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Activation of single heteromeric GABA<sub>A</sub> receptor ion channels by full and partial agonists.
- Published in:
- Journal of Physiology, 2004, v. 557, n. 2, p. 389, doi. 10.1113/jphysiol.2003.054734
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- Publication type:
- Article
Functional pharmacology of cloned heterodimeric GABA<sub>B</sub> receptors expressed in mammalian cells.
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- British Journal of Pharmacology, 1999, v. 128, n. 7, p. 1370, doi. 10.1038/sj.bjp.0702914
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- Publication type:
- Article
Pharmacology of (S)-homoquisqualic acid and (S)-2-amino-5-phosphonopentanoic acid [(S)-AP5] at cloned metabotropic glutamate receptors.
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- British Journal of Pharmacology, 1998, v. 123, n. 2, p. 269, doi. 10.1038/sj.bjp.0701616
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- Publication type:
- Article
Editorial: Die soziale Verantwortung der Wissenschaftler.
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- Angewandte Chemie, 2011, v. 123, n. 46, p. 10926, doi. 10.1002/ange.201105641
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- Publication type:
- Article
Structural Determinants for AMPA Agonist Activity of Aryl or Heteroaryl Substituted AMPA Analogues. Synthesis and Pharmacology.
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- Archiv der Pharmazie, 2001, v. 334, n. 2, p. 62, doi. 10.1002/1521-4184(200102)334:2<62::AID-ARDP62>3.0.CO;2-G
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- Publication type:
- Article
Analogues of Carbacholine: Synthesis and Relationship between Structure and Affinity for Muscarinic and Nicotinic Acetylcholine Receptors.
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- Archiv der Pharmazie, 1996, v. 329, n. 2, p. 95, doi. 10.1002/ardp.19963290207
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- Publication type:
- Article
Specific GABA<sub>A</sub> agonists and partial agonists.
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- Chemical Record, 2002, v. 2, n. 6, p. 419, doi. 10.1002/tcr.10040
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- Publication type:
- Article
Subtype selective kainic acid receptor agonists: Discovery and approaches to rational design.
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- Medicinal Research Reviews, 2009, v. 29, n. 1, p. 3, doi. 10.1002/med.20133
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- Publication type:
- Article
Structural, conformational, and stereochemical requirements of central excitatory amino acid receptors.
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- Medicinal Research Reviews, 1990, v. 10, n. 1, p. 55, doi. 10.1002/med.2610100103
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- Publication type:
- Article
GABA synaptic mechanisms: Stereochemical and conformational requirements.
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- Medicinal Research Reviews, 1988, v. 8, n. 1, p. 27, doi. 10.1002/med.2610080103
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- Publication type:
- Article
Probing the Orthosteric Binding Site of GABA Receptors with Heterocyclic GABA Carboxylic Acid Bioisosteres.
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- Neurochemical Research, 2014, v. 39, n. 6, p. 1005, doi. 10.1007/s11064-013-1226-6
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- Publication type:
- Article
Detecting Protein–Protein Interactions in Living Cells: Development of a Bioluminescence Resonance Energy Transfer Assay to Evaluate the PSD-95/NMDA Receptor Interaction.
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- Neurochemical Research, 2009, v. 34, n. 10, p. 1729, doi. 10.1007/s11064-009-9998-4
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- Publication type:
- Article
Medicinal chemistry education: what is needed and where is it going?
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- Drug Development Research, 2005, v. 66, n. 1, p. 1
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- Publication type:
- Article
Hydroxylated Analogues of 5-Aminovaleric Acid as 4-Aminobutyric AcidB Receptor Antagonists: Stereostructure-Activity Relationships.
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- Journal of Neurochemistry, 1992, v. 58, n. 3, p. 1150, doi. 10.1111/j.1471-4159.1992.tb09374.x
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- Publication type:
- Article
Novel Glutamate Receptor Antagonists Selectively Protect Against Kainic Acid Neurotoxicity in Cultured Cerebral Cortex Neurons.
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- Journal of Neurochemistry, 1990, v. 55, n. 5, p. 1821, doi. 10.1111/j.1471-4159.1990.tb04976.x
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- Publication type:
- Article
Comparative Stereostructure-Activity Studies on GABA<sub>A</sub> and GABA<sub>B</sub> Receptor Sites and GABA Uptake Using Rat Brain Membrane Preparations.
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- Journal of Neurochemistry, 1986, v. 47, n. 3, p. 898, doi. 10.1111/j.1471-4159.1986.tb00695.x
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- Publication type:
- Article
Glycine Antagonists Structurally Related to 4,5,6,7-Tetrahydroisoxazolo[5,4- c]pyridin-3-ol Inhibit Binding of [<sup>3</sup>H]Strychnine to Rat Brain Membranes.
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- Journal of Neurochemistry, 1986, v. 47, n. 3, p. 691, doi. 10.1111/j.1471-4159.1986.tb00667.x
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- Publication type:
- Article
Excitatory Amino Acids: Studies on the Biochemical and Chemical Stability of Ibotenic Acid and Related Compounds.
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- Journal of Neurochemistry, 1985, v. 45, n. 3, p. 725, doi. 10.1111/j.1471-4159.1985.tb04052.x
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- Publication type:
- Article
GABA-Mimetic Activity and Effects on Diazepam Binding of Aminosulphonic Acids Structurally Related to Piperidine-4-Sulphonic Acid.
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- Journal of Neurochemistry, 1985, v. 44, n. 1, p. 68, doi. 10.1111/j.1471-4159.1985.tb07114.x
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- Publication type:
- Article
The Binding of [<sup>3</sup>H]AMPA, a Structural Analogue of Glutamic Acid, to Rat Brain Membranes.
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- Journal of Neurochemistry, 1982, v. 38, n. 1, p. 173, doi. 10.1111/j.1471-4159.1982.tb10868.x
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- Publication type:
- Article
Synthesis, theoretical and structural analyses, and enantiopharmacology of 3‐carboxy homologs of AMPAThis work was supported by grants from the Lundbeck Foundation, the Danish Medical Research Council, and the Danish Natural Science Research Council
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- Chirality, 2004, v. 16, n. 7, p. 452
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- Publication type:
- Article
Stereostructure-activity studies on agonists at the AMPA and kainate subtypes of ionotropic glutamate receptors.
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- Chirality, 2003, v. 15, n. 2, p. 167, doi. 10.1002/chir.10177
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- Publication type:
- Article
Glutamate receptor ligands: Synthesis, stereochemistry, and enantiopharmacology of methylated 2-aminoadipic acid analogs.
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- Chirality, 2002, v. 14, n. 4, p. 351, doi. 10.1002/chir.10104
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- Publication type:
- Article
Resolution, configurational assignment, and enantiopharmacology at glutamate receptors of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) and demethyl-ACPA.
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- Chirality, 2001, v. 13, n. 9, p. 523, doi. 10.1002/chir.1172
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- Publication type:
- Article
Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2 H-tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3- and GluR4-preferring AMPA receptor agonist.
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- Chirality, 2000, v. 12, n. 10, p. 705, doi. 10.1002/1520-636X(2000)12:10<705::AID-CHIR2>3.0.CO;2-9
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- Publication type:
- Article
Solid phase synthesis and biological evaluation of enantiomerically pure wasp toxin analogues PhTX-343 and PhTX-12.
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- Chirality, 2000, v. 12, n. 2, p. 93, doi. 10.1002/(SICI)1520-636X(2000)12:2<93::AID-CHIR6>3.0.CO;2-B
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- Publication type:
- Article
Resolution, absolute stereochemistry, and enantiopharmacology of the GluR1-4 and GluR5 antagonist 2-amino-3-[5- tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid.
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- Chirality, 1999, v. 11, n. 10, p. 752, doi. 10.1002/(SICI)1520-636X(1999)11:10<752::AID-CHIR3>3.0.CO;2-T
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- Publication type:
- Article
Excitatory amino acid receptor antagonists: Resolution, absolute stereochemistry, and pharmacology of (S)- and (R)-2-amino-2-(5- tert-butyl-3-hydroxyisoxazol-4-yl)acetic acid (ATAA).
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- Chirality, 1997, v. 9, n. 5/6, p. 529, doi. 10.1002/(SICI)1520-636X(1997)9:5/6<529::AID-CHIR20>3.0.CO;2-P
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- Publication type:
- Article
AMPA receptor agonists: Resolution, configurational assignment, and pharmacology of (+)-(S)- and (-)-(R)-2-amino-3-[3-hydroxy-5-(2-pyridyl)-isoxazol-4-yl]-propionic acid (2-Py-AMPA).
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- Chirality, 1997, v. 9, n. 3, p. 274, doi. 10.1002/(SICI)1520-636X(1997)9:3<274::AID-CHIR12>3.0.CO;2-K
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- Publication type:
- Article
GABA<sub>B</sub> antagonists: Enantiopharmacology of 5-amino-4-hydroxy-2-methylvaleric acid and X-ray structure of the eutomer.
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- Chirality, 1995, v. 7, n. 7, p. 526, doi. 10.1002/chir.530070706
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- Article
GABA<sub>A</sub> agonists: Resolution and pharmacology of (+)- and (−)-isoguvacine oxide.
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- Chirality, 1995, v. 7, n. 6, p. 434, doi. 10.1002/chir.530070608
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- Publication type:
- Article
GABA<sub>B</sub> antagonists: Resolution, absolute stereochemistry, and pharmacology of (R)- and (S)-phaclofen.
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- Chirality, 1994, v. 6, n. 7, p. 583, doi. 10.1002/chir.530060712
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- Publication type:
- Article
Synaptic and extrasynaptic GABA transporters as targets for anti-epileptic drugs.
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- Journal of Neurochemistry, 2009, v. 109, p. 139, doi. 10.1111/j.1471-4159.2009.05982.x
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- Publication type:
- Article
PHILANTHOTOXIN ANALOGUES CONTAINING ETHER GROUPS DISTINGUISH BETWEEN NICOTINIC ACETYLCHOLINE RECEPTORS AND IONOTROPIC QUISQUALATE RECEPTORS.
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- 1999
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- Publication type:
- Abstract
GABA-A agonists and GABA uptake inhibitors: Structure-activity relationships.
- Published in:
- Drug Development Research, 1990, v. 21, n. 3, p. 169, doi. 10.1002/ddr.430210304
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- Publication type:
- Article
Synthesis of deuterium and tritium labelled ( RS)-2-amino-3-(5- tert-butyl-3-hydroxy-4-isoxazolyl)-propionic acid (ATPA), a selective kainic acid receptor agonist.
- Published in:
- Journal of Labelled Compounds & Radiopharmaceuticals, 1999, v. 42, n. 10, p. 937, doi. 10.1002/(SICI)1099-1344(199910)42:10<937::AID-JLCR252>3.0.CO;2-#
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- Publication type:
- Article
Synthesis of tritiated ( RS)-2-amino-2-(3-hydroxy-5-methylisoxazol-4-yl)acetic acid (AMAA), a potent and selective NMDA agonist.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 1996, v. 38, n. 10, p. 915, doi. 10.1002/(SICI)1099-1344(199610)38:10<915::AID-JLCR903>3.0.CO;2-B
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- Publication type:
- Article
Deuterium labelling of the GABA agonist thiomuscimol.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 1984, v. 21, n. 3, p. 253, doi. 10.1002/jlcr.2580210307
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- Publication type:
- Article
Deuterium labelling of the GABA agonists THIP, piperidine-4-sulphonic acid and the gaba uptake inhibitor THPO.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 1982, v. 19, n. 5, p. 689, doi. 10.1002/jlcr.2580190509
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- Publication type:
- Article
Preparations of deuterium labelled guvacine and isoguvacine.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 1980, v. 17, n. 2, p. 191, doi. 10.1002/jlcr.2580170206
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- Publication type:
- Article
Editorial: Scientific Social Responsibility: A Call to Arms.
- Published in:
- Angewandte Chemie International Edition, 2011, v. 50, n. 46, p. 10738, doi. 10.1002/anie.201105641
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- Publication type:
- Article
Probing α<sub>4</sub>βδ GABAa Receptor Heterogeneity: Differential Regional Effects of a Functionally Selective α<sub>4</sub>β<sub>1</sub>δ/α<sub>4</sub>β<sub>3</sub>δ Receptor Agonist on Tonic and Phasic Inhibition in Rat Brain
- Published in:
- Journal of Neuroscience, 2014, v. 34, n. 49, p. 16256, doi. 10.1523/JNEUROSCI.1495-14.2014
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- Publication type:
- Article