Works by Masurier, Nicolas

Results: 21

Helical Oligomers of Thiazole-Based γ-Amino Acids: Synthesis and Structural Studies.

Published in:

Angewandte Chemie, 2013, v. 125, n. 23, p. 6122, doi. 10.1002/ange.201302106

By:

Mathieu, Loïc;
Legrand, Baptiste;
Deng, Cheng;
Vezenkov, Lubomir;
Wenger, Emmanuel;
Didierjean, Claude;
Amblard, Muriel;
Averlant ‐ Petit, Marie ‐ Christine;
Masurier, Nicolas;
Lisowski, Vincent;
Martinez, Jean;
Maillard, Ludovic T.

Publication type:

Article

1,3‐Diazepine: A privileged scaffold in medicinal chemistry.

Published in:

Medicinal Research Reviews, 2021, v. 41, n. 4, p. 2247, doi. 10.1002/med.21795

By:

Malki, Yohan;
Martinez, Jean;
Masurier, Nicolas

Publication type:

Article

Inhibitors of kallikrein‐related peptidases: An overview.

Published in:

Medicinal Research Reviews, 2018, v. 38, n. 2, p. 655, doi. 10.1002/med.21451

By:

Masurier, Nicolas;
Arama, Dominique P.;
El Amri, Chahrazade;
Lisowski, Vincent

Publication type:

Article

Synthesis of Peptide–Adenine Conjugates as a New Tool for Monitoring Protease Activity.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 1, p. 176, doi. 10.1002/ejoc.201801490

By:

Masurier, Nicolas;
Soualmia, Feryel;
Sanchez, Pierre;
Lefort, Valérie;
Roué, Mia;
Maillard, Ludovic T.;
Subra, Gilles;
Percot, Aline;
El Amri, Chahrazade

Publication type:

Article

Synthesis of Thieno[3,2- e][1,4]diazepin-2-ones: Application of an Uncatalysed Pictet-Spengler Reaction.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 32, p. 7146, doi. 10.1002/ejoc.201500943

By:

Denoyelle, Séverine;
Tambutet, Guillaume;
Masurier, Nicolas;
Maillard, Ludovic T.;
Martinez, Jean;
Lisowski, Vincent

Publication type:

Article

Cross-Claisen Condensation of N-Fmoc-Amino Acids -- A Short Route to Heterocyclic γ-Amino Acids.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 10, p. 2262, doi. 10.1002/ejoc.201500012

By:

Mathieu, Loïc;
Bonnel, Clément;
Masurier, Nicolas;
Maillard, Ludovic T.;
Martinez, Jean;
Lisowski, Vincent

Publication type:

Article

C9/12 Ribbon-Like Structures in Hybrid Peptides Alternating α- and Thiazole-Based γ-Amino Acids.

Published in:

Chemistry - A European Journal, 2017, v. 23, n. 69, p. 17584, doi. 10.1002/chem.201704001

By:

Bonnel, Clément;
Legrand, Baptiste;
Simon, Matthieu;
Martinez, Jean;
Bantignies, Jean‐Louis;
Kang, Young Kee;
Wenger, Emmanuel;
Hoh, Francois;
Masurier, Nicolas;
Maillard, Ludovic T.

Publication type:

Article

1,3‐Diazepine Derivatives: Strategies for Synthesis.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 21, p. 1, doi. 10.1002/ejoc.202100492

By:

Malki, Yohan;
Maillard, Ludovic T.;
Masurier, Nicolas

Publication type:

Article

Solid-Supported Synthesis and 5- HT7/5- HT1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H)-one.

Published in:

Chemical Biology & Drug Design, 2015, v. 86, n. 4, p. 697, doi. 10.1111/cbdd.12539

By:

Grychowska, Katarzyna;
Masurier, Nicolas;
Verdié, Pascal;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Martinez, Jean;
Pawłowski, Maciej;
Subra, Gilles;
Zajdel, Paweł

Publication type:

Article

Thiazole-Based γ-Building Blocks as Reverse-Turn Mimetic to Design a Gramicidin S Analogue: Conformational and Biological Evaluation.

Published in:

Chemistry - A European Journal, 2014, v. 20, n. 22, p. 6713, doi. 10.1002/chem.201402190

By:

Legrand, Baptiste;
Mathieu, Loïc;
Lebrun, Aurélien;
Andriamanarivo, Soahary;
Lisowski, Vincent;
Masurier, Nicolas;
Zirah, Séverine;
Kang, Young Kee;
Martinez, Jean;
Maillard, Ludovic T.

Publication type:

Article

A New Highly Versatile Handle for Chemistry on a Solid Support: The Pipecolic Linker.

Published in:

Chemistry - A European Journal, 2012, v. 18, n. 37, p. 11536, doi. 10.1002/chem.201201452

By:

Masurier, Nicolas;
Zajdel, Paweł;
Verdié, Pascal;
Pawłowski, Maciej;
Amblard, Muriel;
Martinez, Jean;
Subra, Gilles

Publication type:

Article

A New Highly Versatile Handle for Chemistry on a Solid Support: The Pipecolic Linker.

Published in:

Chemistry - A European Journal, 2010, v. 16, n. 25, p. 7547, doi. 10.1002/chem.201000313

By:

Zajdel, Paweł;
Nomezine, Gaël;
Masurier, Nicolas;
Amblard, Muriel;
Pawłowski, Maciej;
Martinez, Jean;
Subra, Gilles

Publication type:

Article

PROteolysis TArgetting Chimeras (PROTACs) Strategy Applied to Kinases: Recent Advances.

Published in:

Advanced Therapeutics, 2020, v. 3, n. 11, p. 1, doi. 10.1002/adtp.202000148

By:

Feral, Anthony;
Laconde, Guillaume;
Amblard, Muriel;
Masurier, Nicolas

Publication type:

Article

Novel N-Arylmethyl-aniline/chalcone hybrids as potential VEGFR inhibitors: synthesis, biological evaluations, and molecular dynamic simulations.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2278022

By:

Haffez, Hesham;
Elsayed, Nosaiba A.;
Ahmed, Marwa F.;
Fatahala, Samar S.;
Khaleel, Eman F.;
Badi, Rehab Mustafa;
Elkaeed, Eslam B.;
El Hassab, Mahmoud A.;
Hammad, Sherif F.;
Eldehna, Wagdy M.;
Masurier, Nicolas;
El-Haggar, Radwan

Publication type:

Article

Design, synthesis, molecular modeling and biological evaluation of novel Benzoxazole-Benzamide conjugates via a 2-Thioacetamido linker as potential anti-proliferative agents, VEGFR-2 inhibitors and apoptotic inducers.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1587, doi. 10.1080/14756366.2022.2081844

By:

Eissa, Ibrahim H.;
El-Haggar, Radwan;
Dahab, Mohammed A.;
Ahmed, Marwa F.;
Mahdy, Hazem A.;
Alsantali, Reem I.;
Elwan, Alaa;
Masurier, Nicolas;
Fatahala, Samar S.

Publication type:

Article

Imidazopyridine-fused [1,3]diazepinones: modulations of positions 2 to 4 and their impacts on the anti-melanoma activity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 935, doi. 10.1080/14756366.2020.1748024

By:

Baccon-Sollier, Paul Le;
Malki, Yohan;
Maye, Morgane;
Ali, Lamiaa M. A.;
Lichon, Laure;
Cuq, Pierre;
Vincent, Laure-Anaïs;
Masurier, Nicolas

Publication type:

Article

Novel hydrazone‐isatin derivatives as potential EGFR inhibitors: Synthesis and in vitro pharmacological profiling.

Published in:

Archiv der Pharmazie, 2023, v. 356, n. 9, p. 1, doi. 10.1002/ardp.202300244

By:

Ahmed, Marwa F.;
El‐Haggar, Radwan;
Almalki, Atiah H.;
Abdullah, Omeima;
El Hassab, Mahmoud A.;
Masurier, Nicolas;
Hammad, Sherif F.

Publication type:

Article

4-Substituted Thieno[3,2- d ]pyrimidines as Dual-Stage Antiplasmodial Derivatives.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 7, p. N.PAG, doi. 10.3390/ph15070820

By:

Lagardère, Prisca;
Mustière, Romain;
Amanzougaghene, Nadia;
Hutter, Sébastien;
Franetich, Jean-François;
Azas, Nadine;
Vanelle, Patrice;
Verhaeghe, Pierre;
Primas, Nicolas;
Mazier, Dominique;
Masurier, Nicolas;
Lisowski, Vincent

Publication type:

Article

AAZTA-Derived Chelators for the Design of Innovative Radiopharmaceuticals with Theranostic Applications.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 2, p. 234, doi. 10.3390/ph15020234

By:

Fersing, Cyril;
Masurier, Nicolas;
Rubira, Léa;
Deshayes, Emmanuel;
Lisowski, Vincent

Publication type:

Article

Thienopyrimidine: A Promising Scaffold to Access Anti-Infective Agents.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 1, p. 35, doi. 10.3390/ph15010035

By:

Lagardère, Prisca;
Fersing, Cyril;
Masurier, Nicolas;
Lisowski, Vincent

Publication type:

Article

Helical Oligomers of Thiazole-Based γ-Amino Acids: Synthesis and Structural Studies.

Published in:

Angewandte Chemie International Edition, 2013, v. 52, n. 23, p. 6006, doi. 10.1002/anie.201302106

By:

Mathieu, Loïc;
Legrand, Baptiste;
Deng, Cheng;
Vezenkov, Lubomir;
Wenger, Emmanuel;
Didierjean, Claude;
Amblard, Muriel;
Averlant‐Petit, Marie‐Christine;
Masurier, Nicolas;
Lisowski, Vincent;
Martinez, Jean;
Maillard, Ludovic T.

Publication type:

Article

Works by Masurier, Nicolas

Helical Oligomers of Thiazole-Based γ-Amino Acids: Synthesis and Structural Studies.

1,3‐Diazepine: A privileged scaffold in medicinal chemistry.

Inhibitors of kallikrein‐related peptidases: An overview.

Synthesis of Peptide–Adenine Conjugates as a New Tool for Monitoring Protease Activity.

Synthesis of Thieno[3,2- e][1,4]diazepin-2-ones: Application of an Uncatalysed Pictet-Spengler Reaction.

Cross-Claisen Condensation of N-Fmoc-Amino Acids -- A Short Route to Heterocyclic γ-Amino Acids.

C<sub>9/12</sub> Ribbon-Like Structures in Hybrid Peptides Alternating α- and Thiazole-Based γ-Amino Acids.

1,3‐Diazepine Derivatives: Strategies for Synthesis.

Solid-Supported Synthesis and 5- HT<sub>7</sub>/5- HT<sub>1A</sub> Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H)-one.

Thiazole-Based γ-Building Blocks as Reverse-Turn Mimetic to Design a Gramicidin S Analogue: Conformational and Biological Evaluation.

A New Highly Versatile Handle for Chemistry on a Solid Support: The Pipecolic Linker.

A New Highly Versatile Handle for Chemistry on a Solid Support: The Pipecolic Linker.

PROteolysis TArgetting Chimeras (PROTACs) Strategy Applied to Kinases: Recent Advances.

Novel N-Arylmethyl-aniline/chalcone hybrids as potential VEGFR inhibitors: synthesis, biological evaluations, and molecular dynamic simulations.

Design, synthesis, molecular modeling and biological evaluation of novel Benzoxazole-Benzamide conjugates via a 2-Thioacetamido linker as potential anti-proliferative agents, VEGFR-2 inhibitors and apoptotic inducers.

Imidazopyridine-fused [1,3]diazepinones: modulations of positions 2 to 4 and their impacts on the anti-melanoma activity.

Novel hydrazone‐isatin derivatives as potential EGFR inhibitors: Synthesis and in vitro pharmacological profiling.

4-Substituted Thieno[3,2- d ]pyrimidines as Dual-Stage Antiplasmodial Derivatives.

AAZTA-Derived Chelators for the Design of Innovative Radiopharmaceuticals with Theranostic Applications.

Thienopyrimidine: A Promising Scaffold to Access Anti-Infective Agents.

Helical Oligomers of Thiazole-Based γ-Amino Acids: Synthesis and Structural Studies.