Works matching AU Ibrahim, Tarek S.
Results: 49
Development of certain benzylidene coumarin derivatives as anti-prostate cancer agents targeting EGFR and PI3Kβ kinases.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2311157
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- Article
Design, synthesis and antitumor evaluation of novel pyrazolo[3,4-d]pyrimidines incorporating different amino acid conjugates as potential DHFR inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 203, doi. 10.1080/14756366.2022.2142786
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- Article
Novel Sunifiram-carbamate hybrids as potential dual acetylcholinesterase inhibitor and NMDAR co-agonist: simulation-guided analogue design and pharmacological screening.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1241, doi. 10.1080/14756366.2022.2068147
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- Article
Novel chalcone/aryl carboximidamide hybrids as potent anti-inflammatory via inhibition of prostaglandin E2 and inducible NO synthase activities: design, synthesis, molecular docking studies and ADMET prediction.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1067, doi. 10.1080/14756366.2021.1929201
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- Article
Discovery of novel quinoline-based analogues of combretastatin A-4 as tubulin polymerisation inhibitors with apoptosis inducing activity and potent anticancer effect.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 802, doi. 10.1080/14756366.2021.1899168
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- Article
Synergistic Benefits: Exploring the Anti-Virulence Effects of Metformin/Vildagliptin Antidiabetic Combination against Pseudomonas aeruginosa via Controlling Quorum Sensing Systems.
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- Biomedicines, 2023, v. 11, n. 5, p. 1442, doi. 10.3390/biomedicines11051442
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- Article
Anti-Quorum Sensing Activities of Gliptins against Pseudomonas aeruginosa and Staphylococcus aureus.
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- Biomedicines, 2022, v. 10, n. 5, p. 1169, doi. 10.3390/biomedicines10051169
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- Article
Redirecting pantoprazole as a metallo-beta-lactamase inhibitor in carbapenem-resistant Klebsiella pneumoniae.
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- Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1366459
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- Article
Efficient synthesis of N-acylbenzotriazoles using tosyl chloride: en route to suberoylanilide hydroxamic acid (SAHA).
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- ARKIVOC: Online Journal of Organic Chemistry, 2016, p. 161, doi. 10.3998/ark.5550190.p009.459
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- Article
Efficient Synthesis and Computational Studies of Useful Guanylating Agents: 1H‐Benzotriazole‐1‐carboximidamides.
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- ChemistrySelect, 2020, v. 5, n. 44, p. 13963, doi. 10.1002/slct.202003796
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- Article
Hiring of the Anti-Quorum Sensing Activities of Hypoglycemic Agent Linagliptin to Alleviate the Pseudomonas aeruginosa Pathogenesis.
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- Microorganisms, 2022, v. 10, n. 12, p. 2455, doi. 10.3390/microorganisms10122455
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- Article
Silencing of Salmonella typhimurium Pathogenesis: Atenolol Acquires Efficient Anti-Virulence Activities.
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- Microorganisms, 2022, v. 10, n. 10, p. 1976, doi. 10.3390/microorganisms10101976
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- Article
Sodium Citrate Alleviates Virulence in Pseudomonas aeruginosa.
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- Microorganisms, 2022, v. 10, n. 5, p. 1046, doi. 10.3390/microorganisms10051046
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- Article
Alteration of Salmonella enterica Virulence and Host Pathogenesis through Targeting sdiA by Using the CRISPR-Cas9 System.
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- Microorganisms, 2021, v. 9, n. 12, p. 2564, doi. 10.3390/microorganisms9122564
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- Article
Xylitol Inhibits Growth and Blocks Virulence in Serratia marcescens.
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- Microorganisms, 2021, v. 9, n. 5, p. 1083, doi. 10.3390/microorganisms9051083
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Repurposing Anti-diabetic Drugs to Cripple Quorum Sensing in Pseudomonas aeruginosa.
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- Microorganisms, 2020, v. 8, n. 9, p. 1285, doi. 10.3390/microorganisms8091285
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- Article
Muting Bacterial Communication: Evaluation of Prazosin Anti-Quorum Sensing Activities against Gram-Negative Bacteria Pseudomonas aeruginosa , Proteus mirabilis , and Serratia marcescens.
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- Biology (2079-7737), 2022, v. 11, n. 9, p. 1349, doi. 10.3390/biology11091349
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- Article
Thymoquinone is a natural antibiofilm and pathogenicity attenuating agent in Pseudomonas aeruginosa.
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- Frontiers in Cellular & Infection Microbiology, 2024, p. 1, doi. 10.3389/fcimb.2024.1382289
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- Article
Benzotriazole-Mediated Synthesis and Antibacterial Activity of Novel N-Acylcephalexins.
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- Scientia Pharmaceutica, 2016, v. 84, n. 3, p. 484, doi. 10.3390/scipharm84030484
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Design, synthesis, antimicrobial, and DNA gyrase inhibitory properties of fluoroquinolone–dichloroacetic acid hybrids.
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- Chemical Biology & Drug Design, 2020, v. 95, n. 2, p. 248, doi. 10.1111/cbdd.13638
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Synthesis and Antiviral Bioassay of New Diphenyl Ether-based Compounds.
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- Chemical Biology & Drug Design, 2016, v. 88, n. 4, p. 511, doi. 10.1111/cbdd.12775
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- Article
Cysteinoyl- and Cysteine-containing Dipeptidoylbenzotriazoles with Free Sulfhydryl Groups: Easy Access to N-terminal and Internal Cysteine Peptides.
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- Chemical Biology & Drug Design, 2012, v. 80, n. 2, p. 194, doi. 10.1111/j.1747-0285.2011.01303.x
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- Article
Elevated Levels of IL-33, IL-17 and IL-25 Indicate the Progression from Chronicity to Hepatocellular Carcinoma in Hepatitis C Virus Patients.
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- Pathogens, 2022, v. 11, n. 1, p. 57, doi. 10.3390/pathogens11010057
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- Article
Tailored Tetrasubstituted Imidazole Carrying the Benzenesulfonamide Fragments as Selective Human Carbonic Anhydrase IX/XII Inhibitors.
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- ChemMedChem, 2024, v. 19, n. 10, p. 1, doi. 10.1002/cmdc.202400004
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- Article
Development of Isatin‐Based Schiff Bases Targeting VEGFR‐2 Inhibition: Synthesis, Characterization, Antiproliferative Properties, and QSAR Studies.
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- ChemMedChem, 2022, v. 17, n. 13, p. 1, doi. 10.1002/cmdc.202200164
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- Article
Characterization of the Anti-Biofilm and Anti-Quorum Sensing Activities of the β-Adrenoreceptor Antagonist Atenolol against Gram-Negative Bacterial Pathogens.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 21, p. 13088, doi. 10.3390/ijms232113088
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- Article
Synthesis of Potential Antiviral Agents for SARS-CoV-2 Using Molecular Hybridization Approach.
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- Molecules, 2022, v. 27, n. 18, p. 5923, doi. 10.3390/molecules27185923
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- Article
Synthesis, Antimicrobial, Anti-Virulence and Anticancer Evaluation of New 5(4 H)-Oxazolone-Based Sulfonamides.
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- Molecules, 2022, v. 27, n. 3, p. 671, doi. 10.3390/molecules27030671
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- Article
Antioxidant Property of the Egyptian Propolis Extract Versus Aluminum Silicate Intoxication on a Rat's Lung: Histopathological Studies.
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- Molecules, 2020, v. 25, n. 24, p. 5821, doi. 10.3390/molecules25245821
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- Article
In Vitro Antimycobacterial Activity and Physicochemical Characterization of Diaryl Ether Triclosan Analogues as Potential InhA Reductase Inhibitors.
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- Molecules, 2020, v. 25, n. 14, p. 3125, doi. 10.3390/molecules25143125
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- Article
An Efficient Greener Approach for N-acylation of Amines in Water Using Benzotriazole Chemistry.
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- Molecules, 2020, v. 25, n. 11, p. 2501, doi. 10.3390/molecules25112501
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- Article
RETRACTED: Awan et al. The Enhanced Cytotoxic and Pro-Apoptotic Effects of Optimized Simvastatin-Loaded Emulsomes on MCF-7 Breast Cancer Cells. Pharmaceutics 2020, 12 , 597.
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- 2024
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- Correction Notice
Development of Carvedilol-Loaded Albumin-Based Nanoparticles with Factorial Design to Optimize In Vitro and In Vivo Performance.
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- Pharmaceutics, 2023, v. 15, n. 5, p. 1425, doi. 10.3390/pharmaceutics15051425
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Repurposing of Sitagliptin- Melittin Optimized Nanoformula against SARS-CoV-2; Antiviral Screening and Molecular Docking Studies.
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- Pharmaceutics, 2021, v. 13, n. 3, p. 307, doi. 10.3390/pharmaceutics13030307
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- Article
The Enhanced Cytotoxic and Pro-Apoptotic Effects of Optimized Simvastatin-Loaded Emulsomes on MCF-7 Breast Cancer Cells.
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- Pharmaceutics, 2020, v. 12, n. 7, p. 597, doi. 10.3390/pharmaceutics12070597
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- Article
Uracil as a Zn-Binding Bioisostere of the Allergic Benzenesulfonamide in the Design of Quinoline–Uracil Hybrids as Anticancer Carbonic Anhydrase Inhibitors.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 5, p. 494, doi. 10.3390/ph15050494
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- Article
Synthesis, Antibacterial Evaluation, and Computational Studies of a Diverse Set of Linezolid Conjugates.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 2, p. 191, doi. 10.3390/ph15020191
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- Article
Computational and Biological Evaluation of β -Adrenoreceptor Blockers as Promising Bacterial Anti-Virulence Agents.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 2, p. 110, doi. 10.3390/ph15020110
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- Article
Design, Synthesis, In Vitro Anticancer Evaluation and Molecular Modelling Studies of 3,4,5-Trimethoxyphenyl-Based Derivatives as Dual EGFR/HDAC Hybrid Inhibitors.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 11, p. 1177, doi. 10.3390/ph14111177
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- Article
New Multi-Targeted Antiproliferative Agents: Design and Synthesis of IC261-Based Oxindoles as Potential Tubulin, CK1 and EGFR Inhibitors.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 11, p. 1114, doi. 10.3390/ph14111114
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- Article
Evaluation of the Antiviral Activity of Sitagliptin-Glatiramer Acetate Nano-Conjugates against SARS-CoV-2 Virus.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 3, p. 178, doi. 10.3390/ph14030178
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- Article
Potent Quinoline-Containing Combretastatin A-4 Analogues: Design, Synthesis, Antiproliferative, and Anti-Tubulin Activity.
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- Pharmaceuticals (14248247), 2020, v. 13, n. 11, p. 393, doi. 10.3390/ph13110393
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- Article
The Anticancer Activity for the Bumetanide-Based Analogs via Targeting the Tumor-Associated Membrane-Bound Human Carbonic Anhydrase-IX Enzyme.
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- Pharmaceuticals (14248247), 2020, v. 13, n. 9, p. 252, doi. 10.3390/ph13090252
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- Article
Not Only Antimicrobial: Metronidazole Mitigates the Virulence of Proteus mirabilis Isolated from Macerated Diabetic Foot Ulcer.
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- Applied Sciences (2076-3417), 2021, v. 11, n. 15, p. 6847, doi. 10.3390/app11156847
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Celastrol boosts fluconazole efficacy against vaginal candidiasis: in vitro and in vivo evidence.
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- AMB Express, 2025, v. 15, n. 1, p. 1, doi. 10.1186/s13568-025-01824-6
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Cilostazol is a promising anti-pseudomonal virulence drug by disruption of quorum sensing.
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- AMB Express, 2024, v. 14, n. 1, p. 1, doi. 10.1186/s13568-024-01740-1
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- Article
Drug repositioning: doxazosin attenuates the virulence factors and biofilm formation in Gram-negative bacteria.
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- Applied Microbiology & Biotechnology, 2023, v. 107, n. 11, p. 3763, doi. 10.1007/s00253-023-12522-3
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- Article
Repurposing α -Adrenoreceptor Blockers as Promising Anti-Virulence Agents in Gram-Negative Bacteria.
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- Antibiotics (2079-6382), 2022, v. 11, n. 2, p. 178, doi. 10.3390/antibiotics11020178
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- Article
Green and catalyst-free synthesis of olsalazine analogs.
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- Green Chemistry Letters & Reviews, 2016, v. 9, n. 2, p. 91, doi. 10.1080/17518253.2016.1163421
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- Article