Works by Kostenis, Evi
Results: 71
Chemisch‐biologischer Werkzeugkasten für die intrazelluläre Bindungsstelle von CCR9: Fluoreszierende Liganden, neue Leitstrukturen und PROTACs.
- Published in:
- Angewandte Chemie, 2022, v. 134, n. 12, p. 1, doi. 10.1002/ange.202116782
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- Publication type:
- Article
Deconvolution of complex G protein–coupled receptor signaling in live cells using dynamic mass redistribution measurements.
- Published in:
- Nature Biotechnology, 2010, v. 28, n. 9, p. 943, doi. 10.1038/nbt.1671
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- Publication type:
- Article
Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity.
- Published in:
- FASEB Journal, 2009, v. 23, n. 2, p. 442, doi. 10.1096/fj.08-114751
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- Publication type:
- Article
Muscarinic Allosteric Modulators: Atypical Structure-Activity-Relationships in Bispyridinium-type Compounds.
- Published in:
- Archiv der Pharmazie, 2006, v. 339, n. 4, p. 207, doi. 10.1002/ardp.200600005
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- Publication type:
- Article
Novel clusters of receptors for sphingosine‐1‐phosphate, sphingosylphosphorylcholine, and (lyso)‐phosphatidic acid: New receptors for “Old” ligands.
- Published in:
- Journal of Cellular Biochemistry, 2004, v. 92, n. 5, p. 923, doi. 10.1002/jcb.20092
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- Publication type:
- Article
The molecular mechanism by which saturated lysophosphatidylcholine attenuates the metastatic capacity of melanoma cells.
- Published in:
- FEBS Open Bio, 2016, v. 6, n. 12, p. 1297, doi. 10.1002/2211-5463.12152
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- Publication type:
- Article
Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling.
- Published in:
- Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-53770-9
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- Publication type:
- Article
GPR55 regulates cannabinoid 2 receptor-mediated responses in human neutrophils.
- Published in:
- 2011
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- Publication type:
- Correction Notice
GPR55 regulates cannabinoid 2 receptor-mediated responses in human neutrophils.
- Published in:
- Cell Research, 2011, v. 21, n. 10, p. 1452, doi. 10.1038/cr.2011.60
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- Publication type:
- Article
G protein-mediated signal transduction: a molecular choreography of G protein activation after GTP binding.
- Published in:
- Signal Transduction & Targeted Therapy, 2024, v. 9, n. 1, p. 1, doi. 10.1038/s41392-024-01903-3
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- Publication type:
- Article
Exploring Biased Agonism at FPR1 as a Means to Encode Danger Sensing †.
- Published in:
- Cells (2073-4409), 2020, v. 9, n. 4, p. 1054, doi. 10.3390/cells9041054
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- Publication type:
- Article
Selective optogenetic control of G<sub>q</sub> signaling using human Neuropsin.
- Published in:
- Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29265-w
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- Publication type:
- Article
Adipocyte G<sub>q</sub> signaling is a regulator of glucose and lipid homeostasis in mice.
- Published in:
- Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29231-6
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- Publication type:
- Article
Direct targeting of Gα<sub>q</sub> and Gα<sub>11</sub> oncoproteins in cancer cells.
- Published in:
- Science Signaling, 2019, v. 12, n. 573, p. N.PAG, doi. 10.1126/scisignal.aau5948
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- Publication type:
- Article
FZD<sub>5</sub> is a Gαq-coupled receptor that exhibits the functional hallmarks of prototypical GPCRs.
- Published in:
- Science Signaling, 2018, v. 11, n. 559, p. 1, doi. 10.1126/scisignal.aar5536
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- Publication type:
- Article
Pharmacological profile of NOP receptors coupled with calcium signaling via the chimeric protein Gα<sub>qi5</sub>.
- Published in:
- Naunyn-Schmiedeberg's Archives of Pharmacology, 2009, v. 379, n. 6, p. 599, doi. 10.1007/s00210-009-0396-x
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- Publication type:
- Article
Effects of human urotensin II in isolated vessels of various species; comparison with other vasoactive agents.
- Published in:
- Naunyn-Schmiedeberg's Archives of Pharmacology, 2002, v. 365, n. 2, p. 141, doi. 10.1007/s00210-001-0503-0
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- Publication type:
- Article
Muscarinic allosteric modulation: M<sub>2</sub>/M<sub>3</sub> subtype selectivity of gallamine is independent of G-protein coupling specificity.
- Published in:
- Naunyn-Schmiedeberg's Archives of Pharmacology, 2001, v. 364, n. 2, p. 172, doi. 10.1007/s002100100441
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- Publication type:
- Article
GRK specificity and Gβγ dependency determines the potential of a GPCR for arrestin-biased agonism.
- Published in:
- Communications Biology, 2024, p. 1, doi. 10.1038/s42003-024-06490-1
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- Publication type:
- Article
Community guidelines for GPCR ligand bias: IUPHAR review 32.
- Published in:
- British Journal of Pharmacology, 2022, v. 179, n. 14, p. 3651, doi. 10.1111/bph.15811
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- Publication type:
- Article
The G<sub>q</sub> signalling pathway inhibits brown and beige adipose tissue.
- Published in:
- Nature Communications, 2016, v. 7, n. 3, p. 10895, doi. 10.1038/ncomms10895
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- Publication type:
- Article
β-Arrestin 2 Inhibits Proinflammatory Chemokine Production and Attenuates Contact Allergic Inflammation in the Skin.
- Published in:
- Journal of Investigative Dermatology, 2014, v. 134, n. 8, p. 2131, doi. 10.1038/jid.2014.117
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- Publication type:
- Article
Mice Lacking Free Fatty Acid Receptor 1 (GPR40/FFAR1) are Protected Against Conjugated Linoleic Acid-Induced Fatty Liver but Develop Inflammation and Insulin Resistance in the Brain.
- Published in:
- Cellular Physiology & Biochemistry (Karger AG), 2015, v. 35, n. 6, p. 2272, doi. 10.1159/000374031
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- Publication type:
- Article
Fluid Shear Stress Differentially Regulates gpr3, gpr6, and gpr12 Expression in Human Umbilical Vein Endothelial Cells.
- Published in:
- Cellular Physiology & Biochemistry (Karger AG), 2003, v. 13, n. 2, p. 75, doi. 10.1159/000070251
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- Publication type:
- Article
Leanness and Low Plasma Leptin in GPR17 Knockout Mice Are Dependent on Strain and Associated With Increased Energy Intake That Is Not Suppressed by Exogenous Leptin.
- Published in:
- Frontiers in Endocrinology, 2021, v. 12, p. 1, doi. 10.3389/fendo.2021.698115
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- Publication type:
- Article
Front Cover: Development of a NanoBRET Assay Platform to Detect Intracellular Ligands for the Chemokine Receptors CCR6 and CXCR1 (ChemMedChem 20/2024).
- Published in:
- ChemMedChem, 2024, v. 19, n. 20, p. 1, doi. 10.1002/cmdc.202482001
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- Publication type:
- Article
Development of a NanoBRET Assay Platform to Detect Intracellular Ligands for the Chemokine Receptors CCR6 and CXCR1.
- Published in:
- ChemMedChem, 2024, v. 19, n. 20, p. 1, doi. 10.1002/cmdc.202400284
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- Publication type:
- Article
The Bacterial G<sub>q</sub> Signal Transduction Inhibitor FR900359 Impairs Soil-Associated Nematodes.
- Published in:
- Journal of Chemical Ecology, 2023, v. 49, n. 9/10, p. 549, doi. 10.1007/s10886-023-01442-1
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- Publication type:
- Article
A Chemical Biology Toolbox Targeting the Intracellular Binding Site of CCR9: Fluorescent Ligands, New Drug Leads and PROTACs.
- Published in:
- Angewandte Chemie International Edition, 2022, v. 61, n. 12, p. 1, doi. 10.1002/anie.202116782
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- Publication type:
- Article
Chemically engineering ligand selectivity at the free fatty acid receptor 2 based on pharmacological variation between species orthologs.
- Published in:
- FASEB Journal, 2012, v. 26, n. 12, p. 4951, doi. 10.1096/fj.12-213314
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- Publication type:
- Article
An optical dynamic mass redistribution assay reveals biased signaling of dualsteric GPCR activators.
- Published in:
- Journal of Receptors & Signal Transduction, 2009, v. 29, n. 3/4, p. 140, doi. 10.1080/10799890903047437
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- Publication type:
- Article
POTENTIATION OF GPCR-SIGNALING VIA MEMBRANE TARGETING OF G PROTEIN α SUBUNITS.
- Published in:
- Journal of Receptors & Signal Transduction, 2002, v. 22, n. 1-4, p. 267, doi. 10.1081/RRS-120014601
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- Publication type:
- Article
Reply to: How carvedilol does not activate β<sub>2</sub>-adrenoceptors.
- Published in:
- 2023
- By:
- Publication type:
- Letter
Author Correction: Selective optogenetic control of G<sub>q</sub> signaling using human Neuropsin.
- Published in:
- 2023
- By:
- Publication type:
- Correction Notice
Selective optogenetic control of G<sub>q</sub> signaling using human Neuropsin.
- Published in:
- Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29265-w
- By:
- Publication type:
- Article
RXFP1 Receptor Activation by Relaxin-2 Induces Vascular Relaxation in Mice via a Gα<sub>i2</sub>-Protein/PI3Kß/γ/Nitric Oxide-Coupled Pathway.
- Published in:
- Frontiers in Physiology, 2018, p. 1, doi. 10.3389/fphys.2018.01234
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- Publication type:
- Article
Targeted inhibition of G<sub>q</sub> signaling induces airway relaxation in mouse models of asthma.
- Published in:
- Science Translational Medicine, 2017, v. 9, n. 407, p. 1, doi. 10.1126/scitranslmed.aag2288
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- Publication type:
- Article
Deciphering Specificity Determinants for FR900359‐Derived G<sub>q</sub>α Inhibitors Based on Computational and Structure–Activity Studies.
- Published in:
- ChemMedChem, 2018, v. 13, n. 16, p. 1634, doi. 10.1002/cmdc.201800304
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- Publication type:
- Article
Front Cover: Deciphering Specificity Determinants for FR900359‐Derived G<sub>q</sub>α Inhibitors Based on Computational and Structure–Activity Studies (ChemMedChem 16/2018).
- Published in:
- ChemMedChem, 2018, v. 13, n. 16, p. 1617, doi. 10.1002/cmdc.201800521
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- Publication type:
- Article
Oxytocin-Modulated Ion Channel Ensemble Controls Depolarization, Integration and Burst Firing in CA2 Pyramidal Neurons.
- Published in:
- Journal of Neuroscience, 2022, v. 42, n. 41, p. 7707, doi. 10.1523/JNEUROSCI.0921-22.2022
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- Publication type:
- Article
Pharmacological Gq inhibition induces strong pulmonary vasorelaxation and reverses pulmonary hypertension.
- Published in:
- EMBO Molecular Medicine, 2024, v. 16, n. 8, p. 1930, doi. 10.1038/s44321-024-00096-0
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- Publication type:
- Article
The D-type prostanoid (DP) receptor enhances the signaling of chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTH2).
- Published in:
- 2011
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- Publication type:
- Abstract
Signalling and function of the human G protein-coupled receptor 55.
- Published in:
- 2010
- By:
- Publication type:
- Abstract
GPR55: signaling pathways and functions.
- Published in:
- BMC Pharmacology, 2009, v. 9, p. 1, doi. 10.1186/1471-2210-9-S2-A3
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- Publication type:
- Article
Tetrahydroimidazo[1,2‐a]pyrazine Derivatives: Synthesis and Evaluation as Gα<sub>q</sub>‐Protein Ligands.
- Published in:
- Chemistry - A European Journal, 2020, v. 26, n. 55, p. 12615, doi. 10.1002/chem.202001446
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- Publication type:
- Article
Disentangling bias between G<sub>q</sub>, GRK2, and arrestin3 recruitment to the M<sub>3</sub> muscarinic acetylcholine receptor.
- Published in:
- eLife, 2021, p. 1, doi. 10.7554/eLife.58442
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- Publication type:
- Article
GPR55 ligands promote receptor coupling to multiple signalling pathways.
- Published in:
- 2010
- By:
- Publication type:
- journal article
Rational design of dualsteric GPCR ligands: quests and promise.
- Published in:
- 2010
- By:
- Publication type:
- journal article
Author Correction: Chemokine receptor trafficking coordinates neutrophil clustering and dispersal at wounds in zebrafish.
- Published in:
- 2020
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- Publication type:
- Correction Notice
Chemokine receptor trafficking coordinates neutrophil clustering and dispersal at wounds in zebrafish.
- Published in:
- Nature Communications, 2019, v. 10, n. 1, p. 1, doi. 10.1038/s41467-019-13107-3
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- Publication type:
- Article