Works by Majer, Pavel

Results: 28

Sphinganine-Like Biogenesis of ( E)-1-Nitropentadec-1-ene in Termite Soldiers of the Genus Prorhinotermes.

Published in:

ChemBioChem, 2014, v. 15, n. 4, p. 533, doi. 10.1002/cbic.201300665

By:

Jirošová, Anna;
Majer, Pavel;
Jančařík, Andrej;
Dolejšová, Klára;
Tykva, Richard;
Šobotník, Jan;
Jiroš, Pavel;
Hanus, Robert

Publication type:

Article

High-affinity Near-infrared Fluorescent Small-molecule Contrast Agents for In Vivo Imaging of Prostate-specific Membrane Antigen.

Published in:

Molecular Imaging, 2005, v. 4, n. 4, p. 448, doi. 10.2310/7290.2005.05163

By:

Humblet, Valerie;
Lapidus, Rena;
Williams, Larry R.;
Tsukamoto, Takashi;
Rojas, Camilo;
Majer, Pavel;
Hin, Bunda;
Ohnishi, Shunsuke;
De Grand, Alec M.;
Zaheer, Atif;
Renze, Jürgen T.;
Nakayama, Akira;
Slusher, Barbara S.;
Frangioni, John V.

Publication type:

Article

Targeting glutamine metabolism enhances tumor-specific immunity by modulating suppressive myeloid cells.

Published in:

2020

By:

Min-Hee Oh;
Im-Hong Sun;
Liang Zhao;
Leone, Robert D.;
Im-Meng Sun;
Wei Xu;
Collins, Samuel L.;
Tam, Ada J.;
Blosser, Richard L.;
Patel, Chirag H.;
Englert, Judson M.;
Arwood, Matthew L.;
Jiayu Wen;
Yee Chan-Li;
Tenora,, Lukáš;
Majer, Pavel;
Rais, Rana;
Slusher, Barbara S.;
Horton, Maureen R.;
Powell, Jonathan D.

Publication type:

journal article

Structure-based specificity mapping of secreted aspartic proteases of Candida parapsilosis, Candida albicans, and Candida tropicalis using peptidomimetic inhibitors and homology modeling.

Published in:

Biological Chemistry, 2006, v. 387, n. 9, p. 1247, doi. 10.1515/BC.2006.154

By:

Majer, Filip;
Pavlíčková, Libuše;
Majer, Pavel;
Hradilek, Martin;
Dolejší, Elena;
Hrušková-Heidingsfeldová, Olga;
Pichová, Iva

Publication type:

Article

Homology modeling and SAR analysis of Schistosoma japonicum cathepsin D (SjCD) with statin inhibitors identify a unique active site steric barrier with potential for the design of specific inhibitors.

Published in:

Biological Chemistry, 2005, v. 386, n. 4, p. 339, doi. 10.1515/BC.2005.041

By:

Caffrey, Conor R.;
Placha, Lenka;
Barinka, Cyril;
Hradilek, Martin;
Dostal, Jiř;í;
Sajid, Mohammed;
McKerrow, James H.;
Majer, Pavel;
Konvalinka, Jan;
Vondrášek, Jiří

Publication type:

Article

Selectivity of Hydroxamate- and Difluoromethyloxadiazole-Based Inhibitors of Histone Deacetylase 6 In Vitro and in Cells.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 5, p. 4720, doi. 10.3390/ijms24054720

By:

Ptacek, Jakub;
Snajdr, Ivan;
Schimer, Jiri;
Kutil, Zsofia;
Mikesova, Jana;
Baranova, Petra;
Havlinova, Barbora;
Tueckmantel, Werner;
Majer, Pavel;
Kozikowski, Alan;
Barinka, Cyril

Publication type:

Article

Synthesis and In Vitro Evaluation of C-7 and C-8 Luteolin Derivatives as Influenza Endonuclease Inhibitors.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 14, p. 7735, doi. 10.3390/ijms22147735

By:

Reiberger, Robert;
Radilová, Kateřina;
Kráľ, Michal;
Zima, Václav;
Majer, Pavel;
Brynda, Jiří;
Dračínský, Martin;
Konvalinka, Jan;
Kožíšek, Milan;
Machara, Aleš

Publication type:

Article

Mapping of CaM, S100A1 and PIP2-Binding Epitopes in the Intracellular N- and C-Termini of TRPM4.

Published in:

International Journal of Molecular Sciences, 2020, v. 21, n. 12, p. 4323, doi. 10.3390/ijms21124323

By:

Bousova, Kristyna;
Barvik, Ivan;
Herman, Petr;
Hofbauerová, Kateřina;
Monincova, Lenka;
Majer, Pavel;
Zouharova, Monika;
Vetyskova, Veronika;
Postulkova, Klara;
Vondrasek, Jiri

Publication type:

Article

JHU-2545 preferentially shields salivary glands and kidneys during PSMA-targeted imaging.

Published in:

European Journal of Nuclear Medicine & Molecular Imaging, 2025, v. 52, n. 5, p. 1631, doi. 10.1007/s00259-024-07044-7

By:

Nedelcovych, Michael T.;
Dash, Ranjeet P.;
Wu, Ying;
Choi, Eun Yong;
Lapidus, Rena S.;
Majer, Pavel;
Jančařík, Andrej;
Abou, Diane;
Penet, Marie-France;
Nikolopoulou, Anastasia;
Amor-Coarasa, Alex;
Babich, John;
Thorek, Daniel L.;
Rais, Rana;
Kratochwil, Clemens;
Slusher, Barbara S.

Publication type:

Article

Substrate binding and specificity of rhomboid intramembrane protease revealed by substrate-peptide complex structures.

Published in:

EMBO Journal, 2014, v. 33, n. 20, p. 2408, doi. 10.15252/embj.201489367

By:

Zoll, Sebastian;
Stanchev, Stancho;
Began, Jakub;
Škerle, Jan;
Lepšík, Martin;
Peclinovská, Lucie;
Majer, Pavel;
Strisovsky, Kvido

Publication type:

Article

Ranking Power of the SQM/COSMO Scoring Function on Carbonic Anhydrase II–Inhibitor Complexes.

Published in:

ChemPhysChem, 2018, v. 19, n. 7, p. 873, doi. 10.1002/cphc.201701104

By:

Pecina, Adam;
Brynda, Jiří;
Vrzal, Lukáš;
Gnanasekaran, Ramachandran;
Hořejší, Magdalena;
Eyrilmez, Saltuk M.;
Řezáč, Jan;
Lepšík, Martin;
Řezáčová, Pavlína;
Hobza, Pavel;
Majer, Pavel;
Veverka, Václav;
Fanfrlík, Jindřich

Publication type:

Article

Smells Like Home: Chemically Mediated Co-Habitation of Two Termite Species in a Single Nest.

Published in:

Journal of Chemical Ecology, 2016, v. 42, n. 10, p. 1070, doi. 10.1007/s10886-016-0756-1

By:

Jirošová, Anna;
Sillam-Dussès, David;
Kyjaková, Pavlína;
Kalinová, Blanka;
Dolejšová, Klára;
Jančařík, Andrej;
Majer, Pavel;
Cristaldo, Paulo;
Hanus, Robert

Publication type:

Article

Structure-based subsite specificity mapping of human cathepsin D using statine-based inhibitors.

Published in:

Protein Science: A Publication of the Protein Society, 1997, v. 6, n. 7, p. 1458, doi. 10.1002/pro.5560060710

By:

Majer, Pavel;
Collins, Jack R.;
Gulnik, Sergei V.;
Erickson, John W.

Publication type:

Article

Engineering the substrate specificity of rhizopuspepsin: The role of Asp 77 of fungal aspartic proteinases in facilitating the cleavage of oligopeptide substrates with lysine in P<sub>1</sub>.

Published in:

Protein Science: A Publication of the Protein Society, 1995, v. 4, n. 4, p. 689, doi. 10.1002/pro.5560040409

By:

Todd Lowther, W.;
Dunn, Ben M.;
Majer, Pavel

Publication type:

Article

Triggering HIV polyprotein processing by light using rapid photodegradation of a tight-binding protease inhibitor.

Published in:

Nature Communications, 2015, v. 6, n. 3, p. 6461, doi. 10.1038/ncomms7461

By:

Schimer, Jiří;
Pávová, Marcela;
Anders, Maria;
Pachl, Petr;
Šácha, Pavel;
Cígler, Petr;
Weber, Jan;
Majer, Pavel;
Řezáčová, Pavlína;
Kräusslich, Hans-Georg;
Müller, Barbara;
Konvalinka, Jan

Publication type:

Article

iBodies: Modular Synthetic Antibody Mimetics Based on Hydrophilic Polymers Decorated with Functional Moieties.

Published in:

Angewandte Chemie, 2016, v. 128, n. 7, p. 2402, doi. 10.1002/ange.201508642

By:

Šácha, Pavel;
Knedlík, Tomáš;
Schimer, Jiří;
Tykvart, Jan;
Parolek, Jan;
Navrátil, Václav;
Dvořáková, Petra;
Sedlák, František;
Ulbrich, Karel;
Strohalm, Jiří;
Majer, Pavel;
Šubr, Vladimír;
Konvalinka, Jan

Publication type:

Article

DNA-linked Inhibitor Antibody Assay (DIANA) for sensitive and selective enzyme detection and inhibitor screening.

Published in:

Nucleic Acids Research, 2017, v. 45, n. 2, p. 1, doi. 10.1093/nar/gkw853

By:

Navrátil, Václav;
Schimer, Jiří;
Tykvart, Jan;
Knedlík, Tomáš;
Vik, Viktor;
Majer, Pavel;
Konvalinka, Jan;
Šácha, Pavel

Publication type:

Article

Structure of glutamate carboxypeptidase II, a drug target in neuronal damage and prostate cancer.

Published in:

EMBO Journal, 2006, v. 25, n. 6, p. 1375, doi. 10.1038/sj.emboj.7600969

By:

Mesters, Jeroen R.;
Barinka, Cyril;
Weixing Li;
Tsukamoto, Takashi;
Majer, Pavel;
Slusher, Barbara S.;
Konvalinka, Jan;
Hilgenfeld, Rolf

Publication type:

Article

The unraveling of substrate specificity of histone deacetylase 6 domains using acetylome peptide microarrays and peptide libraries.

Published in:

FASEB Journal, 2019, v. 33, n. 3, p. 4035, doi. 10.1096/fj.201801680R

By:

Kutil, Zsofia;
Skultetyova, Lubica;
Rauh, David;
Meleshin, Marat;
Snajdr, Ivan;
Novakova, Zora;
Mikesova, Jana;
Pavlicek, Jiri;
Hadzima, Martin;
Baranova, Petra;
Havlinova, Barbora;
Majer, Pavel;
Schutkowski, Mike;
Barinka, Cyril

Publication type:

Article

Biochemical characterization of human glutamate carboxypeptidase III.

Published in:

Journal of Neurochemistry, 2007, v. 101, n. 3, p. 682, doi. 10.1111/j.1471-4159.2006.04341.x

By:

Hlouchová, Klára;
Bařinka, Cyril;
Klusák, Vojtěch;
Šácha, Pavel;
Mlčochová, Petra;
Majer, Pavel;
RulíŠek, Lubomír;
Konvalinka, Jan

Publication type:

Article

Peptide inhibitors of HIV-1 and HIV-2 proteases: a comparative study.

Published in:

Leukemia (08876924), 1997, v. 11, p. 120

By:

PICHOVÁ, Iva;
WEBER, Jan;
LITERA, Jaroslav;
KONVALINKA, Jan;
VONDRÁSEK, JiřI;
SOUČEK, Milan;
STROP, Petr;
MAJER, Pavel;
HEUSER, Anke M.;
KRAEUSSLICH, Hans-Georg

Publication type:

Article

A gut-restricted glutamate carboxypeptidase II inhibitor reduces monocytic inflammation and improves preclinical colitis.

Published in:

Science Translational Medicine, 2023, v. 15, n. 708, p. 1, doi. 10.1126/scitranslmed.abn7491

By:

Peters, Diane E.;
Norris, Lauren D.;
Tenora, Lukáš;
Šnajdr, Ivan;
Ponti, András K.;
Zhu, Xiaolei;
Sakamoto, Shinji;
Veeravalli, Vijayabhaskar;
Pradhan, Manisha;
Alt, Jesse;
Thomas, Ajit G.;
Majer, Pavel;
Rais, Rana;
McDonald, Christine;
Slusher, Barbara S.

Publication type:

Article

Front Cover: 3'‐Dehydroxypurpurogallin‐4‐Carboxamides as Influenza A Endonuclease Inhibitors: Synthesis, Structure‐Activity Relationship Analysis, and Structural Characterization of Protein Complex (ChemMedChem 3/2025).

Published in:

ChemMedChem, 2025, v. 20, n. 3, p. 1, doi. 10.1002/cmdc.202580301

By:

Kráľ, Michal;
Kotačka, Tomáš;
Reiberger, Róbert;
Panýrková, Gabriela;
Radilová, Kateřina;
Osifová, Zuzana;
Flieger, Miroslav;
Konvalinka, Jan;
Majer, Pavel;
Kožíšek, Milan;
Machara, Aleš

Publication type:

Article

3'‐Dehydroxypurpurogallin‐4‐Carboxamides as Influenza A Endonuclease Inhibitors: Synthesis, Structure‐Activity Relationship Analysis, and Structural Characterization of Protein Complex.

Published in:

ChemMedChem, 2025, v. 20, n. 3, p. 1, doi. 10.1002/cmdc.202400577

By:

Kráľ, Michal;
Kotačka, Tomáš;
Reiberger, Róbert;
Panýrková, Gabriela;
Radilová, Kateřina;
Osifová, Zuzana;
Flieger, Miroslav;
Konvalinka, Jan;
Majer, Pavel;
Kožíšek, Milan;
Machara, Aleš

Publication type:

Article

iBodies: Modular Synthetic Antibody Mimetics Based on Hydrophilic Polymers Decorated with Functional Moieties.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 7, p. 2356, doi. 10.1002/anie.201508642

By:

Šácha, Pavel;
Knedlík, Tomáš;
Schimer, Jiří;
Tykvart, Jan;
Parolek, Jan;
Navrátil, Václav;
Dvořáková, Petra;
Sedlák, František;
Ulbrich, Karel;
Strohalm, Jiří;
Majer, Pavel;
Šubr, Vladimír;
Konvalinka, Jan

Publication type:

Article

Mouse brain serine racemase catalyzes specific elimination of L-serine to pyruvate

Published in:

FEBS Letters, 2003, v. 535, n. 1-3, p. 44, doi. 10.1016/S0014-5793(02)03855-3

By:

Střıšovský, Kvido;
Jirásková, Jana;
Bařinka, Cyril;
Majer, Pavel;
Rojas, Camilo;
Slusher, Barbara S.;
Konvalinka, Jan

Publication type:

Article

Shared CaM‐ and S100A1‐binding epitopes in the distal TRPM4 N terminus.

Published in:

FEBS Journal, 2018, v. 285, n. 3, p. 599, doi. 10.1111/febs.14362

By:

Bousova, Kristyna;
Herman, Petr;
Vecer, Jaroslav;
Bednarova, Lucie;
Monincova, Lenka;
Majer, Pavel;
Vyklicky, Ladislav;
Vondrasek, Jiri;
Teisinger, Jan

Publication type:

Article

Integrated Activity and Genetic Profiling of Secreted Peptidases in Cryptococcus neoformans Reveals an Aspartyl Peptidase Required for Low pH Survival and Virulence.

Published in:

PLoS Pathogens, 2016, v. 12, n. 12, p. 1, doi. 10.1371/journal.ppat.1006051

By:

Clarke, Starlynn C.;
O'Donoghue, Anthony J.;
La Greca, Florencia;
Craik, Charles S.;
Dumesic, Phillip A.;
Homer, Christina M.;
Madhani, Hiten D.;
Pallova, Lenka;
Majer, Pavel

Publication type:

Article