Works by Krasavin, Mikhail

Results: 105

Natural products as templates for bioactive compound libraries: synthesis of biaryl derivatives of (±)-vasicine.

Published in:

Natural Product Research, 2006, v. 20, n. 8, p. 735, doi. 10.1080/14786410500247418

By:

Shevyakov, Sergey V.;
Davydova, Olga I.;
Pershin, Dmitry G.;
Krasavin, Mikhail;
Kravchenko, Dmitry V.;
Kiselyov, Alex;
Tkachenko, Sergey E.;
Ivachtchenko, Alexandre V.

Publication type:

Article

Natural products as templates for bioactive compound libraries: Part 2. Novel modifications of vasicine (peganine) core via efficient and regioselective generation of 3-lithiodeoxyvasicine and its stereoselective addition to aliphatic ketones§.

Published in:

Natural Product Research, 2006, v. 20, n. 9, p. 871, doi. 10.1080/14786410500480993

By:

Shevyakov, Sergey V.;
Davydova, Olga I.;
Kiselyov, Alex S.;
Kravchenko, Dmitry V.;
Ivachtchenko, Alexandre V.;
Krasavin, Mikhail

Publication type:

Article

Exploration of the nitrogen heterocyclic periphery around the core of the advanced FFA1 agonist fasiglifam (TAK‐875).

Published in:

Archiv der Pharmazie, 2021, v. 354, n. 4, p. 1, doi. 10.1002/ardp.202000275

By:

Lukin, Alexey;
Bakholdina, Anna;
Zhurilo, Nikolay;
Onopchenko, Oleksandra;
Zhuravel, Elena;
Zozulya, Sergey;
Gureev, Maxim;
Safrygin, Alexander;
Krasavin, Mikhail

Publication type:

Article

Carnosine protects neurons against oxidative stress and modulates the time profile of MAPK cascade signaling.

Published in:

Amino Acids, 2012, v. 43, n. 1, p. 91, doi. 10.1007/s00726-011-1135-4

By:

Kulebyakin, Konstantin;
Karpova, Larisa;
Lakonsteva, Ekaterina;
Krasavin, Mikhail;
Boldyrev, Alexander

Publication type:

Article

Non-covalent interactions observed in nevirapinium pentaiodide hydrate which include the rare I4–I−···O=C halogen bonding.

Published in:

Zeitschrift für Kristallographie. Crystalline Materials, 2019, v. 234, n. 2, p. 101, doi. 10.1515/zkri-2018-2081

By:

Kryukova, Mariya A.;
Sapegin, Alexander V.;
Novikov, Alexander S.;
Krasavin, Mikhail;
Ivanov, Daniil M.

Publication type:

Article

Periphery Exploration around 2,6-Diazaspiro[3.4]octane Core Identifies a Potent Nitrofuran Antitubercular Lead.

Published in:

Molecules, 2023, v. 28, n. 6, p. 2529, doi. 10.3390/molecules28062529

By:

Lukin, Alexei;
Komarova, Kristina;
Vinogradova, Lyubov;
Dogonadze, Marine;
Vinogradova, Tatiana;
Yablonsky, Piotr;
Kazantsev, Alexander;
Krasavin, Mikhail

Publication type:

Article

The Use of Aryl-Substituted Homophthalic Anhydrides in the Castagnoli–Cushman Reaction Provides Access to Novel Tetrahydroisoquinolone Carboxylic Acid Bearing an All-Carbon Quaternary Stereogenic Center.

Published in:

Molecules, 2022, v. 27, n. 23, p. 8462, doi. 10.3390/molecules27238462

By:

Moshnenko, Nazar;
Kazantsev, Alexander;
Bakulina, Olga;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

One-Pot Sequence of Staudinger/aza-Wittig/Castagnoli–Cushman Reactions Provides Facile Access to Novel Natural-like Polycyclic Ring Systems.

Published in:

Molecules, 2022, v. 27, n. 23, p. 8130, doi. 10.3390/molecules27238130

By:

Lebedev, Rodion;
Dar'in, Dmitry;
Kantin, Grigory;
Bakulina, Olga;
Krasavin, Mikhail

Publication type:

Article

Extending the Scope of the New Variant of the Castagnoli–Cushman Cyclocondensation onto o -Methyl Benzoic Acids Bearing Various Electron-Withdrawing Groups in the α-Position.

Published in:

Molecules, 2022, v. 27, n. 21, p. 7211, doi. 10.3390/molecules27217211

By:

Guranova, Natalia;
Yakovleva, Lyudmila;
Bakulina, Olga;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Exploration of Spirocyclic Derivatives of Ciprofloxacin as Antibacterial Agents.

Published in:

Molecules, 2022, v. 27, n. 15, p. 4864, doi. 10.3390/molecules27154864

By:

Lukin, Alexei;
Chudinov, Mikhail;
Vedekhina, Tatiana;
Rogacheva, Elizaveta;
Kraeva, Lyudmila;
Bakulina, Olga;
Krasavin, Mikhail

Publication type:

Article

Conjugates of Iron-Transporting N -Hydroxylactams with Ciprofloxacin.

Published in:

Molecules, 2022, v. 27, n. 12, p. 3910, doi. 10.3390/molecules27123910

By:

Bakulina, Olga;
Bannykh, Anton;
Levashova, Ekaterina;
Krasavin, Mikhail

Publication type:

Article

Dicarboxylic Acid Monoesters in β- and δ-Lactam Synthesis.

Published in:

Molecules, 2022, v. 27, n. 8, p. N.PAG, doi. 10.3390/molecules27082469

By:

Ananeva, Anna;
Bakulina, Olga;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Preparation and Synthetic Applications of Five-to-Seven-Membered Cyclic α-Diazo Monocarbonyl Compounds.

Published in:

Molecules, 2022, v. 27, n. 6, p. 2030, doi. 10.3390/molecules27062030

By:

Zhukovsky, Daniil;
Dar'in, Dmitry;
Bakulina, Olga;
Krasavin, Mikhail

Publication type:

Article

Multicomponent Reactions Involving Diazo Reagents: A 5-Year Update.

Published in:

Molecules, 2021, v. 26, n. 21, p. 6563, doi. 10.3390/molecules26216563

By:

Bakulina, Olga;
Inyutina, Anna;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Diazocarbonyl and Related Compounds in the Synthesis of Azoles.

Published in:

Molecules, 2021, v. 26, n. 9, p. 2530, doi. 10.3390/molecules26092530

By:

Budeev, Anton;
Kantin, Grigory;
Dar'in, Dmitry;
Krasavin, Mikhail;
Zhou, Lei

Publication type:

Article

Two Annulated Azaheterocyclic Cores Readily Available from a Single Tetrahydroisoquinolonic Castagnoli–Cushman Precursor.

Published in:

Molecules, 2020, v. 25, n. 9, p. 2049, doi. 10.3390/molecules25092049

By:

Karchuganova, Elizaveta;
Bakulina, Olga;
Dar'in, Dmitry;
Krasavin, Mikhail;
Bunce, Richard A.;
Belmont, Philippe;
Dehaen, Wim;
Babaev, Eugene

Publication type:

Article

Spirocyclic Motifs in Natural Products.

Published in:

Molecules, 2019, v. 24, n. 22, p. 4165, doi. 10.3390/molecules24224165

By:

Chupakhin, Evgeny;
Babich, Olga;
Prosekov, Alexander;
Asyakina, Lyudmila;
Krasavin, Mikhail;
Tormo, José Rubén

Publication type:

Article

Facile Access to Fe(III)-Complexing Cyclic Hydroxamic Acids in a Three-Component Format.

Published in:

Molecules, 2019, v. 24, n. 5, p. 864, doi. 10.3390/molecules24050864

By:

Chupakhin, Evgeny;
Bakulina, Olga;
Dar'in, Dmitry;
Krasavin, Mikhail;
Bunce, Richard A.;
Belmont, Philippe;
Dehaen, Wim;
Babaev, Eugene

Publication type:

Article

Novel 5-Nitrofuran-Tagged Imidazo-Fused Azines and Azoles Amenable by the Groebke–Blackburn–Bienaymé Multicomponent Reaction: Activity Profile against ESKAPE Pathogens and Mycobacteria.

Published in:

Biomedicines, 2022, v. 10, n. 9, p. 2203, doi. 10.3390/biomedicines10092203

By:

Sapegin, Alexander;
Rogacheva, Elizaveta;
Kraeva, Lyudmila;
Gureev, Maxim;
Dogonadze, Marine;
Vinogradova, Tatiana;
Yablonsky, Petr;
Balalaie, Saeed;
Baykov, Sergey V.;
Krasavin, Mikhail

Publication type:

Article

Synthesis, Structure, and Antiproliferative Action of 2-Pyridyl Urea-Based Cu(II) Complexes.

Published in:

Biomedicines, 2022, v. 10, n. 2, p. 461, doi. 10.3390/biomedicines10020461

By:

Geyl, Kirill K.;
Baykov, Sergey V.;
Kalinin, Stanislav A.;
Bunev, Alexandr S.;
Troshina, Marina A.;
Sharonova, Tatiana V.;
Skripkin, Mikhail Yu.;
Kasatkina, Svetlana O.;
Presnukhina, Sofia I.;
Shetnev, Anton A.;
Krasavin, Mikhail Yu.;
Boyarskiy, Vadim P.

Publication type:

Article

Synthetic Exploration of α‐Diazo γ‐Butyrolactams.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 13, p. 2397, doi. 10.1002/ejoc.201900133

By:

Zhukovsky, Daniil;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Gold‐Catalyzed Oxidation of Internal Alkynes into Benzils and its Application for One‐Pot Synthesis of Five‐, Six‐, and Seven‐Membered Azaheterocycles.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 8, p. 1856, doi. 10.1002/ejoc.201900108

By:

Dubovtsev, Alexey Yu.;
Dar'in, Dmitry V.;
Krasavin, Mikhail;
Kukushkin, Vadim Yu.

Publication type:

Article

RhII‐Catalyzed Cycloaddition of α‐Diazo Homophthalimides and Nitriles Delivers Oxazolo[5,4‐c]isoquinolin‐5(4H)‐one Scaffold.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 35, p. 4857, doi. 10.1002/ejoc.201800955

By:

Kantin, Grigory;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

A General Way to Construct Arene-Fused Seven-Membered Nitrogen Heterocycles.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 3, p. 362, doi. 10.1002/ejoc.201701642

By:

Bakulina, Olga;
Chizhova, Maria;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Sterically Constrained and Encumbered: An Approach to the Naturally Occurring Peptidomimetic Tetrahydropyrazino[1,2- a]indole-1,4-dione Core.

Published in:

European Journal of Organic Chemistry, 2017, v. 2017, n. 13, p. 1740, doi. 10.1002/ejoc.201700152

By:

Golubev, Pavel;
Krasavin, Mikhail

Publication type:

Article

Indoline-Based Constrained Peptidomimetic Motifs Obtained via the Joullié-Ugi Reaction of Indolenines.

Published in:

European Journal of Organic Chemistry, 2016, v. 2016, n. 23, p. 3969, doi. 10.1002/ejoc.201600656

By:

Golubev, Pavel;
Bakulina, Olga;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Efficient Use of 1,2-Dihaloazine Synthons in Transition-Metal-Free Preparation of Diverse Heterocycle-Fused 1,4-Oxazepines.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 6, p. 1333, doi. 10.1002/ejoc.201403397

By:

Sapegin, Alexander V.;
Kalinin, Stanislav A.;
Smirnov, Alexey V.;
Dorogov, Mikhail V.;
Krasavin, Mikhail

Publication type:

Article

Plants of the Russian Federation pharmacopeia: an unexhausted natural products research opportunity?

Published in:

Natural Product Research, 2021, v. 35, n. 21, p. 3525, doi. 10.1080/14786419.2020.1727474

By:

Chupakhin, Evgeny;
Babich, Olga;
Prosekov, Alexander;
Asyakina, Lyudmila;
Gureev, Maxim;
Krasavin, Mikhail

Publication type:

Article

Versatile Diazomethane Sulfonamide for Expedited Exploration of Azole‐Based Carbonic Anhydrase Inhibitors via [3+2] Cycloaddition.

Published in:

ChemMedChem, 2023, v. 18, n. 10, p. 1, doi. 10.1002/cmdc.202200607

By:

Krivovicheva, Vasilisa;
Bubyrev, Andrey;
Kalinin, Stanislav;
Dar'in, Dmitry;
Gureev, Maxim;
Burianova, Valeria;
Vullo, Daniella;
Krasavin, Mikhail;
Supuran, Claudiu T.

Publication type:

Article

Cover Feature: RhII‐Catalyzed De‐symmetrization of Ethane‐1,2‐dithiol and Propane‐1,3‐dithiol Yields Metallo‐β‐lactamase Inhibitors (ChemMedChem 22/2021).

Published in:

ChemMedChem, 2021, v. 16, n. 22, p. 3375, doi. 10.1002/cmdc.202100692

By:

Krasavin, Mikhail;
Zhukovsky, Daniil;
Solovyev, Igor;
Barkhatova, Darina;
Dar'in, Dmitry;
Frank, Denia;
Martinelli, Giada;
Weizel, Lilia;
Proschak, Anna;
Rotter, Marco;
Kramer, Jan S.;
Brunst, Steffen;
Wichelhaus, Thomas A.;
Proschak, Ewgenij

Publication type:

Article

RhII‐Catalyzed De‐symmetrization of Ethane‐1,2‐dithiol and Propane‐1,3‐dithiol Yields Metallo‐β‐lactamase Inhibitors.

Published in:

ChemMedChem, 2021, v. 16, n. 22, p. 3410, doi. 10.1002/cmdc.202100344

By:

Krasavin, Mikhail;
Zhukovsky, Daniil;
Solovyev, Igor;
Barkhatova, Darina;
Dar'in, Dmitry;
Frank, Denia;
Martinelli, Giada;
Weizel, Lilia;
Proschak, Anna;
Rotter, Marco;
Kramer, Jan S.;
Brunst, Steffen;
Wichelhaus, Thomas A.;
Proschak, Ewgenij

Publication type:

Article

Trimethylsilyl Chloride as a Promoter for the Groebke-Blackburn Reaction: Preparation of Imidazo[2,1-b][1,3]Benzothiazoles.

Published in:

Synthetic Communications, 2010, v. 40, n. 1, p. 111, doi. 10.1080/00397910902953331

By:

Tsirulnikov, Sergey;
Kysil, Volodymyr;
Ivachtchenko, Alexandre;
Krasavin, Mikhail

Publication type:

Article

New Crystal Forms for Biologically Active Compounds. Part 2: Anastrozole as N-Substituted 1,2,4-Triazole in Halogen Bonding and Lp-π Interactions with 1,4-Diiodotetrafluorobenzene.

Published in:

Crystals (2073-4352), 2020, v. 10, n. 5, p. 371, doi. 10.3390/cryst10050371

By:

Kryukova, Mariya A.;
Sapegin, Alexander V.;
Novikov, Alexander S.;
Krasavin, Mikhail;
Ivanov, Daniil M.

Publication type:

Article

An improved kilogram-scale preparation of atorvastatin calcium.

Published in:

Chemistry Central Journal, 2015, v. 9, n. 1, p. 1, doi. 10.1186/s13065-015-0082-7

By:

Novozhilov, Yuri V.;
Dorogov, Mikhail V.;
Blumina, Maria V.;
Smirnov, Alexey V.;
Krasavin, Mikhail

Publication type:

Article

Discovery and SAR exploration of N-aryl-N-(3-aryl-1,2,4-oxadiazol-5-yl)amines as potential therapeutic agents for prostate cancer.

Published in:

Chemistry Central Journal, 2010, v. 4, p. 4, doi. 10.1186/1752-153X-4-4

By:

Krasavin, Mikhail;
Rufanov, Konstantin A.;
Sosnov, Andrey V.;
Karapetian, Ruben;
Godovykh, Elena;
Soldatkina, Olga;
Lavrovsky, Yan;
Gakh, Andrei A.

Publication type:

Article

Synthetic Exploration of Novel Sulfamoyl Cyanide N‐Oxides in Heterocycle Synthesis.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 46, p. 1, doi. 10.1002/ejoc.202201162

By:

Krivovicheva, Vasilisa;
Bubyrev, Andrey;
Kalinin, Stanislav;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Steric Push towards the [n+3] Hydrated Imidazoline Ring Expansion (HIRE) of Dibenzo[1.4]oxazepines and Thiazepines.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 35, p. 1, doi. 10.1002/ejoc.202200818

By:

Lavit, Ksenia;
Sapegin, Alexander;
Linnik, Stanislav;
Ryazantsev, Mikhail;
Krasavin, Mikhail

Publication type:

Article

Homophthalic Esters: A New Type of Reagents for the Castagnoli‐Cushman Reaction.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 9, p. 1, doi. 10.1002/ejoc.202101281

By:

Guranova, Natalia;
Bakulina, Olga;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Oxonium Ylides Generated from 1,4‐Disubstituted α‐Diazo Glutaconimides: a Rich Source of Diverse Oxygen Heterocyclic Frameworks.

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 23, p. 3411, doi. 10.1002/ejoc.202100515

By:

Guranova, Natalia;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Cover Feature: Three‐Component Castagnoli‐Cushman Reaction of 3‐Arylglutaconic Acid Anhydrides, Carbonyl Compounds, and Ammonium Acetate: a Quick and Flexible Way to Assemble Polysubstituted NH‐δ‐lactams (Eur. J. Org. Chem. 11/2021)

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 11, p. 1773, doi. 10.1002/ejoc.202100298

By:

Peshkov, Anatoly A.;
Bakulina, Olga;
Dar'in, Dmitry;
Kantin, Grigory;
Bannykh, Anton;
Peshkov, Vsevolod A.;
Krasavin, Mikhail

Publication type:

Article

Three‐Component Castagnoli‐Cushman Reaction of 3‐Arylglutaconic Acid Anhydrides, Carbonyl Compounds, and Ammonium Acetate: a Quick and Flexible Way to Assemble Polysubstituted NH‐δ‐lactams.

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 11, p. 1726, doi. 10.1002/ejoc.202001617

By:

Peshkov, Anatoly A.;
Bakulina, Olga;
Dar'in, Dmitry;
Kantin, Grigory;
Bannykh, Anton;
Peshkov, Vsevolod A.;
Krasavin, Mikhail

Publication type:

Article

Diazo Glutaconimides: an Unexplored Type of Heterocyclic α-Diazocarbonyl Compounds Conveniently Evolved into Pyridine-2,6(1H,3H)-diones and Oxazolo[5,4-b]pyridin-5(4H)-ones.

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 4, p. 623, doi. 10.1002/ejoc.202001451

By:

Guranova, Natalia;
Kantin, Grigory;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Front Cover: An Alternative Approach to the Hydrated Imidazoline Ring Expansion (HIRE) of Diarene‐Fused [1.4]Oxazepines (Eur. J. Org. Chem. 35/2020).

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 35, p. 5635, doi. 10.1002/ejoc.202001186

By:

Grintsevich, Sergey;
Sapegin, Alexander;
Reutskaya, Elena;
Peintner, Stefan;
Erdélyi, Máté;
Krasavin, Mikhail

Publication type:

Article

An Alternative Approach to the Hydrated Imidazoline Ring Expansion (HIRE) of Diarene‐Fused [1.4]Oxazepines.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 35, p. 5664, doi. 10.1002/ejoc.202000789

By:

Grintsevich, Sergey;
Sapegin, Alexander;
Reutskaya, Elena;
Peintner, Stefan;
Erdélyi, Máté;
Krasavin, Mikhail

Publication type:

Article

1,3,5‐Triazinanes as Formaldimine Surrogates in the Ugi Reaction.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 29, p. 4517, doi. 10.1002/ejoc.202000569

By:

Golubev, Pavel;
Guranova, Natalia;
Krasavin, Mikhail

Publication type:

Article

Cover Feature: Synthetic Studies towards CH‐Diazomethane Sulfonamides: a Novel Type of Diazo Reagents (Eur. J. Org. Chem. 27/2020)

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 27, p. 4068, doi. 10.1002/ejoc.202000948

By:

Bubyrev, Andrey;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

From Rare Reagents to Rare Products: Regiospecific Silver-Catalyzed [3+2] Cycloaddition of Aryl-, Alkyl- and Aminosulfonyl Diazomethanes with Arenediazonium Tosylates.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 27, p. 4239, doi. 10.1002/ejoc.202000619

By:

Levashova, Ekaterina;
Bakulina, Olga;
Dar'in, Dmitry;
Bubyrev, Andrey;
Chuprun, Sergey;
Krasavin, Mikhail

Publication type:

Article

Synthetic Studies towards CH-Diazomethane Sulfonamides: a Novel Type of Diazo Reagents.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 27, p. 4112, doi. 10.1002/ejoc.202000446

By:

Bubyrev, Andrey;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Cover Feature: tert‐Butyl 3‐Diazo‐2‐oxopyrrolidine‐1‐carboxylate – A New Reagent for Introduction of the 2‐Oxopyrrolidin‐3‐yl Motif via RhII‐Catalyzed X–H Insertion Reactions (Eur. J. Org. Chem. 20/2020)

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 20, p. 2980, doi. 10.1002/ejoc.202000639

By:

Zhukovsky, Daniil;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

tert‐Butyl 3‐Diazo‐2‐oxopyrrolidine‐1‐carboxylate – A New Reagent for Introduction of the 2‐Oxopyrrolidin‐3‐yl Motif via RhII‐Catalyzed X–H Insertion Reactions.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 20, p. 3013, doi. 10.1002/ejoc.202000067

By:

Zhukovsky, Daniil;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article