Works matching AU Marco‐Contelles, José


Results: 105
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    Synthesis of New Statin Derivatives.

    Published in:
    ChemistrySelect, 2021, v. 6, n. 47, p. 13633, doi. 10.1002/slct.202103544
    By:
    • Chioua, Mourad;
    • Marco‐Contelles, José
    Publication type:
    Article
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    Automated Synthesis of New Quinoxalinetacrines.

    Published in:
    ChemistrySelect, 2020, v. 5, n. 21, p. 6491, doi. 10.1002/slct.202001593
    By:
    • Bautista‐Aguilera, Óscar M.;
    • Ismaili, Lhassane;
    • Chioua, Mourad;
    • Iriepa, Isabel;
    • Ángeles Martinez‐Grau, Marìa;
    • Beadle, Christopher D.;
    • Vetman, Tatiana;
    • López‐Muñoz, Francisco;
    • Marco‐Contelles, José
    Publication type:
    Article
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    Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer's disease therapy.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 479, doi. 10.1080/14756366.2018.1545766
    By:
    • Pachón-Angona, Irene;
    • Refouvelet, Bernard;
    • Andrýs, Rudolf;
    • Martin, Helène;
    • Luzet, Vincent;
    • Iriepa, Isabel;
    • Moraleda, Ignacio;
    • Diez-Iriepa, Daniel;
    • Oset-Gasque, María-Jesús;
    • Marco-Contelles, José;
    • Musilek, Kamil;
    • Ismaili, Lhassane
    Publication type:
    Article
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    Synthesis and biological assessment of KojoTacrines as new agents for Alzheimer's disease therapy.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 163, doi. 10.1080/14756366.2018.1538136
    By:
    • Dgachi, Youssef;
    • Martin, Hélène;
    • Malek, Rim;
    • Jun, Daniel;
    • Janockova, Jana;
    • Sepsova, Vendula;
    • Soukup, Ondrej;
    • Iriepa, Isabel;
    • Moraleda, Ignacio;
    • Maalej, Emna;
    • Carreiras, M. Carmo;
    • Refouvelet, Bernard;
    • Chabchoub, Fakher;
    • Marco-Contelles, José;
    • Ismaili, Lhassane
    Publication type:
    Article
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    Multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer's disease: design, synthesis, biochemical evaluation, ADMET, molecular modeling, and QSAR analysis of novel donepezil-pyridyl hybrids.

    Published in:
    Drug Design, Development & Therapy, 2014, v. 8, p. 1893, doi. 10.2147/DDDT.S69258
    By:
    • Bautista-Aguilera, Oscar M.;
    • Esteban, Gerard;
    • Chioua, Mourad;
    • Nikolic, Katarina;
    • Agbaba, Danica;
    • Moraleda, Ignacio;
    • Iriepa, Isabel;
    • Soriano, Elena;
    • Samadi, Abdelouahid;
    • Unzeta, Mercedes;
    • Marco-Contelles, José
    Publication type:
    Article
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    The Proof-of-Concept of MBA121, a Tacrine–Ferulic Acid Hybrid, for Alzheimer's Disease Therapy.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 15, p. 12254, doi. 10.3390/ijms241512254
    By:
    • Rodríguez-Ruiz, Emelina R.;
    • Herrero-Labrador, Raquel;
    • Fernández-Fernández, Ana P.;
    • Serrano-Masa, Julia;
    • Martínez-Montero, José A.;
    • González-Nieto, Daniel;
    • Hana-Vaish, Mayuri;
    • Benchekroun, Mohamed;
    • Ismaili, Lhassane;
    • Marco-Contelles, José;
    • Martínez-Murillo, Ricardo
    Publication type:
    Article
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    Acetylcholinesterase Inhibition of Diversely Functionalized Quinolinones for Alzheimer's Disease Therapy.

    Published in:
    International Journal of Molecular Sciences, 2020, v. 21, n. 11, p. 3913, doi. 10.3390/ijms21113913
    By:
    • Bautista-Aguilera, Óscar M.;
    • Ismaili, Lhassane;
    • Chioua, Mourad;
    • Andrys, Rudolf;
    • Schmidt, Monika;
    • Bzonek, Petr;
    • Martínez-Grau, María Ángeles;
    • Beadle, Christopher D.;
    • Vetman, Tatiana;
    • López-Muñoz, Francisco;
    • Iriepa, Isabel;
    • Refouvelet, Bernard;
    • Musilek, Kamil;
    • Marco-Contelles, José
    Publication type:
    Article
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    Synthesis of AZA Analogues of TSAO.

    Published in:
    Nucleosides, Nucleotides & Nucleic Acids, 2003, v. 22, n. 5-8, p. 939, doi. 10.1081/NCN-120022690
    By:
    • Nguyen Van Nhien, Albert;
    • Tomassi, Cyrille;
    • Len, Christophe;
    • Marco-Contelles, José Luis;
    • Postel, Denis
    Publication type:
    Article
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    Multi-Target Directed Donepezil-Like Ligands for Alzheimer's Disease.

    Published in:
    Frontiers in Neuroscience, 2016, p. 1, doi. 10.3389/fnins.2016.00205
    By:
    • Unzeta, Mercedes;
    • Esteban, Gerard;
    • Bolea, Irene;
    • Fogel, Wieslawa A.;
    • Ramsay, Rona R.;
    • Youdim, Moussa B. H.;
    • Tipton, Keith F.;
    • Marco-Contelles, José;
    • Grilli, Massimo;
    • Min-Yu Sun
    Publication type:
    Article
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    Synthesis of new 7-azabicyclo[2.2.1]heptane derivatives.

    Published in:
    ARKIVOC: Online Journal of Organic Chemistry, 2010, p. 56
    By:
    • Marco-Contelles, José;
    • Gómez-Sánchez, Elena;
    • Samadi, Abdelouahid;
    • Soriano, Elena;
    • Valderas, Carolina;
    • Álvarez-Pérez, Mónica;
    • Carreiras, María do Carmo
    Publication type:
    Article
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    Updating the CSIC Reaction (2003–2020).

    Published in:
    European Journal of Organic Chemistry, 2021, v. 2021, n. 8, p. 1229, doi. 10.1002/ejoc.202001330
    By:
    • Dobrydnev, Alexey V.;
    • Marco‐Contelles, José
    Publication type:
    Article
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    Synthesis and Biological Assessment of Racemic Benzochromenopyrimidinimines as Antioxidant, Cholinesterase, and Aβ<sub>1−42</sub> Aggregation Inhibitors for Alzheimer's Disease Therapy.

    Published in:
    ChemMedChem, 2016, v. 11, n. 12, p. 1318, doi. 10.1002/cmdc.201500539
    By:
    • Dgachi, Youssef;
    • Ismaili, Lhassane;
    • Knez, Damijan;
    • Benchekroun, Mohamed;
    • Martin, Hélène;
    • Szałaj, Natalia;
    • Wehle, Sarah;
    • Bautista‐Aguilera, Oscar M.;
    • Luzet, Vincent;
    • Bonnet, Alexandre;
    • Malawska, Barbara;
    • Gobec, Stanislav;
    • Chioua, Mourad;
    • Decker, Michael;
    • Chabchoub, Fakher;
    • Marco‐Contelles, José
    Publication type:
    Article
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    Novel Tacrine-Grafted Ugi Adducts as Multipotent Anti-Alzheimer Drugs: A Synthetic Renewal in Tacrine-Ferulic Acid Hybrids.

    Published in:
    ChemMedChem, 2015, v. 10, n. 3, p. 523, doi. 10.1002/cmdc.201402409
    By:
    • Benchekroun, Mohamed;
    • Bartolini, Manuela;
    • Egea, Javier;
    • Romero, Alejandro;
    • Soriano, Elena;
    • Pudlo, Marc;
    • Luzet, Vincent;
    • Andrisano, Vincenza;
    • Jimeno, María‐Luisa;
    • López, Manuela G.;
    • Wehle, Sarah;
    • Gharbi, Tijani;
    • Refouvelet, Bernard;
    • de Andrés, Lucía;
    • Herrera‐Arozamena, Clara;
    • Monti, Barbara;
    • Bolognesi, Maria Laura;
    • Rodríguez‐Franco, María Isabel;
    • Decker, Michael;
    • Marco‐Contelles, José
    Publication type:
    Article
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