Works by Katzenellenbogen, John
Results: 99
Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism.
- Published in:
- Nature Structural Biology, 2002, v. 9, n. 5, p. 359
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- Article
Estrogen regulation of human osteoblast function is determined by the stage of differentiation and the estrogen receptor isoform.
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- Journal of Cellular Biochemistry, 2001, v. 83, n. 3, p. 448, doi. 10.1002/jcb.1242
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- Article
A new fluorescence complementation biosensor for detection of estrogenic compounds.
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- Biotechnology & Bioengineering, 2011, v. 108, n. 12, p. 2794, doi. 10.1002/bit.23254
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- Article
Suppression of FOXM1 activities and breast cancer growth in vitro and in vivo by a new class of compounds.
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- NPJ Breast Cancer, 2019, v. 5, n. 1, p. N.PAG, doi. 10.1038/s41523-019-0141-7
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- Article
Radiosynthesis and Evaluation of Talazoparib and Its Derivatives as PARP-1-Targeting Agents.
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- Biomedicines, 2021, v. 9, n. 5, p. 565, doi. 10.3390/biomedicines9050565
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- Article
Hormone-PAMAM Dendrimer Conjugates: Polymer Dynamics and Tether Structure Affect Ligand Access to Receptors.
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- Angewandte Chemie International Edition, 2006, v. 45, n. 43, p. 7243, doi. 10.1002/anie.200601923
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- Article
1,2-BIS(4-HYDROXYPHENYL)-3,4-DIHYDRO-6-HYDROXYNAPHTHALENE, A PHOTOFLUOROGENIC LIGAND FOR THE ESTROGEN RECEPTOR.
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- Photochemistry & Photobiology, 1986, v. 43, n. 2, p. 121, doi. 10.1111/j.1751-1097.1986.tb09502.x
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- Article
Estrogen Controls Lipolysis by Up-Regulating α2A-Adrenergic Receptors Directly in Human Adipose Tissue through the Estrogen Receptor α. Implications for the Female Fat Distribution.
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- Journal of Clinical Endocrinology & Metabolism, 2004, v. 89, n. 4, p. 1869, doi. 10.1210/jc.2003-031327
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- Article
Book Review: Steroid Receptor MethodsProtocols and Assays. Edited by Benjamin A. Lieberman.
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- ChemBioChem, 2003, v. 4, n. 6, p. 548
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- Article
A mutant form of ERα associated with estrogen insensitivity affects the coupling between ligand binding and coactivator recruitment.
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- Science Signaling, 2020, v. 13, n. 650, p. 1, doi. 10.1126/scisignal.aaw4653
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- Article
Identification of Toll-like receptor signaling inhibitors based on selective activation of hierarchically acting signaling proteins.
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- Science Signaling, 2018, v. 11, n. 543, p. 1, doi. 10.1126/scisignal.aaq1077
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- Article
Respective role of membrane and nuclear estrogen receptor (ER) α in the mandible of growing mice: Implications for ERα modulation.
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- Journal of Bone & Mineral Research, 2018, v. 33, n. 8, p. 1520, doi. 10.1002/jbmr.3434
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- Article
An Efficient, General Synthesis of Alkylsulfinyltoluidides.
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- Synthetic Communications, 1974, v. 4, n. 3, p. 137, doi. 10.1080/00397917408062061
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- Article
Alleviation of extensive visual pathway dysfunction by a remyelinating drug in a chronic mouse model of multiple sclerosis.
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- Brain Pathology, 2021, v. 31, n. 2, p. 312, doi. 10.1111/bpa.12930
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- Article
Estradiol promotes cell survival and induces Greb1 expression in granulosa cell tumors of the ovary through an ERα‐dependent mechanism.
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- Journal of Pathology, 2022, v. 256, n. 3, p. 335, doi. 10.1002/path.5843
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- Article
Imaging Diagnostic and Therapeutic Targets: Steroid Receptors in Breast Cancer.
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- Journal of Nuclear Medicine, 2016, v. 57, p. 75S, doi. 10.2967/jnumed.115.157933
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- Article
Small-Animal PET of Steroid Hormone Receptors Predicts Tumor Response to Endocrine Therapy Using a Preclinical Model of Breast Cancer.
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- Journal of Nuclear Medicine, 2012, v. 53, n. 7, p. 1119, doi. 10.2967/jnumed.112.103465
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- Article
Assessment of Progesterone Receptors in Breast Carcinoma by PET with 21-<sup>18</sup>F-Fluoro-16α,17α-[(R)-(1'-α-furylmethylidene) Dioxy]-19-Norpregn-4-Ene-3,20-Dione.
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- Journal of Nuclear Medicine, 2012, v. 53, n. 3, p. 363, doi. 10.2967/jnumed.111.098319
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- Article
PLASMIN-ACTIVATED ANTICANCER PRODRUGS.
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- Annals of the New York Academy of Sciences, 1982, v. 397, n. 1, p. 324, doi. 10.1111/j.1749-6632.1982.tb43455.x
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- Article
Experimental versus predicted affinities for ligand binding to estrogen receptor: iterative selection and rescoring of docked poses systematically improves the correlation.
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- Journal of Computer-Aided Molecular Design, 2013, v. 27, n. 8, p. 707, doi. 10.1007/s10822-013-9670-6
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- Article
Estrogen Receptor-α Agonists Promote Angiogenesis in Human Myometrial Microvascular Endothelial Cells.
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- Reproductive Sciences, 2004, v. 11, n. 8, p. 529, doi. 10.1016/j.jsgi.2004.06.004
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- Article
Estrogen Receptor Isoform-Specific Induction of Progesterone Receptors in Human Osteoblasts.
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- Journal of Bone & Mineral Research, 2002, v. 17, n. 4, p. 580, doi. 10.1359/jbmr.2002.17.4.580
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- Article
The roles of membrane estrogen receptor subtypes in modulating dopamine transporters in PC-12 cells.
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- Journal of Neurochemistry, 2008, v. 106, n. 4, p. 1525, doi. 10.1111/j.1471-4159.2008.05491.x
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- Article
Pocket similarity identifies selective estrogen receptor modulators as microtubule modulators at the taxane site.
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- Nature Communications, 2019, v. 10, n. 1, p. 1, doi. 10.1038/s41467-019-08965-w
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- Article
PI3K inhibition results in enhanced estrogen receptor function and dependence in hormone receptor–positive breast cancer.
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- Science Translational Medicine, 2015, v. 7, n. 283, p. 1, doi. 10.1126/scitranslmed.aaa4442
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- Article
Dual suppression of estrogenic and inflammatory activities for targeting of endometriosis.
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- Science Translational Medicine, 2015, v. 7, n. 271, p. 1, doi. 10.1126/scitranslmed.3010626
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- Article
Mechanisms enforcing the estrogen receptor β selectivity of botanical estrogens.
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- FASEB Journal, 2013, v. 27, n. 11, p. 4406, doi. 10.1096/fj.13-234617
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- Article
Resistance to FOXM1 inhibitors in breast cancer is accompanied by impeding ferroptosis and apoptotic cell death.
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- Breast Cancer Research & Treatment, 2024, v. 208, n. 2, p. 307, doi. 10.1007/s10549-024-07420-9
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- Article
Exploration of alcohol‐enhanced Cu‐mediated radiofluorination toward practical labeling.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2022, v. 65, n. 1, p. 13, doi. 10.1002/jlcr.3955
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- Article
Meet our advisors: An interview with John Katzenellenbogen.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2021, v. 64, n. 14, p. 527, doi. 10.1002/jlcr.3951
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- Article
Evaluation of aromatic radiobromination by nucleophilic substitution using diaryliodonium salt precursors.
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- 2017
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- Other
Optimization of the preparation of fluorine-18-labeled steroid receptor ligands 16alpha-[<sup>18</sup>F]fluoroestradiol (FES), [<sup>18</sup>F]fluoro furanyl norprogesterone (FFNP), and 16beta-[<sup>18</sup>F]fluoro-5alpha-dihydrotestosterone (FDHT) as radiopharmaceuticals
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2014, v. 57, n. 5, p. 371, doi. 10.1002/jlcr.3191
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- Article
Predominant Role of Nuclear Versus Membrane Estrogen Receptor α in Arterial Protection: Implications for Estrogen Receptor α Modulation in Cardiovascular Prevention/Safety.
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- 2018
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- journal article
Endothelial ERα promotes glucose tolerance by enhancing endothelial insulin transport to skeletal muscle.
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- Nature Communications, 2023, v. 14, n. 1, p. 1, doi. 10.1038/s41467-023-40562-w
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- Article
Triaryl Pyrazole Toll‐Like Receptor Signaling Inhibitors: Structure–Activity Relationships Governing Pan‐ and Selective Signaling Inhibitors.
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- ChemMedChem, 2018, v. 13, n. 20, p. 2208, doi. 10.1002/cmdc.201800417
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- Article
Selenophenes: Introducing a New Element into the Core of Non-Steroidal Estrogen Receptor Ligands.
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- ChemMedChem, 2017, v. 12, n. 3, p. 235, doi. 10.1002/cmdc.201600593
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- Article
Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.
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- ChemMedChem, 2016, v. 11, n. 16, p. 1752, doi. 10.1002/cmdc.201600140
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- Article
Salicylketoximes That Target Glucose Transporter 1 Restrict Energy Supply to Lung Cancer Cells.
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- ChemMedChem, 2015, v. 10, n. 11, p. 1892, doi. 10.1002/cmdc.201500320
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- Article
Development of Selective Estrogen Receptor Modulator (SERM)-Like Activity Through an Indirect Mechanism of Estrogen Receptor Antagonism: Defining the Binding Mode of 7-Oxabicyclo[2.2.1]hept-5-ene Scaffold Core Ligands.
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- ChemMedChem, 2012, v. 7, n. 6, p. 1094, doi. 10.1002/cmdc.201200048
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- Article
Discovering Small-Molecule Estrogen Receptor α/Coactivator Binding Inhibitors: High-Throughput Screening, Ligand Development, and Models for Enhanced Potency.
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- ChemMedChem, 2011, v. 6, n. 4, p. 654, doi. 10.1002/cmdc.201000507
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- Article
THE EFFECT OF ACCEPTOR GROUP VARIATION ON THE SOLVATOCHROMISM OF DONOR-ACCEPTOR FLUOROPHORES.
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- Photochemistry & Photobiology, 1993, v. 58, n. 6, p. 785, doi. 10.1111/j.1751-1097.1993.tb04971.x
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- Article
CHARACTERIZATION OF THE SPECTROSCOPIC PROPERTIES OF A TETRAHYDROCHRYSENE SYSTEM CONTAINING A RIGIDIFIED HYDROXYNITROSTILBENE CHROMOPHORE: AN INHERENTLY FLUORESCENT LIGAND DESIGNED FOR THE ESTROGEN RECEPTOR.
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- Photochemistry & Photobiology, 1993, v. 57, n. 4, p. 616, doi. 10.1111/j.1751-1097.1993.tb02927.x
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- Article
HYDROXYSTILBAZOLES AND HYDROXYAZAPHENANTHRENES: PHOTOCYCLIZATION AND FLUORESCENCE STUDIES.
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- Photochemistry & Photobiology, 1988, v. 47, n. 4, p. 503, doi. 10.1111/j.1751-1097.1988.tb08838.x
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- Article
Estrogen Receptor Beta 1: A Potential Therapeutic Target for Female Triple Negative Breast Cancer.
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- Endocrinology, 2022, v. 163, n. 12, p. 1, doi. 10.1210/endocr/bqac172
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- Article
Differential Actions of Estrogen Receptor α and β via Nongenomic Signaling in Human Prostate Stem and Progenitor Cells.
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- Endocrinology, 2019, v. 160, n. 11, p. 2692, doi. 10.1210/en.2019-00177
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- Article
Effects of Exposure to the Endocrine-Disrupting Chemical Bisphenol A During Critical Windows of Murine Pituitary Development.
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- Endocrinology, 2018, v. 159, n. 1, p. 119, doi. 10.1210/en.2017-00565
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- Article
Structure-Function Relationships in Estrogen Receptors and the Characterization of Novel Selective Estrogen Receptor Modulators with Unique Pharmacological Profiles.
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- Annals of the New York Academy of Sciences, 2001, v. 949, n. 1, p. 6, doi. 10.1111/j.1749-6632.2001.tb03998.x
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- Article
Analogues of ERβ ligand chloroindazole exert immunomodulatory and remyelinating effects in a mouse model of multiple sclerosis.
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- Scientific Reports, 2019, v. 9, n. 1, p. 1, doi. 10.1038/s41598-018-37420-x
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- Article
Transcriptomic analysis identifies gene networks regulated by estrogen receptor α (ERα) and ERβ that control distinct effects of different botanical estrogens.
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- Nuclear Receptor Signaling, 2014, v. 12, p. 1, doi. 10.1621/nrs.12001
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- Article
Hormone–PAMAM Dendrimer Conjugates: Polymer Dynamics and Tether Structure Affect Ligand Access to ReceptorsWe are grateful for support of this research through grants from the National Institutes of Health (PHS 5R37 DK15556). We thank Kathryn Carlson for determining the receptor binding affinities. NMR spectra were obtained in the Varian Oxford Instrument Center for Excellence in NMR Laboratory. Funding for this instrumentation was provided in part by the W. M. Keck Foundation, the National Institutes of Health (PHS 1 S10 RR104444-01), and the National Science Foundation (NSF CHE 96-10502). Mass spectra were obtained on instruments supported by grants from the National Institute of General Medical Sciences (GM 27029), the National Institutes of Health (RR 01575), and the National Science Foundation (PCM 8121494). PAMAM=poly(amide)polyamine.
- Published in:
- Angewandte Chemie, 2006, v. 118, n. 43, p. 7401, doi. 10.1002/ange.200601923
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- Article