Works by Knapp, Stefan

Results: 177
    1
    2
    3

    Ruthenium Half-Sandwich Complexes Bound to Protein Kinase Pim-1We gratefully acknowledge support for this work from the US National Institutes of Health through grant 1 R01 GM071695-01A1 (E.M.). The Structural Genomics Consortium is a registered charity (no. 1097737) funded by the Wellcome Trust, GlaxoSmithKline, Genome Canada, the Canadian Institutes of Health Research, the Ontario Innovation Trust, the Ontario Research and Development Challenge Fund, and the Canadian Foundation for Innovation.

    Published in:
    Angewandte Chemie, 2006, v. 118, n. 10, p. 1610, doi. 10.1002/ange.200503468
    By:
    • Judit É. Debreczeni;
    • Alex N. Bullock;
    • G. Ekin Atilla;
    • Douglas S. Williams;
    • Howard Bregman;
    • Stefan Knapp;
    • Eric Meggers
    Publication type:
    Article
    4
    5
    6
    7

    Inhibition of DYRK1B BY C81 impedes inflammatory processes in leukocytes by reducing STAT3 activity.

    Published in:
    Cellular & Molecular Life Sciences, 2025, v. 82, n. 1, p. 1, doi. 10.1007/s00018-025-05579-y
    By:
    • Ciurus, Sarah;
    • Elewa, Mohammed A. F.;
    • Palmer, Megan A.;
    • Wolf, Anne;
    • Hector, Mandy;
    • Fuhrmann, Dominik C.;
    • Thomas, Dominique;
    • Gurke, Robert;
    • Schwalm, Martin P.;
    • Berger, Lena;
    • Zech, Thomas J.;
    • Burgers, Luisa D.;
    • Marschalek, Rolf;
    • Geisslinger, Gerd;
    • Knapp, Stefan;
    • Langmann, Thomas;
    • Bracher, Franz;
    • Weigert, Andreas;
    • Fürst, Robert
    Publication type:
    Article
    8
    9
    10
    11
    12
    13
    14
    15
    16
    17
    18

    Structural Insights into Pseudokinase Domains of Receptor Tyrosine Kinases.

    Published in:
    FASEB Journal, 2021, v. 35, p. N.PAG, doi. 10.1096/fasebj.2021.35.S1.02446
    By:
    • Sheetz, Joshua;
    • Mathea, Sebastian;
    • Karvonen, Hanna;
    • Malhotra, Ketan;
    • Chatterjee, Deep;
    • Niininen, Wilhelmiina;
    • Perttila, Robert;
    • Preuss, Franziska;
    • Suresh, Krishna;
    • Stayrook, Steven;
    • Tsutsui, Yuko;
    • Radhakrishnan, Ravi;
    • Ungureanu, Daniela;
    • Knapp, Stefan;
    • Lemmon, Mark
    Publication type:
    Article
    19
    20
    21
    22

    Furo[3,2‐b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway.

    Published in:
    Angewandte Chemie, 2019, v. 131, n. 4, p. 1074, doi. 10.1002/ange.201810312
    By:
    • Němec, Václav;
    • Hylsová, Michaela;
    • Maier, Lukáš;
    • Flegel, Jana;
    • Sievers, Sonja;
    • Ziegler, Slava;
    • Schröder, Martin;
    • Berger, Benedict‐Tilman;
    • Chaikuad, Apirat;
    • Valčíková, Barbora;
    • Uldrijan, Stjepan;
    • Drápela, Stanislav;
    • Souček, Karel;
    • Waldmann, Herbert;
    • Knapp, Stefan;
    • Paruch, Kamil
    Publication type:
    Article
    23
    24
    25
    26
    27
    28

    Thermal unfolding of small proteins with SH3 domain folding pattern.

    Published in:
    Proteins, 1998, v. 31, n. 3, p. 309, doi. 10.1002/(SICI)1097-0134(19980515)31:3<309::AID-PROT7>3.0.CO;2-D
    By:
    • Knapp, Stefan;
    • Mattson, Pekka T.;
    • Christova, Petya;
    • Berndt, Kurt D.;
    • Karshikoff, Andrej;
    • Vihinen, Mauno;
    • Smith, C.I. Edvard;
    • Ladenstein, Rudolf
    Publication type:
    Article
    29
    30
    31
    32
    33
    34
    35
    36

    Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1840, doi. 10.1080/14756366.2020.1825408
    By:
    • Elie, Jonathan;
    • Feizbakhsh, Omid;
    • Desban, Nathalie;
    • Josselin, Béatrice;
    • Baratte, Blandine;
    • Bescond, Amandine;
    • Duez, Julien;
    • Fant, Xavier;
    • Bach, Stéphane;
    • Marie, Dominique;
    • Place, Matthieu;
    • Ben Salah, Sami;
    • Chartier, Agnes;
    • Berteina-Raboin, Sabine;
    • Chaikuad, Apirat;
    • Knapp, Stefan;
    • Carles, Fabrice;
    • Bonnet, Pascal;
    • Buron, Frédéric;
    • Routier, Sylvain
    Publication type:
    Article
    37
    38
    39
    40
    41

    Aurora Kinase A Is Involved in Controlling the Localization of Aquaporin-2 in Renal Principal Cells.

    Published in:
    International Journal of Molecular Sciences, 2022, v. 23, n. 2, p. 763, doi. 10.3390/ijms23020763
    By:
    • Baltzer, Sandrine;
    • Bulatov, Timur;
    • Schmied, Christopher;
    • Krämer, Andreas;
    • Berger, Benedict-Tilman;
    • Oder, Andreas;
    • Walker-Gray, Ryan;
    • Kuschke, Christin;
    • Zühlke, Kerstin;
    • Eichhorst, Jenny;
    • Lehmann, Martin;
    • Knapp, Stefan;
    • Weston, John;
    • von Kries, Jens Peter;
    • Süssmuth, Roderich D.;
    • Klussmann, Enno
    Publication type:
    Article
    42

    The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification.

    Published in:
    International Journal of Molecular Sciences, 2021, v. 22, n. 2, p. 566, doi. 10.3390/ijms22020566
    By:
    • Wells, Carrow I.;
    • Al-Ali, Hassan;
    • Andrews, David M.;
    • Asquith, Christopher R. M.;
    • Axtman, Alison D.;
    • Dikic, Ivan;
    • Ebner, Daniel;
    • Ettmayer, Peter;
    • Fischer, Christian;
    • Frederiksen, Mathias;
    • Futrell, Robert E.;
    • Gray, Nathanael S.;
    • Hatch, Stephanie B.;
    • Knapp, Stefan;
    • Lücking, Ulrich;
    • Michaelides, Michael;
    • Mills, Caitlin E.;
    • Müller, Susanne;
    • Owen, Dafydd;
    • Picado, Alfredo
    Publication type:
    Article
    43
    44
    45
    46
    47
    48
    49

    Progress towards a public chemogenomic set for protein kinases and a call for contributions.

    Published in:
    PLoS ONE, 2017, v. 12, n. 8, p. 1, doi. 10.1371/journal.pone.0181585
    By:
    • Drewry, David H.;
    • Wells, Carrow I.;
    • Andrews, David M.;
    • Angell, Richard;
    • Al-Ali, Hassan;
    • Axtman, Alison D.;
    • Capuzzi, Stephen J.;
    • Elkins, Jonathan M.;
    • Ettmayer, Peter;
    • Frederiksen, Mathias;
    • Gileadi, Opher;
    • Gray, Nathanael;
    • Hooper, Alice;
    • Knapp, Stefan;
    • Laufer, Stefan;
    • Luecking, Ulrich;
    • Michaelides, Michael;
    • Müller, Susanne;
    • Muratov, Eugene;
    • Denny, R. Aldrin
    Publication type:
    Article
    50

    Kinase Domain Is a Dynamic Hub for Driving LRRK2 Allostery.

    Published in:
    Frontiers in Molecular Neuroscience, 2020, v. 13, p. N.PAG, doi. 10.3389/fnmol.2020.538219
    By:
    • Taylor, Susan S.;
    • Kaila-Sharma, Pallavi;
    • Weng, Jui-Hung;
    • Aoto, Phillip;
    • Schmidt, Sven H.;
    • Knapp, Stefan;
    • Mathea, Sebastian;
    • Herberg, Friedrich W.
    Publication type:
    Article