Works matching AU Kaniskan, H. Ümit


Results: 10
    1

    A Potent, Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 3 (PRMT3).

    Published in:
    Angewandte Chemie, 2015, v. 127, n. 17, p. 5255, doi. 10.1002/ange.201412154
    By:
    • Kaniskan, H. Ümit;
    • Szewczyk, Magdalena M.;
    • Yu, Zhengtian;
    • Eram, Mohammad S.;
    • Yang, Xiaobao;
    • Schmidt, Keith;
    • Luo, Xiao;
    • Dai, Miao;
    • He, Feng;
    • Zang, Irene;
    • Lin, Ying;
    • Kennedy, Steven;
    • Li, Fengling;
    • Dobrovetsky, Elena;
    • Dong, Aiping;
    • Smil, David;
    • Min, Sun ‐ Joon;
    • Landon, Melissa;
    • Lin ‐ Jones, Jennifer;
    • Huang, Xi ‐ Ping
    Publication type:
    Article
    2

    Inside Back Cover Image, Volume 41, Issue 3.

    Published in:
    Medicinal Research Reviews, 2021, v. 41, n. 3, p. iii, doi. 10.1002/med.21813
    By:
    • Vatansever, Sezen;
    • Schlessinger, Avner;
    • Wacker, Daniel;
    • Kaniskan, H. Ümit;
    • Jin, Jian;
    • Zhou, Ming‐Ming;
    • Zhang, Bin
    Publication type:
    Article
    3
    4
    5

    A selective WDR5 degrader inhibits acute myeloid leukemia in patient-derived mouse models.

    Published in:
    Science Translational Medicine, 2021, v. 13, n. 613, p. 1, doi. 10.1126/scitranslmed.abj1578
    By:
    • Yu, Xufen;
    • Li, Dongxu;
    • Kottur, Jithesh;
    • Shen, Yudao;
    • Kim, Huen Suk;
    • Park, Kwang-Su;
    • Tsai, Yi-Hsuan;
    • Gong, Weida;
    • Wang, Jun;
    • Suzuki, Kyogo;
    • Parker, Joel;
    • Herring, Laura;
    • Kaniskan, H. Ümit;
    • Cai, Ling;
    • Jain, Rinku;
    • Liu, Jing;
    • Aggarwal, Aneel K;
    • Wang, Gang Greg;
    • Jin, Jian
    Publication type:
    Article
    6

    Phenomics‐Based Discovery of Novel Orthosteric Choline Kinase Inhibitors.

    Published in:
    Angewandte Chemie International Edition, 2025, v. 64, n. 7, p. 1, doi. 10.1002/anie.202420149
    By:
    • Bauer, Ludwig G.;
    • Ward, Jennifer A.;
    • Díaz‐Sáez, Laura;
    • Sundström, Yvonne;
    • Tolvanen, Tuomas;
    • Alarcón Barrera, Juan Carlos;
    • Kostidis, Sarantos;
    • Rogers, Catherine M.;
    • Panagakou, Ioanna;
    • Singh, Usha;
    • Rothweiler, Elisabeth M.;
    • Gonzalez Orta, Alejandro;
    • Kaniskan, H. Ümit;
    • Hu, Jianping;
    • Jin, Jian;
    • Sievers, Sonja;
    • Waldmann, Herbert;
    • Giera, Martin;
    • Sundström, Michael;
    • Berg, Louise
    Publication type:
    Article
    7

    A chemical biology toolbox to study protein methyltransferases and epigenetic signaling.

    Published in:
    Nature Communications, 2019, v. 10, n. 1, p. 1, doi. 10.1038/s41467-018-07905-4
    By:
    • Scheer, Sebastian;
    • Ackloo, Suzanne;
    • Medina, Tiago S.;
    • Schapira, Matthieu;
    • Li, Fengling;
    • Ward, Jennifer A.;
    • Lewis, Andrew M.;
    • Northrop, Jeffrey P.;
    • Richardson, Paul L.;
    • Kaniskan, H. Ümit;
    • Shen, Yudao;
    • Liu, Jing;
    • Smil, David;
    • McLeod, David;
    • Zepeda-Velazquez, Carlos A.;
    • Luo, Minkui;
    • Jin, Jian;
    • Barsyte-Lovejoy, Dalia;
    • Huber, Kilian V. M.;
    • De Carvalho, Daniel D.
    Publication type:
    Article
    8

    Phänomik‐basierte Entdeckung neuer orthosterischer Cholinkinase Inhibitoren.

    Published in:
    Angewandte Chemie, 2025, v. 137, n. 7, p. 1, doi. 10.1002/ange.202420149
    By:
    • Bauer, Ludwig G.;
    • Ward, Jennifer A.;
    • Díaz‐Sáez, Laura;
    • Sundström, Yvonne;
    • Tolvanen, Tuomas;
    • Alarcón Barrera, Juan Carlos;
    • Kostidis, Sarantos;
    • Rogers, Catherine M.;
    • Panagakou, Ioanna;
    • Singh, Usha;
    • Rothweiler, Elisabeth M.;
    • Gonzalez Orta, Alejandro;
    • Kaniskan, H. Ümit;
    • Hu, Jianping;
    • Jin, Jian;
    • Sievers, Sonja;
    • Waldmann, Herbert;
    • Giera, Martin;
    • Sundström, Michael;
    • Berg, Louise
    Publication type:
    Article
    9
    10

    A Potent, Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 3 (PRMT3).

    Published in:
    Angewandte Chemie International Edition, 2015, v. 54, n. 17, p. 5166, doi. 10.1002/anie.201412154
    By:
    • Kaniskan, H. Ümit;
    • Szewczyk, Magdalena M.;
    • Yu, Zhengtian;
    • Eram, Mohammad S.;
    • Yang, Xiaobao;
    • Schmidt, Keith;
    • Luo, Xiao;
    • Dai, Miao;
    • He, Feng;
    • Zang, Irene;
    • Lin, Ying;
    • Kennedy, Steven;
    • Li, Fengling;
    • Dobrovetsky, Elena;
    • Dong, Aiping;
    • Smil, David;
    • Min, Sun‐Joon;
    • Landon, Melissa;
    • Lin‐Jones, Jennifer;
    • Huang, Xi‐Ping
    Publication type:
    Article