Works by Guillaumet, Gérald
Results: 58
Design and validation of the first cell-impermeant melatonin receptor agonist.
- Published in:
- 2017
- By:
- Publication type:
- journal article
New insights into homopiperazine-based 5-HT<sub>1A</sub>/5-HT<sub>7</sub>R ligands: synthesis and biological evaluation.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2010, v. 25, n. 3, p. 301, doi. 10.3109/14756360903179393
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- Publication type:
- Article
Synthesis and Cytotoxic Evaluation of Novel Thiazolocarbazoles. Part II1.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2003, v. 18, n. 2, p. 167, doi. 10.1080/1475636032000069837
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- Publication type:
- Article
Synthesis of 5-Substituted-2,3-dihydro-1,4-benzoxathiins: Biological Evaluation as Melatonin Receptors Ligands.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2003, v. 18, n. 2, p. 187, doi. 10.1080/1475636032000096855
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- Publication type:
- Article
Advances in the Synthesis and Biological Applications of Enoxacin-Based Compounds.
- Published in:
- Biomolecules (2218-273X), 2024, v. 14, n. 11, p. 1419, doi. 10.3390/biom14111419
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- Publication type:
- Article
<sup>1</sup>H, <sup>13</sup>C and <sup>15</sup>N NMR spectral assignments for new triazapentalene derivatives.
- Published in:
- Magnetic Resonance in Chemistry, 2009, v. 47, n. 9, p. 752, doi. 10.1002/mrc.2458
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- Publication type:
- Article
Palladium‐Catalyzed Site‐Selective C7 Oxidative Arylation of 4‐EWG‐1H‐Indazoles.
- Published in:
- Asian Journal of Organic Chemistry, 2023, v. 12, n. 8, p. 1, doi. 10.1002/ajoc.202300285
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- Publication type:
- Article
Palladium‐Catalyzed Regioselective C−H Oxidative Arylation of 7‐Azaindazole N‐Oxide at the C6‐Position.
- Published in:
- European Journal of Organic Chemistry, 2023, v. 26, n. 45, p. 1, doi. 10.1002/ejoc.202300730
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- Publication type:
- Article
Synthesis of new pyrazolo[3,4-b]pyridin-3-ones and pyrazolo[1,5-a]pyrimidin-2(1H)-one and study of the pyrazolic nitrogen reactivity.
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- ARKIVOC: Online Journal of Organic Chemistry, 2011, p. 240
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- Publication type:
- Article
Synthesis of aminopyrrolo[1,2-a]thieno[3,2-e]pyrazine derivatives as serotoninergic 5-HT<sub>7</sub> ligands.
- Published in:
- ARKIVOC: Online Journal of Organic Chemistry, 2010, p. 116
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- Publication type:
- Article
Insight on spectral, thermal and biological behaviour of some Cu(II) complexes with saturated pentaazamacrocyclic ligands bearing amino acid residues.
- Published in:
- Journal of Thermal Analysis & Calorimetry, 2021, v. 143, n. 1, p. 173, doi. 10.1007/s10973-020-09259-w
- By:
- Publication type:
- Article
New selective ligands of human cloned melatonin MT<sub>1</sub> and MT<sub>2</sub> receptors.
- Published in:
- Naunyn-Schmiedeberg's Archives of Pharmacology, 2003, v. 367, n. 6, p. 553, doi. 10.1007/s00210-003-0751-2
- By:
- Publication type:
- Article
Synthesis and Functionalization of Imidazo[1,2‐b]Pyridazine by Means of Metal‐Catalyzed Cross‐Coupling Reactions.
- Published in:
- ChemistrySelect, 2021, v. 6, n. 34, p. 8985, doi. 10.1002/slct.202101636
- By:
- Publication type:
- Article
Copper‐Assisted Synthesis of Novel Pyrazolo[3,4‐d]thiazoles.
- Published in:
- ChemCatChem, 2019, v. 11, n. 15, p. 3530, doi. 10.1002/cctc.201900707
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- Publication type:
- Article
Comparison of sulfobutylether- and sulfated-β-cyclodextrins as additives for the chiral separation of basic spirobenzopyrans by capillary electrophoresis.
- Published in:
- Electrophoresis, 1999, v. 20, n. 13, p. 2630, doi. 10.1002/(SICI)1522-2683(19990901)20:13<2630::AID-ELPS2630>3.0.CO;2-9
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- Publication type:
- Article
Design, Synthesis, and Evaluation of EA-Sulfonamides and Indazole-Sulfonamides as Promising Anticancer Agents: Molecular Docking, ADME Prediction, and Molecular Dynamics Simulations.
- Published in:
- Chemistry (2624-8549), 2024, v. 6, n. 6, p. 1396, doi. 10.3390/chemistry6060083
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- Publication type:
- Article
CYTOTOXIC EVALUATION OF ORIGINAL PYRAZOLO[3,4-d]THIAZOLES AND PYRAZOLO[3,4-c]PYRAZOLES.
- Published in:
- Farmacia, 2022, v. 70, n. 2, p. 258, doi. 10.31925/farmacia.2022.2.10
- By:
- Publication type:
- Article
Palladium‐Catalyzed Oxidative Arylation of 1H‐Indazoles with Arenes.
- Published in:
- European Journal of Organic Chemistry, 2020, v. 2020, n. 48, p. 7435, doi. 10.1002/ejoc.202001313
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- Publication type:
- Article
Oxidative Alkenylation of Fused Bicyclic Heterocycles.
- Published in:
- European Journal of Organic Chemistry, 2019, v. 2019, n. 15, p. 2568, doi. 10.1002/ejoc.201900199
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- Publication type:
- Article
Concise and Efficient Access to 5,7-Disubstituted Pyrazolo[1,5-a]pyrimidines by Pd-Catalyzed Sequential Arylation, Alkynylation and SN<sub>Ar</sub>Reaction.
- Published in:
- European Journal of Organic Chemistry, 2017, v. 2017, n. 41, p. 6168, doi. 10.1002/ejoc.201701024
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- Publication type:
- Article
Regioselective Synthesis of 2,4-Substituted Pyrido[1′,2′:1,5]pyrazolo[3,4- d]pyrimidines through Sequential Pd-Catalyzed Arylation and S<sub>N</sub>Ar Reactions.
- Published in:
- European Journal of Organic Chemistry, 2016, v. 2016, n. 21, p. 3550, doi. 10.1002/ejoc.201600356
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- Publication type:
- Article
New Radioligands for Describing the Molecular Pharmacology of MT<sub>1</sub> and MT<sub>2</sub> Melatonin Receptors.
- Published in:
- International Journal of Molecular Sciences, 2013, v. 14, n. 5, p. 8948, doi. 10.3390/ijms14058948
- By:
- Publication type:
- Article
Ecofriendly synthesis of 3-cyanopyridine derivatives by multi-component reaction catalyzed by animal bone meal.
- Published in:
- Environmental Chemistry Letters, 2014, v. 12, n. 4, p. 523, doi. 10.1007/s10311-014-0478-y
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- Publication type:
- Article
Design, Synthesis, Computational Studies, and Anti-Proliferative Evaluation of Novel Ethacrynic Acid Derivatives Containing Nitrogen Heterocycle, Urea, and Thiourea Moieties as Anticancer Agents.
- Published in:
- Molecules, 2024, v. 29, n. 7, p. 1437, doi. 10.3390/molecules29071437
- By:
- Publication type:
- Article
Improvement of the Chemical Reactivity of Michael Acceptor of Ethacrynic Acid Correlates with Antiproliferative Activities.
- Published in:
- Molecules, 2023, v. 28, n. 2, p. 910, doi. 10.3390/molecules28020910
- By:
- Publication type:
- Article
Synthesis, Anticancer Activities and Molecular Docking Studies of a Novel Class of 2-Phenyl-5,6,7,8-tetrahydroimidazo [1,2- b ]pyridazine Derivatives Bearing Sulfonamides.
- Published in:
- Molecules, 2022, v. 27, n. 16, p. 5238, doi. 10.3390/molecules27165238
- By:
- Publication type:
- Article
Regioselective C-H Functionalization of the Six-Membered Ring of the 6,5-Fused Heterocyclic Systems: An Overview.
- Published in:
- Molecules, 2021, v. 26, n. 19, p. 5763, doi. 10.3390/molecules26195763
- By:
- Publication type:
- Article
"On Water" Palladium Catalyzed Direct Arylation of 1H-Indazole and 1H-7-Azaindazole.
- Published in:
- Molecules, 2020, v. 25, n. 12, p. 2820, doi. 10.3390/molecules25122820
- By:
- Publication type:
- Article
Efficient Access to 3,5-Disubstituted 7-(Trifluoromethyl)pyrazolo[1,5-a]pyrimidines Involving SNAr and Suzuki Cross-Coupling Reactions.
- Published in:
- Molecules, 2020, v. 25, n. 9, p. 2062, doi. 10.3390/molecules25092062
- By:
- Publication type:
- Article
Regioselective Synthesis of New 2,4-(Het)aryl-3H-pyrido[1′,2′:1,5]pyrazolo[4,3-d]pyrimidines Involving Palladium-Catalyzed Cross-Coupling Reactions.
- Published in:
- Molecules, 2018, v. 23, n. 11, p. 2740, doi. 10.3390/molecules23112740
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- Publication type:
- Article
2 H-1,5-Benzodioxepin and 3-Halo Derivatives.
- Published in:
- Angewandte Chemie International Edition, 1983, v. 22, n. 1, p. 64, doi. 10.1002/anie.198300641
- By:
- Publication type:
- Article
Intramolecular Metal‐Free N−N Bond Formation with Heteroaromatic Amines: Mild Access to Fused‐Triazapentalene Derivatives.
- Published in:
- Chemistry - A European Journal, 2020, v. 26, n. 7, p. 1525, doi. 10.1002/chem.201905558
- By:
- Publication type:
- Article
Synthesis of 3-Substituted Pyrrolo[2,3- b ]Pyridin-2-one Derivatives.
- Published in:
- Synthetic Communications, 1997, v. 27, n. 22, p. 3861, doi. 10.1080/00397919708005909
- By:
- Publication type:
- Article
New Direct Synthesis of 3-Nitro-2H-chromenes Using Nitroethylene.
- Published in:
- Synthetic Communications, 1990, v. 20, n. 6, p. 783, doi. 10.1080/00397919008052323
- By:
- Publication type:
- Article
A Novel, Unequivocal Synthesis of Polyethylene Glycols.
- Published in:
- Synthetic Communications, 1986, v. 16, n. 1, p. 19, doi. 10.1080/00397918608057683
- By:
- Publication type:
- Article
Efficient Metal-Free Synthesis of Various Pyrido[2′,1′:2,3]imidazo- [4,5- b]quinolines.
- Published in:
- Chemistry - A European Journal, 2013, v. 19, n. 37, p. 12249, doi. 10.1002/chem.201300961
- By:
- Publication type:
- Article
Efficient Synthesis and First Regioselective C-3 Direct Arylation of Imidazo[1,2- b]pyrazoles.
- Published in:
- Chemistry - A European Journal, 2012, v. 18, n. 47, p. 14943, doi. 10.1002/chem.201202593
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- Publication type:
- Article
New Synthetic Approach to Naphtho[1,2 -b]furan and 4′-Oxo-Substituted Spiro[cyclopropane-1,1′(4′ H)-naphthalene] Derivatives.
- Published in:
- Helvetica Chimica Acta, 2001, v. 84, n. 8, p. 2198, doi. 10.1002/1522-2675(20010815)84:8<2198::AID-HLCA2198>3.0.CO;2-J
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- Publication type:
- Article
Synthèse de dioxinocoumarines angulaires.
- Published in:
- Journal of Heterocyclic Chemistry, 1989, v. 26, n. 1, p. 193, doi. 10.1002/jhet.5570260134
- By:
- Publication type:
- Article
Benzodioxines-1,4 disubstituées en position 2,3 par des groupements pharmacophores.
- Published in:
- Journal of Heterocyclic Chemistry, 1987, v. 24, n. 3, p. 609, doi. 10.1002/jhet.5570240313
- By:
- Publication type:
- Article
2H‐1,5‐Benzodioxepin und 3‐Halogen‐Derivate.
- Published in:
- Angewandte Chemie, 1983, v. 95, n. 1, p. 50, doi. 10.1002/ange.19830950112
- By:
- Publication type:
- Article
Regioselective C6‐Arylation of Thieno[3,2‐c]pyrazole Heterocycles with Aryl Iodides.
- Published in:
- Advanced Synthesis & Catalysis, 2024, v. 366, n. 12, p. 2749, doi. 10.1002/adsc.202400141
- By:
- Publication type:
- Article
Front Cover Picture: Palladium‐Catalyzed Regioselective C−H Arylation of 4‐Azaindazole at C3, C5 and C7 Positions (Adv. Synth. Catal. 16/2021).
- Published in:
- Advanced Synthesis & Catalysis, 2021, v. 363, n. 16, p. 3867, doi. 10.1002/adsc.202100859
- By:
- Publication type:
- Article
Palladium‐Catalyzed Regioselective C−H Arylation of 4‐Azaindazole at C3, C5 and C7 Positions.
- Published in:
- Advanced Synthesis & Catalysis, 2021, v. 363, n. 16, p. 3937, doi. 10.1002/adsc.202001421
- By:
- Publication type:
- Article
A Strategy for the Triarylation of Pyrrolopyrimidines by Using Microwave-Promoted Cross-Coupling Reactions.
- Published in:
- European Journal of Organic Chemistry, 2015, v. 2015, n. 29, p. 6547, doi. 10.1002/ejoc.201500625
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- Publication type:
- Article
Synthesis of 1,4-Disubstituted Pyrido[1′,2′:1,5]pyrazolo[3,4- d]pyridazines by Means of S<sub>N</sub>Ar and Palladium-Catalysed Reactions.
- Published in:
- European Journal of Organic Chemistry, 2015, v. 2015, n. 18, p. 4006, doi. 10.1002/ejoc.201500294
- By:
- Publication type:
- Article
Suzuki-Miyaura Reactions of Halospirooxindole Derivatives.
- Published in:
- European Journal of Organic Chemistry, 2015, v. 2015, n. 16, p. 3450, doi. 10.1002/ejoc.201500268
- By:
- Publication type:
- Article
A General and Efficient Method to Access Tetracyclic Spirooxindole Derivatives.
- Published in:
- European Journal of Organic Chemistry, 2015, v. 2015, n. 3, p. 556, doi. 10.1002/ejoc.201403292
- By:
- Publication type:
- Article
First Palladium-Catalyzed Direct Regioselective C-5 (Het)Arylation of Mono- or Disubstituted Thiazolo[3,2- b][1,2,4]triazoles.
- Published in:
- European Journal of Organic Chemistry, 2014, v. 2014, n. 17, p. 3704, doi. 10.1002/ejoc.201402193
- By:
- Publication type:
- Article
Sulfur-Carbon Bond Formation through Ring-Opening of Triazolothiadiazole with Organometallics.
- Published in:
- European Journal of Organic Chemistry, 2014, v. 2014, n. 15, p. 3225, doi. 10.1002/ejoc.201400151
- By:
- Publication type:
- Article