Works by Kostenis, Evi

Results: 71

Tetrahydroimidazo[1,2‐a]pyrazine Derivatives: Synthesis and Evaluation as Gαq‐Protein Ligands.

Published in:

Chemistry - A European Journal, 2020, v. 26, n. 55, p. 12615, doi. 10.1002/chem.202001446

By:

Küppers, Jim;
Benkel, Tobias;
Annala, Suvi;
Kimura, Kenichi;
Reinelt, Lisa;
Fleischmann, Bernd K.;
Kostenis, Evi;
Gütschow, Michael

Publication type:

Article

Leanness and Low Plasma Leptin in GPR17 Knockout Mice Are Dependent on Strain and Associated With Increased Energy Intake That Is Not Suppressed by Exogenous Leptin.

Published in:

Frontiers in Endocrinology, 2021, v. 12, p. 1, doi. 10.3389/fendo.2021.698115

By:

Wargent, Edward T.;
Ahmad, Suhaib J. S.;
Lu, Qing Richard;
Kostenis, Evi;
Arch, Jonathan R. S.;
Stocker, Claire J.

Publication type:

Article

NOP receptor pharmacological profile – A dynamic mass redistribution study.

Published in:

PLoS ONE, 2018, v. 13, n. 8, p. 1, doi. 10.1371/journal.pone.0203021

By:

Malfacini, Davide;
Simon, Katharina;
Trapella, Claudio;
Guerrini, Remo;
Zaveri, Nurulain T.;
Kostenis, Evi;
Calo’, Girolamo

Publication type:

Article

The Bacterial Gq Signal Transduction Inhibitor FR900359 Impairs Soil-Associated Nematodes.

Published in:

Journal of Chemical Ecology, 2023, v. 49, n. 9/10, p. 549, doi. 10.1007/s10886-023-01442-1

By:

Hanke, Wiebke;
Alenfelder, Judith;
Liu, Jun;
Gutbrod, Philipp;
Kehraus, Stefan;
Crüsemann, Max;
Dörmann, Peter;
Kostenis, Evi;
Scholz, Monika;
König, Gabriele M.

Publication type:

Article

Glucose-stimulated insulin secretion depends on FFA1 and Gq in neonatal mouse islets.

Published in:

Diabetologia, 2023, v. 66, n. 8, p. 1501, doi. 10.1007/s00125-023-05932-5

By:

Lorza-Gil, Estela;
Kaiser, Gabriele;
Carlein, Christopher;
Hoffmann, Markus D. A.;
König, Gabriele M.;
Haug, Sieglinde;
Prates Roma, Leticia;
Rexen Ulven, Elisabeth;
Ulven, Trond;
Kostenis, Evi;
Birkenfeld, Andreas L.;
Häring, Hans-Ulrich;
Ullrich, Susanne;
Gerst, Felicia

Publication type:

Article

Detection of free fatty acid receptor 1 expression: the critical role of negative and positive controls.

Published in:

Diabetologia, 2014, v. 57, n. 4, p. 776, doi. 10.1007/s00125-014-3161-8

By:

Teutsch, Charlott-Amelie;
Panse, Madhura;
Grundmann, Manuel;
Kaiser, Gabriele;
Kostenis, Evi;
Häring, Hans-Ulrich;
Ullrich, Susanne

Publication type:

Article

Disentangling bias between Gq, GRK2, and arrestin3 recruitment to the M3 muscarinic acetylcholine receptor.

Published in:

eLife, 2021, p. 1, doi. 10.7554/eLife.58442

By:

Flöser, Anja;
Becker, Katharina;
Kostenis, Evi;
König, Gabriele;
Krasel, Cornelius;
Kolb, Peter;
Bünemann, Moritz

Publication type:

Article

Exploring Biased Agonism at FPR1 as a Means to Encode Danger Sensing †.

Published in:

Cells (2073-4409), 2020, v. 9, n. 4, p. 1054, doi. 10.3390/cells9041054

By:

Gröper, Jieny;
König, Gabriele M.;
Kostenis, Evi;
Gerke, Volker;
Raabe, Carsten A.;
Rescher, Ursula

Publication type:

Article

Selective optogenetic control of Gq signaling using human Neuropsin.

Published in:

Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29265-w

By:

Wagdi, Ahmed;
Malan, Daniela;
Sathyanarayanan, Udhayabhaskar;
Beauchamp, Janosch S.;
Vogt, Markus;
Zipf, David;
Beiert, Thomas;
Mansuroglu, Berivan;
Dusend, Vanessa;
Meininghaus, Mark;
Schneider, Linn;
Kalthof, Bernd;
Wiegert, J. Simon;
König, Gabriele M.;
Kostenis, Evi;
Patejdl, Robert;
Sasse, Philipp;
Bruegmann, Tobias

Publication type:

Article

Adipocyte Gq signaling is a regulator of glucose and lipid homeostasis in mice.

Published in:

Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29231-6

By:

Kimura, Takefumi;
Pydi, Sai P.;
Wang, Lei;
Haspula, Dhanush;
Cui, Yinghong;
Lu, Huiyan;
König, Gabriele M.;
Kostenis, Evi;
Steinberg, Gregory R.;
Gavrilova, Oksana;
Wess, Jürgen

Publication type:

Article

RXFP1 Receptor Activation by Relaxin-2 Induces Vascular Relaxation in Mice via a Gαi2-Protein/PI3Kß/γ/Nitric Oxide-Coupled Pathway.

Published in:

Frontiers in Physiology, 2018, p. 1, doi. 10.3389/fphys.2018.01234

By:

Xiaoming Lian;
Beer-Hammer, Sandra;
König, Gabriele M.;
Kostenis, Evi;
Nürnberg, Bernd;
Gollasch, Maik

Publication type:

Article

Direct targeting of Gαq and Gα11 oncoproteins in cancer cells.

Published in:

Science Signaling, 2019, v. 12, n. 573, p. N.PAG, doi. 10.1126/scisignal.aau5948

By:

Annala, Suvi;
Eryilmaz, Funda;
Patt, Julian;
Pfeil, Eva M.;
Häberlein, Felix;
Schrage, Ramona;
Heycke, Nina;
Rick, Ulrike;
Kostenis, Evi;
Feng, Xiaodong;
Gutkind, J. Silvio;
Shridhar, Naveen;
Slodczyk, Tanja;
Tüting, Thomas;
Gaffal, Evelyn;
Yang, JuHee;
Pfeifer, Alexander;
Cervantes-Villagrana, Rodolfo Daniel;
Vázquez-Prado, José;
Inoue, Asuka

Publication type:

Article

FZD5 is a Gαq-coupled receptor that exhibits the functional hallmarks of prototypical GPCRs.

Published in:

Science Signaling, 2018, v. 11, n. 559, p. 1, doi. 10.1126/scisignal.aar5536

By:

Wright, Shane C.;
Cañizal, Maria Consuelo Alonso;
Benkel, Tobias;
Simon, Katharina;
Le Gouill, Christian;
Matricon, Pierre;
Namkung, Yoon;
Lukasheva, Viktoria;
König, Gabriele M.;
Laporte, Stéphane A.;
Carlsson, Jens;
Kostenis, Evi;
Bouvier, Michel;
Schulte, Gunnar;
Hoffmann, Carsten

Publication type:

Article

PGH1, the Precursor for the Anti-Inflammatory Prostaglandins of the 1-series, Is a Potent Activator of the Pro-Inflammatory Receptor CRTH2/DP2.

Published in:

PLoS ONE, 2012, v. 7, n. 3, p. 1, doi. 10.1371/journal.pone.0033329

By:

Schröder, Ralf;
Luzheng Xue;
Konya, Viktoria;
Martini, Lene;
Kampitsch, Nora;
Whistler, Jennifer L.;
Ulven, Trond;
Heinemann, Akos;
Pettipher, Roy;
Kostenis, Evi

Publication type:

Article

Chemically engineering ligand selectivity at the free fatty acid receptor 2 based on pharmacological variation between species orthologs.

Published in:

FASEB Journal, 2012, v. 26, n. 12, p. 4951, doi. 10.1096/fj.12-213314

By:

Hudson, Brian D.;
Christiansen, Elisabeth;
Tikhonova, Irina G.;
Grundmann, Manuel;
Kostenis, Evi;
Adams, David R.;
Ulven, Trond;
Milligan, Graeme

Publication type:

Article

Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity.

Published in:

FASEB Journal, 2009, v. 23, n. 2, p. 442, doi. 10.1096/fj.08-114751

By:

Antony, Johannes;
Kellershohn, Kerstin;
Mohr-Andrä, Marion;
Kebig, Anna;
Prilla, Stefanie;
Muth, Mathias;
Heller, Eberhard;
Disingrini, Teresa;
Dallanoce, Clelia;
Bertoni, Simona;
Schrobang, Jasmin;
Tränkle, Christian;
Kostenis, Evi;
Christopoulos, Arthur;
Höltje, Hans-Dieter;
Barocelli, Elisabetta;
De Amici, Marco;
Holzgrabe, Ulrike;
Mohr, Klaus

Publication type:

Article

GPR55 ligands promote receptor coupling to multiple signalling pathways.

Published in:

2010

By:

Henstridge, Christopher M;
Balenga, Nariman AB;
Schröder, Ralf;
Kargl, Julia K;
Platzer, Wolfgang;
Martini, Lene;
Arthur, Simon;
Penman, June;
Whistler, Jennifer L;
Kostenis, Evi;
Waldhoer, Maria;
Irving, Andrew J;
Schröder, Ralf

Publication type:

journal article

Rational design of dualsteric GPCR ligands: quests and promise.

Published in:

2010

By:

Mohr, Klaus;
Tränkle, Christian;
Kostenis, Evi;
Barocelli, Elisabetta;
De Amici, Marco;
Holzgrabe, Ulrike;
Tränkle, Christian

Publication type:

journal article

Reply to: How carvedilol does not activate β2-adrenoceptors.

Published in:

2023

By:

Kostenis, Evi;
Gomeza, Jesus;
Miess-Tanneberg, Elke;
Blum, Nina Kathleen;
Benkel, Tobias;
Chevigné, Andy;
Hoffmann, Carsten;
Kolb, Peter;
Nikolaev, Viacheslav;
Waldhoer, Maria;
Szpakowska, Martyna;
Inoue, Asuka;
Schulz, Stefan

Publication type:

Letter

Author Correction: Selective optogenetic control of Gq signaling using human Neuropsin.

Published in:

2023

By:

Wagdi, Ahmed;
Malan, Daniela;
Sathyanarayanan, Udhayabhaskar;
Beauchamp, Janosch S.;
Vogt, Markus;
Zipf, David;
Beiert, Thomas;
Mansuroglu, Berivan;
Dusend, Vanessa;
Meininghaus, Mark;
Schneider, Linn;
Kalthof, Bernd;
Wiegert, J. Simon;
König, Gabriele M.;
Kostenis, Evi;
Patejdl, Robert;
Sasse, Philipp;
Bruegmann, Tobias

Publication type:

Correction Notice

Selective optogenetic control of Gq signaling using human Neuropsin.

Published in:

Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29265-w

By:

Wagdi, Ahmed;
Malan, Daniela;
Sathyanarayanan, Udhayabhaskar;
Beauchamp, Janosch S.;
Vogt, Markus;
Zipf, David;
Beiert, Thomas;
Mansuroglu, Berivan;
Dusend, Vanessa;
Meininghaus, Mark;
Schneider, Linn;
Kalthof, Bernd;
Wiegert, J. Simon;
König, Gabriele M.;
Kostenis, Evi;
Patejdl, Robert;
Sasse, Philipp;
Bruegmann, Tobias

Publication type:

Article

A Chemical Biology Toolbox Targeting the Intracellular Binding Site of CCR9: Fluorescent Ligands, New Drug Leads and PROTACs.

Published in:

Angewandte Chemie International Edition, 2022, v. 61, n. 12, p. 1, doi. 10.1002/anie.202116782

By:

Huber, Max E.;
Toy, Lara;
Schmidt, Maximilian F.;
Vogt, Hannah;
Budzinski, Julian;
Wiefhoff, Martin F. J.;
Merten, Nicole;
Kostenis, Evi;
Weikert, Dorothee;
Schiedel, Matthias

Publication type:

Article

Novel clusters of receptors for sphingosine‐1‐phosphate, sphingosylphosphorylcholine, and (lyso)‐phosphatidic acid: New receptors for “Old” ligands.

Published in:

Journal of Cellular Biochemistry, 2004, v. 92, n. 5, p. 923, doi. 10.1002/jcb.20092

By:

Evi Kostenis

Publication type:

Article

Mice Lacking Free Fatty Acid Receptor 1 (GPR40/FFAR1) are Protected Against Conjugated Linoleic Acid-Induced Fatty Liver but Develop Inflammation and Insulin Resistance in the Brain.

Published in:

Cellular Physiology & Biochemistry (Karger AG), 2015, v. 35, n. 6, p. 2272, doi. 10.1159/000374031

By:

Sartorius, Tina;
Drescher, andrea;
Panse, Madhura;
Lastovicka, Petr;
Peter, andreas;
Weigert, Cora;
Kostenis, Evi;
Ullrich, Susanne;
Häring, Hans-Ulrich

Publication type:

Article

Fluid Shear Stress Differentially Regulates gpr3, gpr6, and gpr12 Expression in Human Umbilical Vein Endothelial Cells.

Published in:

Cellular Physiology & Biochemistry (Karger AG), 2003, v. 13, n. 2, p. 75, doi. 10.1159/000070251

By:

Uhlenbrock, Kirsten;
Huber, Jochen;
Ardati, Ali;
Busch, Andreas E.;
Kostenis, Evi

Publication type:

Article

GRK specificity and Gβγ dependency determines the potential of a GPCR for arrestin-biased agonism.

Published in:

Communications Biology, 2024, p. 1, doi. 10.1038/s42003-024-06490-1

By:

Matthees, Edda S. F.;
Filor, Jenny C.;
Jaiswal, Natasha;
Reichel, Mona;
Youssef, Noureldine;
D'Uonnolo, Giulia;
Szpakowska, Martyna;
Drube, Julia;
König, Gabriele M.;
Kostenis, Evi;
Chevigné, Andy;
Godbole, Amod;
Hoffmann, Carsten

Publication type:

Article

Pseudomonas aeruginosa ExoY, a cyclic GMP- and cyclic UMP-generating nucleotidyl cyclase.

Published in:

2013

By:

Seifert, Roland;
Hartwig, Christina;
Wolter, Sabine;
Reinecke, Daniel;
Burhenne, Heike;
Kaever, Volkhard;
Munder, Antje;
Tümmler, Burkhard;
Schwede, Frank;
Grundmann, Manuel;
Kostenis, Evi;
Frank, Dara W.;
Beckert, Ulrike

Publication type:

Abstract

Heterotrimeric G-proteins: a short history.

Published in:

British Journal of Pharmacology, 2006, p. S46, doi. 10.1038/sj.bjp.0706405

By:

Milligan, Graeme;
Kostenis, Evi

Publication type:

Article

Regulated and constitutive activation of specific signalling pathways by the human S1P5 receptor.

Published in:

British Journal of Pharmacology, 2003, v. 138, n. 3, p. 481, doi. 10.1038/sj.bjp.0705055

By:

Niedernberg, Anke;
Blaukat, Andree;
Schoneberg, Torsten;
Kostenis, Evi

Publication type:

Article

Deconvolution of complex G protein–coupled receptor signaling in live cells using dynamic mass redistribution measurements.

Published in:

Nature Biotechnology, 2010, v. 28, n. 9, p. 943, doi. 10.1038/nbt.1671

By:

Schröder, Ralf;
Janssen, Nicole;
Schmidt, Johannes;
Kebig, Anna;
Merten, Nicole;
Hennen, Stephanie;
Müller, Anke;
Blättermann, Stefanie;
Mohr-Andrä, Marion;
Zahn, Sabine;
Wenzel, Jörg;
Smith, Nicola J.;
Gomeza, Jesús;
Drewke, Christel;
Milligan, Graeme;
Mohr, Klaus;
Kostenis, Evi

Publication type:

Article

FFA2-, but not FFA3-agonists inhibit GSIS of human pseudoislets: a comparative study with mouse islets and rat INS-1E cells.

Published in:

Scientific Reports, 2020, v. 10, n. 1, p. N.PAG, doi. 10.1038/s41598-020-73467-5

By:

Lorza-Gil, Estela;
Kaiser, Gabriele;
Rexen Ulven, Elisabeth;
König, Gabriele M.;
Gerst, Felicia;
Oquendo, Morgana Barroso;
Birkenfeld, Andreas L.;
Häring, Hans-Ulrich;
Kostenis, Evi;
Ulven, Trond;
Ullrich, Susanne

Publication type:

Article

The molecular mechanism by which saturated lysophosphatidylcholine attenuates the metastatic capacity of melanoma cells.

Published in:

FEBS Open Bio, 2016, v. 6, n. 12, p. 1297, doi. 10.1002/2211-5463.12152

By:

Ross, Thomas;
Jakubzig, Bastian;
Grundmann, Manuel;
Massing, Ulrich;
Kostenis, Evi;
Schlesinger, Martin;
Bendas, Gerd

Publication type:

Article

Thioesterase-mediated side chain transesterification generates potent Gq signaling inhibitor FR900359.

Published in:

Nature Communications, 2021, v. 12, n. 1, p. 1, doi. 10.1038/s41467-020-20418-3

By:

Hermes, Cornelia;
Richarz, René;
Wirtz, Daniel A.;
Patt, Julian;
Hanke, Wiebke;
Kehraus, Stefan;
Voß, Jan Hendrik;
Küppers, Jim;
Ohbayashi, Tsubasa;
Namasivayam, Vigneshwaran;
Alenfelder, Judith;
Inoue, Asuka;
Mergaert, Peter;
Gütschow, Michael;
Müller, Christa E.;
Kostenis, Evi;
König, Gabriele M.;
Crüsemann, Max

Publication type:

Article

The atypical chemokine receptor ACKR3/CXCR7 is a broad-spectrum scavenger for opioid peptides.

Published in:

Nature Communications, 2020, v. 11, n. 1, p. 1, doi. 10.1038/s41467-020-16664-0

By:

Meyrath, Max;
Szpakowska, Martyna;
Zeiner, Julian;
Massotte, Laurent;
Merz, Myriam P.;
Benkel, Tobias;
Simon, Katharina;
Ohnmacht, Jochen;
Turner, Jonathan D.;
Krüger, Rejko;
Seutin, Vincent;
Ollert, Markus;
Kostenis, Evi;
Chevigné, Andy

Publication type:

Article

Reactivation of Gαi‐coupled formyl peptide receptors is inhibited by Gαq‐selective inhibitors when induced by signals generated by the platelet‐activating factor receptor.

Published in:

Journal of Leukocyte Biology, 2017, v. 102, n. 3, p. 871, doi. 10.1189/jlb.2A0317-086RR

By:

Holdfeldt, André;
Dahlstrand Rudin, Agnes;
Gabl, Michael;
Rajabkhani, Zahra;
König, Gabriele M.;
Kostenis, Evi;
Dahlgren, Claes;
Forsman, Huamei

Publication type:

Article

Muscarinic Allosteric Modulators: Atypical Structure-Activity-Relationships in Bispyridinium-type Compounds.

Published in:

Archiv der Pharmazie, 2006, v. 339, n. 4, p. 207, doi. 10.1002/ardp.200600005

By:

Ulf Sürig;
Klaudia Gaal;
Evi Kostenis;
Christian Tränkle;
Klaus Mohr

Publication type:

Article

An optical dynamic mass redistribution assay reveals biased signaling of dualsteric GPCR activators.

Published in:

Journal of Receptors & Signal Transduction, 2009, v. 29, n. 3/4, p. 140, doi. 10.1080/10799890903047437

By:

Kebig, Anna;
Kostenis, Evi;
Mohr, Klaus;
Mohr-Andrä, Marion

Publication type:

Article

POTENTIATION OF GPCR-SIGNALING VIA MEMBRANE TARGETING OF G PROTEIN α SUBUNITS.

Published in:

Journal of Receptors & Signal Transduction, 2002, v. 22, n. 1-4, p. 267, doi. 10.1081/RRS-120014601

By:

Kostenis, Evi

Publication type:

Article

G protein-mediated signal transduction: a molecular choreography of G protein activation after GTP binding.

Published in:

Signal Transduction & Targeted Therapy, 2024, v. 9, n. 1, p. 1, doi. 10.1038/s41392-024-01903-3

By:

Kostenis, Evi;
Jürgenliemke, Lars;
Alenfelder, Judith

Publication type:

Article

Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling.

Published in:

Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-53770-9

By:

Holze, Janine;
Lauber, Felicitas;
Soler, Sofía;
Kostenis, Evi;
Weindl, Günther

Publication type:

Article

Pharmacological Gq inhibition induces strong pulmonary vasorelaxation and reverses pulmonary hypertension.

Published in:

EMBO Molecular Medicine, 2024, v. 16, n. 8, p. 1930, doi. 10.1038/s44321-024-00096-0

By:

Seidinger, Alexander;
Roberts, Richard;
Bai, Yan;
Müller, Marion;
Pfeil, Eva;
Matthey, Michaela;
Rieck, Sarah;
Alenfelder, Judith;
König, Gabriele M;
Pfeifer, Alexander;
Kostenis, Evi;
Klinke, Anna;
Fleischmann, Bernd K;
Wenzel, Daniela

Publication type:

Article

Development of a NanoBRET Assay Platform to Detect Intracellular Ligands for the Chemokine Receptors CCR6 and CXCR1.

Published in:

ChemMedChem, 2024, v. 19, n. 20, p. 1, doi. 10.1002/cmdc.202400284

By:

Huber, Max E.;
Wurnig, Silas L.;
Moumbock, Aurélien F. A.;
Toy, Lara;
Kostenis, Evi;
Alonso Bartolomé, Ana;
Szpakowska, Martyna;
Chevigné, Andy;
Günther, Stefan;
Hansen, Finn K.;
Schiedel, Matthias

Publication type:

Article

Front Cover: Development of a NanoBRET Assay Platform to Detect Intracellular Ligands for the Chemokine Receptors CCR6 and CXCR1 (ChemMedChem 20/2024).

Published in:

ChemMedChem, 2024, v. 19, n. 20, p. 1, doi. 10.1002/cmdc.202482001

By:

Huber, Max E.;
Wurnig, Silas L.;
Moumbock, Aurélien F. A.;
Toy, Lara;
Kostenis, Evi;
Alonso Bartolomé, Ana;
Szpakowska, Martyna;
Chevigné, Andy;
Günther, Stefan;
Hansen, Finn K.;
Schiedel, Matthias

Publication type:

Article

β-Arrestin 2 Inhibits Proinflammatory Chemokine Production and Attenuates Contact Allergic Inflammation in the Skin.

Published in:

Journal of Investigative Dermatology, 2014, v. 134, n. 8, p. 2131, doi. 10.1038/jid.2014.117

By:

Gaffal, Evelyn;
Jakobs, Mira;
Glodde, Nicole;
Schröder, Ralf;
Kostenis, Evi;
Tüting, Thomas

Publication type:

Article

The D-type prostanoid (DP) receptor enhances the signaling of chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTH2).

Published in:

2011

By:

Sedej, Miriam;
Schröder, Ralf;
Bell, Kathrin;
Platzer, Wolfgang;
Kostenis, Evi;
Heinemann, Ákos;
Waldhoer, Maria

Publication type:

Abstract

Signalling and function of the human G protein-coupled receptor 55.

Published in:

2010

By:

Balenga, Nariman;
Kargl, Julia;
Schröder, Ralf;
Heinemann, Ákos;
Kostenis, Evi;
Waldhoer, Maria

Publication type:

Abstract

GPR55: signaling pathways and functions.

Published in:

BMC Pharmacology, 2009, v. 9, p. 1, doi. 10.1186/1471-2210-9-S2-A3

By:

Balenga, Nariman;
Schröder, Ralf;
Kargl, Julia;
Platzer, Wolfgang;
Blättermann, Stefanie;
Heinemann, Ákos;
Kostenis, Evi;
Waldhoer, Maria

Publication type:

Article

Novel Insights Into Appropriate Encapsulation Methods for Bioactive Compounds Into Polymers: A Study With Peptides and HDAC Inhibitors.

Published in:

Macromolecular Bioscience, 2014, v. 14, n. 1, p. 69, doi. 10.1002/mabi.201300213

By:

Hennig, Dorle;
Schubert, Stephanie;
Dargatz, Harald;
Kostenis, Evi;
Fahr, Alfred;
Schubert, Ulrich S.;
Heinzel, Thorsten;
Imhof, Diana

Publication type:

Article

Chemisch‐biologischer Werkzeugkasten für die intrazelluläre Bindungsstelle von CCR9: Fluoreszierende Liganden, neue Leitstrukturen und PROTACs.

Published in:

Angewandte Chemie, 2022, v. 134, n. 12, p. 1, doi. 10.1002/ange.202116782

By:

Huber, Max E.;
Toy, Lara;
Schmidt, Maximilian F.;
Vogt, Hannah;
Budzinski, Julian;
Wiefhoff, Martin F. J.;
Merten, Nicole;
Kostenis, Evi;
Weikert, Dorothee;
Schiedel, Matthias

Publication type:

Article

Heterologe Expression, Biosynthese und ökologische Funktion des selektiven Gq‐Signaltransduktionsinhibitors FR900359.

Published in:

Angewandte Chemie, 2018, v. 130, n. 3, p. 844, doi. 10.1002/ange.201707996

By:

Crüsemann, Max;
Reher, Raphael;
Schamari, Isabella;
Brachmann, Alexander O.;
Ohbayashi, Tsubasa;
Kuschak, Markus;
Malfacini, Davide;
Seidinger, Alexander;
Pinto‐Carbó, Marta;
Richarz, René;
Reuter, Tatjana;
Kehraus, Stefan;
Hallab, Asis;
Attwood, Misty;
Schiöth, Helgi B.;
Mergaert, Peter;
Kikuchi, Yoshitomo;
Schäberle, Till F.;
Kostenis, Evi;
Wenzel, Daniela

Publication type:

Article