Works by Kartsev, Victor

Results: 30

Synthesis and antimicrobial activity of new 2‐piperazin‐1‐yl‐N‐1,3‐thiazol‐2‐ylacetamides of cyclopenta[c]pyridines and pyrano[3,4‐c]pyridines.

Published in:

Archiv der Pharmazie, 2021, v. 354, n. 1, p. 1, doi. 10.1002/ardp.202000208

By:

Sirakanyan, Samvel;
Kartsev, Victor;
Spinelli, Domenico;
Geronikaki, Athina;
Petrou, Anthi;
Ivanov, Marija;
Glamoclija, Jasmina;
Sokovic, Marina;
Hakobyan, Elmira;
Hovakimyan, Anush

Publication type:

Article

Discovery of Novel EGFR Inhibitor Targeting Wild-Type and Mutant Forms of EGFR: In Silico and In Vitro Study.

Published in:

Molecules, 2023, v. 28, n. 7, p. 3014, doi. 10.3390/molecules28073014

By:

Todsaporn, Duangjai;
Zubenko, Alexander;
Kartsev, Victor;
Aiebchun, Thitinan;
Mahalapbutr, Panupong;
Petrou, Anthi;
Geronikaki, Athina;
Divaeva, Liudmila;
Chekrisheva, Victoria;
Yildiz, Ilkay;
Choowongkomon, Kiattawee;
Rungrotmongkol, Thanyada

Publication type:

Article

New Bicyclic Pyridine-Based Hybrids Linked to the 1,2,3-Triazole Unit: Synthesis via Click Reaction and Evaluation of Neurotropic Activity and Molecular Docking.

Published in:

Molecules, 2023, v. 28, n. 3, p. 921, doi. 10.3390/molecules28030921

By:

Sirakanyan, Samvel N.;
Spinelli, Domenico;
Petrou, Anthi;
Geronikaki, Athina;
Kartsev, Victor G.;
Hakobyan, Elmira K.;
Yegoryan, Hasmik A.;
Zuppiroli, Luca;
Zuppiroli, Riccardo;
Ayvazyan, Armen G.;
Paronikyan, Ruzanna G.;
Arakelyan, Tatevik A.;
Hovakimyan, Anush A.

Publication type:

Article

Benzothiazole and Chromone Derivatives as Potential ATR Kinase Inhibitors and Anticancer Agents.

Published in:

Molecules, 2022, v. 27, n. 14, p. N.PAG, doi. 10.3390/molecules27144637

By:

Frasinyuk, Mykhaylo;
Chhabria, Dimple;
Kartsev, Victor;
Dilip, Haritha;
Sirakanyan, Samvel N.;
Kirubakaran, Sivapriya;
Petrou, Anthi;
Geronikaki, Athina;
Spinelli, Domenico

Publication type:

Article

Synthesis, Biological Evaluation and Molecular Docking Studies of 5-Indolylmethylen-4-oxo-2-thioxothiazolidine Derivatives.

Published in:

Molecules, 2022, v. 27, n. 3, p. 1068, doi. 10.3390/molecules27031068

By:

Horishny, Volodymyr;
Geronikaki, Athina;
Kartsev, Victor;
Matiychuk, Vasyl;
Petrou, Anthi;
Pogodin, Pavel;
Poroikov, Vladimir;
Papadopoulou, Theodora A.;
Vizirianakis, Ioannis S.;
Kostic, Marina;
Ivanov, Marija;
Sokovic, Marina

Publication type:

Article

Carbonic Anhydrase Inhibition with Sulfonamides Incorporating Pyrazole- and Pyridazinecarboxamide Moieties Provides Examples of Isoform-Selective Inhibitors.

Published in:

Molecules, 2021, v. 26, n. 22, p. 7023, doi. 10.3390/molecules26227023

By:

Angeli, Andrea;
Kartsev, Victor;
Petrou, Anthi;
Pinteala, Mariana;
Brovarets, Volodymyr;
Vydzhak, Roman;
Panchishin, Svitlana;
Geronikaki, Athina;
Supuran, Claudiu T.

Publication type:

Article

Synthesis and Neurotropic Activity of New Heterocyclic Systems: Pyridofuro[3,2- d ]pyrrolo[1,2- a ]pyrimidines, Pyridofuro[3,2- d ]pyrido[1,2- a ]pyrimidines and Pyridofuro[3′,2′:4,5]pyrimido[1,2- a ]azepines.

Published in:

Molecules, 2021, v. 26, n. 11, p. 3320, doi. 10.3390/molecules26113320

By:

Sirakanyan, Samvel N.;
Spinelli, Domenico;
Geronikaki, Athina;
Kartsev, Victor;
Hakobyan, Elmira K.;
Petrou, Anthi;
Paronikyan, Ruzanna G.;
Nazaryan, Ivetta M.;
Akopyan, Hasmik H.;
Hovakimyan, Anush A.

Publication type:

Article

5-(1H-Indol-3-ylmethylene)-4-oxo-2-thioxothiazolidin-3-yl)alkancarboxylic Acids as Antimicrobial Agents: Synthesis, Biological Evaluation, and Molecular Docking Studies.

Published in:

Molecules, 2020, v. 25, n. 8, p. 1964, doi. 10.3390/molecules25081964

By:

Horishny, Volodymyr;
Kartsev, Victor;
Geronikaki, Athina;
Matiychuk, Vasyl;
Petrou, Anthi;
Glamoclija, Jasmina;
Ciric, Ana;
Sokovic, Marina;
Catto, Marco;
Altomare, Cosimo Damiano

Publication type:

Article

Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation.

Published in:

Molecules, 2019, v. 24, n. 19, p. 3580, doi. 10.3390/molecules24193580

By:

Kartsev, Victor;
Geronikaki, Athina;
Bua, Silvia;
Nocentini, Alessio;
Petrou, Anthi;
Lichitsky, Boris;
Frasinyuk, Mykhaylo;
Leitans, Janis;
Kazaks, Andris;
Tars, Kaspars;
Supuran, Claudiu T.

Publication type:

Article

Application of Docking Analysis in the Prediction and Biological Evaluation of the Lipoxygenase Inhibitory Action of Thiazolyl Derivatives of Mycophenolic Acid.

Published in:

Molecules, 2018, v. 23, n. 7, p. 1621, doi. 10.3390/molecules23071621

By:

Tsolaki, Evangelia;
Eleftheriou, Phaedra;
Kartsev, Victor;
Geronikaki, Athina;
Saxena, Anil K.

Publication type:

Article

Synthesis, biological evaluation, and molecular docking studies of thiazolo[4,5‐b]pyridin‐5‐ones as antimicrobial agents.

Published in:

Journal of Heterocyclic Chemistry, 2022, v. 59, n. 9, p. 1573, doi. 10.1002/jhet.4491

By:

Kartsev, Victor;
Geronikaki, Athina;
Lichitsky, Boris;
Komogortsev, Andrey;
Petrou, Anthi;
Ivanov, Marija;
Glamočlija, Jasmina;
Soković, Marina

Publication type:

Article

Synthesis and Rearrangement of New 1,3-Diamino-2,7-naphthyridines and 1-Amino-3-oxo-2,7-naphthyridines.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 22, p. 11977, doi. 10.3390/ijms252211977

By:

Sirakanyan, Samvel N.;
Spinelli, Domenico;
Mattioli, Edoardo Jun;
Calvaresi, Matteo;
Geronikaki, Athina;
Kartsev, Victor G.;
Hakobyan, Elmira K.;
Yegoryan, Hasmik A.;
Jughetsyan, Hasmik V.;
Manukyan, Mariam E.;
Hovakimyan, Anush A.

Publication type:

Article

Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 3, p. 2802, doi. 10.3390/ijms24032802

By:

Angeli, Andrea;
Petrou, Anthi;
Kartsev, Victor;
Lichitsky, Boris;
Komogortsev, Andrey;
Capasso, Clemente;
Geronikaki, Athina;
Supuran, Claudiu T.

Publication type:

Article

Synthesis of 1-Amino-3-oxo-2,7-naphthyridines via Smiles Rearrangement: A New Approach in the Field of Chemistry of Heterocyclic Compounds.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 11, p. 5904, doi. 10.3390/ijms23115904

By:

Sirakanyan, Samvel N.;
Spinelli, Domenico;
Geronikaki, Athina;
Zuppiroli, Luca;
Zuppiroli, Riccardo;
Kartsev, Victor G.;
Hakobyan, Elmira K.;
Yegoryan, Hasmik A.;
Hovakimyan, Anush A.

Publication type:

Article

Chromene-Containing Aromatic Sulfonamides with Carbonic Anhydrase Inhibitory Properties.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 10, p. 5082, doi. 10.3390/ijms22105082

By:

Angeli, Andrea;
Kartsev, Victor;
Petrou, Anthi;
Pinteala, Mariana;
Brovarets, Volodymyr;
Slyvchuk, Sergii;
Pilyo, Stepan;
Geronikaki, Athina;
Supuran, Claudiu T.;
Christov, Christo Z.

Publication type:

Article

Disruption of the Complex between GAPDH and Hsp70 Sensitizes C6 Glioblastoma Cells to Hypoxic Stress.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 4, p. 1520, doi. 10.3390/ijms22041520

By:

Mikeladze, Marina A.;
Dutysheva, Elizaveta A.;
Kartsev, Victor G.;
Margulis, Boris A.;
Guzhova, Irina V.;
Lazarev, Vladimir F.;
Nikolaidis, Nikolas

Publication type:

Article

Identification of Novel Antibacterials Using Machine Learning Techniques.

Published in:

Frontiers in Pharmacology, 2019, p. 1, doi. 10.3389/fphar.2019.00913

By:

Ivanenkov, Yan A.;
Zhavoronkov, Alex;
Yamidanov, Renat S.;
Osterman, Ilya A.;
Sergiev, Petr V.;
Aladinskiy, Vladimir A.;
Aladinskaya, Anastasia V.;
Terentiev, Victor A.;
Veselov, Mark S.;
Ayginin, Andrey A.;
Kartsev, Victor G.;
Skvortsov, Dmitry A.;
Chemeris, Alexey V.;
Baimiev, Alexey Kh.;
Sofronova, Alina A.;
Malyshev, Alexander S.;
Filkov, Gleb I.;
Bezrukov, Dmitry S.;
Zagribelnyy, Bogdan A.;
Putin, Evgeny O.

Publication type:

Article

Madumycin II inhibits peptide bond formation by forcing the peptidyl transferase center into an inactive state.

Published in:

Nucleic Acids Research, 2017, v. 45, n. 12, p. 7507, doi. 10.1093/nar/gkx413

By:

Osterman, Ilya A.;
Khabibullina, Nelli F.;
Komarova, Ekaterina S.;
Kasatsky, Pavel;
Kartsev, Victor G.;
Bogdanov, Alexey A.;
Dontsova, Olga A.;
Konevega, Andrey L.;
Sergiev, Petr V.;
Polikanov, Yury S.

Publication type:

Article

Synthesis of 3,3-dimethyl-6-oxopyrano[3,4-c]pyridines and their antiplatelet and vasodilatory activity.

Published in:

Journal of Pharmacy & Pharmacology, 2022, v. 74, n. 6, p. 887, doi. 10.1093/jpp/rgab075

By:

Sirakanyan, Samvel N;
Hrubša, Marcel;
Spinelli, Domenico;
Dias, Patrícia;
Kartsev, Victor;
Carazo, Alejandro;
Hovakimyan, Anush A;
Pourová, Jana;
Hakobyan, Elmira K;
Karlíčková, Jana;
Parvin, Shamima;
Fadraersada, Jaka;
Macáková, Kateřina;
Geronikaki, Athina;
Mladěnka, Přemysl

Publication type:

Article

Synthesis and Neurotropic Activity of New 5-Piperazinopyrazolo[3,4- c ]-2,7-naphthyridines and Isoxazolo[5,4- c ]-2,7-naphthyridines.

Published in:

Pharmaceuticals (14248247), 2025, v. 18, n. 4, p. 597, doi. 10.3390/ph18040597

By:

Sirakanyan, Samvel N.;
Hakobyan, Elmira K.;
Geronikaki, Athina;
Spinelli, Domenico;
Petrou, Anthi;
Kartsev, Victor G.;
Yegoryan, Hasmik A.;
Jughetsyan, Hasmik V.;
Manukyan, Mariam E.;
Paronikyan, Ruzanna G.;
Araqelyan, Tatevik A.;
Hovakimyan, Anush A.

Publication type:

Article

N -Derivatives of (Z)-Methyl 3-(4-Oxo-2-thioxothiazolidin-5-ylidene)methyl)-1 H -indole-2-carboxylates as Antimicrobial Agents—In Silico and In Vitro Evaluation.

Published in:

Pharmaceuticals (14248247), 2023, v. 16, n. 1, p. 131, doi. 10.3390/ph16010131

By:

Petrou, Anthi;
Geronikaki, Athina;
Kartsev, Victor;
Kousaxidis, Antonios;
Papadimitriou-Tsantarliotou, Aliki;
Kostic, Marina;
Ivanov, Marija;
Sokovic, Marina;
Nicolaou, Ioannis;
Vizirianakis, Ioannis S.

Publication type:

Article

Pyrazolo[4,3-c]pyridine Sulfonamides as Carbonic Anhydrase Inhibitors: Synthesis, Biological and In Silico Studies.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 3, p. 316, doi. 10.3390/ph15030316

By:

Angeli, Andrea;
Kartsev, Victor;
Petrou, Anthi;
Lichitsky, Boris;
Komogortsev, Andrey;
Pinteala, Mariana;
Geronikaki, Athina;
Supuran, Claudiu T.

Publication type:

Article

4-(Indol-3-yl)thiazole-2-amines and 4-ιndol-3-yl)thiazole Acylamines as Νovel Antimicrobial Agents: Synthesis, In Silico and In Vitro Evaluation.

Published in:

Pharmaceuticals (14248247), 2021, v. 14, n. 11, p. 1096, doi. 10.3390/ph14111096

By:

Simakov, Sergei;
Kartsev, Victor;
Petrou, Anthi;
Nicolaou, Ioannis;
Geronikaki, Athina;
Ivanov, Marija;
Kostic, Marina;
Glamočlija, Jasmina;
Soković, Marina;
Talea, Despoina;
Vizirianakis, Ioannis S.

Publication type:

Article

New Sulfanilamide Derivatives Incorporating Heterocyclic Carboxamide Moieties as Carbonic Anhydrase Inhibitors.

Published in:

Pharmaceuticals (14248247), 2021, v. 14, n. 8, p. 828, doi. 10.3390/ph14080828

By:

Angeli, Andrea;
Kartsev, Victor;
Petrou, Anthi;
Pinteala, Mariana;
Vydzhak, Roman M.;
Panchishin, Svitlana Y.;
Brovarets, Volodymyr;
De Luca, Viviana;
Capasso, Clemente;
Geronikaki, Athina;
Supuran, Claudiu T.

Publication type:

Article

3-Amino-5-(indol-3-yl)methylene-4-oxo-2-thioxothiazolidine Derivatives as Antimicrobial Agents: Synthesis, Computational and Biological Evaluation.

Published in:

Pharmaceuticals (14248247), 2020, v. 13, n. 9, p. 229, doi. 10.3390/ph13090229

By:

Horishny, Volodymyr;
Kartsev, Victor;
Matiychuk, Vasyl;
Geronikaki, Athina;
Anthi, Petrou;
Pogodin, Pavel;
Poroikov, Vladimir;
Ivanov, Marija;
Kostic, Marina;
Soković, Marina D.;
Eleftheriou, Phaedra

Publication type:

Article

Synthesis and Antimicrobial Activity of New Heteroaryl(aryl) Thiazole Derivatives Molecular Docking Studies.

Published in:

Antibiotics (2079-6382), 2022, v. 11, n. 10, p. N.PAG, doi. 10.3390/antibiotics11101337

By:

Kartsev, Victor;
Geronikaki, Athina;
Zubenko, Alexander;
Petrou, Anthi;
Ivanov, Marija;
Glamočlija, Jasmina;
Sokovic, Marina;
Divaeva, Lyudmila;
Morkovnik, Anatolii;
Klimenko, Alexander

Publication type:

Article

In silico Design, Synthesis and Biological Evaluation of Novel Thieno[3,2‐d]pyrimidine Derivatives for Cancer Therapy – A Preliminary Study on the Inhibitory Potential towards ATR Kinase Domain and PIKK Family.

Published in:

Chemistry & Biodiversity, 2024, v. 21, n. 3, p. 1, doi. 10.1002/cbdv.202302071

By:

Sirakanyan, Samvel N.;
Dilip, Haritha;
Geronikaki, Athina;
Spinelli, Domenico;
Kirubakaran, Sivapriya;
Petrou, Anthi;
Hakobyan, Elmira K.;
Kartsev, Victor G.;
Paronikyan, Ervand G.;
Yegoryan, Hasmik A.;
Yermalovyan, Lilit V.;
Hovakimyan, Anush A.

Publication type:

Article

Synthesis of Alkaloid Sinomenine Derivatives Containing a Pyrimidine Substituent in Ring A.

Published in:

Chemistry of Heterocyclic Compounds, 2021, v. 57, n. 9, p. 934, doi. 10.1007/s10593-021-03003-4

By:

Finke, Anastasiya O.;
Kartsev, Victor G.;
Shults, Elvira E.

Publication type:

Article

Synthesis and antimicrobial evaluation of novel polyheterocyclic systems derived from cyclopenta[4',5']pyrido[3',2':4,5]furo[3,2-d]pyrimidine.

Published in:

Chemistry of Heterocyclic Compounds, 2021, v. 57, n. 1, p. 75, doi. 10.1007/s10593-021-02870-1

By:

Sirakanyan, Samvel N.;
Spinelli, Domenico;
Geronikaki, Athina;
Kartsev, Victor G.;
Stepanyan, Hrachya M.;
Hakobyan, Elmira K.;
Hovakimyan, Anush A.

Publication type:

Article

Novel isatin-derived molecules activate p53 via interference with Mdm2 to promote apoptosis.

Published in:

Cell Cycle, 2018, v. 17, n. 15, p. 1917, doi. 10.1080/15384101.2018.1506664

By:

Fedorova, Olga;
Daks, Alexandra;
Petrova, Varvara;
Petukhov, Alexey;
Lezina, Larissa;
Shuvalov, Oleg;
Davidovich, Pavel;
Kriger, Darya;
Lomert, Ekaterina;
Tentler, Dmitry;
Kartsev, Victor;
Uyanik, Burhan;
Tribulovich, Vyacheslav;
Demidov, Oleg;
Melino, Gerry;
Barlev, Nickolai A.

Publication type:

Article