Works by Kothayer, Hend

Results: 11

Design, computational studies, synthesis and in vitro antimicrobial evaluation of benzimidazole based thio-oxadiazole and thio-thiadiazole analogues.

Published in:

BMC Chemistry, 2021, v. 15, n. 1, p. 1, doi. 10.1186/s13065-021-00785-8

By:

Noureldin, Nada A.;
Richards, Jennifer;
Kothayer, Hend;
Baraka, Mohammed M.;
Eladl, Sobhy M.;
Wootton, Mandy;
Simons, Claire

Publication type:

Article

The neuroprotective effect of a novel 1,4‐Dihydroquinazolin‐3(2H)‐yl benzamide derivative against chronic constriction injury‐induced neuropathic pain in rats.

Published in:

FASEB Journal, 2022, v. 36, p. N.PAG, doi. 10.1096/fasebj.2022.36.S1.R6301

By:

Rezq, Samar;
Sakr, Asmaa;
Kothayer, Hend;
Hassan, Nancy H.;
Alsemeh, Amira

Publication type:

Article

Triple targeting of mutant EGFR<sup>L858R/T790M</sup>, COX-2, and 15-LOX: design and synthesis of novel quinazolinone tethered phenyl urea derivatives for anti-inflammatory and anticancer evaluation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2199166

By:

Kothayer, Hend;
Rezq, Samar;
Abdelkhalek, Ahmed S.;
Romero, Damian G.;
Elbaramawi, Samar S.

Publication type:

Article

Design and synthesis of novel quinazolinones conjugated ibuprofen, indole acetamide, or thioacetohydrazide as selective COX-2 inhibitors: anti-inflammatory, analgesic and anticancer activities.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1810, doi. 10.1080/14756366.2021.1956912

By:

Sakr, Asmaa;
Rezq, Samar;
Ibrahim, Samy M.;
Soliman, Eman;
Baraka, Mohamed M.;
Romero, Damian G.;
Kothayer, Hend

Publication type:

Article

Synthesis, in vivo and in silico evaluation of novel 2,3‐dihydroquinazolin‐4(1H)‐one derivatives as potential anticonvulsant agents.

Published in:

Drug Development Research, 2019, v. 80, n. 3, p. 343, doi. 10.1002/ddr.21506

By:

Kothayer, Hend;
Ibrahim, Samy M.;
Soltan, Moustafa K.;
Rezq, Samar;
Mahmoud, Shireen S.

Publication type:

Article

Novel 2‐[thio]acetamide linked quinazoline/1,2,4‐triazole/chalcone hybrids: Design, synthesis, and anticancer activity as EGFR inhibitors and apoptotic inducers.

Published in:

Archiv der Pharmazie, 2024, v. 357, n. 7, p. 1, doi. 10.1002/ardp.202300627

By:

Abdelkhalek, Ahmed S.;
Kothayer, Hend;
Soltan, Mostafa K.;
Ibrahim, Samy M.;
Elbaramawi, Samar S.

Publication type:

Article

Synthesis of 1,2,4‐triazole and 1,3,4‐oxadiazole derivatives as inhibitors for STAT3 enzymes of breast cancer.

Published in:

Archiv der Pharmazie, 2023, v. 356, n. 11, p. 1, doi. 10.1002/ardp.202300345

By:

Fawzy, Sherif M.;
Loksha, Yasser M.;
El‐Sadek, Mohamed;
Ibrahim, Samy M.;
Beshay, Botros Y.;
Shamaa, Marium M.;
Kothayer, Hend

Publication type:

Article

Quinazoline‐tethered hydrazone: A versatile scaffold toward dual anti‐TB and EGFR inhibition activities in NSCLC.

Published in:

Archiv der Pharmazie, 2021, v. 354, n. 12, p. 1, doi. 10.1002/ardp.202100281

By:

Emam, Aya M.;
Dahal, Achyut;
Singh, Sitanshu S.;
Tosso, Rodrigo D.;
Ibrahim, Samy M.;
El‐Sadek, Mohamed;
Jois, Seetharama D.;
Enriz, Ricardo D.;
Kothayer, Hend

Publication type:

Article

Synthesis, Anticonvulsant Activity, and SAR Study of Novel 4-Quinazolinone Derivatives.

Published in:

Archiv der Pharmazie, 2017, v. 350, n. 2, p. n/a, doi. 10.1002/ardp.201600332

By:

Noureldin, Nada A.;
Kothayer, Hend;
Lashine, El ‐ Sayed M.;
Baraka, Mohamed M.;
El ‐ Eraky, Wafaa;
Awdan, Sally A. El

Publication type:

Article

Vitamin D3 mitigates myopathy and metabolic dysfunction in rats with metabolic syndrome: the potential role of dipeptidyl peptidase-4.

Published in:

Naunyn-Schmiedeberg's Archives of Pharmacology, 2025, v. 398, n. 4, p. 3697, doi. 10.1007/s00210-024-03439-3

By:

Shoier, Nourhan O.;
Ghareib, Salah A.;
Kothayer, Hend;
Alsemeh, Amira Ebrahim;
El-Sayed, Shaimaa S.

Publication type:

Article

Synthesis of New 2,3-Dihydroquinazolin-4(1 H)-one Derivatives for Analgesic and Anti-inflammatory Evaluation.

Published in:

Archiv der Pharmazie, 2010, v. 343, n. 5, p. 274, doi. 10.1002/ardp.200900220

By:

El-Sabbagh, Osama I.;
Ibrahim, Samy M.;
Baraka, Mohamed M.;
Kothayer, Hend

Publication type:

Article