Works matching AU Kovaříková, Petra


Results: 17
    1

    Structure-Activity Relationships of Novel Salicylaldehyde Isonicotinoyl Hydrazone (SIH) Analogs: Iron Chelation, Anti-Oxidant and Cytotoxic Properties.

    Published in:
    PLoS ONE, 2014, v. 9, n. 11, p. 1, doi. 10.1371/journal.pone.0112059
    By:
    • Potůčková, Eliška;
    • Hrušková, Kateřina;
    • Bureš, Jan;
    • Kovaříková, Petra;
    • Špirková, Iva A.;
    • Pravdíková, Kateřina;
    • Kolbabová, Lucie;
    • Hergeselová, Tereza;
    • Hašková, Pavlína;
    • Jansová, Hana;
    • Macháček, Miloslav;
    • Jirkovská, Anna;
    • Richardson, Vera;
    • Lane, Darius J. R.;
    • Kalinowski, Danuta S.;
    • Richardson, Des R.;
    • Vávrová, Kateřina;
    • Šimůnek, Tomáš
    Publication type:
    Article
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    Development of water-soluble prodrugs of the bisdioxopiperazine topoisomerase IIβ inhibitor ICRF-193 as potential cardioprotective agents against anthracycline cardiotoxicity.

    Published in:
    Scientific Reports, 2021, v. 11, n. 1, p. 1, doi. 10.1038/s41598-021-83688-x
    By:
    • Bavlovič Piskáčková, Hana;
    • Jansová, Hana;
    • Kubeš, Jan;
    • Karabanovich, Galina;
    • Váňová, Nela;
    • Kollárová-Brázdová, Petra;
    • Melnikova, Iuliia;
    • Jirkovská, Anna;
    • Lenčová-Popelová, Olga;
    • Chládek, Jaroslav;
    • Roh, Jaroslav;
    • Šimůnek, Tomáš;
    • Štěrba, Martin;
    • Štěrbová-Kovaříková, Petra
    Publication type:
    Article
    5

    A hit expansion of 3‐benzamidopyrazine‐2‐carboxamide: Toward inhibitors of prolyl‐tRNA synthetase with antimycobacterial activity.

    Published in:
    Archiv der Pharmazie, 2024, v. 357, n. 8, p. 1, doi. 10.1002/ardp.202400171
    By:
    • Pallabothula, Vinod Sukanth Kumar;
    • Abdalrahman, Nechirwan Taimur;
    • Mori, Matteo;
    • Fekri, Amir Hossein;
    • Janďourek, Ondřej;
    • Konečná, Klára;
    • Paterová, Pavla;
    • Novák, Martin;
    • Dudášová‐Hatoková, Paulína;
    • Štěrbová‐Kovaříková, Petra;
    • Castellano, Carlo;
    • Meneghetti, Fiorella;
    • Villa, Stefania;
    • Kuneš, Jiří;
    • Juhás, Martin;
    • Zitko, Jan
    Publication type:
    Article
    6

    Topobexin targets the Topoisomerase II ATPase domain for beta isoform-selective inhibition and anthracycline cardioprotection.

    Published in:
    Nature Communications, 2025, v. 16, n. 1, p. 1, doi. 10.1038/s41467-025-60167-9
    By:
    • Kubeš, Jan;
    • Karabanovich, Galina;
    • Cong, Anh T. Q.;
    • Melnikova, Iuliia;
    • Lenčová, Olga;
    • Kollárová, Petra;
    • Bavlovič Piskáčková, Hana;
    • Keresteš, Veronika;
    • Applová, Lenka;
    • Arrouye, Lise C. M.;
    • Alvey, Julia R.;
    • Paluncic, Jasmina;
    • Witter, Taylor L.;
    • Jirkovská, Anna;
    • Kuneš, Jiří;
    • Štěrbová-Kovaříková, Petra;
    • Austin, Caroline A.;
    • Štěrba, Martin;
    • Šimůnek, Tomáš;
    • Roh, Jaroslav
    Publication type:
    Article
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    9

    Novel SPME fibers based on a plastic support for determination of plasma protein binding of thiosemicarbazone metal chelators: a case example of DpC, an anti-cancer drug that entered clinical trials.

    Published in:
    Analytical & Bioanalytical Chemistry, 2019, v. 411, n. 11, p. 2383, doi. 10.1007/s00216-019-01681-w
    By:
    • Reimerová, Petra;
    • Stariat, Ján;
    • Bavlovič Piskáčková, Hana;
    • Jansová, Hana;
    • Roh, Jaroslav;
    • Kalinowski, Danuta S.;
    • Macháček, Miloslav;
    • Šimůnek, Tomáš;
    • Richardson, Des R.;
    • Štěrbová-Kovaříková, Petra
    Publication type:
    Article
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    15

    Simultaneous determination of the novel thiosemicarbazone anti-cancer agent, Bp4eT, and its main phase I metabolites in plasma: Application to a pilot pharmacokinetic study in rats.

    Published in:
    Biomedical Chromatography, 2014, v. 28, n. 5, p. 621, doi. 10.1002/bmc.3080
    By:
    • Stariat, Ján;
    • Suprunová, Vlasta;
    • Roh, Jaroslav;
    • Šesták, Vít;
    • Eisner, Tomáš;
    • Filipský, Tomáš;
    • Mladěnka, Přemysl;
    • Nobilis, Milan;
    • Šimůnek, Tomáš;
    • Klimeš, Jiří;
    • Kalinowski, Danuta S.;
    • Richardson, Des R.;
    • Kovaříková, Petra
    Publication type:
    Article
    16

    Prodrug of ICRF-193 provides promising protective effects against chronic anthracycline cardiotoxicity in a rabbit model in vivo.

    Published in:
    Clinical Science, 2021, v. 135, n. 15, p. 1897, doi. 10.1042/CS20210311
    By:
    • Kollárová-Brázdová, Petra;
    • Lenčová-Popelová, Olga;
    • Karabanovich, Galina;
    • Kocu'rová-Lengvarská, Júlia;
    • Kubeš, Jan;
    • Váňová, Nela;
    • Mazurová, Yvona;
    • Adamcová, Michaela;
    • Jirkovská, Anna;
    • Holečková, Magdalena;
    • Šimůnek, Tomáš;
    • Štěrbová-Kovaříková, Petra;
    • Roh, Jaroslav;
    • Štěrba, Martin
    Publication type:
    Article
    17

    Exploring the effects of topoisomerase II inhibitor XK469 on anthracycline cardiotoxicity and DNA damage.

    Published in:
    Toxicological Sciences, 2024, v. 198, n. 2, p. 288, doi. 10.1093/toxsci/kfae008
    By:
    • Keresteš, Veronika;
    • Kubeš, Jan;
    • Applová, Lenka;
    • Kollárová, Petra;
    • Lenčová-Popelová, Olga;
    • Melnikova, Iuliia;
    • Karabanovich, Galina;
    • Khazeem, Mushtaq M;
    • Bavlovič-Piskáčková, Hana;
    • Štěrbová-Kovaříková, Petra;
    • Austin, Caroline A;
    • Roh, Jaroslav;
    • Štěrba, Martin;
    • Šimůnek, Tomáš;
    • Jirkovská, Anna
    Publication type:
    Article