Works matching AU Krasavin, Mikhail

Results: 105

Natural‐Like Spirocyclic Δα,β‐Butenolides Obtained from Diazo Homophthalimides.

Published in:

Chemistry - A European Journal, 2021, v. 27, n. 31, p. 8221, doi. 10.1002/chem.202100880

By:

Dar'in, Dmitry;
Kantin, Grigory;
Chupakhin, Evgeny;
Sharoyko, Vladimir;
Krasavin, Mikhail

Publication type:

Article

Carnosine protects neurons against oxidative stress and modulates the time profile of MAPK cascade signaling.

Published in:

Amino Acids, 2012, v. 43, n. 1, p. 91, doi. 10.1007/s00726-011-1135-4

By:

Kulebyakin, Konstantin;
Karpova, Larisa;
Lakonsteva, Ekaterina;
Krasavin, Mikhail;
Boldyrev, Alexander

Publication type:

Article

Gold‐Catalyzed Oxidation of Internal Alkynes into Benzils and its Application for One‐Pot Synthesis of Five‐, Six‐, and Seven‐Membered Azaheterocycles.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 8, p. 1856, doi. 10.1002/ejoc.201900108

By:

Dubovtsev, Alexey Yu.;
Dar'in, Dmitry V.;
Krasavin, Mikhail;
Kukushkin, Vadim Yu.

Publication type:

Article

RhII‐Catalyzed Cycloaddition of α‐Diazo Homophthalimides and Nitriles Delivers Oxazolo[5,4‐c]isoquinolin‐5(4H)‐one Scaffold.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 35, p. 4857, doi. 10.1002/ejoc.201800955

By:

Kantin, Grigory;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

A General Way to Construct Arene-Fused Seven-Membered Nitrogen Heterocycles.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 3, p. 362, doi. 10.1002/ejoc.201701642

By:

Bakulina, Olga;
Chizhova, Maria;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Sterically Constrained and Encumbered: An Approach to the Naturally Occurring Peptidomimetic Tetrahydropyrazino[1,2- a]indole-1,4-dione Core.

Published in:

European Journal of Organic Chemistry, 2017, v. 2017, n. 13, p. 1740, doi. 10.1002/ejoc.201700152

By:

Golubev, Pavel;
Krasavin, Mikhail

Publication type:

Article

Indoline-Based Constrained Peptidomimetic Motifs Obtained via the Joullié-Ugi Reaction of Indolenines.

Published in:

European Journal of Organic Chemistry, 2016, v. 2016, n. 23, p. 3969, doi. 10.1002/ejoc.201600656

By:

Golubev, Pavel;
Bakulina, Olga;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Efficient Use of 1,2-Dihaloazine Synthons in Transition-Metal-Free Preparation of Diverse Heterocycle-Fused 1,4-Oxazepines.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 6, p. 1333, doi. 10.1002/ejoc.201403397

By:

Sapegin, Alexander V.;
Kalinin, Stanislav A.;
Smirnov, Alexey V.;
Dorogov, Mikhail V.;
Krasavin, Mikhail

Publication type:

Article

Trimethylsilyl Chloride as a Promoter for the Groebke-Blackburn Reaction: Preparation of Imidazo[2,1-b][1,3]Benzothiazoles.

Published in:

Synthetic Communications, 2010, v. 40, n. 1, p. 111, doi. 10.1080/00397910902953331

By:

Tsirulnikov, Sergey;
Kysil, Volodymyr;
Ivachtchenko, Alexandre;
Krasavin, Mikhail

Publication type:

Article

Preparation and Chemical Behavior of 2‐(tert‐Butoxycarbonyl)amino‐3‐bromomethyl Pyridine, a Novel Alkylating Agent.

Published in:

Synthetic Communications, 2006, v. 36, n. 2, p. 181, doi. 10.1080/00397910500334371

By:

Krasavin, Mikhail;
Shkavrov, Sergey;
Kravchenko, Dmitry

Publication type:

Article

Synthesis and Practical Use of 1H ‐1,2,3‐Benzotriazole‐5‐carboxaldehyde for Reductive Amination.

Published in:

Synthetic Communications, 2005, v. 35, n. 19, p. 2587, doi. 10.1080/00397910500214151

By:

Krasavin, Mikhail;
Pershin, Dmitry;
Larkin, Denis;
Kravchenko, Dmitry

Publication type:

Article

A Convenient Synthesis of 1-Amino-7-(Piperidin-4-yl)Isoquinoline.

Published in:

Synthetic Communications, 2005, v. 35, n. 5, p. 725, doi. 10.1081/SCC-200050372

By:

Shkavrov, Sergey;
Popov, Sergey;
Kravchenko, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Cyclic Hydroxamic Acid Analogues of Bacterial Siderophores as Iron-Complexing Agents prepared through the Castagnoli-Cushman Reaction of Unprotected Oximes.

Published in:

Chemistry - A European Journal, 2017, v. 23, n. 70, p. 17667, doi. 10.1002/chem.201704389

By:

Bakulina, Olga;
Bannykh, Anton;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Mutually Isomeric 2- and 4-(3-Nitro-1,2,4-triazol-1-yl)pyrimidines Inspired by an Antimycobacterial Screening Hit: Synthesis and Biological Activity against the ESKAPE Panel of Pathogens.

Published in:

Antibiotics (2079-6382), 2020, v. 9, n. 10, p. 666, doi. 10.3390/antibiotics9100666

By:

Chuprun, Sergey;
Dar'in, Dmitry;
Rogacheva, Elizaveta;
Kraeva, Liudmila;
Levin, Oleg;
Manicheva, Olga;
Dogonadze, Marine;
Vinogradova, Tatiana;
Bakulina, Olga;
Krasavin, Mikhail

Publication type:

Article

Catalyst Loading Controls Chemoselectivity: Unusual Effect in Rhodium(II) Carbene Insertion Reactions with Tetrahydrofuran †.

Published in:

Catalysts (2073-4344), 2023, v. 13, n. 2, p. 428, doi. 10.3390/catal13020428

By:

Kazantsev, Alexander;
Rodionov, Ivan A.;
Bakulina, Olga;
Kantin, Grigory;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Synthetic Exploration of Novel Sulfamoyl Cyanide N‐Oxides in Heterocycle Synthesis.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 46, p. 1, doi. 10.1002/ejoc.202201162

By:

Krivovicheva, Vasilisa;
Bubyrev, Andrey;
Kalinin, Stanislav;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Steric Push towards the [n+3] Hydrated Imidazoline Ring Expansion (HIRE) of Dibenzo[1.4]oxazepines and Thiazepines.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 35, p. 1, doi. 10.1002/ejoc.202200818

By:

Lavit, Ksenia;
Sapegin, Alexander;
Linnik, Stanislav;
Ryazantsev, Mikhail;
Krasavin, Mikhail

Publication type:

Article

Homophthalic Esters: A New Type of Reagents for the Castagnoli‐Cushman Reaction.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 9, p. 1, doi. 10.1002/ejoc.202101281

By:

Guranova, Natalia;
Bakulina, Olga;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Oxonium Ylides Generated from 1,4‐Disubstituted α‐Diazo Glutaconimides: a Rich Source of Diverse Oxygen Heterocyclic Frameworks.

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 23, p. 3411, doi. 10.1002/ejoc.202100515

By:

Guranova, Natalia;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Cover Feature: Three‐Component Castagnoli‐Cushman Reaction of 3‐Arylglutaconic Acid Anhydrides, Carbonyl Compounds, and Ammonium Acetate: a Quick and Flexible Way to Assemble Polysubstituted NH‐δ‐lactams (Eur. J. Org. Chem. 11/2021)

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 11, p. 1773, doi. 10.1002/ejoc.202100298

By:

Peshkov, Anatoly A.;
Bakulina, Olga;
Dar'in, Dmitry;
Kantin, Grigory;
Bannykh, Anton;
Peshkov, Vsevolod A.;
Krasavin, Mikhail

Publication type:

Article

Three‐Component Castagnoli‐Cushman Reaction of 3‐Arylglutaconic Acid Anhydrides, Carbonyl Compounds, and Ammonium Acetate: a Quick and Flexible Way to Assemble Polysubstituted NH‐δ‐lactams.

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 11, p. 1726, doi. 10.1002/ejoc.202001617

By:

Peshkov, Anatoly A.;
Bakulina, Olga;
Dar'in, Dmitry;
Kantin, Grigory;
Bannykh, Anton;
Peshkov, Vsevolod A.;
Krasavin, Mikhail

Publication type:

Article

Diazo Glutaconimides: an Unexplored Type of Heterocyclic α-Diazocarbonyl Compounds Conveniently Evolved into Pyridine-2,6(1H,3H)-diones and Oxazolo[5,4-b]pyridin-5(4H)-ones.

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 4, p. 623, doi. 10.1002/ejoc.202001451

By:

Guranova, Natalia;
Kantin, Grigory;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Front Cover: An Alternative Approach to the Hydrated Imidazoline Ring Expansion (HIRE) of Diarene‐Fused [1.4]Oxazepines (Eur. J. Org. Chem. 35/2020).

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 35, p. 5635, doi. 10.1002/ejoc.202001186

By:

Grintsevich, Sergey;
Sapegin, Alexander;
Reutskaya, Elena;
Peintner, Stefan;
Erdélyi, Máté;
Krasavin, Mikhail

Publication type:

Article

An Alternative Approach to the Hydrated Imidazoline Ring Expansion (HIRE) of Diarene‐Fused [1.4]Oxazepines.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 35, p. 5664, doi. 10.1002/ejoc.202000789

By:

Grintsevich, Sergey;
Sapegin, Alexander;
Reutskaya, Elena;
Peintner, Stefan;
Erdélyi, Máté;
Krasavin, Mikhail

Publication type:

Article

1,3,5‐Triazinanes as Formaldimine Surrogates in the Ugi Reaction.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 29, p. 4517, doi. 10.1002/ejoc.202000569

By:

Golubev, Pavel;
Guranova, Natalia;
Krasavin, Mikhail

Publication type:

Article

Cover Feature: Synthetic Studies towards CH‐Diazomethane Sulfonamides: a Novel Type of Diazo Reagents (Eur. J. Org. Chem. 27/2020)

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 27, p. 4068, doi. 10.1002/ejoc.202000948

By:

Bubyrev, Andrey;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

From Rare Reagents to Rare Products: Regiospecific Silver-Catalyzed [3+2] Cycloaddition of Aryl-, Alkyl- and Aminosulfonyl Diazomethanes with Arenediazonium Tosylates.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 27, p. 4239, doi. 10.1002/ejoc.202000619

By:

Levashova, Ekaterina;
Bakulina, Olga;
Dar'in, Dmitry;
Bubyrev, Andrey;
Chuprun, Sergey;
Krasavin, Mikhail

Publication type:

Article

Synthetic Studies towards CH-Diazomethane Sulfonamides: a Novel Type of Diazo Reagents.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 27, p. 4112, doi. 10.1002/ejoc.202000446

By:

Bubyrev, Andrey;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Cover Feature: tert‐Butyl 3‐Diazo‐2‐oxopyrrolidine‐1‐carboxylate – A New Reagent for Introduction of the 2‐Oxopyrrolidin‐3‐yl Motif via RhII‐Catalyzed X–H Insertion Reactions (Eur. J. Org. Chem. 20/2020)

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 20, p. 2980, doi. 10.1002/ejoc.202000639

By:

Zhukovsky, Daniil;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

tert‐Butyl 3‐Diazo‐2‐oxopyrrolidine‐1‐carboxylate – A New Reagent for Introduction of the 2‐Oxopyrrolidin‐3‐yl Motif via RhII‐Catalyzed X–H Insertion Reactions.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 20, p. 3013, doi. 10.1002/ejoc.202000067

By:

Zhukovsky, Daniil;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Cover Feature: Convenient Approach to 2‐Substituted (Thio)morpholin‐3‐ones from α‐Diazoacetates via X‐H Carbene Insertion – Lactamization Sequence (Eur. J. Org. Chem. 45/2019).

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 45, p. 7400, doi. 10.1002/ejoc.201901632

By:

Solovyov, Igor;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Convenient Approach to 2‐Substituted (Thio)morpholin‐3‐ones from α‐Diazoacetates via X‐H Carbene Insertion – Lactamization Sequence.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 45, p. 7432, doi. 10.1002/ejoc.201901238

By:

Solovyov, Igor;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Employing α‐Diazocarbonyl Compound Chemistry in the Assembly of Medicinally Important Aryl(alkyl)thiolactam Scaffold.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 33, p. 5798, doi. 10.1002/ejoc.201900944

By:

Barkhatova, Darina;
Zhukovsky, Daniil;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Convenient Assembly of Privileged (Hetero)Arene‐Fused Benzo[1.4]oxazepines by Two Tandem SNAr Events. Part 2 – The Use of o‐[N‐(Hetero)aryl]aminomethyl Phenols.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 31/32, p. 5242, doi. 10.1002/ejoc.201900264

By:

Firsov, Andrey;
Sapegin, Alexander;
Krasavin, Mikhail

Publication type:

Article

Convenient Assembly of Privileged (Hetero)Arene‐Fused Benzo[1.4]oxazepines via Two Tandem SNAr Events. Part 1 – On the Importance of the Intermittent Smiles Rearrangement.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 31/32, p. 5234, doi. 10.1002/ejoc.201900263

By:

Sapegin, Alexander;
Krasavin, Mikhail

Publication type:

Article

α‐Diazo‐β‐oxosulfones as Partners in the Wolff 1,2,3‐Triazole Synthesis and the Wolff Rearrangement in the Presence of Aromatic Amines.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 29, p. 4721, doi. 10.1002/ejoc.201900698

By:

Safrygin, Alexander;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Rh2(esp)2‐Catalyzed Coupling of α‐Diazo‐γ‐butyrolactams with Aromatic Amines.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 27, p. 4377, doi. 10.1002/ejoc.201900565

By:

Zhukovsky, Daniil;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Synthetic Exploration of α‐Diazo γ‐Butyrolactams.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 13, p. 2397, doi. 10.1002/ejoc.201900133

By:

Zhukovsky, Daniil;
Dar'in, Dmitry;
Kantin, Grigory;
Krasavin, Mikhail

Publication type:

Article

Ligands for cereblon: 2017–2021 patent overview.

Published in:

Expert Opinion on Therapeutic Patents, 2022, v. 32, n. 2, p. 171, doi. 10.1080/13543776.2022.1999415

By:

Kazantsev, Alexander;
Krasavin, Mikhail

Publication type:

Article

Thioredoxin reductase inhibitors: updated patent review (2017-present).

Published in:

Expert Opinion on Therapeutic Patents, 2021, v. 31, n. 8, p. 745, doi. 10.1080/13543776.2021.1899160

By:

Chupakhin, Evgeny;
Krasavin, Mikhail

Publication type:

Article

Natural products as templates for bioactive compound libraries: Part 2. Novel modifications of vasicine (peganine) core via efficient and regioselective generation of 3-lithiodeoxyvasicine and its stereoselective addition to aliphatic ketones§.

Published in:

Natural Product Research, 2006, v. 20, n. 9, p. 871, doi. 10.1080/14786410500480993

By:

Shevyakov, Sergey V.;
Davydova, Olga I.;
Kiselyov, Alex S.;
Kravchenko, Dmitry V.;
Ivachtchenko, Alexandre V.;
Krasavin, Mikhail

Publication type:

Article

Natural products as templates for bioactive compound libraries: synthesis of biaryl derivatives of (±)-vasicine.

Published in:

Natural Product Research, 2006, v. 20, n. 8, p. 735, doi. 10.1080/14786410500247418

By:

Shevyakov, Sergey V.;
Davydova, Olga I.;
Pershin, Dmitry G.;
Krasavin, Mikhail;
Kravchenko, Dmitry V.;
Kiselyov, Alex;
Tkachenko, Sergey E.;
Ivachtchenko, Alexandre V.

Publication type:

Article

Castagnoli‐Cushman Reaction of 3‐Aryl Glutaric Acids: A Convenient, Diastereoselective Reaction for 6‐Oxo‐2,4‐diarylpiperidine‐3‐carboxylic Acid Scaffold.

Published in:

ChemistrySelect, 2022, v. 7, n. 3, p. 1, doi. 10.1002/slct.202104011

By:

Paramonova, Polina;
Bakulina, Olga;
Nabiyev, Alem;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Catalyst‐Free Synthesis of Diastereomerically Pure 3‐Cyanoazetidin‐2‐ones via Thermally Promoted Tandem Wolff Rearrangement–Staudinger [2+2] Cycloaddition.

Published in:

ChemistrySelect, 2021, v. 6, n. 47, p. 13582, doi. 10.1002/slct.202103446

By:

Levashova, Ekaterina;
Bakulina, Olga;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Replacing the phthalimide core in thalidomide with benzotriazole.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 527, doi. 10.1080/14756366.2021.2024525

By:

Krasavin, Mikhail;
Bubyrev, Andrey;
Kazantsev, Alexander;
Heim, Christopher;
Maiwald, Samuel;
Zhukovsky, Daniil;
Dar'in, Dmitry;
Hartmann, Marcus D.;
Bunev, Alexander

Publication type:

Article

Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 857, doi. 10.1080/14756366.2022.2051023

By:

Sharonova, Tatiana;
Zhmurov, Petr;
Kalinin, Stanislav;
Nocentini, Alessio;
Angeli, Andrea;
Ferraroni, Marta;
Korsakov, Mikhail;
Supuran, Claudiu T.;
Krasavin, Mikhail

Publication type:

Article

5-(Sulfamoyl)thien-2-yl 1,3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1005, doi. 10.1080/14756366.2022.2056733

By:

Kalinin, Stanislav;
Kovalenko, Alexander;
Valtari, Annika;
Nocentini, Alessio;
Gureev, Maxim;
Urtti, Arto;
Korsakov, Mikhail;
Supuran, Claudiu T.;
Krasavin, Mikhail

Publication type:

Article

1-Oxo-3,4-dihydroisoquinoline-4-carboxamides as novel druglike inhibitors of poly(ADP-ribose) polymerase (PARP) with favourable ADME characteristics.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1968, doi. 10.1080/14756366.2021.1972993

By:

Safrygin, Alexander;
Zhmurov, Petr;
Dar'in, Dmitry;
Silonov, Sergey;
Kasatkina, Mariia;
Zonis, Yulia;
Gureev, Maxim;
Krasavin, Mikhail

Publication type:

Article

Three-component Castagnoli-Cushman reaction with ammonium acetate delivers 2-unsubstituted isoquinol-1-ones as potent inhibitors of poly(ADP-ribose) polymerase (PARP).

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1916, doi. 10.1080/14756366.2021.1969386

By:

Safrygin, Alexander;
Zhmurov, Petr;
Dar'in, Dmitry;
Silonov, Sergey;
Kasatkina, Mariia;
Zonis, Yulia;
Gureev, Maxim;
Krasavin, Mikhail

Publication type:

Article

Strained contacts with the cell membrane may influence ligand affinity to G protein coupled receptors: a case of free fatty acid receptor 1 agonists.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1650, doi. 10.1080/14756366.2021.1955874

By:

Lukin, Alexey;
Bakholdina, Anna;
Chudinov, Mikhail;
Onopchenko, Oleksandra;
Zhuravel, Elena;
Zozulya, Sergey;
Gureev, Maxim;
Krasavin, Mikhail

Publication type:

Article