Works by Lozach, Olivier

Results: 12

Design and Microwave Synthesis of New (5 Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5 Z) 2-Amino-5-arylidene-1,3-thiazol-4(5 H)-one as New Inhibitors of Protein Kinase DYRK1A.

Published in:

Pharmaceuticals (14248247), 2021, v. 14, n. 11, p. 1086, doi. 10.3390/ph14111086

By:

Bourahla, Khadidja;
Guihéneuf, Solène;
Limanton, Emmanuelle;
Paquin, Ludovic;
Le Guével, Rémy;
Charlier, Thierry;
Rahmouni, Mustapha;
Durieu, Emilie;
Lozach, Olivier;
Carreaux, François;
Meijer, Laurent;
Bazureau, Jean-Pierre

Publication type:

Article

Combined Virtual and Experimental Screening for CK1 Inhibitors Identifies a Modulator of p53 and Reveals Important Aspects of in Silico Screening Performance.

Published in:

International Journal of Molecular Sciences, 2017, v. 18, n. 10, p. 2102, doi. 10.3390/ijms18102102

By:

Myrianthopoulos, Vassilios;
Lozach, Olivier;
Zareifi, Danae;
Alexopoulos, Leonidas;
Meijer, Laurent;
Gorgoulis, Vassilis G.;
Mikros, Emmanuel

Publication type:

Article

Polyprenyl-hydroquinones and -furans from three marine sponges inhibit the cell cycle regulating phosphatase CDC25A.

Published in:

Natural Product Research, 2004, v. 18, n. 1, p. 1, doi. 10.1080/1478641031000111534

By:

Erdogan-Orhan*, Ilkay;
Sener, Bilge;
De Rosa, Salvatore;
Perez-Baz, Julia;
Lozach, Olivier;
Leost, Maryse;
Rakhilin, Sergei;
Meijer, Laurent

Publication type:

Article

Lipid‐Based Quaternary Ammonium Sophorolipid Amphiphiles with Antimicrobial and Transfection Activities.

Published in:

ChemSusChem, 2019, v. 12, n. 15, p. 3642, doi. 10.1002/cssc.201900721

By:

Delbeke, Elisabeth I. P.;
Everaert, Jonas;
Lozach, Olivier;
Le Gall, Tony;
Berchel, Mathieu;
Montier, Tristan;
Jaffrès, Paul‐Alain;
Rigole, Petra;
Coenye, Tom;
Brennich, Martha;
Baccile, Niki;
Roelants, Sophie L. K. W.;
Soetaert, Wim;
Van Bogaert, Inge N. A.;
Van Geem, Kevin M.;
Stevens, Christian V.

Publication type:

Article

Several Human Cyclin-Dependent Kinase Inhibitors, Structurally Related to Roscovitine, As New Anti-Malarial Agents.

Published in:

Molecules, 2014, v. 19, n. 9, p. 15237, doi. 10.3390/molecules190915237

By:

Houzé, Sandrine;
Nha-Thu Hoang;
Lozach, Olivier;
Le Bras, Jacques;
Meijer, Laurent;
Galons, Hervé;
Demange, Luc

Publication type:

Article

Natural Aristolactams and Aporphine Alkaloids as Inhibitors of CDK1/Cyclin B and DYRK1A.

Published in:

Molecules, 2013, v. 18, n. 3, p. 3018, doi. 10.3390/molecules18033018

By:

Marti, Guillaume;
Eparvier, Véronique;
Morleo, Barbara;
Le Ven, Jessica;
Apel, Cécile;
Bodo, Bernard;
Amand, Séverine;
Dumontet, Vincent;
Lozach, Olivier;
Meijer, Laurent;
Guéritte, Françoise;
Litaudon, Marc

Publication type:

Article

A Practical Approach to New (5Z) 2-Alkylthio-5-arylmethylene-1-methyl-1,5-dihydro-4H-imidazol-4-one Derivatives.

Published in:

Molecules, 2011, v. 16, n. 9, p. 7377, doi. 10.3390/molecules16097377

By:

Bourahla, Khadidja;
Paquin, Ludovic;
Lozach, Olivier;
Meijer, Laurent;
Carreaux, François;
Bazureau, Jean Pierre

Publication type:

Article

Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2005, v. 20, n. 6, p. 557, doi. 10.1080/14756360500212399

By:

Testard, Alexandra;
Picot, Laurent;
Lozach, Olivier;
Blairvacq, Melina;
Meijer, Laurent;
Murillo, Laurence;
Piot, Jean-Marie;
Thiéry, Valérie;
Besson, Thierry

Publication type:

Article

Biosynthesis of New Indigoid Inhibitors of Protein Kinases Using Recombinant Cytochrome P450 2A6.

Published in:

Chemistry & Biodiversity, 2005, v. 2, n. 1, p. 51, doi. 10.1002/cbdv.200490166

By:

Wu, Zhongliu-Liu;
Aryal, Pramod;
Lozach, Olivier;
Meijer, Laurent;
Guengerich, F. Peter

Publication type:

Article

First BRET-based screening assay performed in budding yeast leads to the discovery of CDK5/p25 interaction inhibitors.

Published in:

Biotechnology Journal, 2011, v. 6, n. 7, p. 860, doi. 10.1002/biot.201100138

By:

Corbel, Caroline;
Wang, Qian;
Bousserouel, Hadjira;
Hamdi, Amel;
Zhang, Bing;
Lozach, Olivier;
Ferandin, Yoan;
Tan, Vincent B. C.;
Guéritte, Françoise;
Colas, Pierre;
Couturier, Cyril;
Bach, Stéphane

Publication type:

Article

Catalyst-free synthesis of quinazolin-4-ones from (hetero)aryl-guanidines: application to the synthesis of pyrazolo[4,3- f]quinazolin-9-ones, a new family of DYRK1A inhibitors.

Published in:

Molecular Diversity, 2012, v. 16, n. 4, p. 659, doi. 10.1007/s11030-012-9397-7

By:

Debray, Julien;
Bonte, Simon;
Lozach, Olivier;
Meijer, Laurent;
Demeunynck, Martine

Publication type:

Article

Access to Paullone Analogues by Intramolecular Heck Reaction.

Published in:

Helvetica Chimica Acta, 2007, v. 90, n. 4, p. 753, doi. 10.1002/hlca.200790076

By:

Lionel Joucla;
Florence Popowycz;
Olivier Lozach;
Laurent Meijer;
Benoît Joseph

Publication type:

Article