Works by Guillaumet, Gérald

Results: 59

Design and validation of the first cell-impermeant melatonin receptor agonist.

Published in:

2017

By:

Gbahou, Florence;
Cecon, Erika;
Viault, Guillaume;
Gerbier, Romain;
Jean ‐ Alphonse, Frederic;
Karamitri, Angeliki;
Guillaumet, Gérald;
Delagrange, Philippe;
Friedlander, Robert M;
Vilardaga, Jean ‐ Pierre;
Suzenet, Franck;
Jockers, Ralf;
Jean-Alphonse, Frederic;
Guillaumet, Gérald;
Vilardaga, Jean-Pierre

Publication type:

journal article

Ecofriendly synthesis of 3-cyanopyridine derivatives by multi-component reaction catalyzed by animal bone meal.

Published in:

Environmental Chemistry Letters, 2014, v. 12, n. 4, p. 523, doi. 10.1007/s10311-014-0478-y

By:

Riadi, Yassine;
Mamouni, Rachid;
Routier, Sylvain;
Guillaumet, Gérald;
Lazar, Saïd

Publication type:

Article

2H‐1,5‐Benzodioxepin und 3‐Halogen‐Derivate.

Published in:

Angewandte Chemie, 1983, v. 95, n. 1, p. 50, doi. 10.1002/ange.19830950112

By:

Guillaumet, Gérald;
Coudert, Gérard;
Loubinoux, Bernard

Publication type:

Article

Regioselective C6‐Arylation of Thieno[3,2‐c]pyrazole Heterocycles with Aryl Iodides.

Published in:

Advanced Synthesis & Catalysis, 2024, v. 366, n. 12, p. 2749, doi. 10.1002/adsc.202400141

By:

Ait Lfakir, Noura;
Jismy, Badr;
Guillaumet, Gérald;
Akssira, Mohamed;
El Hakmaoui, Ahmed;
Guillot, Régis;
Tikad, Abdellatif;
Abarbri, Mohamed

Publication type:

Article

Front Cover Picture: Palladium‐Catalyzed Regioselective C−H Arylation of 4‐Azaindazole at C3, C5 and C7 Positions (Adv. Synth. Catal. 16/2021).

Published in:

Advanced Synthesis & Catalysis, 2021, v. 363, n. 16, p. 3867, doi. 10.1002/adsc.202100859

By:

Faarasse, Soukaina;
El Kazzouli, Saïd;
Bourzikat, Otmane;
Bourg, Stéphane;
Aci‐Sèche, Samia;
Bonnet, Pascal;
Suzenet, Franck;
Guillaumet, Gérald

Publication type:

Article

Palladium‐Catalyzed Regioselective C−H Arylation of 4‐Azaindazole at C3, C5 and C7 Positions.

Published in:

Advanced Synthesis & Catalysis, 2021, v. 363, n. 16, p. 3937, doi. 10.1002/adsc.202001421

By:

Faarasse, Soukaina;
El Kazzouli, Saïd;
Bourzikat, Otmane;
Bourg, Stéphane;
Aci‐Sèche, Samia;
Bonnet, Pascal;
Suzenet, Franck;
Guillaumet, Gérald

Publication type:

Article

Synthesis and Functionalization of Imidazo[1,2‐b]Pyridazine by Means of Metal‐Catalyzed Cross‐Coupling Reactions.

Published in:

ChemistrySelect, 2021, v. 6, n. 34, p. 8985, doi. 10.1002/slct.202101636

By:

El Akkaoui, Ahmed;
Koubachi, Jamal;
Guillaumet, Gérald;
El Kazzouli, Saïd

Publication type:

Article

New Radioligands for Describing the Molecular Pharmacology of MT1 and MT2 Melatonin Receptors.

Published in:

International Journal of Molecular Sciences, 2013, v. 14, n. 5, p. 8948, doi. 10.3390/ijms14058948

By:

Legros, Céline;
Matthey, Ulrich;
Grelak, Teresa;
Pedragona-Moreau, Sandrine;
Hassler, Werner;
Yous, Saïd;
Thomas, Emmanuel;
Suzenet, Franck;
Folleas, Benoît;
Lefoulon, François;
Berthelot, Pascal;
Caignard, Daniel-Henri;
Guillaumet, Gérald;
Delagrange, Philippe;
Brayer, Jean-Louis;
Nosjean, Olivier;
Boutin, Jean A.

Publication type:

Article

1H, 13C and 15N NMR spectral assignments for new triazapentalene derivatives.

Published in:

Magnetic Resonance in Chemistry, 2009, v. 47, n. 9, p. 752, doi. 10.1002/mrc.2458

By:

Palmas, Pascal;
Nyffenegger, Coralie;
Pasquinet, Eric;
Guillaumet, Gérald

Publication type:

Article

New selective ligands of human cloned melatonin MT1 and MT2 receptors.

Published in:

Naunyn-Schmiedeberg's Archives of Pharmacology, 2003, v. 367, n. 6, p. 553, doi. 10.1007/s00210-003-0751-2

By:

Audinot, Valérie;
Mailliet, François;
Lahaye-Brasseur, Chantal;
Bonnaud, Anne;
Le Gall, Aude;
Amossé, Christophe;
Dromaint, Sandra;
Rodriguez, Marianne;
Nagel, Nadine;
Galizzi, Jean-Pierre;
xEE;t#Malpaux, Beno&;
Guillaumet, Gérald;
Lesieur, Daniel;
Lefoulon, François;
Renard, Pierre;
Delagrange, Philippe;
Boutin, Jean A.

Publication type:

Article

CYTOTOXIC EVALUATION OF ORIGINAL PYRAZOLO[3,4-d]THIAZOLES AND PYRAZOLO[3,4-c]PYRAZOLES.

Published in:

Farmacia, 2022, v. 70, n. 2, p. 258, doi. 10.31925/farmacia.2022.2.10

By:

OSTACHE, NICU-COSMIN;
PARIS, ARNAUD;
HIEBEL, MARIE-AUDE;
FÎNARU, ADRIANALUMINIȚA;
DANIELLOU, RICHARD;
SUZENET, FRANCK;
GUILLAUMET, GÉRALD

Publication type:

Article

Concise and Efficient Access to 5,7-Disubstituted Pyrazolo[1,5-a]pyrimidines by Pd-Catalyzed Sequential Arylation, Alkynylation and SNArReaction.

Published in:

European Journal of Organic Chemistry, 2017, v. 2017, n. 41, p. 6168, doi. 10.1002/ejoc.201701024

By:

Jismy, Badr;
Guillaumet, Gérald;
Allouchi, Hassan;
Akssira, Mohamed;
Abarbri, Mohamed

Publication type:

Article

Regioselective Synthesis of 2,4-Substituted Pyrido[1′,2′:1,5]pyrazolo[3,4- d]pyrimidines through Sequential Pd-Catalyzed Arylation and SNAr Reactions.

Published in:

European Journal of Organic Chemistry, 2016, v. 2016, n. 21, p. 3550, doi. 10.1002/ejoc.201600356

By:

Belaroussi, Rabia;
El Hakmaoui, Ahmed;
Akssira, Mohamed;
Guillaumet, Gérald;
Routier, Sylvain

Publication type:

Article

A Strategy for the Triarylation of Pyrrolopyrimidines by Using Microwave-Promoted Cross-Coupling Reactions.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 29, p. 6547, doi. 10.1002/ejoc.201500625

By:

Prieur, Vanessa;
Pujol, M. Dolors;
Guillaumet, Gérald

Publication type:

Article

Synthesis of 1,4-Disubstituted Pyrido[1′,2′:1,5]pyrazolo[3,4- d]pyridazines by Means of SNAr and Palladium-Catalysed Reactions.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 18, p. 4006, doi. 10.1002/ejoc.201500294

By:

Belaroussi, Rabia;
El Hakmaoui, Ahmed;
Percina, Nathalie;
Chartier, Agnes;
Marchivie, Mathieu;
Massip, Stéphane;
Jarry, Christian;
Akssira, Mohamed;
Guillaumet, Gérald;
Routier, Sylvain

Publication type:

Article

Suzuki-Miyaura Reactions of Halospirooxindole Derivatives.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 16, p. 3450, doi. 10.1002/ejoc.201500268

By:

El Bouakher, Abderrahman;
Allouchi, Hassan;
Abrunhosa‐Thomas, Isabelle;
Troin, Yves;
Guillaumet, Gérald

Publication type:

Article

A General and Efficient Method to Access Tetracyclic Spirooxindole Derivatives.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 3, p. 556, doi. 10.1002/ejoc.201403292

By:

El Bouakher, Abderrahman;
Massip, Stéphane;
Jarry, Christian;
Troin, Yves;
Abrunhosa‐Thomas, Isabelle;
Guillaumet, Gérald

Publication type:

Article

First Palladium-Catalyzed Direct Regioselective C-5 (Het)Arylation of Mono- or Disubstituted Thiazolo[3,2- b][1,2,4]triazoles.

Published in:

European Journal of Organic Chemistry, 2014, v. 2014, n. 17, p. 3704, doi. 10.1002/ejoc.201402193

By:

Le Meur, Mikaël;
Bourg, Stéphane;
Massip, Stéphane;
Marchivie, Mathieu;
Jarry, Christian;
Guillaumet, Gérald;
Routier, Sylvain

Publication type:

Article

Sulfur-Carbon Bond Formation through Ring-Opening of Triazolothiadiazole with Organometallics.

Published in:

European Journal of Organic Chemistry, 2014, v. 2014, n. 15, p. 3225, doi. 10.1002/ejoc.201400151

By:

Othman, Raja Ben;
Massip, Stéphane;
Marchivie, Mathieu;
Jarry, Christian;
Vercouillie, Johnny;
Chalon, Sylvie;
Guillaumet, Gérald;
Suzenet, Franck;
Routier, Sylvain

Publication type:

Article

Microwave-Assisted Synthesis of Substituted Pyrrolo[2,3- d]pyrimidines.

Published in:

European Journal of Organic Chemistry, 2014, v. 2014, n. 7, p. 1514, doi. 10.1002/ejoc.201301496

By:

Prieur, Vanessa;
Rubio‐Martínez, Jaime;
Font‐Bardia, Mercè;
Guillaumet, Gérald;
Pujol, M. Dolors

Publication type:

Article

Access to Imidazo[1,2- a]imidazolin-2-ones and Functionalization through Suzuki-Miyaura Cross-Coupling Reactions.

Published in:

European Journal of Organic Chemistry, 2013, v. 2013, n. 19, p. 4146, doi. 10.1002/ejoc.201300268

By:

Grosse, Sandrine;
Pillard, Christelle;
Himbert, Franck;
Massip, Stéphane;
Léger, Jean Michel;
Jarry, Christian;
Bernard, Philippe;
Guillaumet, Gérald

Publication type:

Article

Extending the Scope of the Aza-Fischer Synthesis of 4- and 6-Azaindoles.

Published in:

European Journal of Organic Chemistry, 2013, v. 2013, n. 16, p. 3328, doi. 10.1002/ejoc.201300167

By:

Thomae, David;
Jeanty, Matthieu;
Coste, Jérome;
Guillaumet, Gérald;
Suzenet, Franck

Publication type:

Article

Direct C-3-Arylations of 1 H-Indazoles.

Published in:

European Journal of Organic Chemistry, 2012, v. 2012, n. 36, p. 7075, doi. 10.1002/ejoc.201200860

By:

Ben-Yahia, Ali;
Naas, Mohammed;
El Kazzouli, Saïd;
Essassi, El Mokhtar;
Guillaumet, Gérald

Publication type:

Article

Regiocontroled SNAr and Palladium Cross-Coupling Reactions of 2,4,7-Trichloropyrido[3,2- d]pyrimidine.

Published in:

European Journal of Organic Chemistry, 2012, v. 2012, n. 24, p. 4523, doi. 10.1002/ejoc.201200521

By:

Tikad, Abdellatif;
Akssira, Mohamed;
Massip, Stéphane;
Léger, Jean-Michel;
Jarry, Christian;
Guillaumet, Gérald;
Routier, Sylvain

Publication type:

Article

Catalyst- and Base-Controlled Site-Selective sp2 and sp3 Direct Arylation of 5,7-Dimethyl-2-phenylpyrazolo[1,5- a]pyrimidine Using Aryl Bromides.

Published in:

European Journal of Organic Chemistry, 2012, v. 2012, n. 13, p. 2572, doi. 10.1002/ejoc.201101833

By:

Bassoude, Ibtissam;
Berteina-Raboin, Sabine;
Massip, Stéphane;
Leger, Jean-Michel;
Jarry, Christian;
Essassi, El Mokhtar;
Guillaumet, Gérald

Publication type:

Article

Influence of an Alkoxy Group on Bis-Triazinyl-Pyridines for Selective Extraction of Americium(III).

Published in:

Solvent Extraction & Ion Exchange, 2013, v. 31, n. 3, p. 253, doi. 10.1080/07366299.2012.757160

By:

Dupont, Carine;
Hill, Clément;
Suzenet, Franck;
Guillaumet, Gérald

Publication type:

Article

Insight on spectral, thermal and biological behaviour of some Cu(II) complexes with saturated pentaazamacrocyclic ligands bearing amino acid residues.

Published in:

Journal of Thermal Analysis & Calorimetry, 2021, v. 143, n. 1, p. 173, doi. 10.1007/s10973-020-09259-w

By:

Pătraşcu, Elena;
Badea, Mihaela;
Čelan Korošin, Nataša;
Cerc Korošec, Romana;
Ruţă, Lavinia L.;
Farcaşanu, Ileana C.;
Grecu, Maria Nicoleta;
Guillaumet, Gérald;
Olar, Rodica

Publication type:

Article

Synthesis of new pyrazolo[3,4-b]pyridin-3-ones and pyrazolo[1,5-a]pyrimidin-2(1H)-one and study of the pyrazolic nitrogen reactivity.

Published in:

ARKIVOC: Online Journal of Organic Chemistry, 2011, p. 240

By:

Fadel, Salah;
Hamri, Salha;
Hajbi, Youssef;
Suzenet, Franck;
Hafid, Abderrafia;
Rakib, El-Mostapha;
Khouili, Mostafa;
Pujol, Maria D.;
Guillaumet, Gérald

Publication type:

Article

Synthesis of aminopyrrolo[1,2-a]thieno[3,2-e]pyrazine derivatives as serotoninergic 5-HT7 ligands.

Published in:

ARKIVOC: Online Journal of Organic Chemistry, 2010, p. 116

By:

Pavé, Grégoire;
Lazar, Saïd;
Lesnard, Aurélien;
Rault, Sylvain;
Guillaumet, Gérald

Publication type:

Article

Intramolecular Metal‐Free N−N Bond Formation with Heteroaromatic Amines: Mild Access to Fused‐Triazapentalene Derivatives.

Published in:

Chemistry - A European Journal, 2020, v. 26, n. 7, p. 1525, doi. 10.1002/chem.201905558

By:

Daniel, Matthieu;
Hiebel, Marie‐Aude;
Guillaumet, Gérald;
Pasquinet, Eric;
Suzenet, Franck

Publication type:

Article

Advances in the Synthesis and Biological Applications of Enoxacin-Based Compounds.

Published in:

Biomolecules (2218-273X), 2024, v. 14, n. 11, p. 1419, doi. 10.3390/biom14111419

By:

Suleiman, Garba;
El Brahmi, Nabil;
Guillaumet, Gérald;
El Kazzouli, Saïd

Publication type:

Article

Palladium‐Catalyzed Regioselective C−H Oxidative Arylation of 7‐Azaindazole N‐Oxide at the C6‐Position.

Published in:

European Journal of Organic Chemistry, 2023, v. 26, n. 45, p. 1, doi. 10.1002/ejoc.202300730

By:

Nassiri, Sarah;
Bousmina, Mostapha;
Suzenet, Franck;
Guillaumet, Gérald;
El Kazzouli, Saïd

Publication type:

Article

Palladium‐Catalyzed Oxidative Arylation of 1H‐Indazoles with Arenes.

Published in:

European Journal of Organic Chemistry, 2020, v. 2020, n. 48, p. 7435, doi. 10.1002/ejoc.202001313

By:

Gambouz, Khadija;
Abbouchi, Abdelmoula El;
Nassiri, Sarah;
Suzenet, Franck;
Bousmina, Mostapha;
Akssira, Mohamed;
Guillaumet, Gérald;
El Kazzouli, Saïd

Publication type:

Article

Oxidative Alkenylation of Fused Bicyclic Heterocycles.

Published in:

European Journal of Organic Chemistry, 2019, v. 2019, n. 15, p. 2568, doi. 10.1002/ejoc.201900199

By:

Koubachi, Jamal;
El Brahmi, Nabil;
Guillaumet, Gérald;
El Kazzouli, Saïd

Publication type:

Article

Attempted synthesis of ethyl 3,4-dihydro-2 H-1,4-benzoxazine-3-carboxylate and 3-acetate derivatives.

Published in:

Journal of Heterocyclic Chemistry, 2001, v. 38, n. 1, p. 221, doi. 10.1002/jhet.5570380133

By:

Mayer, Stanislas;
Arrault, Axelle;
Guillaumet, GÉRald;
Mérour, Jean-Yves

Publication type:

Article

A straightforward route to 4 H-1,4-Benzoxazine-2-carbaldehydes by swern oxidation.

Published in:

Journal of Heterocyclic Chemistry, 1996, v. 33, n. 1, p. 191, doi. 10.1002/jhet.5570330133

By:

Bourlot, Anne-Sophie;
Guillaumet, Gérald;
Mérour, Jean-Yves

Publication type:

Article

Synthèse de dioxinocoumarines angulaires.

Published in:

Journal of Heterocyclic Chemistry, 1989, v. 26, n. 1, p. 193, doi. 10.1002/jhet.5570260134

By:

Guillaumet, Gérald;
Hretani, Mohamed;
Coudert, Gérard

Publication type:

Article

Benzodioxines-1,4 disubstituées en position 2,3 par des groupements pharmacophores.

Published in:

Journal of Heterocyclic Chemistry, 1987, v. 24, n. 3, p. 609, doi. 10.1002/jhet.5570240313

By:

Coudert, Gérard;
Borredon-Watrin, Corinne;
Guillaumet, Gérald

Publication type:

Article

Efficient Metal-Free Synthesis of Various Pyrido[2′,1′:2,3]imidazo- [4,5- b]quinolines.

Published in:

Chemistry - A European Journal, 2013, v. 19, n. 37, p. 12249, doi. 10.1002/chem.201300961

By:

Arnould, Mathieu;
Hiebel, Marie‐Aude;
Massip, Stéphane;
Léger, Jean Michel;
Jarry, Christian;
Berteina‐Raboin, Sabine;
Guillaumet, Gérald

Publication type:

Article

Efficient Synthesis and First Regioselective C-3 Direct Arylation of Imidazo[1,2- b]pyrazoles.

Published in:

Chemistry - A European Journal, 2012, v. 18, n. 47, p. 14943, doi. 10.1002/chem.201202593

By:

Grosse, Sandrine;
Pillard, Christelle;
Massip, Stéphane;
Léger, Jean Michel;
Jarry, Christian;
Bourg, Stéphane;
Bernard, Philippe;
Guillaumet, Gérald

Publication type:

Article

Design, Synthesis, and Evaluation of EA-Sulfonamides and Indazole-Sulfonamides as Promising Anticancer Agents: Molecular Docking, ADME Prediction, and Molecular Dynamics Simulations.

Published in:

Chemistry (2624-8549), 2024, v. 6, n. 6, p. 1396, doi. 10.3390/chemistry6060083

By:

Saghdani, Nassima;
El Brahmi, Nabil;
El Abbouchi, Abdelmoula;
Haloui, Rachid;
Elkhattabi, Souad;
Guillaumet, Gérald;
El Kazzouli, Saïd

Publication type:

Article

Palladium‐Catalyzed Site‐Selective C7 Oxidative Arylation of 4‐EWG‐1H‐Indazoles.

Published in:

Asian Journal of Organic Chemistry, 2023, v. 12, n. 8, p. 1, doi. 10.1002/ajoc.202300285

By:

Ouazzani Chahdi, Chaimae;
Boujdi, Khalid;
El Brahmi, Nabil;
Mathé‐Allainmat, Monique;
Mouhi Eddine, Hachim;
Akssira, Mohamed;
Guillaumet, Gérald;
Lebreton, Jacques;
Koubachi, Jamal;
El Kazzouli, Saïd

Publication type:

Article

2 H-1,5-Benzodioxepin and 3-Halo Derivatives.

Published in:

Angewandte Chemie International Edition, 1983, v. 22, n. 1, p. 64, doi. 10.1002/anie.198300641

By:

Guillaumet, Gérald;
Coudert, Gérard;
Loubinoux, Bernard

Publication type:

Article

Synthesis of 3-Substituted Pyrrolo[2,3- b ]Pyridin-2-one Derivatives.

Published in:

Synthetic Communications, 1997, v. 27, n. 22, p. 3861, doi. 10.1080/00397919708005909

By:

Marie-Claude, Viaud;
Patricia, Jamoneau;
Gérald, Guillaumet

Publication type:

Article

New Direct Synthesis of 3-Nitro-2H-chromenes Using Nitroethylene.

Published in:

Synthetic Communications, 1990, v. 20, n. 6, p. 783, doi. 10.1080/00397919008052323

By:

Neirabeyeh, Mamdouh Ai;
Koussini, Rafik;
Guillaumet, Gérald

Publication type:

Article

A Novel, Unequivocal Synthesis of Polyethylene Glycols.

Published in:

Synthetic Communications, 1986, v. 16, n. 1, p. 19, doi. 10.1080/00397918608057683

By:

Coudert, GÉRard;
Mpassi, Michel;
Guillaumet, GÉRald;
Selve, Claude

Publication type:

Article

New insights into homopiperazine-based 5-HT1A/5-HT7R ligands: synthesis and biological evaluation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2010, v. 25, n. 3, p. 301, doi. 10.3109/14756360903179393

By:

Badarau, Eduard;
Putey, Aurélien;
Suzenet, Franck;
Joseph, Benoit;
Bojarski, Andrzej;
Finaru, Adriana;
Guillaumet, Gérald

Publication type:

Article

Synthesis and Cytotoxic Evaluation of Novel Thiazolocarbazoles. Part II1.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2003, v. 18, n. 2, p. 167, doi. 10.1080/1475636032000069837

By:

Chabane, Hadjila;
Lamazzi, Christelle;
Thiery, Valerie;
Pierre, Alain;
Leonce, Stephane;
Pfeiffer, Bruno;
Renard, Pierre;
Guillaumet, Gérald;
Besson, Thierry

Publication type:

Article

Synthesis of 5-Substituted-2,3-dihydro-1,4-benzoxathiins: Biological Evaluation as Melatonin Receptors Ligands.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2003, v. 18, n. 2, p. 187, doi. 10.1080/1475636032000096855

By:

Charton, Isabelle;
Suzenet, Franck;
Boutin, Jean A.;
Audinot, Valérie;
Delagrange, Philippe;
Bennejean, Caroline;
Renard, Pierre;
Guillaumet, Gérald

Publication type:

Article

Copper‐Assisted Synthesis of Novel Pyrazolo[3,4‐d]thiazoles.

Published in:

ChemCatChem, 2019, v. 11, n. 15, p. 3530, doi. 10.1002/cctc.201900707

By:

Ostache, Nicu‐Cosmin;
Hiebel, Marie‐Aude;
Fînaru, Adriana‐Luminiţa;
Guillaumet, Gérald;
Suzenet, Franck

Publication type:

Article