Works by Holota, Yuliia


Results: 10
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    2

    Integrated workflow for the identification of new GABA<sub>A</sub>R positive allosteric modulators based on the in silico screening with further in vitro validation. Case study using Enamine's stock chemical space.

    Published in:
    Molecular Informatics, 2024, v. 43, n. 2, p. 1, doi. 10.1002/minf.202300156
    By:
    • Platonov, Maksym;
    • Maximyuk, Oleksandr;
    • Rayevsky, Alexey;
    • Iegorova, Olena;
    • Hurmach, Vasyl;
    • Holota, Yuliia;
    • Bulgakov, Elijah;
    • Cherninskyi, Andrii;
    • Karpov, Pavel;
    • Ryabukhin, Sergey;
    • Krishtal, Oleg;
    • Volochnyuk, Dmitriy
    Publication type:
    Article
    3

    Front Cover: 3,3‐Difluorooxetane–A Versatile Functional Group for Bioisosteric Replacements in Drug Discovery (Chem. Eur. J. 72/2024).

    Published in:
    Chemistry - A European Journal, 2024, v. 30, n. 72, p. 1, doi. 10.1002/chem.202487201
    By:
    • Liashuk, Oleksandr S.;
    • Fedinchyk, Anastasiya;
    • Melnykov, Kostiantyn P.;
    • Herasymchuk, Maksym;
    • Alieksieieva, Diana;
    • Lesyk, Dmytro;
    • Bas, Yuliia P.;
    • Keda, Tetiana Ye.;
    • Yatsymyrskiy, Andriy V.;
    • Holota, Yuliia;
    • Borysko, Petro;
    • Yarmolchuk, Volodymyr S.;
    • Grygorenko, Oleksandr O.
    Publication type:
    Article
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    7

    "Angular" Spirocyclic Azetidines: Synthesis, Characterization, and Evaluation in Drug Discovery.

    Published in:
    Angewandte Chemie, 2025, v. 137, n. 7, p. 1, doi. 10.1002/ange.202418850
    By:
    • Kirichok, Alexander A.;
    • Tkachuk, Hennadii;
    • Levchenko, Kostiantyn;
    • Granat, Dmitry;
    • Yegorova, Tetyana;
    • Lesyk, Dmytro;
    • Anisiforova, Anna;
    • Holota, Yuliia;
    • Zomchak, Viktoriia;
    • Bodenchuk, Iryna;
    • Kosach, Viktoriia;
    • Borysko, Petro;
    • Korzh, Rodion A.;
    • Al‐Maali, Galeb;
    • Kubyshkin, Vladimir;
    • Rzepa, Henry S.;
    • Mykhailiuk, Pavel K.
    Publication type:
    Article
    8
    9

    2-Oxabicyclo[2.2.2]octane as a new bioisostere of the phenyl ring.

    Published in:
    Nature Communications, 2023, v. 14, n. 1, p. 1, doi. 10.1038/s41467-023-41298-3
    By:
    • Levterov, Vadym V.;
    • Panasiuk, Yaroslav;
    • Sahun, Kateryna;
    • Stashkevych, Oleksandr;
    • Badlo, Valentyn;
    • Shablykin, Oleh;
    • Sadkova, Iryna;
    • Bortnichuk, Lina;
    • Klymenko-Ulianov, Oleksii;
    • Holota, Yuliia;
    • Lachmann, Leonid;
    • Borysko, Petro;
    • Horbatok, Kateryna;
    • Bodenchuk, Iryna;
    • Bas, Yuliia;
    • Dudenko, Dmytro;
    • Mykhailiuk, Pavel K.
    Publication type:
    Article
    10

    "Angular" Spirocyclic Azetidines: Synthesis, Characterization, and Evaluation in Drug Discovery.

    Published in:
    Angewandte Chemie International Edition, 2025, v. 64, n. 7, p. 1, doi. 10.1002/anie.202418850
    By:
    • Kirichok, Alexander A.;
    • Tkachuk, Hennadii;
    • Levchenko, Kostiantyn;
    • Granat, Dmitry;
    • Yegorova, Tetyana;
    • Lesyk, Dmytro;
    • Anisiforova, Anna;
    • Holota, Yuliia;
    • Zomchak, Viktoriia;
    • Bodenchuk, Iryna;
    • Kosach, Viktoriia;
    • Borysko, Petro;
    • Korzh, Rodion A.;
    • Al‐Maali, Galeb;
    • Kubyshkin, Vladimir;
    • Rzepa, Henry S.;
    • Mykhailiuk, Pavel K.
    Publication type:
    Article