Works by Jean-Michel Chezal

Results: 28

99mTc-NTP 15-5 Imaging for Cartilage Involvement in Experimental Rheumatoid Arthritis: Comparison with Routinely Used Molecular Imaging Methods and Sensitivity to Chronic Nonsteroidal Antiinflammatory Drug Treatment.

Published in:

Journal of Nuclear Medicine, 2015, v. 56, n. 5, p. 798, doi. 10.2967/jnumed.114.151415

By:

Khairnar, Amit;
Marchand, Fabien;
Vidal, Aurélien;
Etienne, Monique;
Miladi, Imen;
Auzeloux, Philippe;
Cachin, Florent;
Eschalier, Alain;
Chezal, Jean-Michel;
Ardid, Denis;
Miot-Noirault, Elisabeth

Publication type:

Article

First Preclinical Imaging of Primary Cartilage Neoplasm and Its Local Recurrence Using 99mTc-NTP 15-5 Radiotracer.

Published in:

Journal of Nuclear Medicine, 2009, v. 50, n. 9, p. 1541, doi. 10.2967/jnumed.108.056721

By:

Miot-Noirault, Elisabeth;
Gouin, François;
Vidal, Aurélien;
Rapp, Maryse;
Maublant, Jean;
Askienazy, Serge;
Chezal, Jean-Michel;
Heymann, Dominique;
Redini, Françoise;
Moins, Nicole

Publication type:

Article

Annexin A1 in primary tumors promotes melanoma dissemination.

Published in:

Clinical & Experimental Metastasis, 2014, v. 31, n. 7, p. 749, doi. 10.1007/s10585-014-9665-2

By:

Boudhraa, Zied;
Rondepierre, Fabien;
Ouchchane, Lemlih;
Kintossou, Roselyne;
Trzeciakiewicz, Anna;
Franck, Frederic;
Kanitakis, Jean;
Labeille, Bruno;
Joubert-Zakeyh, Juliette;
Bouchon, Bernadette;
Perrot, Jean;
Mansard, Sandrine;
Papon, Janine;
Dechelotte, Pierre;
Chezal, Jean-Michel;
Miot-Noirault, Elisabeth;
Bonnet, Mathilde;
D'Incan, Michel;
Degoul, Françoise

Publication type:

Article

A Convenient Route to New (Radio)Fluorinated and (Radio)Iodinated Cyclic Tyrosine Analogs.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 2, p. 162, doi. 10.3390/ph15020162

By:

Chao, Maria Noelia;
Chezal, Jean-Michel;
Debiton, Eric;
Canitrot, Damien;
Witkowski, Tiffany;
Levesque, Sophie;
Degoul, Françoise;
Tarrit, Sébastien;
Wenzel, Barbara;
Miot-Noirault, Elisabeth;
Serre, Audrey;
Maisonial-Besset, Aurélie

Publication type:

Article

Development of a New Radiofluorinated Quinoline Analog for PET Imaging of Phosphodiesterase 5 (PDE5) in Brain.

Published in:

Pharmaceuticals (14248247), 2016, v. 9, n. 2, p. 22, doi. 10.3390/ph9020022

By:

Jianrong Liu;
Wenzel, Barbara;
Dukic-Stefanovic, Sladjana;
Teodoro, Rodrigo;
Ludwig, Friedrich-Alexander;
Deuther-Conrad, Winnie;
Schröder, Susann;
Chezal, Jean-Michel;
Moreau, Emmanuel;
Brust, Peter;
Maisonial-Besset, Aurélie

Publication type:

Article

Doxycycline and its quaternary ammonium derivative for adjuvant therapies of chondrosarcoma.

Published in:

2017

By:

Miladi, Imen;
Vivier, Magali;
Dauplat, Marie-Mélanie;
Chatard, Morgane;
Besse, Sophie;
Vidal, Aurélien;
Chassain, Karine;
Jean, Betty;
Forestier, Christiane;
Chezal, Jean-Michel;
Rédini, Francoise;
Degoul, Francoise;
Miot-Noirault, Elisabeth;
Dauplat, Marie-Mélanie;
Vidal, Aurélien;
Rédini, Francoise

Publication type:

journal article

Radiation dosimetry of [131I]ICF01012 in rabbits: Application to targeted radionuclide therapy for human melanoma treatment.

Published in:

Medical Physics, 2018, v. 45, n. 11, p. 5251, doi. 10.1002/mp.13165

By:

Jouberton, Elodie;
Perrot, Yann;
Dirat, Béatrice;
Billoux, Tommy;
Auzeloux, Philippe;
Cachin, Florent;
Chezal, Jean‐Michel;
Filaire, Marc;
Labarre, Pierre;
Miot‐Noirault, Elisabeth;
Millardet, Corinne;
Valla, Clémence;
Vidal, Aurélien;
Degoul, Françoise;
Maigne, Lydia

Publication type:

Article

Phase I study of [131I] ICF01012, a targeted radionuclide therapy, in metastatic melanoma: MELRIV-1 protocol.

Published in:

2022

By:

Thivat, Emilie;
Rouanet, Jacques;
Auzeloux, Philippe;
Sas, Nicolas;
Jouberton, Elodie;
Levesque, Sophie;
Billoux, Tommy;
Mansard, Sandrine;
Molnar, Ioana;
Chanchou, Marion;
Fois, Giovanna;
Maigne, Lydia;
Chezal, Jean-Michel;
Miot-Noirault, Elisabeth;
D'Incan, Michel;
Durando, Xavier;
Cachin, Florent

Publication type:

journal article

Early detection and longitudinal monitoring of experimental primary and disseminated melanoma using [F]ICF01006, a highly promising melanoma PET tracer.

Published in:

European Journal of Nuclear Medicine & Molecular Imaging, 2012, v. 39, n. 9, p. 1449, doi. 10.1007/s00259-012-2168-y

By:

Rbah-Vidal, Latifa;
Vidal, Aurélien;
Besse, Sophie;
Cachin, Florent;
Bonnet, Mathilde;
Audin, Laurent;
Askienazy, Serge;
Dollé, Frédéric;
Degoul, Françoise;
Miot-Noirault, Elisabeth;
Moins, Nicole;
Auzeloux, Philippe;
Chezal, Jean-Michel

Publication type:

Article

Improved automated one-pot two-step radiosynthesis of (S)-[18F]FETrp, a radiotracer for PET imaging of indoleamine 2,3-dioxygenase 1 (IDO1).

Published in:

EJNMMI Radiopharmacy & Chemistry, 2024, v. 9, n. 1, p. 1, doi. 10.1186/s41181-024-00256-0

By:

Maisonial-Besset, Aurélie;
Kryza, David;
Kopka, Klaus;
Levesque, Sophie;
Moreau, Emmanuel;
Wenzel, Barbara;
Chezal, Jean-Michel

Publication type:

Article

Development and characterization of a human three-dimensional chondrosarcoma culture for in vitro drug testing.

Published in:

PLoS ONE, 2017, v. 12, n. 7, p. 1, doi. 10.1371/journal.pone.0181340

By:

Voissiere, Aurélien;
Jouberton, Elodie;
Maubert, Elise;
Degoul, Françoise;
Peyrode, Caroline;
Chezal, Jean-Michel;
Miot-Noirault, Élisabeth

Publication type:

Article

First ex vivo study demonstrating that Tc-NTP 15-5 radiotracer binds to human articular cartilage.

Published in:

European Journal of Nuclear Medicine & Molecular Imaging, 2011, v. 38, n. 11, p. 2077, doi. 10.1007/s00259-011-1890-1

By:

Cachin, Florent;
Boisgard, Stéphane;
Vidal, Aurélien;
Filaire, Marc;
Auzeloux, Philippe;
Culot, Damien;
Askienazy, Serge;
Madelmont, Jean-Claude;
Chezal, Jean-Michel;
Miot-Noirault, Elisabeth

Publication type:

Article

From netrin‐1‐targeted SPECT/CT to internal radiotherapy for management of advanced solid tumors.

Published in:

EMBO Molecular Medicine, 2023, v. 15, n. 4, p. 1, doi. 10.15252/emmm.202216732

By:

Kryza, David;
Wischhusen, Jennifer;
Richaud, Mathieu;
Hervieu, Maëva;
Sidi Boumedine, Jacqueline;
Delcros, Jean‐Guy;
Besse, Sophie;
Baudier, Thomas;
Laval, Pierre‐Alexandre;
Breusa, Silvia;
Boutault, Erwan;
Clermidy, Hugo;
Rama, Nicolas;
Ducarouge, Benjamin;
Devouassoux‐Shisheboran, Mojgan;
Chezal, Jean‐Michel;
Giraudet, Anne‐Laure;
Walter, Thomas;
Mehlen, Patrick;
Sarrut, David

Publication type:

Article

Relevance of the combination of external beam radiotherapy with the hypoxia-activated prodrug ICF05016 in an experimental model of extraskeletal myxoid chondrosarcoma.

Published in:

Investigational New Drugs, 2021, v. 39, n. 2, p. 295, doi. 10.1007/s10637-020-01002-4

By:

Maubert, Elise;
Weber, Valérie;
Voissière, Aurélien;
Gérard, Yvain;
Dedieu, Véronique;
Degoul, Françoise;
Chezal, Jean-Michel;
Chautard, Emmanuel;
Miot-Noirault, Elisabeth

Publication type:

Article

Evaluation of two I-radiolabeled acridine derivatives for Auger-electron radionuclide therapy of melanoma.

Published in:

Investigational New Drugs, 2014, v. 32, n. 4, p. 587, doi. 10.1007/s10637-014-0086-5

By:

Gardette, Maryline;
Viallard, Claire;
Paillas, Salomé;
Guerquin-Kern, Jean-Luc;
Papon, Janine;
Moins, Nicole;
Labarre, Pierre;
Desbois, Nicolas;
Wong-Wah-Chung, Pascal;
Palle, Sabine;
Wu, Ting-Di;
Pouget, Jean-Pierre;
Miot-Noirault, Elisabeth;
Chezal, Jean-Michel;
Degoul, Francoise

Publication type:

Article

Evaluation of new iodinated acridine derivatives for targeted radionuclide therapy of melanoma using (125)I, an Auger electron emitter.

Published in:

2011

By:

Gardette, Maryline;
Papon, Janine;
Bonnet, Mathilde;
Desbois, Nicolas;
Labarre, Pierre;
Wu, Ting-Dee;
Miot-Noirault, Elisabeth;
Madelmont, Jean-Claude;
Guerquin-Kern, Jean-Luc;
Chezal, Jean-Michel;
Moins, Nicole

Publication type:

Journal Article

Evaluation of new iodinated acridine derivatives for targeted radionuclide therapy of melanoma using I, an Auger electron emitter.

Published in:

Investigational New Drugs, 2011, v. 29, n. 6, p. 1253, doi. 10.1007/s10637-010-9471-x

By:

Gardette, Maryline;
Papon, Janine;
Bonnet, Mathilde;
Desbois, Nicolas;
Labarre, Pierre;
Wu, Ting-Dee;
Miot-Noirault, Elisabeth;
Madelmont, Jean-Claude;
Guerquin-Kern, Jean-Luc;
Chezal, Jean-Michel;
Moins, Nicole

Publication type:

Article

Preclinical investigation of tolerance and antitumour activity of new fluorodeoxyglucose-coupled chlorambucil alkylating agents.

Published in:

Investigational New Drugs, 2011, v. 29, n. 3, p. 424, doi. 10.1007/s10637-009-9371-0

By:

Miot-Noirault, Elisabeth;
Reux, Bastien;
Debiton, Eric;
Madelmont, Jean-Claude;
Chezal, Jean-Michel;
Coudert, Pascal;
Weber, Valérie

Publication type:

Article

New compounds from the essential oil of Vetiveria nigritana roots from Mali.

Published in:

Flavour & Fragrance Journal, 2007, v. 22, n. 6, p. 488, doi. 10.1002/ffj.1828

By:

Champagnat, Pascal;
Bessière, Jean-Marie;
Chezal, Jean-Michel;
Chalchat, Jean-Claude;
Carnat, André-Paul

Publication type:

Article

In vivo efficacy of melanoma internal radionuclide therapy with a 131I-labelled melanin-targeting heteroarylcarboxamide molecule.

Published in:

International Journal of Cancer, 2013, v. 133, n. 5, p. 1042, doi. 10.1002/ijc.28103

By:

Degoul, Françoise;
Borel, Michèle;
Jacquemot, Nathalie;
Besse, Sophie;
Communal, Yves;
Mishellany, Florence;
Papon, Janine;
Penault‐Llorca, Frédérique;
Donnarieix, Denise;
Doly, Michel;
Maigne, Lydia;
Miot‐Noirault, Elisabeth;
Cayre, Anne;
Cluzel, Jacques;
Moins, Nicole;
Chezal, Jean‐Michel;
Bonnet, Mathilde

Publication type:

Article

Targeted radionuclide therapy of melanoma: Anti-tumoural efficacy studies of a new.

Published in:

International Journal of Cancer, 2009, v. 125, n. 3, p. 708, doi. 10.1002/ijc.24413

By:

Bonnet-Duquennoy, Mathilde;
Papon, Janine;
Mishellany, Florence;
Labarre, Pierre;
Guerquin-Kern, Jean-Luc;
Wu, Ting-Di;
Gardette, Maryline;
Maublant, Jean;
Penault-Llorca, Frédérique;
Miot-Noirault, Elisabeth;
Cayre, Anne;
Madelmont, Jean-Claude;
Chezal, Jean-Michel;
Moins, Nicole

Publication type:

Article

Base/Cryptand/Metal‐Free Automated Nucleophilic Radiofluorination of [18F]FDOPA from Iodonium Salts: Importance of Hydrogen Carbonate Counterion.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 48, p. 7058, doi. 10.1002/ejoc.201801608

By:

Maisonial‐Besset, Aurélie;
Serre, Audrey;
Ouadi, Ali;
Schmitt, Sébastien;
Canitrot, Damien;
Léal, Fernand;
Miot‐Noirault, Elisabeth;
Brasse, David;
Marchand, Patrice;
Chezal, Jean‐Michel

Publication type:

Article

[18F]ML-10 PET imaging fails to assess early response to neoadjuvant chemotherapy in a preclinical model of triple negative breast cancer.

Published in:

EJNMMI Research, 2020, v. 10, n. 1, p. 1, doi. 10.1186/s13550-019-0587-5

By:

Jouberton, Elodie;
Schmitt, Sébastien;
Chautard, Emmanuel;
Maisonial-Besset, Aurélie;
Roy, Marie;
Radosevic-Robin, Nina;
Chezal, Jean-Michel;
Miot-Noirault, Elisabeth;
Bouvet, Yann;
Cachin, Florent

Publication type:

Article

PHOTOCHEMISTRY OF POLYHALOGENATED HETEROCYCLIC ENAMINONES: COMPETITION BETWEEN CYCLIZATION AND DEHALOGENATION.

Published in:

Heterocyclic Communications, 2003, v. 9, n. 2, p. 189

By:

Aragon, Pierre-Jean;
Chezal, Jean-Michel;
Chavignon, Olivier;
Teulade, Jean-Claude;
Chapat, Jean-Pierre;
Blache, Yves

Publication type:

Article

CONVERSION OF IMIDAZO[1,2-a]PYRIDINES INTO PYRIDO[1,2-e]PURINES.

Published in:

Heterocyclic Communications, 1996, v. 2, n. 3, p. 241

By:

Gueiffier, Alain;
Chavignon, Olivier;
Mavel, Sylvie;
Chezal, Jean-Michel;
Teulade, Jean-Claude;
Blache, Yves;
Chapat, Jean-Pierre

Publication type:

Article

In Vitro and in Vivo Antimalarial Activity of Derivatives of 1,10-Phenanthroline Framework.

Published in:

Archiv der Pharmazie, 2006, v. 339, n. 4, p. 201, doi. 10.1002/ardp.200500246

By:

Ange-Désiré Yapi;
Alexis Valentin;
Jean-Michel Chezal;
Olivier Chavignon;
Bernard Chaillot;
Roseline Gerhardt;
Jean-Claude Teulade

Publication type:

Article

Synthesis and In Vitro Comparison of DOTA, NODAGA and 15-5 Macrocycles as Chelators for the 64 Cu-Labelling of Immunoconjugates.

Published in:

Molecules, 2023, v. 28, n. 1, p. 75, doi. 10.3390/molecules28010075

By:

Maisonial-Besset, Aurélie;
Witkowski, Tiffany;
Quintana, Mercedes;
Besse, Sophie;
Gaumet, Vincent;
Cordonnier, Axel;
Alliot, Cyrille;
Vidal, Aurélien;
Denevault-Sabourin, Caroline;
Tarrit, Sébastien;
Levesque, Sophie;
Miot-Noirault, Elisabeth;
Chezal, Jean-Michel

Publication type:

Article

Novel Radioiodinated and Radiofluorinated Analogues of FT-2102 for SPECT or PET Imaging of mIDH1 Mutant Tumours.

Published in:

Molecules, 2022, v. 27, n. 12, p. 3766, doi. 10.3390/molecules27123766

By:

Weber, Valérie;
Arnaud, Lucie;
Dukic-Stefanovic, Sladjana;
Wenzel, Barbara;
Roux, Valérie;
Chezal, Jean-Michel;
Lai, Thu-Hang;
Teodoro, Rodrigo;
Kopka, Klaus;
Miot-Noirault, Elisabeth;
Deuther-Conrad, Winnie;
Maisonial-Besset, Aurélie

Publication type:

Article

Works by Jean-Michel Chezal

<sup>99m</sup>Tc-NTP 15-5 Imaging for Cartilage Involvement in Experimental Rheumatoid Arthritis: Comparison with Routinely Used Molecular Imaging Methods and Sensitivity to Chronic Nonsteroidal Antiinflammatory Drug Treatment.

First Preclinical Imaging of Primary Cartilage Neoplasm and Its Local Recurrence Using <sup>99m</sup>Tc-NTP 15-5 Radiotracer.

Annexin A1 in primary tumors promotes melanoma dissemination.

A Convenient Route to New (Radio)Fluorinated and (Radio)Iodinated Cyclic Tyrosine Analogs.

Development of a New Radiofluorinated Quinoline Analog for PET Imaging of Phosphodiesterase 5 (PDE5) in Brain.

Doxycycline and its quaternary ammonium derivative for adjuvant therapies of chondrosarcoma.

Radiation dosimetry of [<sup>131</sup>I]ICF01012 in rabbits: Application to targeted radionuclide therapy for human melanoma treatment.

Phase I study of [<sup>131</sup>I] ICF01012, a targeted radionuclide therapy, in metastatic melanoma: MELRIV-1 protocol.

Early detection and longitudinal monitoring of experimental primary and disseminated melanoma using [F]ICF01006, a highly promising melanoma PET tracer.

Improved automated one-pot two-step radiosynthesis of (S)-[<sup>18</sup>F]FETrp, a radiotracer for PET imaging of indoleamine 2,3-dioxygenase 1 (IDO1).

Development and characterization of a human three-dimensional chondrosarcoma culture for in vitro drug testing.

First ex vivo study demonstrating that Tc-NTP 15-5 radiotracer binds to human articular cartilage.

From netrin‐1‐targeted SPECT/CT to internal radiotherapy for management of advanced solid tumors.

Relevance of the combination of external beam radiotherapy with the hypoxia-activated prodrug ICF05016 in an experimental model of extraskeletal myxoid chondrosarcoma.

Evaluation of two I-radiolabeled acridine derivatives for Auger-electron radionuclide therapy of melanoma.

Evaluation of new iodinated acridine derivatives for targeted radionuclide therapy of melanoma using (125)I, an Auger electron emitter.

Evaluation of new iodinated acridine derivatives for targeted radionuclide therapy of melanoma using I, an Auger electron emitter.

Preclinical investigation of tolerance and antitumour activity of new fluorodeoxyglucose-coupled chlorambucil alkylating agents.

New compounds from the essential oil of Vetiveria nigritana roots from Mali.

In vivo efficacy of melanoma internal radionuclide therapy with a <sup>131</sup>I-labelled melanin-targeting heteroarylcarboxamide molecule.

Targeted radionuclide therapy of melanoma: Anti-tumoural efficacy studies of a new.

Base/Cryptand/Metal‐Free Automated Nucleophilic Radiofluorination of [<sup>18</sup>F]FDOPA from Iodonium Salts: Importance of Hydrogen Carbonate Counterion.

[18F]ML-10 PET imaging fails to assess early response to neoadjuvant chemotherapy in a preclinical model of triple negative breast cancer.

PHOTOCHEMISTRY OF POLYHALOGENATED HETEROCYCLIC ENAMINONES: COMPETITION BETWEEN CYCLIZATION AND DEHALOGENATION.

CONVERSION OF IMIDAZO[1,2-a]PYRIDINES INTO PYRIDO[1,2-e]PURINES.

In Vitro and in Vivo Antimalarial Activity of Derivatives of 1,10-Phenanthroline Framework.

Synthesis and In Vitro Comparison of DOTA, NODAGA and 15-5 Macrocycles as Chelators for the 64 Cu-Labelling of Immunoconjugates.

Novel Radioiodinated and Radiofluorinated Analogues of FT-2102 for SPECT or PET Imaging of mIDH1 Mutant Tumours.