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Heterologe Expression, Biosynthese und ökologische Funktion des selektiven Gq‐Signaltransduktionsinhibitors FR900359.
- Published in:
- Angewandte Chemie, 2018, v. 130, n. 3, p. 844, doi. 10.1002/ange.201707996
- By:
- Publication type:
- Article
Novel clusters of receptors for sphingosine‐1‐phosphate, sphingosylphosphorylcholine, and (lyso)‐phosphatidic acid: New receptors for “Old” ligands.
- Published in:
- Journal of Cellular Biochemistry, 2004, v. 92, n. 5, p. 923, doi. 10.1002/jcb.20092
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- Publication type:
- Article
Glucose-stimulated insulin secretion depends on FFA1 and Gq in neonatal mouse islets.
- Published in:
- Diabetologia, 2023, v. 66, n. 8, p. 1501, doi. 10.1007/s00125-023-05932-5
- By:
- Publication type:
- Article
Exploring Biased Agonism at FPR1 as a Means to Encode Danger Sensing †.
- Published in:
- Cells (2073-4409), 2020, v. 9, n. 4, p. 1054, doi. 10.3390/cells9041054
- By:
- Publication type:
- Article
GPR55 ligands promote receptor coupling to multiple signalling pathways.
- Published in:
- 2010
- By:
- Publication type:
- journal article
Rational design of dualsteric GPCR ligands: quests and promise.
- Published in:
- 2010
- By:
- Publication type:
- journal article
Reply to: How carvedilol does not activate β<sub>2</sub>-adrenoceptors.
- Published in:
- 2023
- By:
- Publication type:
- Letter
Author Correction: Selective optogenetic control of G<sub>q</sub> signaling using human Neuropsin.
- Published in:
- 2023
- By:
- Publication type:
- Correction Notice
NOP receptor pharmacological profile – A dynamic mass redistribution study.
- Published in:
- PLoS ONE, 2018, v. 13, n. 8, p. 1, doi. 10.1371/journal.pone.0203021
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- Publication type:
- Article
Chemically engineering ligand selectivity at the free fatty acid receptor 2 based on pharmacological variation between species orthologs.
- Published in:
- FASEB Journal, 2012, v. 26, n. 12, p. 4951, doi. 10.1096/fj.12-213314
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- Publication type:
- Article
Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity.
- Published in:
- FASEB Journal, 2009, v. 23, n. 2, p. 442, doi. 10.1096/fj.08-114751
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- Publication type:
- Article
GRK specificity and Gβγ dependency determines the potential of a GPCR for arrestin-biased agonism.
- Published in:
- Communications Biology, 2024, p. 1, doi. 10.1038/s42003-024-06490-1
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- Publication type:
- Article
G protein-mediated signal transduction: a molecular choreography of G protein activation after GTP binding.
- Published in:
- Signal Transduction & Targeted Therapy, 2024, v. 9, n. 1, p. 1, doi. 10.1038/s41392-024-01903-3
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- Publication type:
- Article
Pseudomonas aeruginosa ExoY, a cyclic GMP- and cyclic UMP-generating nucleotidyl cyclase.
- Published in:
- 2013
- By:
- Publication type:
- Abstract
The G<sub>q</sub> signalling pathway inhibits brown and beige adipose tissue.
- Published in:
- Nature Communications, 2016, v. 7, n. 3, p. 10895, doi. 10.1038/ncomms10895
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- Publication type:
- Article
Targeted inhibition of G<sub>q</sub> signaling induces airway relaxation in mouse models of asthma.
- Published in:
- Science Translational Medicine, 2017, v. 9, n. 407, p. 1, doi. 10.1126/scitranslmed.aag2288
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- Publication type:
- Article
Direct targeting of Gα<sub>q</sub> and Gα<sub>11</sub> oncoproteins in cancer cells.
- Published in:
- Science Signaling, 2019, v. 12, n. 573, p. N.PAG, doi. 10.1126/scisignal.aau5948
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- Publication type:
- Article
FZD<sub>5</sub> is a Gαq-coupled receptor that exhibits the functional hallmarks of prototypical GPCRs.
- Published in:
- Science Signaling, 2018, v. 11, n. 559, p. 1, doi. 10.1126/scisignal.aar5536
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- Publication type:
- Article
Front Cover: Deciphering Specificity Determinants for FR900359‐Derived G<sub>q</sub>α Inhibitors Based on Computational and Structure–Activity Studies (ChemMedChem 16/2018).
- Published in:
- ChemMedChem, 2018, v. 13, n. 16, p. 1617, doi. 10.1002/cmdc.201800521
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- Publication type:
- Article
Deciphering Specificity Determinants for FR900359‐Derived G<sub>q</sub>α Inhibitors Based on Computational and Structure–Activity Studies.
- Published in:
- ChemMedChem, 2018, v. 13, n. 16, p. 1634, doi. 10.1002/cmdc.201800304
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- Publication type:
- Article
Reevaluation of fatty acid receptor 1 as a drug target for the stimulation of insulin secretion in humans.
- Published in:
- 2013
- By:
- Publication type:
- journal article
Reevaluation of Fatty Acid Receptor 1 as a Drug Target for the Stimulation of Insulin Secretion in Humans.
- Published in:
- Diabetes, 2013, v. 62, n. 6, p. 2106, doi. 10.2337/db12-1249
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- Publication type:
- Article
Muscarinic Allosteric Modulators: Atypical Structure-Activity-Relationships in Bispyridinium-type Compounds.
- Published in:
- Archiv der Pharmazie, 2006, v. 339, n. 4, p. 207, doi. 10.1002/ardp.200600005
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- Publication type:
- Article
Disentangling bias between G<sub>q</sub>, GRK2, and arrestin3 recruitment to the M<sub>3</sub> muscarinic acetylcholine receptor.
- Published in:
- eLife, 2021, p. 1, doi. 10.7554/eLife.58442
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- Publication type:
- Article
The molecular mechanism by which saturated lysophosphatidylcholine attenuates the metastatic capacity of melanoma cells.
- Published in:
- FEBS Open Bio, 2016, v. 6, n. 12, p. 1297, doi. 10.1002/2211-5463.12152
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- Publication type:
- Article
Pharmacological Gq inhibition induces strong pulmonary vasorelaxation and reverses pulmonary hypertension.
- Published in:
- EMBO Molecular Medicine, 2024, v. 16, n. 8, p. 1930, doi. 10.1038/s44321-024-00096-0
- By:
- Publication type:
- Article
Heterologous Expression, Biosynthetic Studies, and Ecological Function of the Selective Gq‐Signaling Inhibitor FR900359.
- Published in:
- Angewandte Chemie International Edition, 2018, v. 57, n. 3, p. 836, doi. 10.1002/anie.201707996
- By:
- Publication type:
- Article
Tetrahydroimidazo[1,2‐a]pyrazine Derivatives: Synthesis and Evaluation as Gα<sub>q</sub>‐Protein Ligands.
- Published in:
- Chemistry - A European Journal, 2020, v. 26, n. 55, p. 12615, doi. 10.1002/chem.202001446
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- Publication type:
- Article
Leanness and Low Plasma Leptin in GPR17 Knockout Mice Are Dependent on Strain and Associated With Increased Energy Intake That Is Not Suppressed by Exogenous Leptin.
- Published in:
- Frontiers in Endocrinology, 2021, v. 12, p. 1, doi. 10.3389/fendo.2021.698115
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- Publication type:
- Article
Deconvolution of complex G protein–coupled receptor signaling in live cells using dynamic mass redistribution measurements.
- Published in:
- Nature Biotechnology, 2010, v. 28, n. 9, p. 943, doi. 10.1038/nbt.1671
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- Publication type:
- Article
A Chemical Biology Toolbox Targeting the Intracellular Binding Site of CCR9: Fluorescent Ligands, New Drug Leads and PROTACs.
- Published in:
- Angewandte Chemie International Edition, 2022, v. 61, n. 12, p. 1, doi. 10.1002/anie.202116782
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- Publication type:
- Article
Thioesterase-mediated side chain transesterification generates potent Gq signaling inhibitor FR900359.
- Published in:
- Nature Communications, 2021, v. 12, n. 1, p. 1, doi. 10.1038/s41467-020-20418-3
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- Publication type:
- Article
PGH<sub>1</sub>, the Precursor for the Anti-Inflammatory Prostaglandins of the 1-series, Is a Potent Activator of the Pro-Inflammatory Receptor CRTH2/DP2.
- Published in:
- PLoS ONE, 2012, v. 7, n. 3, p. 1, doi. 10.1371/journal.pone.0033329
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- Publication type:
- Article
Heterotrimeric G-proteins: a short history.
- Published in:
- British Journal of Pharmacology, 2006, p. S46, doi. 10.1038/sj.bjp.0706405
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- Publication type:
- Article
Regulated and constitutive activation of specific signalling pathways by the human S1P5 receptor.
- Published in:
- British Journal of Pharmacology, 2003, v. 138, n. 3, p. 481, doi. 10.1038/sj.bjp.0705055
- By:
- Publication type:
- Article
Selective optogenetic control of G<sub>q</sub> signaling using human Neuropsin.
- Published in:
- Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29265-w
- By:
- Publication type:
- Article
Selective optogenetic control of G<sub>q</sub> signaling using human Neuropsin.
- Published in:
- Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29265-w
- By:
- Publication type:
- Article
Adipocyte G<sub>q</sub> signaling is a regulator of glucose and lipid homeostasis in mice.
- Published in:
- Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-29231-6
- By:
- Publication type:
- Article
Oxytocin-Modulated Ion Channel Ensemble Controls Depolarization, Integration and Burst Firing in CA2 Pyramidal Neurons.
- Published in:
- Journal of Neuroscience, 2022, v. 42, n. 41, p. 7707, doi. 10.1523/JNEUROSCI.0921-22.2022
- By:
- Publication type:
- Article
Platelet P2Y<sub>1</sub> receptor exhibits constitutive G protein signaling and β-arrestin 2 recruitment.
- Published in:
- BMC Biology, 2023, v. 21, n. 1, p. 1, doi. 10.1186/s12915-023-01528-y
- By:
- Publication type:
- Article
Detection of free fatty acid receptor 1 expression: the critical role of negative and positive controls.
- Published in:
- Diabetologia, 2014, v. 57, n. 4, p. 776, doi. 10.1007/s00125-014-3161-8
- By:
- Publication type:
- Article
FFA2-, but not FFA3-agonists inhibit GSIS of human pseudoislets: a comparative study with mouse islets and rat INS-1E cells.
- Published in:
- Scientific Reports, 2020, v. 10, n. 1, p. N.PAG, doi. 10.1038/s41598-020-73467-5
- By:
- Publication type:
- Article
Novel Insights Into Appropriate Encapsulation Methods for Bioactive Compounds Into Polymers: A Study With Peptides and HDAC Inhibitors.
- Published in:
- Macromolecular Bioscience, 2014, v. 14, n. 1, p. 69, doi. 10.1002/mabi.201300213
- By:
- Publication type:
- Article
Effects of human urotensin II in isolated vessels of various species; comparison with other vasoactive agents.
- Published in:
- Naunyn-Schmiedeberg's Archives of Pharmacology, 2002, v. 365, n. 2, p. 141, doi. 10.1007/s00210-001-0503-0
- By:
- Publication type:
- Article
Muscarinic allosteric modulation: M<sub>2</sub>/M<sub>3</sub> subtype selectivity of gallamine is independent of G-protein coupling specificity.
- Published in:
- Naunyn-Schmiedeberg's Archives of Pharmacology, 2001, v. 364, n. 2, p. 172, doi. 10.1007/s002100100441
- By:
- Publication type:
- Article
Mice Lacking Free Fatty Acid Receptor 1 (GPR40/FFAR1) are Protected Against Conjugated Linoleic Acid-Induced Fatty Liver but Develop Inflammation and Insulin Resistance in the Brain.
- Published in:
- Cellular Physiology & Biochemistry (Karger AG), 2015, v. 35, n. 6, p. 2272, doi. 10.1159/000374031
- By:
- Publication type:
- Article
Fluid Shear Stress Differentially Regulates gpr3, gpr6, and gpr12 Expression in Human Umbilical Vein Endothelial Cells.
- Published in:
- Cellular Physiology & Biochemistry (Karger AG), 2003, v. 13, n. 2, p. 75, doi. 10.1159/000070251
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- Publication type:
- Article
Community guidelines for GPCR ligand bias: IUPHAR review 32.
- Published in:
- British Journal of Pharmacology, 2022, v. 179, n. 14, p. 3651, doi. 10.1111/bph.15811
- By:
- Publication type:
- Article
The atypical chemokine receptor ACKR3/CXCR7 is a broad-spectrum scavenger for opioid peptides.
- Published in:
- Nature Communications, 2020, v. 11, n. 1, p. 1, doi. 10.1038/s41467-020-16664-0
- By:
- Publication type:
- Article
Author Correction: Chemokine receptor trafficking coordinates neutrophil clustering and dispersal at wounds in zebrafish.
- Published in:
- 2020
- By:
- Publication type:
- Correction Notice