterocyclic Ynones and Ynediones by In Situ Activation of Carboxylic Acids with Oxalyl Chloride.
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- Angewandte Chemie International Edition, 2011, v. 50, n. 44, p. 10448, doi. 10.1002/anie.201103296
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- Publication type:
- Article
18
Three-Component Synthesis of Ynediones by a Glyoxylation/Stephens-Castro Coupling Sequence.
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- Angewandte Chemie International Edition, 2011, v. 50, n. 13, p. 2966, doi. 10.1002/anie.201007194
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- Article